pyrazole and oxadiazoles

pyrazole has been researched along with oxadiazoles in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (9.09)29.6817
2010's9 (81.82)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Hamersak, Z; Minidis, AB; Svensson, MA; Vallin, KS; Wensbo Posaric, D1
Gong, ZL; Liu, WY; Lv, HS; Xie, YS; Zhao, BX1
Buridipad, SK; Chikkanna, C; Poojary, B; Puthiyapurayil, P1
Beck, H; Bhargava, A; Boyer, S; Ellinghaus, P; Greschat-Schade, S; Härter, M; Hess-Stumpp, H; Thierauch, KH; Unterschemmann, K1
Appa Rao, C; Krishna Tilak, T; Mallikarjuna Reddy, G; Muralikrishna, A; Padmaja, A; Padmavathi, V1
Bhadraiah, UK; Doddaramappa, SD; Javarasetty, C; Keshavamurthy, S; Ningaiah, S1
Duan, GY; Ge, YQ; Jia, J; Sun, HW; Wang, JW; Wang, T1
Gupta, S; Jain, N; Kamal, A; Krishna, KV; Kumar, GB; Mishra, RK; Nagabhushana, A; Polepalli, S; Reddy, VS; Shaik, AB1
Akhtar, M; Akhtar, W; Alam, MM; Ali, A; Ali, I; Chashoo, G; Khan, MF; Shaquiquzzaman, M; Verma, G1
Gulnaz, AR; Khanum, SA; Mohammed, YHE1
Ganapathi, T; Kamal, A; Khan, I; Kumar, CG; Rehman, MM; Shareef, MA1

Other Studies

11 other study(ies) available for pyrazole and oxadiazoles

ArticleYear
Efficient chemoenzymatic dynamic kinetic resolution of 1-heteroaryl ethanols.
    The Journal of organic chemistry, 2009, Dec-18, Volume: 74, Issue:24

    Topics: Biocatalysis; Enzymes, Immobilized; Ethanol; Fungal Proteins; Heterocyclic Compounds; Hydrogenation; Imidazoles; Isoxazoles; Kinetics; Lipase; Molecular Dynamics Simulation; Oxadiazoles; Pyrazoles; Ruthenium; Stereoisomerism

2009
Synthesis, X-ray crystal structures and optical properties of novel substituted pyrazoly 1,3,4-oxadiazole derivatives.
    Journal of fluorescence, 2011, Volume: 21, Issue:4

    Topics: Crystallography, X-Ray; Fluorescence; Models, Molecular; Molecular Structure; Optical Phenomena; Oxadiazoles; Pyrazoles; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet; Stereoisomerism

2011
Design, synthesis and biological evaluation of a novel series of 1,3,4-oxadiazole bearing N-methyl-4-(trifluoromethyl)phenyl pyrazole moiety as cytotoxic agents.
    European journal of medicinal chemistry, 2012, Volume: 53

    Topics: Antineoplastic Agents; Cell Line, Tumor; Chemistry Techniques, Synthetic; Drug Design; Humans; Inhibitory Concentration 50; Oxadiazoles; Pyrazoles; Time Factors

2012
Inhibition of hypoxia-induced gene transcription by substituted pyrazolyl oxadiazoles: initial lead generation and structure-activity relationships.
    ChemMedChem, 2014, Volume: 9, Issue:1

    Topics: Administration, Oral; Amides; Animals; Cell Hypoxia; Cell Line, Tumor; Cell Survival; Half-Life; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Injections, Intravenous; Oxadiazoles; Pyrazoles; Rats; Structure-Activity Relationship; Transcription, Genetic

2014
Synthesis and antioxidant activity of styrylsulfonylmethyl 1,3,4-oxadiazoles, pyrazolyl/isoxazolyl-1,3,4-oxadiazoles.
    Chemical & pharmaceutical bulletin, 2013, Volume: 61, Issue:12

    Topics: Antioxidants; Biphenyl Compounds; Hydrogen Peroxide; Methylation; Nitric Oxide; Oxadiazoles; Picrates; Pyrazoles; Sulfones

2013
Novel pyrazole integrated 1,3,4-oxadiazoles: synthesis, characterization and antimicrobial evaluation.
    Bioorganic & medicinal chemistry letters, 2014, Jan-01, Volume: 24, Issue:1

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Dose-Response Relationship, Drug; Fungi; Microbial Sensitivity Tests; Molecular Structure; Oxadiazoles; Pyrazoles; Structure-Activity Relationship

2014
The synthesis, characterization and optical properties of novel 5-(3-aryl-1H-pyrazol-5-yl)-2-(3-butyl-1-chloroimidazo[1,5-a]pyridin-7-yl)-1,3,4-oxadiazole.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2014, Apr-05, Volume: 123

    Topics: Crystallography, X-Ray; Halogenation; Magnetic Resonance Spectroscopy; Models, Molecular; Oxadiazoles; Pyrazoles; Pyridines; Spectrometry, Fluorescence; Spectrophotometry, Infrared; Spectrophotometry, Ultraviolet

2014
Pyrazole-oxadiazole conjugates: synthesis, antiproliferative activity and inhibition of tubulin polymerization.
    Organic & biomolecular chemistry, 2014, Oct-28, Volume: 12, Issue:40

    Topics: Animals; Antineoplastic Agents; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; HeLa Cells; Humans; MCF-7 Cells; Models, Molecular; Molecular Structure; Oxadiazoles; Polymerization; Pyrazoles; Structure-Activity Relationship; Tubulin; Zebrafish

2014
Synthesis of pyrazole acrylic acid based oxadiazole and amide derivatives as antimalarial and anticancer agents.
    Bioorganic chemistry, 2018, Volume: 77

    Topics: Acrylates; Amides; Antimalarials; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Molecular Docking Simulation; Molecular Structure; Oxadiazoles; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyrazoles; Structure-Activity Relationship

2018
Design, synthesis and molecular docking of benzophenone conjugated with oxadiazole sulphur bridge pyrazole pharmacophores as anti inflammatory and analgesic agents.
    Bioorganic chemistry, 2019, Volume: 92

    Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzophenones; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Drug Design; Edema; Formaldehyde; Humans; Mice; Molecular Docking Simulation; Molecular Structure; Oxadiazoles; Pain; Pain Measurement; Pyrazoles; Rats; Structure-Activity Relationship

2019
New indenopyrazole linked oxadiazole conjugates as anti-pancreatic cancer agents: Design, synthesis, in silico studies including 3D-QSAR analysis.
    Bioorganic & medicinal chemistry letters, 2021, 07-15, Volume: 44

    Topics: Antineoplastic Agents; Apoptosis; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Humans; Molecular Docking Simulation; Molecular Structure; Oxadiazoles; Pancreatic Neoplasms; Pyrazoles; Quantitative Structure-Activity Relationship

2021