Page last updated: 2024-08-21

pyridazine and azetidine

pyridazine has been researched along with azetidine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fotsch, C; St Jean, DJ1
Hohman, TC; Malamas, MS1
Brandon, NJ; Bridges, TM; Byers, FW; Chang, S; Cho, HP; Conn, PJ; Duggan, ME; Engers, DW; Jones, CK; Lamsal, A; Lindsley, CW; Luscombe, VB; Melancon, BJ; Niswender, CM; Noetzel, MJ; Rodriguez, AL; Tarr, JC; Wood, MR; Wood, MW1

Reviews

1 review(s) available for pyridazine and azetidine

ArticleYear
Mitigating heterocycle metabolism in drug discovery.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats

2012

Other Studies

2 other study(ies) available for pyridazine and azetidine

ArticleYear
N-substituted spirosuccinimide, spiropyridazine, spiroazetidine, and acetic acid aldose reductase inhibitors derived from isoquinoline-1,3-diones. 2.
    Journal of medicinal chemistry, 1994, Jun-24, Volume: 37, Issue:13

    Topics: Acetates; Acetic Acid; Administration, Oral; Aldehyde Reductase; Animals; Azetidines; Galactosemias; In Vitro Techniques; Isoquinolines; Lens, Crystalline; Magnetic Resonance Spectroscopy; Pyridazines; Rats; Sciatic Nerve; Structure-Activity Relationship; Succinimides

1994
Challenges in the development of an M
    Bioorganic & medicinal chemistry letters, 2017, 12-01, Volume: 27, Issue:23

    Topics: Allosteric Regulation; Amides; Azetidines; Drug Evaluation, Preclinical; Humans; Protein Binding; Pyridazines; Receptor, Muscarinic M4; Structure-Activity Relationship

2017