pyrazole and pyrimidinones

pyrazole has been researched along with pyrimidinones in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Agarwal, JK; Dash, RP; Nivsarkar, M; Pandya, DH; Sagar, SR; Vasu, KK1
Abeywickrema, P; Cabalu, TD; Chen, Y; Crespo, A; Dwyer, MP; Ginetti, AT; Lu, J; Morriello, GJ; Paone, DV; Sinz, C; Stachel, SJ; Wang, D; Wilson, JE; Xu, S1

Other Studies

2 other study(ies) available for pyrazole and pyrimidinones

ArticleYear
Design, synthesis and biological evaluation of novel pyrazolo-pyrimidinones as DPP-IV inhibitors in diabetes.
    Bioorganic & medicinal chemistry letters, 2015, Oct-15, Volume: 25, Issue:20

    Topics: Animals; Blood Glucose; Diabetes Mellitus, Experimental; Dipeptidyl Peptidase 4; Dose-Response Relationship, Drug; Drug Design; Hyperglycemia; Hypoglycemic Agents; Male; Models, Molecular; Molecular Structure; Pyrazoles; Pyrimidinones; Rats; Rats, Wistar; Structure-Activity Relationship

2015
Discovery of novel N-1 substituted pyrazolopyrimidinones as potent, selective PDE2 inhibitors.
    Bioorganic & medicinal chemistry letters, 2021, 07-15, Volume: 44

    Topics: Crystallography, X-Ray; Cyclic Nucleotide Phosphodiesterases, Type 2; Dose-Response Relationship, Drug; Drug Discovery; Humans; Models, Molecular; Molecular Structure; Phosphodiesterase Inhibitors; Pyrazoles; Pyrimidinones; Structure-Activity Relationship

2021