Page last updated: 2024-08-21

pyridazine and imidazole

pyridazine has been researched along with imidazole in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hayashi, M; Iguchi, Y; Iizuka, K; Kajiwara, I; Kawamura, M; Miyamoto, T; Nakazawa, M; Ohyama, I; Okada, T; Taniguchi, K; Tanouchi, T1
Fotsch, C; St Jean, DJ1
Ashida, Y; Fukuda, S; Gyoten, M; Kamei, T; Kawano, Y; Midoro, K; Nagaya, H1
Andrews, PS; Boezio, AA; Boezio, CM; Bush, TL; Cai, T; Cheng, AC; Choquette, D; Coats, JR; Colletti, AE; Copeland, KW; DuPont, M; Graceffa, R; Grubinska, B; Kim, JL; La, DS; Lewis, RT; Liu, J; Mullady, EL; Peterson, EA; Potashman, MH; Romero, K; Shaffer, PL; Stanton, MK; Stellwagen, JC; Teffera, Y; Yi, S1

Reviews

1 review(s) available for pyridazine and imidazole

ArticleYear
Mitigating heterocycle metabolism in drug discovery.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats

2012

Other Studies

3 other study(ies) available for pyridazine and imidazole

ArticleYear
Highly selective inhibitors of thromboxane synthetase. 2. Pyridine derivatives.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:10

    Topics: Animals; Oxidoreductases; Pyridines; Sheep; Structure-Activity Relationship; Thromboxane-A Synthase

1981
Inhibition of allergic dermal inflammation by the novel imidazopyridazine derivative TAK-427 in a guinea pig experimental model of eczema.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:3

    Topics: Animals; Anti-Allergic Agents; Anti-Inflammatory Agents, Non-Steroidal; Cytokines; Dermatitis, Allergic Contact; Dexamethasone; Disease Models, Animal; Eczema; Female; Guinea Pigs; Histamine H1 Antagonists; Imidazoles; Male; Pyridazines; RNA, Messenger

2002
Discovery and optimization of potent and selective imidazopyridine and imidazopyridazine mTOR inhibitors.
    Bioorganic & medicinal chemistry letters, 2012, Aug-01, Volume: 22, Issue:15

    Topics: Animals; Benzimidazoles; Binding Sites; Binding, Competitive; Crystallography, X-Ray; Drug Design; Drug Evaluation, Preclinical; Half-Life; Humans; Imidazoles; Male; Mice; Microsomes, Liver; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Protein Structure, Tertiary; Pyridazines; Pyridines; Rats, Sprague-Dawley; Signal Transduction; Structure-Activity Relationship; TOR Serine-Threonine Kinases

2012