Page last updated: 2024-08-16

propranolol and quinacrine

propranolol has been researched along with quinacrine in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19907 (23.33)18.7374
1990's6 (20.00)18.2507
2000's7 (23.33)29.6817
2010's10 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Fitos, I; Mády, G; Visy, J; Zsila, F1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Glen, RC; Lowe, R; Mitchell, JB1
Atzpodien, EA; Csato, M; Doessegger, L; Fischer, H; Lenz, B; Schmitt, G; Singer, T1
Fijorek, K; Glinka, A; Mendyk, A; Polak, S; Wiśniowska, B1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Brun, R; Buckner, FS; Chatterjee, AK; Creason, SA; Duster, NA; Gelb, MH; Gillespie, JR; Glynne, R; Hulverson, MA; McQueen, J; Molteni, V; Nagendar, P; Nagle, A; Norcross, NR; Ranade, RM; Supek, F; Tatipaka, HB; Wenzler, T1
Buckner, FS; Gelb, MH; Gillespie, JR; Herbst, ZM; Montanari, CA; Nguyen, UTT; Ranade, RM; Silva, DG1
Buchynskyy, A; Buckner, FS; Gelb, MH; Gillespie, JR; Herbst, ZM; Ranade, RM1
Abdalla, S; Khalili, F1
Abdalla, S; Afifi, F; al-Khalil, S1
Abdalla, S; Abu-Zarga, M; Sabri, S1
Fassina, G; Froldi, G; Ragazzi, E1
Andrenyak, DM; Epstein, PM; Feinstein, MB; Sha'afi, RI; Volpi, M1
Andrenyak, D; Epstein, PM; Feinstein, MB; Sha'afi, RI; Volpi, M1
Abdel-Latif, AA; Akhtar, RA; Smith, JP1
Lasslo, A1
García-Sancho, J; Herreros, B; Sanchez, A1
Babb, RR1
D'Amore, PA; Dethlefsen, SM; Shepro, D1
Kozawa, O; Oiso, Y; Saito, H; Shinoda, J; Suzuki, A; Watanabe-Tomita, Y1
Dohi, S; Kozawa, O; Matsuno, H; Niwa, M; Tanabe, K; Uematsu, T1
Choi, HJ; Han, JS; Kim, JM; Kim, SC; Lee, KS; Lee, SC; Min, do S; Oh, DY; Oh, KJ1
Cho, JH; Choi, HJ; Han, JS; Lee, JH; Park, SY1
Chen, RK; Jiang, B; Li, XY; Lu, YB; Luo, JY; Wang, Q; Wu, M1

Reviews

2 review(s) available for propranolol and quinacrine

ArticleYear
Blood platelet function, medicinal agents, and other chemical entities.
    Federation proceedings, 1984, Volume: 43, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Amines; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Blood Vessels; Calcium; Cell Membrane; Chlorpromazine; Dipyridamole; Humans; Papaverine; Phospholipids; Platelet Aggregation; Propranolol; Quinacrine; Structure-Activity Relationship; Tretoquinol

1984
Giardiasis. Taming this pervasive parasitic infection.
    Postgraduate medicine, 1995, Volume: 98, Issue:2

    Topics: Antiprotozoal Agents; Giardiasis; Humans; Intestinal Secretions; Metronidazole; Parasite Egg Count; Propranolol; Quinacrine

1995

Other Studies

28 other study(ies) available for propranolol and quinacrine

ArticleYear
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Selective plasma protein binding of antimalarial drugs to alpha1-acid glycoprotein.
    Bioorganic & medicinal chemistry, 2008, Apr-01, Volume: 16, Issue:7

    Topics: Antimalarials; Binding Sites; Chromatography, Affinity; Circular Dichroism; Humans; Molecular Structure; Orosomucoid; Protein Binding; Serum Albumin; Spectrophotometry; Stereoisomerism; Structure-Activity Relationship

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Predicting phospholipidosis using machine learning.
    Molecular pharmaceutics, 2010, Oct-04, Volume: 7, Issue:5

    Topics: Animals; Artificial Intelligence; Databases, Factual; Drug Discovery; Humans; Lipidoses; Models, Biological; Phospholipids; Support Vector Machine

2010
In silico assay for assessing phospholipidosis potential of small druglike molecules: training, validation, and refinement using several data sets.
    Journal of medicinal chemistry, 2012, Jan-12, Volume: 55, Issue:1

    Topics: Animals; Cattle; Cells, Cultured; Computer Simulation; Cornea; Drug-Related Side Effects and Adverse Reactions; Fibroblasts; Lipidoses; Lysosomal Storage Diseases; Models, Molecular; Pharmaceutical Preparations; Phospholipids; Structure-Activity Relationship; Thermodynamics

2012
Predictive model for L-type channel inhibition: multichannel block in QT prolongation risk assessment.
    Journal of applied toxicology : JAT, 2012, Volume: 32, Issue:10

    Topics: Artificial Intelligence; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Computational Biology; Computer Simulation; Drugs, Investigational; Ether-A-Go-Go Potassium Channels; Expert Systems; Heart Rate; Humans; Models, Biological; Myocytes, Cardiac; NAV1.5 Voltage-Gated Sodium Channel; Potassium Channel Blockers; Quantitative Structure-Activity Relationship; Risk Assessment; Shaker Superfamily of Potassium Channels; Torsades de Pointes; Voltage-Gated Sodium Channel Blockers

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Substituted 2-phenylimidazopyridines: a new class of drug leads for human African trypanosomiasis.
    Journal of medicinal chemistry, 2014, Feb-13, Volume: 57, Issue:3

    Topics: Administration, Oral; Animals; Biological Availability; Cell Line, Tumor; Cell Membrane Permeability; Databases, Chemical; Dogs; Female; Humans; Imidazoles; Madin Darby Canine Kidney Cells; Mice; Microsomes, Liver; Pyridines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2014
New Class of Antitrypanosomal Agents Based on Imidazopyridines.
    ACS medicinal chemistry letters, 2017, Jul-13, Volume: 8, Issue:7

    Topics:

2017
1-Benzyl-3-aryl-2-thiohydantoin Derivatives as New Anti-
    ACS medicinal chemistry letters, 2017, Aug-10, Volume: 8, Issue:8

    Topics:

2017
Effects of dichloroglyoxime on isolated guinea-pig smooth muscle and atrium.
    Drug and chemical toxicology, 1992, Volume: 15, Issue:2

    Topics: Animals; Epinephrine; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth, Vascular; Oximes; Propranolol; Quinacrine

1992
Observations on the pharmacology of thalicminine, an oxyaporphine alkaloid from Thalictrum isopyroides.
    General pharmacology, 1991, Volume: 22, Issue:2

    Topics: Animals; Aorta, Thoracic; Aporphines; Arachidonic Acid; Arachidonic Acids; Blood Pressure; Epinephrine; Guinea Pigs; Heart Rate; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Plants, Medicinal; Propranolol; Pulmonary Artery; Quinacrine; Trachea

1991
Preliminary observations on the pharmacology of petaline chloride, a quaternary alkaloid from Leontice leontopetalum.
    General pharmacology, 1989, Volume: 20, Issue:5

    Topics: Alkaloids; Animals; Blood Pressure; Cardiotonic Agents; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Myocardial Contraction; Plants, Medicinal; Propranolol; Quinacrine; Rats

1989
Resveratrol activity on guinea pig isolated trachea from normal and albumin-sensitized animals.
    Pharmacological research communications, 1988, Volume: 20 Suppl 5

    Topics: Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; Guinea Pigs; Immunization; In Vitro Techniques; Male; Masoprocol; Muscle Contraction; Ovalbumin; Propranolol; Quinacrine; Resveratrol; Stilbenes; Trachea

1988
Local anesthetics, mepacrine, and propranolol are antagonists of calmodulin.
    Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Anesthetics, Local; Animals; Brain; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Cyclic Nucleotide Phosphodiesterases, Type 1; Dibucaine; Drug Antagonism; Enzyme Activation; Erythrocyte Membrane; Erythrocytes; Humans; Kinetics; Propranolol; Quinacrine; Rats

1981
Antagonism of calmodulin by local anesthetics, mepacrine, and propranolol.
    Annals of the New York Academy of Sciences, 1980, Volume: 356

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Anesthetics, Local; Animals; Brain; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Drug Antagonism; Enzyme Activation; Erythrocyte Membrane; Humans; Kinetics; Propranolol; Quinacrine; Rats

1980
Studies on the mechanism of alteration by propranolol and mepacrine of the metabolism of phosphoinositides and other glycerolipids in the rabbit iris muscle.
    Biochemical pharmacology, 1983, Dec-15, Volume: 32, Issue:24

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; In Vitro Techniques; Iris; Microsomes; Muscle, Smooth; Phosphatidylinositols; Phospholipids; Propranolol; Quinacrine; Rabbits

1983
Effects of several inhibitors on the K+ efflux induced by activation of the Ca2+-dependent channel and by valinomycin in the human red cell.
    FEBS letters, 1980, Jan-28, Volume: 110, Issue:1

    Topics: Antimycin A; Calcimycin; Chlorides; Chlorpromazine; Dipyridamole; Erythrocytes; Humans; Ion Channels; Oligomycins; Potassium; Propranolol; Quinacrine; Sodium; Valinomycin

1980
Arachidonic acid metabolites in bFGF-, PDGF-, and serum-stimulated vascular cell growth.
    Experimental cell research, 1994, Volume: 212, Issue:2

    Topics: Animals; Arachidonic Acid; Cattle; Cell Division; Cells, Cultured; Cyclooxygenase Inhibitors; Endothelium, Vascular; Fibroblast Growth Factor 2; Flavanones; Flavonoids; In Vitro Techniques; Lipoxygenase Inhibitors; Masoprocol; Muscle, Smooth, Vascular; Phospholipase D; Phospholipases A; Phospholipases A2; Platelet-Derived Growth Factor; Propranolol; Quinacrine; Signal Transduction

1994
Mechanism of thrombin-induced arachidonic acid release in osteoblast-like cells.
    Prostaglandins, leukotrienes, and essential fatty acids, 1997, Volume: 56, Issue:6

    Topics: 3T3 Cells; Animals; Arachidonic Acid; Cyclohexanones; Dinoprostone; Enzyme Inhibitors; Estrenes; Lipoprotein Lipase; Mice; Osteoblasts; Phosphatidate Phosphatase; Phospholipases A; Phospholipases A2; Propranolol; Pyrrolidinones; Quinacrine; Thrombin; Type C Phospholipases

1997
Effect of propofol on arachidonate cascade by vasopressin in aortic smooth muscle cells: inhibition of PGI2 synthesis.
    Anesthesiology, 1999, Volume: 90, Issue:1

    Topics: Anesthetics, Intravenous; Animals; Aorta, Thoracic; Arachidonic Acid; Arginine Vasopressin; Cells, Cultured; Choline; Enzyme Inhibitors; Epoprostenol; Estrenes; Humans; Inositol Phosphates; Muscle, Smooth, Vascular; Phospholipases; Propofol; Propranolol; Pyrrolidinones; Quinacrine; Rats; Vasoconstrictor Agents; Vasopressins

1999
Role of phospholipase D2 in anti-apoptotic signaling through increased expressions of Bcl-2 and Bcl-xL.
    Journal of cellular biochemistry, 2007, Aug-15, Volume: 101, Issue:6

    Topics: Animals; Antihypertensive Agents; Apoptosis; bcl-X Protein; Cell Line; Cell Survival; Cyclooxygenase 2; Enzyme Inhibitors; fas Receptor; Mice; Palmitates; Phosphatidic Acids; Phospholipase D; Propranolol; Proto-Oncogene Proteins c-bcl-2; Quinacrine; Signal Transduction

2007
STAT3 is involved in phosphatidic acid-induced Bcl-2 expression in HeLa cells.
    Experimental & molecular medicine, 2009, Feb-28, Volume: 41, Issue:2

    Topics: Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; HeLa Cells; Humans; Mitogen-Activated Protein Kinase Kinases; Phosphatidic Acids; Propranolol; Proto-Oncogene Proteins c-bcl-2; Quinacrine; RNA, Small Interfering; STAT3 Transcription Factor

2009
Activation of phospholipase D involved in both injury and survival in A549 alveolar epithelial cells exposed to H2O2.
    Toxicology letters, 2010, Jul-15, Volume: 196, Issue:3

    Topics: Cell Survival; Cells, Cultured; Enzyme Activation; Epithelial Cells; Humans; Hydrogen Peroxide; Phosphatidic Acids; Phospholipase D; Propranolol; Pulmonary Alveoli; Quinacrine; Reactive Oxygen Species

2010