Compounds > pyrazole

pyrazole and piperidine

pyrazole has been researched along with piperidine in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19901 (20.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (60.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Hayashi, M; Iguchi, Y; Iizuka, K; Kajiwara, I; Kawamura, M; Miyamoto, T; Nakazawa, M; Ohyama, I; Okada, T; Taniguchi, K; Tanouchi, T1
Fotsch, C; St Jean, DJ1
Bader, SJ; Bagley, SW; Bernhardson, DJ; Cabral, S; Edmonds, DJ; Griffith, DA; Kung, DW; Polivkova, J; Rose, CR; Southers, JA; Yang, X1
Bonin, PD; Cai, C; Chen, Y; Cornelius, P; DeNinno, MP; Futatsugi, K; Gao, H; Guimarães, CR; Hamilton, MD; Hank, R; Harris, AR; Kalgutkar, AS; Kung, DW; Lavergne, SY; Lefker, BA; Lopaze, MG; Mascitti, V; McClure, KF; Morishita, N; Munchhof, MJ; Preville, C; Robinson, RP; Wright, SW1
Alexander, R; Espiritu, C; Flores, OA; Hartman, GD; Klumpp, K; Kuduk, SD; Lam, AM; Lau, V; Stoops, B; Vogel, R1

Reviews

1 review(s) available for pyrazole and piperidine

ArticleYear
Mitigating heterocycle metabolism in drug discovery.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats

2012

Other Studies

4 other study(ies) available for pyrazole and piperidine

ArticleYear
Highly selective inhibitors of thromboxane synthetase. 2. Pyridine derivatives.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:10

    Topics: Animals; Oxidoreductases; Pyridines; Sheep; Structure-Activity Relationship; Thromboxane-A Synthase

1981
Synthesis of 7-oxo-dihydrospiro[indazole-5,4'-piperidine] acetyl-CoA carboxylase inhibitors.
    The Journal of organic chemistry, 2012, Feb-03, Volume: 77, Issue:3

    Topics: Acetyl-CoA Carboxylase; Alkenes; Alkylation; Chemistry Techniques, Synthetic; Enzyme Inhibitors; Indazoles; Ketones; Piperidines; Pyrazoles; Stereoisomerism; Substrate Specificity

2012
From partial to full agonism: identification of a novel 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole as a full agonist of the human GPR119 receptor.
    Bioorganic & medicinal chemistry letters, 2013, Jan-01, Volume: 23, Issue:1

    Topics: Carbamates; Humans; Piperidines; Protein Binding; Pyrazoles; Receptors, G-Protein-Coupled; Structure-Activity Relationship

2013
Identification of a new class of HBV capsid assembly modulator.
    Bioorganic & medicinal chemistry letters, 2021, 05-01, Volume: 39

    Topics: Antiviral Agents; Capsid Proteins; Dose-Response Relationship, Drug; Hepatitis B virus; Microbial Sensitivity Tests; Molecular Structure; Piperidines; Pyrazoles; Structure-Activity Relationship

2021