pyrazole and am 251

pyrazole has been researched along with am 251 in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Krishnamurthy, M; Li, W; Moore, BM1
Fong, O; Fong, TM; Muise, ES; Qian, S; Thompson, JR; Weingarth, D; Zhao, W1

Other Studies

2 other study(ies) available for pyrazole and am 251

ArticleYear
Synthesis, biological evaluation, and structural studies on N1 and C5 substituted cycloalkyl analogues of the pyrazole class of CB1 and CB2 ligands.
    Bioorganic & medicinal chemistry, 2004, Jan-15, Volume: 12, Issue:2

    Topics: Animals; Biochemistry; CHO Cells; Cricetinae; Drug Evaluation, Preclinical; Humans; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Structure-Activity Relationship

2004
Genome-wide expression profiling revealed peripheral effects of cannabinoid receptor 1 inverse agonists in improving insulin sensitivity and metabolic parameters.
    Molecular pharmacology, 2010, Volume: 78, Issue:3

    Topics: Adipose Tissue; Animals; Cannabinoid Receptor Agonists; Down-Regulation; Homozygote; Insulin; Insulin Resistance; Liver; Male; Mice; Mice, Knockout; Mice, Obese; Piperidines; PPAR alpha; PPAR gamma; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Cannabinoid; Signal Transduction; Sterol Regulatory Element Binding Protein 1; Transcriptional Activation

2010