Page last updated: 2024-08-21

pyrazines and l 689660

pyrazines has been researched along with l 689660 in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Freedman, SB; Hargreaves, RJ; Harley, EA; Hutson, PH; McKnight, AT; Newberry, NR; Patel, S; Scholey, K; Semark, JE; Street, LJ1
Iversen, SD; Rupniak, NM; Tye, SJ1
Bymaster, FP; Calligaro, DO; Deeter, JB; Merritt, L; Mitch, CH; Olesen, PH; Peters, SC; Sauerberg, P; Sawyer, BD; Shannon, HE; Sheardown, MJ; Swedberg, MD; Ward, JS1
Bayley, P; Channell, S; Dawson, GR; Iversen, SD1
Dawson, GR; Iversen, SD1
Aagaard, P; McKinney, M1

Other Studies

6 other study(ies) available for pyrazines and l 689660

ArticleYear
L-689,660, a novel cholinomimetic with functional selectivity for M1 and M3 muscarinic receptors.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Ganglia, Sympathetic; Lacrimal Apparatus; Male; Myocardium; Parasympathomimetics; Pyrazines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Succinimides; Thiophenes

1992
Comparison of the effects of selective and nonselective muscarinic agonists on cognition and thermoregulation in primates.
    Journal of the neurological sciences, 1992, Volume: 110, Issue:1-2

    Topics: Animals; Body Temperature Regulation; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cognition; Macaca mulatta; Male; Memory; Parasympathomimetics; Piperazines; Pyrazines; Quinuclidines; Receptors, Muscarinic; Saimiri; Scopolamine; Space Perception; Succinimides; Thiophenes

1992
Functionally selective M1 muscarinic agonists. 3. Side chains and azacycles contributing to functional muscarinic selectivity among pyrazinylazacycles.
    Journal of medicinal chemistry, 1995, Sep-01, Volume: 38, Issue:18

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Male; Mice; Muscarinic Agonists; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Structure-Activity Relationship; Thiadiazoles

1995
A comparison of the effects of the novel muscarinic receptor agonists L-689,660 and AF102B in tests of reference and working memory.
    Psychopharmacology, 1994, Volume: 113, Issue:3-4

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Conditioning, Operant; Drinking Behavior; Male; Memory; Memory, Short-Term; Mice; Mice, Inbred Strains; Muscarinic Agonists; Pain Measurement; Parasympathomimetics; Pyrazines; Quinuclidines; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Scopolamine; Thiophenes

1994
The effects of novel cholinesterase inhibitors and selective muscarinic receptor agonists in tests of reference and working memory.
    Behavioural brain research, 1993, Nov-30, Volume: 57, Issue:2

    Topics: Animals; Avoidance Learning; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Conditioning, Classical; Discrimination Learning; Donepezil; Dose-Response Relationship, Drug; Indans; Learning; Memory; Mice; Oxadiazoles; Pain Threshold; Parasympathomimetics; Physostigmine; Piperidines; Pyrazines; Quinuclidines; Rats; Receptors, Muscarinic; Thiophenes

1993
Pharmacological characterization of the novel cholinomimetic L-689,660 at cloned and native brain muscarinic receptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:3

    Topics: Acetylcholine; Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cloning, Molecular; Cyclic AMP; Hippocampus; Humans; Male; Muscarinic Antagonists; Parasympathomimetics; Phosphatidylinositols; Pyrazines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic

1993