propranolol has been researched along with cgp 20712a in 34 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (5.88) | 18.7374 |
1990's | 14 (41.18) | 18.2507 |
2000's | 15 (44.12) | 29.6817 |
2010's | 3 (8.82) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL | 1 |
Baker, JG | 1 |
Duke, BJ; Jackman, GP; Louis, SN; Louis, WJ; Machida, CA; Nero, TL; Rezmann-Vitti, LA | 1 |
Cantillon, DM; Derudas, M; Huckvale, R; Kenyon, EJ; Kirkwood, NK; Kros, CJ; O'Reilly, M; Richardson, GP; Waddell, SJ; Ward, SE | 1 |
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P | 1 |
Choi, AL; Martínez de la Escalera, G; Weiner, RI | 1 |
Blanksma, PK; Bouwer, J; Elsinga, PH; Lie, KI; Meeder, JG; Paans, AM; Vaalburg, W; van Waarde, A; Visser, GM | 1 |
Grino, M; Oliver, C | 1 |
Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
Holzer, G; Künster, A; Wessler, I | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Hadcock, JR; Malbon, CC | 1 |
MacDonald, A; McKean, J | 1 |
Collins, S; Daniel, KW; Kozak, LP; Premont, RT; Rohlfs, EM | 1 |
Collins, S; Daniel, KW; Gettys, TW; Ramkumar, V; Rohlfs, EM; Taylor, IL | 1 |
Doze, P; Elsinga, PH; Ensing, K; Kraan, J; Vaalburg, W; van der Mark, TW; van Waarde, A; Visser, TJ | 1 |
Antunes, E; Brain, SD; Costa, SK; de Nucci, G; Hyslop, S; Nathan, LP; Zanesco, A | 1 |
Atgié, C; Berlan, M; Carpéné, C; Fontana, E; Galitzky, J; Lafontan, M | 1 |
Carson, PE | 1 |
Brawley, L; MacDonald, A; Shaw, AM | 1 |
Beiler, RJ; Commins, SP; Gettys, TW; Levin, N; Watson, PM | 1 |
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S | 1 |
Santos, IN; Spadari-Bratfisch, RC | 1 |
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K; Yoshida, K | 1 |
Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
Corleto, VD; Delle Fave, G; Romano, G; Severi, C; Tattoli, I | 1 |
Christ, T; Kaumann, A; Molenaar, P; Ravens, U | 1 |
Horinouchi, T; Koike, K; Michikawa, H; Tanaka, Y; Yamashita, Y | 1 |
Chartier, D; Ehrlich, JR; Hébert, TE; Nattel, S; Qi, X; Yeh, YH | 1 |
Chen, P; Liu, Z; Ma, K; Yang, H; Zhang, Y; Zhou, C | 1 |
Gong, KZ; Guo, JH; Song, Y; Xia, Y; Xu, M; Zhang, P; Zhang, YY | 1 |
Cho, KW; Choi, DH; Choi, HR; Cui, HZ; Kang, DG; Lee, HS | 1 |
Barnes, JL; Ghosh, PM; Ikeno, Y; Kamat, A; Katz, MS; Lu, Z; Shu, ZJ; Yeh, CK; Zhang, BX; Zhu, B | 1 |
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB | 1 |
1 review(s) available for propranolol and cgp 20712a
Article | Year |
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Beta-blocker therapy in heart failure: pathophysiology and clinical results.
Topics: Adrenergic beta-Antagonists; Aged; Bisoprolol; Carbazoles; Carvedilol; Clinical Trials as Topic; Exercise; Heart Failure; Heart Rate; Hemodynamics; Humans; Imidazoles; Male; Metoprolol; Middle Aged; Propanolamines; Propranolol; Quality of Life; Stroke Volume; Time Factors; Vasodilator Agents; Xamoterol | 1999 |
33 other study(ies) available for propranolol and cgp 20712a
Article | Year |
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LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea | 1999 |
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2005 |
Role of Tyr(356(7.43)) and Ser(190(4.57)) in antagonist binding in the rat beta1-adrenergic receptor.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Models, Molecular; Mutagenesis, Site-Directed; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Serine; Stereoisomerism; Transfection; Tyrosine | 2006 |
Design, Synthesis, and Biological Evaluation of a New Series of Carvedilol Derivatives That Protect Sensory Hair Cells from Aminoglycoside-Induced Damage by Blocking the Mechanoelectrical Transducer Channel.
Topics: Aminoglycosides; Animals; Carvedilol; Chemistry Techniques, Synthetic; Cytoprotection; Dose-Response Relationship, Drug; Drug Design; Electrophysiological Phenomena; Hair Cells, Auditory; Mechanotransduction, Cellular; Mice; Zebrafish | 2019 |
Influence of age on the beta 1- and beta 2-adrenergic receptors in rat liver.
Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Cell Membrane; Imidazoles; Liver; Liver Glycogen; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1992 |
Beta 1-adrenergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via receptors positively coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Line; Cyclic AMP; Gonadotropin-Releasing Hormone; Imidazoles; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Neurons; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, LHRH | 1992 |
Suitability of CGP-12177 and CGP-26505 for quantitative imaging of beta-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Imidazoles; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Time Factors; Tissue Distribution; Tritium | 1992 |
Ontogeny of insulin-induced hypoglycemia stimulation of adrenocorticotropin secretion in the rat: role of catecholamines.
Topics: Adrenergic beta-Antagonists; Adrenocorticotropic Hormone; Aging; Animals; Arginine Vasopressin; Catecholamines; Hypoglycemia; Imidazoles; Immunization, Passive; Insulin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1992 |
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection | 1991 |
Stimulation of beta 1-adrenoceptors enhances electrically evoked [3H]-acetylcholine release from rat phrenic nerve.
Topics: Acetylcholine; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Female; Fenoterol; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Phentolamine; Phrenic Nerve; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Tritium | 1990 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Down-regulation of beta-adrenergic receptors: agonist-induced reduction in receptor mRNA levels.
Topics: Adrenergic beta-Antagonists; Animals; Cell Line; Cricetinae; Cyclic AMP; DNA; Endonucleases; Imidazoles; Isoproterenol; Kinetics; Male; Nucleic Acid Hybridization; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA, Messenger; Single-Strand Specific DNA and RNA Endonucleases; Vas Deferens | 1988 |
Contributions of beta-adrenoceptor subtypes to responses to isoprenaline in rat isolated distal colon.
Topics: Animals; Colon; Imidazoles; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1995 |
Regulation of the uncoupling protein gene (Ucp) by beta 1, beta 2, and beta 3-adrenergic receptor subtypes in immortalized brown adipose cell lines.
Topics: Adenylyl Cyclases; Adipocytes; Adipose Tissue, Brown; Animals; Base Sequence; Binding, Competitive; Carrier Proteins; Cell Line; Cell Membrane; Dioxoles; DNA Primers; Gene Expression; Imidazoles; Ion Channels; Isoenzymes; Kinetics; Lipid Metabolism; Membrane Proteins; Mice; Mice, Inbred C57BL; Mitochondrial Proteins; Molecular Sequence Data; Norepinephrine; Propranolol; Receptors, Adrenergic, beta; RNA, Messenger; Uncoupling Protein 1 | 1995 |
Impaired expression and functional activity of the beta 3- and beta 1-adrenergic receptors in adipose tissue of congenitally obese (C57BL/6J ob/ob) mice.
Topics: Adenylyl Cyclases; Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Activation; Epinephrine; Gene Expression Regulation; Hyperglycemia; Imidazoles; Lipolysis; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Obesity; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA Splicing; RNA, Messenger | 1994 |
Characterisation of beta2-adrenoceptors, using the agonist [11C]formoterol and positron emission tomography.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbon Radioisotopes; Ethanolamines; Formoterol Fumarate; Imidazoles; Isoproterenol; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta-2; Tissue Distribution; Tomography, Emission-Computed | 1998 |
Activation by Phoneutria nigriventer spider venom of autonomic nerve fibers in the isolated rat heart.
Topics: Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Animals; Anti-Arrhythmia Agents; Arachnida; Atropine; Autonomic Nervous System; Butoxamine; Capsaicin; Cardiac Output; Heart; Hypertension; Hypotension; Imidazoles; In Vitro Techniques; Male; Propranolol; Rats; Rats, Wistar; Reserpine; Spider Venoms | 1998 |
Selective activation of beta3-adrenoceptors by octopamine: comparative studies in mammalian fat cells.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adult; Animals; Binding, Competitive; Biogenic Amines; Bupranolol; CHO Cells; Cricetinae; Dioxoles; Dogs; Ethanolamines; Female; Gene Expression; Guinea Pigs; Humans; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lipolysis; Male; Mammals; Mesocricetus; Norepinephrine; Octopamine; Oxygen Consumption; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Species Specificity | 1999 |
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents | 2000 |
Central leptin regulates the UCP1 and ob genes in brown and white adipose tissue via different beta-adrenoceptor subtypes.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Carrier Proteins; Cell Membrane; Cerebral Ventricles; Gene Expression Regulation; Imidazoles; Injections, Intraventricular; Ion Channels; Leptin; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Mitochondrial Proteins; Propanolamines; Propranolol; Receptors, Adrenergic, beta-3; Receptors, Leptin; RNA, Messenger; Transcription, Genetic; Uncoupling Protein 1 | 2000 |
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes | 2000 |
Chronotropic response to (+/-)-CGP12177 in right atria of stressed rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Heart Atria; Heart Rate; Imidazoles; In Vitro Techniques; Male; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Physiological; Time Factors | 2001 |
Role of beta-adrenoceptor subtypes in mediating relaxation of the pig bladder trigonal muscle in vitro.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Swine; Urinary Bladder | 2003 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Beta3-adrenoceptors: relaxant function and mRNA detection in smooth muscle cells isolated from the human colon.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Colon; Gastrointestinal Motility; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Myocytes, Smooth Muscle; Propranolol; Receptors, Adrenergic, beta-3; RNA, Messenger; Tetrahydronaphthalenes | 2004 |
Carvedilol blocks beta2- more than beta1-adrenoceptors in human heart.
Topics: Adrenergic beta-Antagonists; Calcium Channels, L-Type; Carbazoles; Carvedilol; Dose-Response Relationship, Drug; Epinephrine; Heart Atria; Heart Failure; Heart Ventricles; Humans; Imidazoles; In Vitro Techniques; Metoprolol; Myocardial Contraction; Myocardium; Norepinephrine; Patch-Clamp Techniques; Propanolamines; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 2006 |
Pharmacological characterization of the beta-adrenoceptor that mediates the relaxant response to noradrenaline in guinea-pig tracheal smooth muscle.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Albuterol; Animals; Atenolol; Bupranolol; Butoxamine; Desipramine; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Trachea | 2007 |
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes.
Topics: Acetylcholine; Action Potentials; Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bee Venoms; Clonidine; Cyclic AMP-Dependent Protein Kinases; Dihydropyridines; Dogs; Dose-Response Relationship, Drug; Estrenes; Heart Atria; Imidazoles; Indoles; Isoproterenol; Isoquinolines; Maleimides; Myocytes, Cardiac; Patch-Clamp Techniques; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Potassium Channels; Prazosin; Propanolamines; Propranolol; Protein Kinase C; Pyrrolidinones; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Sulfonamides; Type C Phospholipases | 2007 |
Mouse embryonic stem cell-derived cardiomyocytes express functional adrenoceptors.
Topics: Animals; Cell Differentiation; Cell Line; Embryonic Stem Cells; Extracellular Signal-Regulated MAP Kinases; Gene Expression; Imidazoles; Isoproterenol; Mice; Myocytes, Cardiac; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptor, Muscarinic M2; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Tyrosine 3-Monooxygenase | 2008 |
Regulation of gap-junction protein connexin 43 by beta-adrenergic receptor stimulation in rat cardiomyocytes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Cells, Cultured; Connexin 43; Cyclic AMP-Dependent Protein Kinases; Gap Junctions; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Imidazoles; Isoproterenol; Myocytes, Cardiac; Pertussis Toxin; Propranolol; Protein Isoforms; Protein Phosphatase 2; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Signal Transduction | 2009 |
Aqueous extract of Zanthoxylum schinifolium elicits contractile and secretory responses via beta1-adrenoceptor activation in beating rabbit atria.
Topics: Animals; Atrial Natriuretic Factor; Blood Pressure; Carbazoles; Cardiotonic Agents; Cardiovascular Agents; Cyclic AMP; Diltiazem; Heart Atria; Hemodynamics; Imidazoles; Plant Extracts; Plant Leaves; Plant Stems; Propanolamines; Propranolol; Pyrroles; Rabbits; Receptors, Adrenergic, beta-1; Stroke Volume; Zanthoxylum | 2009 |
Role of β-adrenergic receptors in regulation of hepatic fat accumulation during aging.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Cells, Cultured; Enzyme Activation; Fats; Hepatocytes; Imidazoles; Isoproterenol; Lipids; Liver; Male; Mice; Mice, Inbred C57BL; Propanolamines; Propranolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Time Factors | 2012 |
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei | 2012 |