Page last updated: 2024-08-21

pyrazines and capsaicin

pyrazines has been researched along with capsaicin in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.78)18.7374
1990's1 (2.78)18.2507
2000's14 (38.89)29.6817
2010's20 (55.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Govindarajan, VS1
Advenier, C; Bakdach, H; Bonnet, PA; Cui, YY; Michel, A; Naline, E1
Bristol, DR; Harrison, JE; Mark, L; Pomonis, JD; Valenzano, KJ; Walker, K1
Anthes, JC; Correll, CC; Phelps, PT1
Fujiuchi, A; Hara, T; Imai, A; Kanai, Y; Nakazato, E1
Gavva, NR; Klionsky, L; Louis, JC; Norman, MH; Tamir, R; Treanor, JJ; Wild, KD1
Christoph, T; Erdmann, VA; Frank, R; Gillen, C; Grünweller, A; Kurreck, J; Mika, J; Schäfer, MK; Wade, EJ; Weihe, E1
Briggs, MA; Bruton, G; Calver, AR; Chessell, I; Crook, B; Davis, JB; Davis, RP; Foley, AG; Heslop, T; Hirst, WD; Medhurst, AD; Medhurst, SJ; Ociepka, S; Orlek, B; Ray, A; Regan, CM; Sargent, B; Schogger, J; Stean, TO; Trail, BK; Upton, N; White, T; Wilson, DM1
Aggarwal, BB; Bhutani, M; Guha, S; Kunnumakkara, AB; Nair, AS; Pathak, AK; Sethi, G1
De Man, JG; De Schepper, HU; De Winter, BY; Deiteren, A; Herman, AG; Martinet, W; Pelckmans, PA; Ruyssers, NE; Timmermans, JP; Van Nassauw, L1
Reilly, CA; Sabnis, AS; Shadid, M; Yost, GS1
Bandell, M; Dhaka, A; Dubin, AE; Mathur, J; Patapoutian, A; Petrus, M; Uzzell, V1
Bredenoord, AJ; De Man, JG; De Schepper, HU; De Winter, BY; Pelckmans, PA; Timmermans, JP; Van Nassauw, L1
Horie, S; Hosoya, T; Kurosawa, E; Matsumoto, K; Murayama, T; Priestley, JV; Tashima, K; Terui, H1
Beltrán, C; Castellano, LE; Chirinos, M; Darszon, A; De Blas, GA; Hernández-González, EO; Larrea, F; Ocampo, AY; Serrano, CJ; Treviño, CL1
Fernández-Ballester, G; Ferrer-Montiel, A; Malkia, A; Pertusa, M; Viana, F1
Brennan, FX; Bryant, RW; Devantier, HR; Long, DJ; Palmer, RK; Salemme, FR1
Fujihara, H; Hashimoto, H; Nagatomo, T; Ohbuchi, T; Otsubo, H; Saito, T; Suzuki, H; Ueta, Y; Yokoyama, T1
Bakthavatchalam, R; Blum, CA; Boyce, S; Brielmann, H; Burnaby-Davies, N; Caldwell, T; Capitosti, S; Chenard, BL; Conley, R; Cortright, D; Crandall, M; De Lombaert, S; Hodgetts, KJ; Jones, AB; Kershaw, MT; Krause, JE; Martin, WJ; Mason, G; Matson, D; Murphy, BA; Perrett, H; Rycroft, W; Zheng, X1
Appenzeller, M; Bigliardi, P; Buclin, T; Grouzmann, E; Pannatier, A1
Beltrán, C; Darszon, A; De Blas, G; de la Vega-Beltrán, JL; Gibbs, GM; Martínez-López, P; Monroy, E; O'Bryan, MK; Orta, G; Treviño, CL1
Bartho, L; Benko, R; Illényi, L; Kelemen, D; Papp, A; Papp, R1
Beattie, RE; Beck, JP; Blanco, MJ; Broad, LM; Folly, EA; Mill, CE; Mogg, AJ1
Mutoh, T; Taki, Y; Tsubone, H1
Baek, HH; Kang, KM1
Baumann, K; Belmaáti, MS; Christensen, RE; Claesson, MH; Diemer, S; Hvarness, T; Pedersen, AE1
Carlin, KP; Crumley, G; Ilyin, VI; Patel, A; Wu, G1
Asano, A; Dayanithi, G; Forostyak, O; Hosaka, YZ; Ichimura, M; Kayano, T; Kitamura, N; Moriya, T; Shibasaki, R; Shibuya, I; Takebuchi, N; Verkhratsky, A1
Bartho, L; Bencsik, T; Sandor, Z1
Fujita, T; Jiang, CY; Kumamoto, E; Wang, C; Xu, ZH1
Andrade, VA; Araujo, IG; Barbosa-Filho, JM; Braz, AL; Chaves, CG; Correia, Nde A; Cruz, Jdos S; de Albuquerque, JG; de Almeida, MM; de Medeiros, IA; Gomes, MA; Leite, Mde F; Nunes, XP; Pesquero, JL; Pinho-da-Silva, L; Silva, DF1
Dhandapani, P; Grötzinger, C; Huimann, P; Khajavi, N; Köhrle, J; Ljubojevic, N; Lucius, A; Mergler, S; Reinach, PS1
Ide, S; Kojima, S; Nakanishi, Y; Nishino, K; Tanamachi, K; Tanuma, S; Tsukimoto, M1
Fujita, T; Kumamoto, E; Piao, LH; Yu, T1
Fischer, MJM; Namer, B; Reeh, PW; Schwarz, MG1
Cai, DS; Chen, HS; Cui, HR; Guo, WB; Huang, XM; Jia, XH; Lei, HM; Qi, JC; Wang, H; Wang, PL; Xu, B; Yang, YQ; Zhang, WX; Zhou, F1

Reviews

1 review(s) available for pyrazines and capsaicin

ArticleYear
Capsicum--production, technology, chemistry, and quality. Part III. Chemistry of the color, aroma, and pungency stimuli.
    Critical reviews in food science and nutrition, 1986, Volume: 24, Issue:3

    Topics: Capsaicin; Capsicum; Carotenoids; Chemical Phenomena; Chemistry; Chromatography; Food Preservation; Food Technology; Hot Temperature; Ketones; Light; Molecular Conformation; Odorants; Pigmentation; Plants, Edible; Plants, Medicinal; Pyrazines; Smell; Taste; Volatilization; Xanthophylls

1986

Trials

2 trial(s) available for pyrazines and capsaicin

ArticleYear
Substance P-induced skin inflammation is not modulated by a single dose of sitagliptin in human volunteers.
    Biological chemistry, 2011, Volume: 392, Issue:3

    Topics: Capsaicin; Carbonated Beverages; Cross-Over Studies; Dipeptidyl Peptidase 4; Dipeptidyl-Peptidase IV Inhibitors; Dose-Response Relationship, Drug; Double-Blind Method; Drug Eruptions; Edema; Erythema; Humans; Injections, Intradermal; Male; Pain; Pyrazines; Sitagliptin Phosphate; Skin; Substance P; Triazoles; Vasodilation

2011
TRPA1 and TRPV1 Antagonists Do Not Inhibit Human Acidosis-Induced Pain.
    The journal of pain, 2017, Volume: 18, Issue:5

    Topics: Acid Sensing Ion Channel Blockers; Acidosis; Adult; Amiloride; Analgesics; Analysis of Variance; Capsaicin; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Middle Aged; Oximes; Pain; Pain Measurement; Pyrazines; Pyridines; TRPA1 Cation Channel; TRPV Cation Channels

2017

Other Studies

33 other study(ies) available for pyrazines and capsaicin

ArticleYear
Effects of SCA40 on human bronchi and on guinea pig main bronchi in vitro. Comparison with cromakalim.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Acetylcholine; Animals; Benzopyrans; Bronchi; Bronchodilator Agents; Capsaicin; Charybdotoxin; Cromakalim; Electric Stimulation; Female; Glyburide; Guinea Pigs; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Neurokinin A; Nitroprusside; Osmolar Concentration; Parasympatholytics; Potassium Channel Blockers; Potassium Channels; Pyrazines; Pyrroles; Tetraethylammonium; Tetraethylammonium Compounds

1996
N-(4-Tertiarybutylphenyl)-4-(3-cholorphyridin-2-yl)tetrahydropyrazine -1(2H)-carbox-amide (BCTC), a novel, orally effective vanilloid receptor 1 antagonist with analgesic properties: II. in vivo characterization in rat models of inflammatory and neuropath
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 306, Issue:1

    Topics: Analgesics; Animals; Ataxia; Capsaicin; Hyperalgesia; Inflammation; Male; Nerve Tissue; Pain; Pain Threshold; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Drug

2003
Cloning and functional characterization of dog transient receptor potential vanilloid receptor-1 (TRPV1).
    European journal of pharmacology, 2005, Apr-18, Volume: 513, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Biological Transport; Calcium; Capsaicin; Cell Line; Cloning, Molecular; Diterpenes; DNA, Complementary; Dogs; Dopamine; Dose-Response Relationship, Drug; Fluorometry; Genetic Vectors; Genotype; Humans; Molecular Sequence Data; Mutation, Missense; Phorbol Esters; Phylogeny; Pyrazines; Pyridines; Receptors, Drug; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Transfection

2005
Involvement of an increased spinal TRPV1 sensitization through its up-regulation in mechanical allodynia of CCI rats.
    Neuropharmacology, 2005, Volume: 49, Issue:7

    Topics: Animals; Blotting, Western; Calcitonin Gene-Related Peptide; Capsaicin; In Vitro Techniques; Injections, Spinal; Male; Nerve Tissue Proteins; Neuropeptides; Pain; Pain Measurement; Physical Stimulation; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Spinal Cord; Spinal Cord Injuries; Substance P; TRPV Cation Channels; Up-Regulation

2005
Proton activation does not alter antagonist interaction with the capsaicin-binding pocket of TRPV1.
    Molecular pharmacology, 2005, Volume: 68, Issue:6

    Topics: Animals; Binding Sites; Capsaicin; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Protein Binding; Protein Conformation; Protons; Pyrazines; Pyridines; Rabbits; Rats; TRPV Cation Channels

2005
Silencing of vanilloid receptor TRPV1 by RNAi reduces neuropathic and visceral pain in vivo.
    Biochemical and biophysical research communications, 2006, Nov-10, Volume: 350, Issue:1

    Topics: Animals; Base Sequence; Capsaicin; Chlorocebus aethiops; Colitis; COS Cells; Disease Models, Animal; Humans; Male; Mice; Molecular Sequence Data; Nervous System Diseases; Pain; Pyrazines; Pyridines; Rats; RNA Interference; Sequence Alignment; Sequence Homology, Amino Acid; TRPV Cation Channels

2006
Structurally novel histamine H3 receptor antagonists GSK207040 and GSK334429 improve scopolamine-induced memory impairment and capsaicin-induced secondary allodynia in rats.
    Biochemical pharmacology, 2007, Apr-15, Volume: 73, Issue:8

    Topics: Analgesics; Animals; Avoidance Learning; Azepines; Benzazepines; Capsaicin; Central Nervous System; Drinking; Histamine Agonists; Histamine Antagonists; Humans; Male; Memory Disorders; Neuralgia; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Scopolamine

2007
Capsaicin is a novel blocker of constitutive and interleukin-6-inducible STAT3 activation.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2007, May-15, Volume: 13, Issue:10

    Topics: Antineoplastic Agents; Apoptosis; bcl-X Protein; Boronic Acids; Bortezomib; Capsaicin; Caspase 3; Caspase Inhibitors; Cell Line, Tumor; Cell Proliferation; Cyclin D1; DNA; Extracellular Signal-Regulated MAP Kinases; G1 Phase; Humans; Inhibitor of Apoptosis Proteins; Interleukin-6; Janus Kinase 1; Microtubule-Associated Proteins; Multiple Myeloma; Neoplasm Proteins; Phosphorylation; Poly(ADP-ribose) Polymerases; Protein Tyrosine Phosphatases; Proto-Oncogene Proteins c-bcl-2; Pyrazines; STAT3 Transcription Factor; Survivin; Thalidomide; Vascular Endothelial Growth Factor A

2007
TRPV1 receptor signaling mediates afferent nerve sensitization during colitis-induced motility disorders in rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2008, Volume: 294, Issue:1

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Colitis; Disease Models, Animal; Dose-Response Relationship, Drug; Ganglia, Spinal; Gastric Emptying; Gastrointestinal Motility; Gastroparesis; Intestinal Mucosa; Intestines; Male; Muscle Relaxation; Neurons, Afferent; Peptide Fragments; Pyrazines; Pyridines; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; RNA, Messenger; Signal Transduction; Time Factors; Trinitrobenzenesulfonic Acid; TRPV Cation Channels

2008
Human lung epithelial cells express a functional cold-sensing TRPM8 variant.
    American journal of respiratory cell and molecular biology, 2008, Volume: 39, Issue:4

    Topics: Amino Acid Sequence; Animals; Bronchi; Capsaicin; Cell Line; Cold Temperature; Cytokines; Endoplasmic Reticulum; Epithelial Cells; Humans; Lung; Menthol; Molecular Sequence Data; Pyrazines; Pyridines; Thapsigargin; Thermoreceptors; Thermosensing; TRPM Cation Channels

2008
TRPV1 is activated by both acidic and basic pH.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Jan-07, Volume: 29, Issue:1

    Topics: Acids; Ammonium Chloride; Animals; Calcium; Capsaicin; Cell Line, Transformed; Ganglia, Spinal; Humans; Hydrogen-Ion Concentration; Luminescent Proteins; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Biological; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Pyrazines; Pyridines; Sensory Receptor Cells; Sensory System Agents; Transfection; TRPV Cation Channels

2009
Involvement of afferent neurons in the pathogenesis of endotoxin-induced ileus in mice: role of CGRP and TRPV1 receptors.
    European journal of pharmacology, 2009, Aug-01, Volume: 615, Issue:1-3

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Gastric Emptying; Gastrointestinal Transit; Hexamethonium; Ileus; Lipopolysaccharides; Male; Mice; Neurons, Afferent; Peptide Fragments; Pyrazines; Pyridines; Receptors, Calcitonin Gene-Related Peptide; Sepsis; TRPV Cation Channels

2009
Localization of TRPV1 and contractile effect of capsaicin in mouse large intestine: high abundance and sensitivity in rectum and distal colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2009, Volume: 297, Issue:2

    Topics: Animals; Atropine; Capsaicin; Colon; Dose-Response Relationship, Drug; Gastrointestinal Motility; Immunohistochemistry; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Neurokinin A; Pyrazines; Pyridines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Rectum; Substance P; Tetrodotoxin; Time Factors; TRPV Cation Channels; Ubiquitin Thiolesterase

2009
TRPM8, a versatile channel in human sperm.
    PloS one, 2009, Jun-30, Volume: 4, Issue:6

    Topics: Acrosome Reaction; Calcium; Capsaicin; Chemotaxis; Fluorescent Antibody Technique, Indirect; Humans; Male; Models, Biological; Progesterone; Pyrazines; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Sperm Motility; Spermatozoa; TRPM Cation Channels

2009
Differential role of the menthol-binding residue Y745 in the antagonism of thermally gated TRPM8 channels.
    Molecular pain, 2009, Nov-03, Volume: 5

    Topics: Animals; Capsaicin; Clotrimazole; Cold Temperature; Humans; Imidazoles; Ion Channel Gating; Menthol; Mice; Models, Molecular; Molecular Dynamics Simulation; Mutant Proteins; Mutation; Phenotype; Pyrazines; Pyridines; Structure-Activity Relationship; TRPM Cation Channels; Tyrosine

2009
Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:2

    Topics: Acrylamides; Administration, Oral; Alkaloids; Anilides; Animals; Avoidance Learning; Benzodioxoles; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cinnamates; Diterpenes; Dose-Response Relationship, Drug; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Polyunsaturated Alkamides; Pyrazines; Pyridines; Taste; TRPM Cation Channels; TRPV Cation Channels

2010
TRPV1 gene deficiency attenuates miniature EPSC potentiation induced by mannitol and angiotensin II in supraoptic magnocellular neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Jan-20, Volume: 30, Issue:3

    Topics: Analysis of Variance; Angiotensin II; Anilides; Animals; Capsaicin; Chelating Agents; Cinnamates; Diuretics, Osmotic; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; In Vitro Techniques; Male; Mannitol; Mice; Mice, Inbred C57BL; Mice, Knockout; Miniature Postsynaptic Potentials; Neurons; Piperidines; Pyrazines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Signal Transduction; Supraoptic Nucleus; TRPV Cation Channels; Vasoconstrictor Agents

2010
Discovery of novel 6,6-heterocycles as transient receptor potential vanilloid (TRPV1) antagonists.
    Journal of medicinal chemistry, 2010, Apr-22, Volume: 53, Issue:8

    Topics: Analgesics; Animals; Biological Availability; Capsaicin; Chlorocebus aethiops; COS Cells; Hot Temperature; Humans; Hyperalgesia; In Vitro Techniques; Inflammation; Microsomes, Liver; Naphthyridines; Pain; Pyrazines; Pyridines; Pyrimidines; Quinazolines; Quinolines; Rats; Structure-Activity Relationship; TRPV Cation Channels

2010
TRPM8 in mouse sperm detects temperature changes and may influence the acrosome reaction.
    Journal of cellular physiology, 2011, Volume: 226, Issue:6

    Topics: Acrosome Reaction; Animals; Capsaicin; Humans; Ion Channel Gating; Male; Menthol; Mice; Mice, Knockout; Pyrazines; Pyridines; Pyrimidinones; Spermatozoa; Temperature; Testis; TRPM Cation Channels

2011
Use and limitations of three TRPV-1 receptor antagonists on smooth muscles of animals and man: a vote for BCTC.
    European journal of pharmacology, 2012, Jan-05, Volume: 674, Issue:1

    Topics: Animals; Capsaicin; Female; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Kidney Pelvis; Male; Mice; Muscle Contraction; Muscle, Smooth; Organ Specificity; Pyrazines; Pyridines; Rats; Trachea; TRPV Cation Channels; Urinary Bladder

2012
Altered pharmacology of native rodent spinal cord TRPV1 after phosphorylation.
    British journal of pharmacology, 2013, Volume: 168, Issue:4

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Phosphorylation; Protein Kinase C; Pyrazines; Pyridines; Rats; Rats, Inbred Strains; Spinal Cord; TRPV Cation Channels

2013
Desflurane but not sevoflurane augments laryngeal C-fiber inputs to nucleus tractus solitarii neurons by activating transient receptor potential-A1.
    Life sciences, 2013, May-02, Volume: 92, Issue:14-16

    Topics: Acetanilides; Anesthetics, Inhalation; Animals; Capsaicin; Desflurane; Guinea Pigs; Isoflurane; Isothiocyanates; Laryngeal Nerves; Larynx; Male; Methyl Ethers; Nerve Fibers; Neurons; Purines; Pyrazines; Pyridines; Sevoflurane; Solitary Nucleus; Time Factors; Transient Receptor Potential Channels

2013
Aroma quality assessment of Korean fermented red pepper paste (gochujang) by aroma extract dilution analysis and headspace solid-phase microextraction-gas chromatography-olfactometry.
    Food chemistry, 2014, Feb-15, Volume: 145

    Topics: Capsaicin; Capsicum; Chromatography, Gas; Food Analysis; Odorants; Olfactometry; Pyrazines; Republic of Korea; Solid Phase Microextraction

2014
Antiproliferative effects of TRPV1 ligands on nonspecific and enteroantigen-specific T cells from wild-type and Trpv1 KO mice.
    Inflammatory bowel diseases, 2014, Volume: 20, Issue:6

    Topics: Animals; Antigens; Antipruritics; beta 2-Microglobulin; Capsaicin; CD4-Positive T-Lymphocytes; Cell Proliferation; Colitis; Cytokines; Disease Models, Animal; Ligands; Lymphoid Tissue; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Knockout; Mice, SCID; Pyrazines; Pyridines; Signal Transduction; TRPV Cation Channels

2014
Phenylarsine oxide as a redox modulator of transient receptor potential vanilloid type 1 channel function.
    Journal of neuroscience research, 2015, Volume: 93, Issue:2

    Topics: Adult; Animals; Arsenicals; Calcium; Capsaicin; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ganglia, Spinal; Humans; Membrane Potentials; Neurons; Oxidation-Reduction; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Sensory System Agents; TRPV Cation Channels

2015
Full-length transient receptor potential vanilloid 1 channels mediate calcium signals and possibly contribute to osmoreception in vasopressin neurones in the rat supraoptic nucleus.
    Cell calcium, 2015, Volume: 57, Issue:1

    Topics: Action Potentials; Animals; Calcium Signaling; Capsaicin; Cells, Cultured; HEK293 Cells; Humans; Male; Mannitol; Neurons; Osmolar Concentration; Oxytocin; Pyrazines; Pyridines; Rats; Rats, Transgenic; Rats, Wistar; Supraoptic Nucleus; Temperature; TRPV Cation Channels

2015
High-Concentration Piperine: Capsaicin-Sensitive and -Insensitive Effects on Isolated Organs.
    Pharmacology, 2015, Volume: 96, Issue:1-2

    Topics: Acetanilides; Alkaloids; Animals; Benzodioxoles; Capsaicin; Dose-Response Relationship, Drug; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Nifedipine; Piperidines; Polyunsaturated Alkamides; Purines; Pyrazines; Pyridines; Trachea; TRPV Cation Channels; Urinary Bladder

2015
Action of thymol on spontaneous excitatory transmission in adult rat spinal substantia gelatinosa neurons.
    Neuroscience letters, 2015, Oct-08, Volume: 606

    Topics: Acetanilides; Animals; Capsaicin; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Neurons; Purines; Pyrazines; Pyridines; Rats, Sprague-Dawley; Sodium Channel Blockers; Substantia Gelatinosa; Synaptic Transmission; Tetrodotoxin; Thymol; TRPA1 Cation Channel; TRPC Cation Channels; TRPM Cation Channels

2015
TRPM8 Channel Activation Induced by Monoterpenoid Rotundifolone Underlies Mesenteric Artery Relaxation.
    PloS one, 2015, Volume: 10, Issue:11

    Topics: Animals; Blotting, Western; Calcium; Calcium Signaling; Capsaicin; Cold Temperature; Cytosol; In Vitro Techniques; Ion Channel Gating; Male; Menthol; Mesenteric Arteries; Monoterpenes; Pyrazines; Pyridines; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Ruthenium Red; TRPM Cation Channels; TRPV Cation Channels; Vasodilation

2015
3-Iodothyronamine increases transient receptor potential melastatin channel 8 (TRPM8) activity in immortalized human corneal epithelial cells.
    Cellular signalling, 2016, Volume: 28, Issue:3

    Topics: Calcium; Capsaicin; Cell Line; Epithelial Cells; Humans; Interleukin-6; Membrane Potentials; Patch-Clamp Techniques; Pyrazines; Pyridines; Pyrimidinones; Thyronines; TRPM Cation Channels; TRPV Cation Channels

2016
Radiosensitizing Effect of TRPV1 Channel Inhibitors in Cancer Cells.
    Biological & pharmaceutical bulletin, 2016, Jul-01, Volume: 39, Issue:7

    Topics: Acrylamides; Anilides; Animals; Apoptosis; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cell Line, Tumor; Cell Survival; Cinnamates; DNA Damage; Gamma Rays; Humans; Mice; Necrosis; Neoplasms; Pyrazines; Pyridines; Radiation-Sensitizing Agents; TRPV Cation Channels

2016
Presynaptic facilitation by tetracaine of glutamatergic spontaneous excitatory transmission in the rat spinal substantia gelatinosa - Involvement of TRPA1 channels.
    Brain research, 2017, 02-15, Volume: 1657

    Topics: Acetanilides; Amides; Anesthetics, Local; Animals; Bupivacaine; Capsaicin; Excitatory Postsynaptic Potentials; Glutamic Acid; Levobupivacaine; Male; Neurotransmitter Agents; Pain; Patch-Clamp Techniques; Presynaptic Terminals; Prilocaine; Purines; Pyrazines; Pyridines; Rats, Sprague-Dawley; Ropivacaine; Ruthenium Red; Substantia Gelatinosa; Tetracaine; Tetrodotoxin; Tissue Culture Techniques; TRPA1 Cation Channel; TRPC Cation Channels

2017
Design, synthesis and biological evaluation of cinnamic acid derivatives with synergetic neuroprotection and angiogenesis effect.
    European journal of medicinal chemistry, 2019, Dec-01, Volume: 183

    Topics: Angiogenesis Inducing Agents; Apoptosis; Capsaicin; Cell Line; Cell Survival; Cinnamates; Dose-Response Relationship, Drug; Drug Design; Humans; Membrane Potential, Mitochondrial; Molecular Structure; Neuroprotective Agents; Oxidative Stress; Pyrazines; RNA, Messenger; Structure-Activity Relationship; Vascular Endothelial Growth Factor Receptor-2

2019