Page last updated: 2024-08-21

pyrazines and ketanserin

pyrazines has been researched along with ketanserin in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19907 (43.75)18.7374
1990's3 (18.75)18.2507
2000's5 (31.25)29.6817
2010's1 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anderson, EG; Todorovic, SM1
Brazell, C; Dourish, CT; King, BH; Middlemiss, DN1
Barrett, JE; Bolger, GT; Mansbach, RS; Skolnick, P; Weissman, B; Witkin, JM1
Barrett, JE; Brady, LS1
Clineschmidt, BV; Pettibone, DJ; Reiss, DR; Robinson, JL1
Barrett, JE; Mansbach, RS1
Gudelsky, GA; Koenig, JI; Meltzer, HY2
Battaglia, G; Brownfield, MS; Cabrera, TM; Levy, AD; Li, Q; Rittenhouse, PA; van de Kar, LD1
Fiorella, D; Helsley, S; Rabin, RA; Winter, JC1
Basura, GJ; Goshgarian, HG; Zhou, SY1
Cunningham, KA; Filip, M; McCreary, AC1
Goto, F; Obata, H; Saito, S; Sakurazawa, S; Sasaki, M; Usui, T1
Egashira, N; Fujiwara, M; Iwasaki, K; Koushi, E; Mishima, K; Oishi, R1
Levesque, P; Li, D; Li, J; Miller, KJ; Robl, JA; Rossi, KA; Varnes, JG; Wacker, DA; Wu, GY1
Biggers, WJ; Burns, RT; Lehman, C; Pechenik, JA; Scavo, G1

Other Studies

16 other study(ies) available for pyrazines and ketanserin

ArticleYear
Pharmacological characterization of 5-hydroxytryptamine2 and 5-hydroxytryptamine3 receptors in rat dorsal root ganglion cells.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Ganglia, Spinal; Indoles; Ketanserin; Male; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tropanes; Tropisetron

1990
MK-212 increases rat plasma ACTH concentration by activation of the 5-HT1C receptor subtype.
    Neuroscience letters, 1989, Oct-23, Volume: 105, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Animals; Antiparkinson Agents; Ergolines; Ketanserin; Male; Metergoline; Pindolol; Piperazines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1989
Behavioral studies with anxiolytic drugs. IV. Serotonergic involvement in the effects of buspirone on punished behavior of pigeons.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Buspirone; Columbidae; Dose-Response Relationship, Drug; Ketanserin; Male; Punishment; Pyrazines; Pyrimidines; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Tritium

1987
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri

1985
Characterization of 5-hydroxytryptamine receptors in rat stomach fundus.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Gastric Fundus; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperazines; Piperidines; Propranolol; Pyrazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1985
Effects of MK-212 (6-chloro-2[1-piperazinyl]pyrazine) on schedule-controlled behavior and their reversal by 5-HT antagonists in the pigeon.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: Animals; Columbidae; Conditioning, Operant; Cues; Generalization, Stimulus; Ketanserin; Male; Metergoline; Methysergide; Piperidines; Pyrazines; Receptors, Serotonin; Reinforcement Schedule

1986
Thermoregulatory responses to serotonin (5-HT) receptor stimulation in the rat. Evidence for opposing roles of 5-HT2 and 5-HT1A receptors.
    Neuropharmacology, 1986, Volume: 25, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature Regulation; Ketanserin; Male; Methoxydimethyltryptamines; Pindolol; Piperidines; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Tetrahydronaphthalenes

1986
Stimulation of corticosterone and beta-endorphin secretion in the rat by selective 5-HT receptor subtype activation.
    European journal of pharmacology, 1987, May-07, Volume: 137, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; beta-Endorphin; Corticosterone; Endorphins; Ketanserin; Male; Pindolol; Pyrazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spiperone; Tetrahydronaphthalenes

1987
Long-term treatment with the antidepressants fluoxetine and desipramine potentiates endocrine responses to the serotonin agonists 6-chloro-2-[1-piperazinyl]-pyrazine (MK-212) and (+-)-1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane HCl (DOI).
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Adrenocorticotropic Hormone; Amphetamines; Animals; Desipramine; Drug Synergism; Fluoxetine; Hormones; Ketanserin; Male; Pyrazines; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Vasopressins

1993
5-HT2C receptor-mediated phosphoinositide turnover and the stimulus effects of m-chlorophenylpiperazine.
    Psychopharmacology, 1995, Volume: 122, Issue:3

    Topics: Animals; Choroid Plexus; Conditioning, Operant; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drug Interactions; Ketanserin; Lysergic Acid Diethylamide; Ondansetron; Phosphatidylinositols; Piperazines; Pyrazines; Quipazine; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Serotonin(2) receptors mediate respiratory recovery after cervical spinal cord hemisection in adult rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2001, Volume: 91, Issue:6

    Topics: Amphetamines; Animals; Asphyxia; Cervical Vertebrae; Female; Ketanserin; Phrenic Nerve; Pyrazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Respiratory Physiological Phenomena; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord Injuries; Spiro Compounds; Sulfonamides

2001
Discriminative stimulus properties of (+/-)-fenfluramine: the role of 5-HT2 receptor subtypes.
    Behavioral neuroscience, 2003, Volume: 117, Issue:2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Fenfluramine; Fluorobenzenes; Indoles; Ketanserin; Male; Piperidines; Pyrazines; Pyridines; Rats; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfonamides; Thiophenes

2003
Antiallodynic effects of intrathecally administered 5-HT(2C) receptor agonists in rats with nerve injury.
    Pain, 2004, Volume: 108, Issue:1-2

    Topics: Amphetamines; Animals; Indoles; Injections, Spinal; Ketanserin; Ligation; Lumbar Vertebrae; Male; Neuralgia; Nociceptors; Piperazines; Pyrazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Serotonin; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Nerves; Spiro Compounds; Sulfonamides; Thiophenes

2004
2,5-Dimethoxy-4-iodoamphetamine (DOI) inhibits Delta9-tetrahydrocannabinol-induced catalepsy-like immobilization in mice.
    Journal of pharmacological sciences, 2007, Volume: 105, Issue:4

    Topics: Aminopyridines; Amphetamines; Analysis of Variance; Animals; Animals, Outbred Strains; Behavior, Animal; Dose-Response Relationship, Drug; Dronabinol; Freezing Reaction, Cataleptic; Indoles; Injections, Intraperitoneal; Ketanserin; Male; Mice; Pyrazines; Quinoxalines; Serotonin 5-HT2 Receptor Agonists; Serotonin Receptor Agonists; Time Factors

2007
Position 5.46 of the serotonin 5-HT2A receptor contributes to a species-dependent variation for the 5-HT2C agonist (R)-9-ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: impact on selectivity and toxicological evaluation.
    Molecular pharmacology, 2009, Volume: 76, Issue:6

    Topics: Animals; Binding, Competitive; Blood Pressure; Calcium; Cell Line; Dogs; Genetic Variation; Humans; Isoindoles; Ketanserin; Macaca fascicularis; Male; Motor Activity; Mutagenesis, Site-Directed; Protein Binding; Pyrazines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Sequence Homology, Amino Acid; Serotonin 5-HT2 Receptor Agonists; Serotonin Antagonists; Species Specificity; Structural Homology, Protein

2009
The B vitamins nicotinamide (B3) and riboflavin (B2) stimulate metamorphosis in larvae of the deposit-feeding polychaete Capitella teleta: implications for a sensory ligand-gated ion channel.
    PloS one, 2014, Volume: 9, Issue:11

    Topics: Animals; Biological Assay; Calcium; Imidazoles; Ketanserin; Larva; Ligand-Gated Ion Channels; Metamorphosis, Biological; Niacinamide; Polychaeta; Pyrazines; Pyridines; Riboflavin; Seawater

2014