proline and sdz nkt 343

proline has been researched along with sdz nkt 343 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brown, MC; Buchheit, KH; Campbell, EA; Docherty, R; Ewan, S; Hedley, L; James, IF; Ko, S; McIntyre, P; Urban, LA; Walpole, CS1
Beattie, D; Brown, M; Campbell, E; Dickenson, F; Ewan, S; Hughes, GA; Ko, SY; Lemaire, M; Lerpiniere, J; Patel, S; Urban, L; Walpole, C1
Rees, H; Sluka, KA; Urban, L; Walpole, CJ; Willis, WD1
Campbell, EA; Gentry, CT; Panesar, MS; Patel, S; Urban, L; Walpole, CS1
Campbell, EA; Cruwys, S; Fox, AJ; Gentry, C; Kidd, B; Patel, S; Urban, L1

Other Studies

5 other study(ies) available for proline and sdz nkt 343

ArticleYear
Comparative, general pharmacology of SDZ NKT 343, a novel, selective NK1 receptor antagonist.
    British journal of pharmacology, 1998, Volume: 124, Issue:1

    Topics: Animals; Base Sequence; Binding Sites; Cell Line; COS Cells; DNA Primers; Ganglia, Spinal; Gerbillinae; Guinea Pigs; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Naphthalenes; Neurokinin-1 Receptor Antagonists; Proline; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Recombinant Proteins; Substance P

1998
2-Nitrophenylcarbamoyl-(S)-prolyl-(S)-3-(2-naphthyl)alanyl-N-benzyl-N - methylamide (SDZ NKT 343), a potent human NK1 tachykinin receptor antagonist with good oral analgesic activity in chronic pain models.
    Journal of medicinal chemistry, 1998, Aug-13, Volume: 41, Issue:17

    Topics: Analgesics; Animals; Aspirin; Binding, Competitive; Brain; Drug Design; Guinea Pigs; Humans; Hyperalgesia; Kinetics; Molecular Structure; Naphthalenes; Neurokinin-1 Receptor Antagonists; Pain; Phenylthiourea; Proline; Rabbits; Rats; Receptors, Neurokinin-1; Spectrometry, Mass, Fast Atom Bombardment; Structure-Activity Relationship

1998
The effects of SDZ NKT 343, a potent NK1 receptor antagonist, on cutaneous responses of primate spinothalamic tract neurones sensitized by intradermal capsaicin injection.
    Experimental brain research, 1998, Volume: 121, Issue:3

    Topics: Action Potentials; Animals; Capsaicin; Electrophysiology; Haplorhini; Injections, Intradermal; Male; Naphthalenes; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Proline; Skin; Spinothalamic Tracts; Substance P

1998
Selective neurokinin-1 receptor antagonists are anti-hyperalgesic in a model of neuropathic pain in the guinea-pig.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: Administration, Oral; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Guinea Pigs; Hyperalgesia; Indoles; Injections, Spinal; Isoindoles; Naphthalenes; Nerve Fibers; Neuralgia; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Piperidines; Proline; Receptors, Neurokinin-1; Spinal Cord

1998
Oral anti-hyperalgesic and anti-inflammatory activity of NK(1) receptor antagonists in models of inflammatory hyperalgesia of the guinea-pig.
    Pain, 2000, Volume: 87, Issue:3

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Carrageenan; Disease Models, Animal; Female; Freund's Adjuvant; Guinea Pigs; Humans; Hyperalgesia; Indoles; Isoindoles; Male; Naphthalenes; Neurokinin-1 Receptor Antagonists; Piperidines; Proline; Quinuclidines

2000