Page last updated: 2024-09-04

pumosetrag and granisetron

pumosetrag has been researched along with granisetron in 1 studies

Compound Research Comparison

Studies
(pumosetrag)
Trials
(pumosetrag)
Recent Studies (post-2010)
(pumosetrag)
Studies
(granisetron)
Trials
(granisetron)
Recent Studies (post-2010) (granisetron)
84359016

Protein Interaction Comparison

ProteinTaxonomypumosetrag (IC50)granisetron (IC50)
Solute carrier family 22 member 2Homo sapiens (human)4.3
DRattus norvegicus (Norway rat)3.8019
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)3.8019
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)3.8019
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)3.8019
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)3.8019
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)1.76
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.7702
Multidrug and toxin extrusion protein 1Homo sapiens (human)5
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)1.76

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, NM; Brady, CA; Butler, AS; Choo, SH; Cioffi, CL; Cohen, ML; Dobritsa, S; Earley, WG; Fitzpatrick, K; Guo, C; Guzzo, PR; Hassler, C; Manning, DD; Masih, L; Naginskaya, J; Ryan, KN; Sikkander, MI; Usyatinsky, A; Wierschke, JD; Zhang, Z1

Other Studies

1 other study(ies) available for pumosetrag and granisetron

ArticleYear
Novel serotonin type 3 receptor partial agonists for the potential treatment of irritable bowel syndrome.
    Bioorganic & medicinal chemistry letters, 2011, Jan-01, Volume: 21, Issue:1

    Topics: Animals; Cell Line; Disease Models, Animal; Humans; Imidazoles; Indoles; Irritable Bowel Syndrome; Mice; Microsomes, Liver; Receptors, Serotonin, 5-HT3; Serotonin 5-HT3 Receptor Agonists

2011