Page last updated: 2024-08-21

pyrazines and carbachol

pyrazines has been researched along with carbachol in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19906 (46.15)18.7374
1990's7 (53.85)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beleta, J; Berga, P; Bou, J; Cardelús, I; Fernández, AG; Gristwood, RW; Llenas, J1
Antunes-Rodrigues, J; Ramalho, MJ; Reis, LC1
Blinks, JR; Endoh, M; Taira, N; Yanagisawa, T1
English, TA; Gristwood, RW; Owen, DA; Sampford, KA; Wallwork, J1
Dhasmana, KM; Dixit, KS; Tangri, KK1
Endoh, M; Taira, N; Yanagisawa, T1
Bonting, SL; De Pont, JJ; Fleuren-Jakobs, AM; Kuijpers, GA; Rodrigues de Miranda, JF; Van Nooy, IG1
Ando, H; Kobayashi-Ando, S; Takeya, K; Yajima, M1
Bonnet, PA; Boucard, M; Chapat, JP; Laurent, F; Michel, A1
Ando, H; Ando, S; Nomura, H; Takeya, K; Yajima, M1
Miyoshi, Y; Nakaya, Y; Nomura, M; Saito, K; Shono, M; Wakatsuki, T1
Fozard, JR; Müller-Schweinitzer, E1
Abou-Gharbia, M; Boast, CA; Husbands, GM; Moyer, JA; Sabb, AL; Stein, RP; Tasse, RP; Tokolics, J1

Other Studies

13 other study(ies) available for pyrazines and carbachol

ArticleYear
Studies on the cardiac actions of flosequinan in vitro.
    British journal of pharmacology, 1992, Volume: 105, Issue:4

    Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Action Potentials; Animals; Carbachol; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Pyrazines; Pyrrolidinones; Quinolines; Rolipram; Vasodilator Agents

1992
Central serotonergic modulation of drinking behavior induced by angiotensin II and carbachol in normally hydrated rats: effect of intracerebroventricular injection of MK-212.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1990, Volume: 23, Issue:12

    Topics: Angiotensin II; Animals; Carbachol; Drinking Behavior; Injections, Intraventricular; Male; Pyrazines; Rats; Serotonin

1990
Effects of new inotropic agents on cyclic nucleotide metabolism and calcium transients in canine ventricular muscle.
    Circulation, 1986, Volume: 73, Issue:3 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aequorin; Aminopyridines; Amrinone; Animals; Calcium; Carbachol; Cardiotonic Agents; Colforsin; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Enoximone; Female; Imidazoles; Male; Milrinone; Myocardial Contraction; Myocardium; Nifedipine; Nucleotides, Cyclic; Pyrazines; Pyridones; Quinolines; Time Factors

1986
Analysis of responses to a selective phosphodiesterase III inhibitor, SK&F 94120, on isolated myocardium, including human ventricular myocardium from "end-stage" failure patients.
    Journal of cardiovascular pharmacology, 1987, Volume: 9, Issue:6

    Topics: Animals; Carbachol; Cats; Female; Guinea Pigs; Heart Failure; Heart Ventricles; Humans; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Phosphodiesterase Inhibitors; Pyrazines; Swine

1987
An analysis of the central vasomotor effects of monoamine oxidase inhibitor, modaline sulphate.
    Japanese journal of pharmacology, 1972, Volume: 22, Issue:5

    Topics: Animals; Atropine; Blood Pressure; Carbachol; Carotid Arteries; Cerebral Ventricles; Dogs; Female; Hemicholinium 3; Injections; Male; Phenoxybenzamine; Propranolol; Pyrazines; Stimulation, Chemical; Tachyphylaxis; Tetrabenazine; Transducers; Vagus Nerve; Vasomotor System

1972
Involvement of cyclic AMP in the positive inotropic effect of OPC-8212, a new cardiotonic agent, on the canine ventricular muscle.
    Japanese journal of pharmacology, 1984, Volume: 36, Issue:3

    Topics: Animals; Atenolol; Carbachol; Cardiotonic Agents; Cyclic AMP; Dogs; Female; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Myocardium; Pyrazines; Quinolines; Stimulation, Chemical; Thiophenes

1984
Amiloride is a cholinergic antagonist in the rabbit pancreas.
    Biochimica et biophysica acta, 1984, Jun-19, Volume: 804, Issue:2

    Topics: Acetylcholine; Amiloride; Amylases; Animals; Calcium; Carbachol; In Vitro Techniques; Kinetics; Pancreas; Pancreatic Juice; Pyrazines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic

1984
Positive inotropic effect of 3,4-dihydro-6-[4-(3,4-dimethoxybenzoyl)-1 -piperazinyl]-2(1H)-quinolinone (OPC-8212) and mechanism of action in guinea pig ventricular myocardium.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:3A

    Topics: Animals; Carbachol; Cardiotonic Agents; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Myocardial Contraction; Propranolol; Pyrazines; Quinolines; Reserpine

1984
Evaluation of the relaxant effects of SCA40, a novel charybdotoxin-sensitive potassium channel opener, in guinea-pig isolated trachealis.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Animals; Carbachol; Charybdotoxin; Glyburide; Guinea Pigs; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Potassium Channels; Potassium Chloride; Pyrazines; Scorpion Venoms; Trachea

1993
Relaxing effect of vesnarinone (OPC-8212) on the tracheal muscle strips isolated from guinea pigs.
    Japanese journal of pharmacology, 1993, Volume: 62, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Airway Resistance; Animals; Carbachol; Drug Interactions; Female; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Potassium; Propranolol; Pyrazines; Quinolines; Reserpine; Trachea

1993
Effects of vesnarinone (OPC-8212) on Ca(2+)-activated K channels and cytosolic Ca2+ in cultured smooth muscle cells from porcine coronary artery.
    Japanese heart journal, 1994, Volume: 35, Issue:1

    Topics: Amrinone; Animals; Arteries; Calcium; Carbachol; Cardiotonic Agents; Cells, Cultured; Coronary Vessels; Cyclic AMP; Cytosol; Muscle, Smooth, Vascular; Potassium Channels; Pyrazines; Quinolines; Swine

1994
SCA 40: studies of the relaxant effects on cryopreserved human airway and vascular smooth muscle.
    British journal of pharmacology, 1997, Volume: 120, Issue:7

    Topics: Albuterol; Bronchi; Carbachol; Cryopreservation; Drug Interactions; Humans; Imidazoles; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium; Pyrazines

1997
Discovery of a highly potent, functionally-selective muscarinic M1 agonist, WAY-132983 using rational drug design and receptor modelling.
    Bioorganic & medicinal chemistry letters, 1999, Jul-19, Volume: 9, Issue:14

    Topics: Administration, Oral; Animals; Bridged-Ring Compounds; Carbachol; Cerebral Cortex; CHO Cells; Cognition Disorders; Computer Simulation; Cricetinae; Crystallography, X-Ray; Drug Design; Drug Evaluation, Preclinical; Humans; Macaca mulatta; Maze Learning; Models, Molecular; Muscarinic Agonists; Phosphatidylinositols; Protein Conformation; Pyrazines; Pyridines; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Salivation; Structure-Activity Relationship; Thiadiazoles

1999