pyrazole and indazoles

pyrazole has been researched along with indazoles in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (28.57)29.6817
2010's4 (57.14)24.3611
2020's1 (14.29)2.80

Authors

AuthorsStudies
Daidone, G; Maggio, B; Plescia, F; Raffa, D; Schillaci, D; Torta, L1
Arion, VB; Büchel, GE; Hejl, M; Jakupec, MA; Keppler, BK; Stepanenko, IN1
Abad, MC; Gibbs, AC; Kuo, GH; Kuo, LC; Song, F; Sui, Z; Sun, W; Xiang, A; Zhang, X1
Cheng, Y; Hu, J; Rao, Y; Yang, Y1
Bader, SJ; Bagley, SW; Bernhardson, DJ; Cabral, S; Edmonds, DJ; Griffith, DA; Kung, DW; Polivkova, J; Rose, CR; Southers, JA; Yang, X1
Huang, J; Jiang, H; Jin, F; Li, C; Li, J; Liu, G; Lu, W; Tang, Y; Wang, W; Wu, D; Zhu, J1
Ghosh, A; Ghosh, D; Ghosh, S; Hajra, A; Majumder, S; Pyne, P1

Reviews

1 review(s) available for pyrazole and indazoles

ArticleYear
Visible light-induced functionalization of indazole and pyrazole: a recent update.
    Chemical communications (Cambridge, England), 2022, Apr-05, Volume: 58, Issue:28

    Topics: Catalysis; Indazoles; Light; Pyrazoles

2022

Other Studies

6 other study(ies) available for pyrazole and indazoles

ArticleYear
Synthesis and antifungal activity of new N-(1-phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides.
    Farmaco (Societa chimica italiana : 1989), 2002, Volume: 57, Issue:3

    Topics: Antifungal Agents; Benzamides; Colony Count, Microbial; Fungi; Indazoles; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Pyrazoles; Spectrophotometry, Infrared

2002
[Os(IV)Cl(5)(Hazole)](-) complexes: synthesis, structure, spectroscopic properties, and antiproliferative activity.
    Inorganic chemistry, 2009, Nov-16, Volume: 48, Issue:22

    Topics: Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Electrochemistry; Humans; Hydrolysis; Indazoles; Magnetic Resonance Spectroscopy; Magnetics; Organometallic Compounds; Osmium; Pyrazoles; Solubility; Water

2009
Optimization of a pyrazole hit from FBDD into a novel series of indazoles as ketohexokinase inhibitors.
    Bioorganic & medicinal chemistry letters, 2011, Aug-15, Volume: 21, Issue:16

    Topics: Crystallography, X-Ray; Dose-Response Relationship, Drug; Drug Discovery; Fructokinases; Indazoles; Models, Molecular; Molecular Structure; Pyrazoles; Stereoisomerism; Structure-Activity Relationship

2011
A general and efficient approach to 2H-indazoles and 1H-pyrazoles through copper-catalyzed intramolecular N-N bond formation under mild conditions.
    Chemical communications (Cambridge, England), 2011, Sep-28, Volume: 47, Issue:36

    Topics: Catalysis; Copper; Cyclization; Indazoles; Pyrazoles

2011
Synthesis of 7-oxo-dihydrospiro[indazole-5,4'-piperidine] acetyl-CoA carboxylase inhibitors.
    The Journal of organic chemistry, 2012, Feb-03, Volume: 77, Issue:3

    Topics: Acetyl-CoA Carboxylase; Alkenes; Alkylation; Chemistry Techniques, Synthetic; Enzyme Inhibitors; Indazoles; Ketones; Piperidines; Pyrazoles; Stereoisomerism; Substrate Specificity

2012
Synthesis, structure-activity relationship, and pharmacophore modeling studies of pyrazole-3-carbohydrazone derivatives as dipeptidyl peptidase IV inhibitors.
    Chemical biology & drug design, 2012, Volume: 79, Issue:6

    Topics: Binding Sites; Computer Simulation; Dipeptidyl Peptidase 4; Dipeptidyl-Peptidase IV Inhibitors; Humans; Hydrazones; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Indazoles; Naphthalenes; Protein Structure, Tertiary; Pyrazoles; Structure-Activity Relationship

2012