Page last updated: 2024-08-18

pyrazolanthrone and h 89

pyrazolanthrone has been researched along with h 89 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (40.00)29.6817
2010's6 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A1
Hanada, K; Iwasaki, Y; Kageyama, K; Nigawara, T; Sakihara, S; Suda, T; Takayasu, S1
Boulukos, K; Clavel, S; Coldefy, AS; Dérijard, B; Pisani, DF; Siffroi-Fernandez, S1
Fernández-Galilea, M; Martinez, JA; Moreno-Aliaga, MJ; Pérez-Matute, P; Prieto-Hontoria, PL1
Cao, JP; Chen, CQ; Jiang, ZM; Li, CL; Lin, D; Liu, S; Ma, DC; Pu, FF; Xing, SN; Yang, JG; Zhao, S; Zhao, YS1
Li, C; Liu, S; Ma, D; Pu, F; Xing, S; Yang, J; Yu, Y; Zhao, S1
Li, C; Liu, S; Ma, D; Wang, L; Xing, S; Yang, J; Yu, Y; Zhao, S1

Other Studies

10 other study(ies) available for pyrazolanthrone and h 89

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
    The Biochemical journal, 2013, Apr-15, Volume: 451, Issue:2

    Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase

2013
Involvement of regulatory elements on corticotropin-releasing factor gene promoter in hypothalamic 4B cells.
    Journal of endocrinological investigation, 2008, Volume: 31, Issue:12

    Topics: Anthracenes; Cell Line; Chromones; Colforsin; Corticotropin-Releasing Hormone; Dexamethasone; Flavonoids; Genes, Reporter; Humans; Hypothalamus; Imidazoles; Isoquinolines; Morpholines; Promoter Regions, Genetic; Protein Kinase Inhibitors; Pyridines; Regulatory Elements, Transcriptional; Sequence Deletion; Sulfonamides; Transfection

2008
Regulation of the intracellular localization of Foxo3a by stress-activated protein kinase signaling pathways in skeletal muscle cells.
    Molecular and cellular biology, 2010, Volume: 30, Issue:2

    Topics: Animals; Anthracenes; Cell Line; Cell Nucleus; Chromones; Exportin 1 Protein; Forkhead Box Protein O3; Forkhead Transcription Factors; Humans; Isoquinolines; Karyopherins; MAP Kinase Kinase 3; MAP Kinase Kinase 4; Mice; Mitogen-Activated Protein Kinase Kinases; Morpholines; Muscle Cells; Muscle Fibers, Skeletal; Muscle Proteins; Muscular Atrophy; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Receptors, Cytoplasmic and Nuclear; Signal Transduction; SKP Cullin F-Box Protein Ligases; Sulfonamides; Thiophenes; Transfection

2010
Effects of lipoic acid on lipolysis in 3T3-L1 adipocytes.
    Journal of lipid research, 2012, Volume: 53, Issue:11

    Topics: 3T3-L1 Cells; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Anthracenes; Carrier Proteins; Chromones; Isoquinolines; JNK Mitogen-Activated Protein Kinases; Lipase; Lipolysis; Mice; Morpholines; Perilipin-1; Phosphoproteins; Phosphorylation; Quinolones; Ribonucleotides; Sterol Esterase; Sulfonamides; Thioctic Acid

2012
Phosphorylation of ribosomal protein S6 kinase 1 at Thr421/Ser424 and dephosphorylation at Thr389 regulates SP600125-induced polyploidization of megakaryocytic cell lines.
    PloS one, 2014, Volume: 9, Issue:12

    Topics: Anthracenes; Cell Line; Cell Proliferation; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Humans; Isoquinolines; Megakaryocytes; Models, Molecular; Molecular Conformation; Mutation; Phosphorylation; Polyploidy; Protein Binding; Protein Interaction Domains and Motifs; Protein Kinase Inhibitors; Ribosomal Protein S6 Kinases, 70-kDa; Sulfonamides

2014
[Protein kinase A inhibitor H-89 blocks polyploidization of SP600125-induced CMK cells by regulating phosphorylation of ribosomal protein S6 kinase 1].
    Xi bao yu fen zi mian yi xue za zhi = Chinese journal of cellular and molecular immunology, 2016, Volume: 32, Issue:10

    Topics: Anthracenes; Cell Line; Humans; Isoquinolines; Megakaryocytes; Molecular Docking Simulation; Phosphorylation; Polyploidy; Protein Kinase Inhibitors; Ribosomal Protein S6 Kinases, 90-kDa; Sulfonamides

2016
[SP600125-induced polyploidization of megakaryocytic leukemia cell lines by ribosomal protein S6 kinase 1 depends on the degree of cell differentiation].
    Xi bao yu fen zi mian yi xue za zhi = Chinese journal of cellular and molecular immunology, 2016, Volume: 32, Issue:10

    Topics: Anthracenes; Cell Differentiation; Cell Line; Humans; Isoquinolines; Leukemia, Megakaryoblastic, Acute; Megakaryocytes; Phosphorylation; Polyploidy; Ribosomal Protein S6 Kinases; Sulfonamides

2016