pyrazines has been researched along with l 689660 in 6 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Freedman, SB; Hargreaves, RJ; Harley, EA; Hutson, PH; McKnight, AT; Newberry, NR; Patel, S; Scholey, K; Semark, JE; Street, LJ | 1 |
Iversen, SD; Rupniak, NM; Tye, SJ | 1 |
Bymaster, FP; Calligaro, DO; Deeter, JB; Merritt, L; Mitch, CH; Olesen, PH; Peters, SC; Sauerberg, P; Sawyer, BD; Shannon, HE; Sheardown, MJ; Swedberg, MD; Ward, JS | 1 |
Bayley, P; Channell, S; Dawson, GR; Iversen, SD | 1 |
Dawson, GR; Iversen, SD | 1 |
Aagaard, P; McKinney, M | 1 |
6 other study(ies) available for pyrazines and l 689660
Article | Year |
---|---|
L-689,660, a novel cholinomimetic with functional selectivity for M1 and M3 muscarinic receptors.
Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Ganglia, Sympathetic; Lacrimal Apparatus; Male; Myocardium; Parasympathomimetics; Pyrazines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Succinimides; Thiophenes | 1992 |
Comparison of the effects of selective and nonselective muscarinic agonists on cognition and thermoregulation in primates.
Topics: Animals; Body Temperature Regulation; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cognition; Macaca mulatta; Male; Memory; Parasympathomimetics; Piperazines; Pyrazines; Quinuclidines; Receptors, Muscarinic; Saimiri; Scopolamine; Space Perception; Succinimides; Thiophenes | 1992 |
Functionally selective M1 muscarinic agonists. 3. Side chains and azacycles contributing to functional muscarinic selectivity among pyrazinylazacycles.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Male; Mice; Muscarinic Agonists; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Structure-Activity Relationship; Thiadiazoles | 1995 |
A comparison of the effects of the novel muscarinic receptor agonists L-689,660 and AF102B in tests of reference and working memory.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Conditioning, Operant; Drinking Behavior; Male; Memory; Memory, Short-Term; Mice; Mice, Inbred Strains; Muscarinic Agonists; Pain Measurement; Parasympathomimetics; Pyrazines; Quinuclidines; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Scopolamine; Thiophenes | 1994 |
The effects of novel cholinesterase inhibitors and selective muscarinic receptor agonists in tests of reference and working memory.
Topics: Animals; Avoidance Learning; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Conditioning, Classical; Discrimination Learning; Donepezil; Dose-Response Relationship, Drug; Indans; Learning; Memory; Mice; Oxadiazoles; Pain Threshold; Parasympathomimetics; Physostigmine; Piperidines; Pyrazines; Quinuclidines; Rats; Receptors, Muscarinic; Thiophenes | 1993 |
Pharmacological characterization of the novel cholinomimetic L-689,660 at cloned and native brain muscarinic receptors.
Topics: Acetylcholine; Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cloning, Molecular; Cyclic AMP; Hippocampus; Humans; Male; Muscarinic Antagonists; Parasympathomimetics; Phosphatidylinositols; Pyrazines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic | 1993 |