proglumide and sincalide
proglumide has been researched along with sincalide in 176 studies
Research
Studies (176)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 67 (38.07) | 18.7374 |
1990's | 78 (44.32) | 18.2507 |
2000's | 26 (14.77) | 29.6817 |
2010's | 4 (2.27) | 24.3611 |
2020's | 1 (0.57) | 2.80 |
Authors
Authors | Studies |
---|---|
Collins, KA; Suh, HH; Tseng, LF | 1 |
Rozengurt, E; Sethi, T | 1 |
Brenner, L; Ritter, RC; Yox, DP | 1 |
Bishop, LA; Black, JW; Gerskowitch, VP; Hull, RA; Shankley, NP | 1 |
Berry, P; Botella, A; Bueno, L; Delvaux, M; Frexinos, J | 1 |
Almegård, B; Bill, A; Stjernschantz, J | 1 |
Nagy, I; Pap, A; Takács, T; Varró, V | 2 |
Fujii, N; Funakoshi, A; Miyasaka, K; Shinozaki, H; Wakasugi, H | 1 |
Galas, MC; Lignon, MF; Martinez, J; Nagain, C; Rodriguez, M; Rozé, C | 1 |
Giovanetti, R; Makovec, F; Mennuni, L; Peris, W; Revel, L; Rovati, LC | 1 |
De Saint Hilaire-Kafi, Z; Gaillard, JM; Vallet, PG | 1 |
Chang, TM; Chey, WY; Jo, YH; Lee, KY | 1 |
Han, JS; Wang, XH; Wang, XJ | 2 |
Gaginella, TS; Kachur, JF; Phillips, GS | 1 |
Colton, DG; Dodds, WJ; Hanyu, N; Hogan, WJ; Layman, RD | 1 |
Andrus, C; Kaminski, DL; Schlarman, D; Westfall, S | 1 |
Bennett, A; D'Amato, M; Stamford, IF | 1 |
Kellstein, DE; Mayer, DJ; Price, DD | 1 |
Bennet, L; Gluckman, PD; Johnston, BM | 1 |
Suh, HH; Tseng, LF | 1 |
Brandonisio, R; Chiloiro, M; Di Ciaula, A; Maggi, V; Palasciano, G; Portincasa, P | 1 |
Agnati, LF; Ferraro, L; Fuxe, K; Tanganelli, S; Ungerstedt, U; von Euler, G | 1 |
Baba, H; Fujimura, M; Toda, N | 1 |
Konda, Y; Matozaki, T; Nagao, M; Nakano, O; Nishisaki, H; Sakamoto, C | 1 |
Gardner, JD; Howard, JM; Jensen, RT; Jones, SW; Murphy, RB; Schneider, LH; Trampota, M | 1 |
Johnson, LR; Tabata, K; Yamaguchi, T | 1 |
Murase, K; Randić, M; Urban, L; Willetts, J | 1 |
Grendell, JH; Niederau, C; Niederau, M; Williams, JA | 1 |
Gardner, JD; Jensen, RT; Jones, SW; Murphy, RB; Rovati, LA; Setnikar, I; Zhou, ZC | 1 |
Burks, TF; Shook, JE | 1 |
Iwamoto, Y; Kuzuya, T; Yamamoto, R | 1 |
Grendell, JH; Liddle, RA; Niederau, C; Williams, JA | 1 |
Hill, RG; Hughes, J; Rodriguez, RE | 1 |
Liang, JP; Louie, DS; Owyang, C | 1 |
Baba, S; Fujii, M; Fujisawa, T; Koide, M; Nakamura, T; Okabayashi, Y; Otsuki, M; Tani, S | 3 |
Chang, JH; Moriyoshi, Y; Shimizu, K; Shiratori, K; Takeuchi, T; Watanabe, S | 1 |
Gardner, JD; Jensen, RT; Maton, PN; Menozzi, D | 1 |
Gomez, G; Green, D; Rajaraman, S; Thompson, JC; Townsend, CM; Uchida, T | 1 |
Debas, HT; Mulholland, MW | 1 |
Bednar, I; Forsberg, G; Lindén, A; Södersten, P; Uvnäs-Moberg, K | 1 |
Guo, YS; Houston, CW; Jin, GF | 1 |
Baba, S; Inui, A; Sakatani, N | 1 |
Brinn, JE; Fletcher, DJ; Pabst, SJ; Rowley, WH | 1 |
de Jong, AJ; Douglas, BR; Jansen, JB; Lamers, CB; Rovati, LC; Woutersen, RA | 1 |
Han, JS; Li, Y | 1 |
Bogdal, J; Konturek, JW; Konturek, SJ; Kurek, A; Oleksy, J; Rovati, L | 1 |
Altar, AC; Cosi, C; Wood, PL | 1 |
Aprahamian, M; Damgé, C; Hajri, A | 1 |
Sinton, CM | 2 |
Murphy, RB; Schneider, LH; Smith, GP | 1 |
Stabile, BE; Stubbs, RS | 1 |
Bitar, KN; Makhlouf, GM | 1 |
Furukawa, T; Harada, T; Katsuragi, T | 1 |
Barone, FC; Bondinell, WE; Labosh, TJ; Ormsbee, HS; White, RF | 1 |
Itoh, S; Katsuura, G | 2 |
Chang, RS; Chen, TB; Lotti, VJ | 1 |
Goyal, RK; Rattan, S | 1 |
Crawley, JN; Hommer, DW; Paul, SM; Skirboll, LR; Stivers, JA | 1 |
Bani, M; Chisté, R; Makovec, F; Revel, L; Rovati, LA; Rovati, LC | 1 |
Ammon, HP; Goldfine, ID; Verspohl, EJ; Williams, JA; Wunderle, G | 1 |
Davison, JS; Kerrin, JP; MacVicar, BA | 1 |
Aitken, PG; Jaffe, DB; Nadler, JV | 1 |
Jiang, LH; Kasser, RJ; Wang, RY | 1 |
Funakoshi, A; Kitani, K; Miyasaka, K; Nakamura, R | 1 |
Chase, TN; Nilaver, G; Tamminga, CA; Tanimoto, K | 1 |
Fujimura, M; Gomez, G; Greeley, GH; Guo, YS; Lluis, F; Lonovics, J; Thompson, JC; Townsend, CM | 1 |
Beglinger, C; Gyr, K; Hildebrand, P; Köhler, E; Setnikar, I | 1 |
Bani, M; Chistè, R; Makovec, F; Revel, L; Rovati, LC; Setnikar, I | 1 |
Baba, S; Inoue, T; Inui, A; Morioka, H; Oya, M; Sakatani, N | 1 |
Izzo, RS; Praissman, M | 1 |
Bednar, I; Forsberg, G; Hansen, S; Lindén, A; Södersten, P; Uvnäs-Moberg, K | 1 |
Deupree, D; Hsiao, S | 1 |
Biziere, K; Briet, C; Castro, B; Martinez, J; Worms, P | 1 |
Go, VL; Schick, RR; Yaksh, TL | 1 |
Cerino, DJ; Change, RS; Kling, PJ; Lotti, VJ | 1 |
Grider, JR; Makhlouf, GM | 1 |
Korc, M; Magun, BE | 1 |
Hsiao, S; Itoh, S; Katsuura, G | 1 |
Collins, SM; Conover, KL; Forsyth, PA; Weingarten, HP | 1 |
Nemeth, PR; Wood, JD; Zafirov, DH | 1 |
Schneider, LH | 1 |
Ambrose, FG; Autry, WL; Barbaz, BS; Gerber, R; Liebman, JM | 1 |
Magnani, M; Mantovani, P; Pepeu, G | 1 |
Wang, RY; White, FJ | 1 |
Akanuma, Y; Iwamoto, Y; Nakamura, R | 1 |
Collins, SM; Gardner, JD | 1 |
Da Silva, AM; Garvey, TQ; Gillis, RA; Hamosh, P; Jensen, RT; Pagani, FD; Quest, JA; Souza, JD | 1 |
Ito, H; Kadowaki, M; Matsuo, M; Nakarai, T; Sato, Y; Sogabe, H; Tokoro, K; Tomoi, M; Yoshida, K | 1 |
Chan, MY; Tang, F | 1 |
Williams, JA; Yule, DI | 1 |
Kashima, K; Kataoka, K; Kato, M; Kuriyama, K; Mukainaka, T; Ohkuma, S | 1 |
Moriyoshi, Y; Shiratori, K; Takeuchi, T; Watanabe, S | 1 |
Gaw, AJ; Hills, DM; Spraggs, CF | 1 |
Chen, JH; Wang, XC; Wu, FM; Zhang, WN; Zheng, YL | 1 |
De Pont, JJ; Hoenderop, JG; Van Emst-De Vries, SE; Van Hoof, HJ; Van Mackelenbergh, MG; Willems, PH | 1 |
Fölsch, UR; Höcker, M; Hughes, J; Schmidt, WE | 1 |
Fujii, K; Haruma, K; Kajiyama, G; Kishimoto, S; Kobayashi, H; Machino, H; Miyoshi, A | 1 |
Chey, WY; Imamura, M; Yamauchi, H | 1 |
Bourin, M; Bradwejn, J; Harro, J; Lang, A; Vasar, E | 1 |
Aufderhaar, U; Bauerfeind, P; Beglinger, C; Burckhardt, B; Delco, F; Ensinck, JW; Gyr, K; Ketterer, S; Meier, R | 1 |
Nakano, S; Otsuki, M; Tachibana, I | 1 |
Wang, SX | 1 |
Akiyama, T; Otsuki, M | 1 |
Beglinger, C | 1 |
Bekkering, M; Chua, AS; Keeling, PW; Rovati, LC | 1 |
Ohtsuka, T; Yokose, K | 1 |
Han, JS; Mei, L | 1 |
Fukumoto, M; Hayashi, H; Imamura, M; Kawabata, K; Manabe, T; Masai, Y; Morimoto, H; Nio, Y; Tsubono, M | 1 |
Albus, K; Baumfalk, U; Hicks, TP; Kaneko, T | 1 |
Aprahamian, M; Damgé, C; Doffoël, M; Garaud, JC; Hajri, A; Karsenty, L | 1 |
Choi, YS; Kim, YH; Song, DK; Suh, HW | 1 |
Funakoshi, A; Miyasaka, K; Nakamura, E; Teraoka, H | 1 |
Rakovska, A | 2 |
Brotschi, EA; Hilbinger, CL; Kahl, EA; Midis, NA; Vaules, WA | 1 |
Arii, S; Funaki, N; Imamura, M; Imamura, T; Kohmoto, M; Ohshio, G; Okada, N; Sasaoki, T; Tanaka, J; Tanaka, T; Wang, ZH; Yoshida, M | 1 |
Akiyama, T; Hirohata, Y; Otsuki, M; Shirohara, H; Tachibana, I; Yamamoto, M | 1 |
Dickenson, JM; Hill, SJ | 1 |
D'Amato, M; Kisfalvi, I; Scarpignato, C; Varga, G | 1 |
Endo, T; Nagasaki, M; Taniguchi, H; Yazaki, N | 1 |
Beglinger, C; Hartel, M; Niebergall-Roth, E; Riepl, RL; Singer, MV; Teyssen, S; Wetzel, D | 1 |
Endo, T; Nagasaki, M; Shikano, T; Taniguchi, H; Yazaki, N; Yomota, E | 1 |
Hanada, K; Hirata, M; Itoh, M; Kajiyama, G; Ooishi, H; Tsuchida, A | 1 |
Cheeseman, CI; Hirsh, AJ; Kammila, S; Tsang, R | 1 |
Kondo, T; Liu, F; Naruse, S; Ozaki, T; Sazi, T; Toda, Y | 1 |
Corp, ES; Curcio, M; Gibbs, J; Smith, GP | 1 |
Dunlop, J; Evans, N; Zhang, Y | 1 |
Adler, G; Beckh, K; Dirks, A; Koop, H; Koop, I | 1 |
Iwaki, N; Kato, S; Kogishi, K; Mineo, H; Onaga, T; Zabielski, R | 1 |
Kihara, Y; Nakano, S; Otsuki, M | 1 |
Hayashi, K; Kannbe, M; Kishimoto, S | 1 |
Azpiroz, F; Clavé, P; Cussó, X; D'Amato, M; Farré, A; González, A; Lluís, F; López, R; Moreno, A | 1 |
Johnson, AK; Menani, JV | 1 |
Akagi, Y; Eguchi, R; Itoh, N; Muto, N; Tanaka, K | 1 |
Domschke, W; Hengst, K; Konturek, JW; Konturek, SJ; Sito, E; Stachura, J | 1 |
Brzozowska, I; Brzozowski, T; Hahn, EG; Konturek, PC; Konturek, SJ; Kwiecién, S; Pajdo, R | 1 |
Akiyama, T; Hirohata, Y; Kihara, Y; Otsuki, M; Tashiro, M | 1 |
Brzozowski, T; Drozdowicz, D; Hahn, EG; Konturek, PC; Konturek, SJ; Kwiecień, S; Pajdo, R | 1 |
Edwards, GL; Power, JD | 1 |
Beglinger, C; Drewe, J; Gutzwiller, JP; Hildebrand, P; Ketterer, S; Krautheim, A | 1 |
Capellà, G; Clavé, P; Farré, R; González, AA; Monés, J | 1 |
De Luca, LA; Fratucci De Gobbi, JI; Johnson, AK; Menani, JV | 1 |
Aloe, L; Lundeberg, T; Manni, L; Tirassa, P | 1 |
Ivanov, AI; Kulchitsky, VA; Romanovsky, AA | 1 |
Akiyama, T; Fukumitsu, K; Jia, DM; Otani, M; Otsuki, M; Yamamoto, M; Yoshikawa, H | 1 |
Guimarães, FS; Netto, CF | 1 |
He, RR; Liu, YX; Ma, HJ; Zhang, H | 1 |
Cox, JE; Kelm, GR; Meller, ST; Randich, A | 1 |
Mostofsky, DI; Yehuda, S | 1 |
Bartolomé-Nebreda, JM; Cenarruzabeitia, E; Del Río, J; García-López, MT; González-Muñiz, R; Herranz, R; Latorre, M | 1 |
Cong, B; Gao, WJ; Gu, ZY; Xu, SJ; Yao, YX | 1 |
Baptista, V; Coleman, FH; Rogers, RC; Travagli, RA; Zheng, ZL | 1 |
Acuña-Castroviejo, D; Escames, G; García-Navarro, A; González-Puga, C; León, J; López-Cantarero, M; Ros, E | 1 |
Thavanathan, R; Volkoff, H | 1 |
Cong, B; Gao, WJ; Gu, ZY; Li, SJ; Ling, YL; Ma, CL; Xu, SJ; Yao, YX | 1 |
Micevych, P; Quesada, A | 1 |
Cong, B; Gao, F; Gu, ZY; Ling, YL; Liu, X; Ma, LQ; Ping, J; Wang, XY; Xu, JR; Yan, YX; Zhao, L | 1 |
Aloj, L; De Luca, S; Lassiani, L; Morelli, G; Saviano, M; Stefanidou, P; Varnavas, A; Yannakopoulou, K | 1 |
Cruz-Vera, J; Diaz-Zagoya, JC; Flores-Murrieta, FJ; Granados-Soto, V; Juárez-Rojop, IE; Ortíz-López, JU; Torres-López, JE | 1 |
Travagli, RA; Viard, E; Wan, S; Zheng, Z | 1 |
Coleman, FH; Travagli, RA; Wan, S | 1 |
Davidson, WS; Liu, M; Lo, CM; Ma, L; Pearson, K; Raybould, HE; Sakai, RR; Sun, W; Tso, P; Woods, SC; Zhang, DM | 1 |
Doong, ML; Wang, PS; Wu, CL | 1 |
Gao, LP; Liu, JF; Lu, HL; Sun, J; Wang, QZ; Wen, SW; Zhang, J; Zhang, SW | 1 |
Hara, I; Hayashi, H; Kagawa, K; Kirisawa, R; Onaga, T; Sugita, A; Wakaiki, R | 1 |
Cevik-Aras, H; Ekström, J | 1 |
Crespo, I; Gómez de Heras, R; López-Moreno, JA; Orio, L; Reyes-Cabello, C; Rodríguez de Fonseca, F | 1 |
Drew, PA; Liu, JF; Liu, XB; Zhang, J | 1 |
Arnold, M; Liu, M; Lo, CC; Shen, L; Tso, P; Wang, DQ; Woods, SC | 1 |
Konno, N; Matsuda, K; Nakamachi, T; Watanabe, K; Yokobori, E; Yoshida, D | 1 |
Reviews
2 review(s) available for proglumide and sincalide
Article | Year |
---|---|
Effect of cholecystokinin on gastric motility in humans.
Topics: Benzodiazepinones; Cholecystokinin; Colon; Devazepide; Digestive System; Digestive System Physiological Phenomena; Duodenum; Gastric Emptying; Gastrointestinal Motility; Humans; Ileum; Infusions, Intravenous; Proglumide; Receptors, Cholecystokinin; Sincalide | 1994 |
[Cholecystokinin receptor antagonists].
Topics: Amino Acid Sequence; Animals; Benzodiazepinones; Cholecystokinin; Furans; Indoles; Meglumine; Molecular Sequence Data; Proglumide; Receptors, Cholecystokinin; Sincalide; Thiophenes | 1993 |
Trials
4 trial(s) available for proglumide and sincalide
Article | Year |
---|---|
Cholecystokinin is a physiological regulator of gastric acid secretion in man.
Topics: Adult; Cholecystokinin; Dose-Response Relationship, Drug; Drug Interactions; Eating; Gastric Acid; Gastric Mucosa; Gastrins; Homeostasis; Hormones; Humans; Male; Middle Aged; Proglumide; Sincalide; Somatostatin | 1994 |
Clinical efficacy and prokinetic effect of the CCK-A antagonist loxiglumide in nonulcer dyspepsia.
Topics: Adult; Analysis of Variance; Double-Blind Method; Dyspepsia; Female; Gastric Emptying; Humans; Male; Middle Aged; Proglumide; Receptors, Cholecystokinin; Sincalide; Time Factors | 1994 |
Physiological role of cholecystokinin in gastroprotection in humans.
Topics: Adult; Cholecystokinin; Double-Blind Method; Duodenum; Ethanol; Gastric Mucosa; Gastroscopy; Hormone Antagonists; Humans; Injections, Intravenous; Male; Oleic Acid; Proglumide; Sincalide; Somatostatin; Stomach | 1998 |
Interaction between CCK and a preload on reduction of food intake is mediated by CCK-A receptors in humans.
Topics: Adult; Cholecystokinin; Cross-Over Studies; Double-Blind Method; Eating; Energy Intake; Humans; Hunger; Infusions, Intravenous; Male; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Satiety Response; Sincalide | 2000 |
Other Studies
170 other study(ies) available for proglumide and sincalide
Article | Year |
---|---|
Intrathecal cholecystokinin octapeptide attenuates the antinociception and release of immunoreactive Met-enkephalin induced by intraventricular beta-endorphin in the rat.
Topics: Animals; beta-Endorphin; Depression, Chemical; Enkephalin, Methionine; Injections, Intraventricular; Injections, Spinal; Narcotic Antagonists; Pain; Proglumide; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Receptors, Opioid, delta; Reflex; Secretory Rate; Sincalide; Spinal Cord; Tail | 1992 |
Gastrin stimulates Ca2+ mobilization and clonal growth in small cell lung cancer cells.
Topics: Benzamides; Calcium; Carcinoma, Small Cell; Cell Division; Gastrins; Humans; Lung Neoplasms; Proglumide; Sincalide; Tumor Cells, Cultured | 1992 |
CCK-receptor antagonists attenuate suppression of sham feeding by intestinal nutrients.
Topics: Amylases; Animal Nutritional Physiological Phenomena; Animals; Benzodiazepinones; Catheterization; Cholecystokinin; Devazepide; Duodenum; Eating; Intestines; Male; Maltose; Oleic Acid; Oleic Acids; Phenylalanine; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Satiety Response; Sincalide; Stomach | 1992 |
Combined dose-ratio analysis of cholecystokinin receptor antagonists, devazepide, lorglumide and loxiglumide in the guinea-pig gall bladder.
Topics: Analysis of Variance; Animals; Benzodiazepinones; Binding, Competitive; Biological Assay; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Gallbladder; Guinea Pigs; Muscle, Smooth; Pentagastrin; Proglumide; Receptors, Cholecystokinin; Sincalide | 1992 |
Cholecystokinin and gastrin induce cell contraction in pig ileum by interacting with different receptor subtypes.
Topics: Animals; Calcium; Cholecystokinin; Dose-Response Relationship, Drug; Gastrins; Ileum; In Vitro Techniques; Male; Muscle Contraction; Pentagastrin; Peptide Fragments; Proglumide; Receptors, Cholecystokinin; Sincalide; Swine; Tetragastrin | 1992 |
Cholecystokinin contracts isolated human and monkey iris sphincters; a study with CCK receptor antagonists.
Topics: Aged; Aged, 80 and over; Animals; Cholecystokinin; Female; Humans; In Vitro Techniques; Iris; Macaca fascicularis; Male; Middle Aged; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide | 1992 |
The effect of long-term administration of lorglumide (CR 1409) on rat pancreatic growth and enzyme composition.
Topics: Amylases; Animals; Chymotrypsinogen; DNA; Lipase; Male; Organ Size; Pancreas; Proglumide; Proteins; Rats; Rats, Inbred Strains; Sincalide; Trypsinogen | 1990 |
Bioactivity of synthetic human cholecystokinin (CCK)-33 in vitro and in vivo.
Topics: Amylases; Animals; Cholecystokinin; Hormones; Humans; Male; Pancreas; Pancreatic Juice; Proglumide; Rats; Sincalide; Species Specificity; Swine | 1991 |
Synthetic CCK8 analogs with antagonist activity on pancreatic receptors: in vivo study in the rat, compared to non-peptidic antagonists.
Topics: Amino Acid Sequence; Amylases; Animals; Benzodiazepinones; Devazepide; Male; Molecular Sequence Data; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide | 1991 |
Structure-antigastrin activity relationships of new (R)-4-benzamido-5-oxopentanoic acid derivatives.
Topics: Animals; Binding, Competitive; Cats; Cholecystokinin; Dogs; Gastric Acid; Gastrins; Male; Models, Molecular; Pentanoic Acids; Proglumide; Rabbits; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide; Stereoisomerism; Structure-Activity Relationship | 1992 |
Hypnotic action of flunitrazepam is reversed by proglumide in rats.
Topics: Animals; Ceruletide; Electroencephalography; Electromyography; Flunitrazepam; Hypnotics and Sedatives; Male; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Sleep; Sleep, REM | 1991 |
Role of cholecystokinin in pancreatic bicarbonate secretion in dogs.
Topics: Animals; Bicarbonates; Body Water; Cholecystokinin; Corn Oil; Dogs; Female; Infusions, Parenteral; Male; Pancreas; Proglumide; Secretin; Sincalide | 1991 |
Cholecystokinin octapeptide antagonized opioid analgesia mediated by mu- and kappa- but not delta-receptors in the spinal cord of the rat.
Topics: Animals; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Narcotic Antagonists; Pain; Pain Measurement; Peptide Fragments; Proglumide; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sincalide; Spinal Cord | 1990 |
[Cholecystokinin octapeptide (CCK-8) antagonized analgesia mediated by mu and kappa opioid receptors].
Topics: Analgesics; Animals; Dynorphins; Endorphins; Injections, Spinal; Male; Pain; Peptide Fragments; Proglumide; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sensory Thresholds; Sincalide; Spinal Cord | 1990 |
Neuromodulation of guinea pig intestinal electrolyte transport by cholecystokinin octapeptide.
Topics: Animals; Atropine; Biological Transport; Bumetanide; Calcium; Culture Media; Dose-Response Relationship, Drug; Electrolytes; Electrophysiology; Guinea Pigs; Ileum; Intestinal Mucosa; Intestines; Male; Proglumide; Receptors, Cholecystokinin; Sincalide; Tetrodotoxin | 1991 |
Effect of two new cholecystokinin antagonists on gallbladder emptying in opossums.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Female; Gallbladder; Kinetics; Male; Opossums; Proglumide; Sincalide | 1991 |
The effect of cholecystokinin-receptor antagonists on cholecystokinin-stimulated bile flow in dogs.
Topics: Animals; Anti-Ulcer Agents; Benzamides; Bile; Bile Acids and Salts; Cholecystokinin; Corn Oil; Dogs; Electrolytes; Female; Glucagon; Insulin; Kinetics; Proglumide; Receptors, Cholecystokinin; Sincalide; Taurocholic Acid | 1991 |
Studies of three non-peptide cholecystokinin antagonists (devazepide, lorglumide and loxiglumide) in human isolated alimentary muscle and guinea-pig ileum.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Digestive System; Digestive System Physiological Phenomena; Female; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide | 1991 |
Cholecystokinin and its antagonist lorglumide respectively attenuate and facilitate morphine-induced inhibition of C-fiber evoked discharges of dorsal horn nociceptive neurons.
Topics: Animals; Cholecystokinin; Electric Stimulation; Evoked Potentials; Male; Morphine; Nerve Fibers; Neurons; Pain; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Spinal Cord | 1991 |
Apneic effects of cholecystokinin in unanaesthetized fetal sheep.
Topics: Animals; Apnea; Dose-Response Relationship, Drug; Injections, Intraventricular; Proglumide; Respiratory Mechanics; Sheep; Sincalide; Sleep Stages | 1990 |
Differential effects of sulfated cholecystokinin octapeptide and proglumide injected intrathecally on antinociception induced by beta-endorphin and morphine administered intracerebroventricularly in mice.
Topics: Analgesics; Animals; beta-Endorphin; Glutamine; Injections, Intraventricular; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Morphine; Proglumide; Reaction Time; Sincalide | 1990 |
The effect of a novel CCK-antagonist (lorglumide) on human and guinea pig gallbladder strips: a tensiometric study.
Topics: Adult; Aged; Animals; Dose-Response Relationship, Drug; Gallbladder; Guinea Pigs; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Proglumide; Receptors, Cholecystokinin; Sincalide; Species Specificity | 1990 |
Involvement of cholecystokinin receptors in the control of striatal dopamine autoreceptors.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Brain Chemistry; Corpus Striatum; Dialysis; Dopamine; Homovanillic Acid; Male; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Receptors, Dopamine; Sincalide | 1990 |
The effect of CR 1409, a potent CCK receptor antagonist, on basal and stimulated pancreatic secretion in rat.
Topics: Animals; Bicarbonates; Dose-Response Relationship, Drug; Glutamine; Male; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Secretory Rate; Sincalide | 1990 |
Mechanism of inhibitory action of peptide YY on cholecystokinin-induced contractions of isolated dog ileum.
Topics: Animals; Cholecystokinin; Dogs; Female; Gallbladder; Glutamine; Ileum; Isometric Contraction; Male; Muscle Contraction; Peptide YY; Peptides; Proglumide; Sincalide | 1990 |
Effects of CCK-receptor antagonists on CCK-stimulated pepsinogen secretion and calcium increase in isolated guinea pig gastric chief cells.
Topics: Animals; Benzodiazepinones; Calcium; Cells, Cultured; Cholecystokinin; Devazepide; Dibutyryl Cyclic GMP; Dose-Response Relationship, Drug; Gastric Mucosa; Guinea Pigs; In Vitro Techniques; Male; Pepsinogens; Proglumide; Receptors, Cholecystokinin; Signal Transduction; Sincalide | 1990 |
Proglumide analogues: potent cholecystokinin receptor antagonists.
Topics: Amylases; Animals; Glutamine; Guinea Pigs; In Vitro Techniques; Male; Mice; Pancreas; Proglumide; Rats; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide; Structure-Activity Relationship | 1985 |
Effect of proglumide on rat pancreatic growth.
Topics: Animals; Cholecystokinin; DNA; Gastrins; Glutamine; Male; Organ Size; Pancreas; Proglumide; Proteins; Rats; Rats, Inbred Strains; RNA; Sincalide | 1985 |
Actions of cholecystokinin octapeptide on rat spinal dorsal horn neurons.
Topics: Animals; Calcium; Ganglia, Spinal; In Vitro Techniques; Membrane Potentials; Neurons; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Spinal Cord; Substance P; Tetraethylammonium Compounds; Tetrodotoxin | 1985 |
New proglumide-analogue CCK receptor antagonists: very potent and selective for peripheral tissues.
Topics: Amylases; Animals; Biological Assay; Cerebral Cortex; Cholecystokinin; Glutamine; Male; Mice; Pancreas; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide | 1986 |
Structural features of various proglumide-related cholecystokinin receptor antagonists.
Topics: Amylases; Animals; Cholecystokinin; Glutamine; Guinea Pigs; Kinetics; Male; Mice; Pancreas; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide; Structure-Activity Relationship | 1986 |
A novel bioassay for the NK-2 neurokinin receptor: the guinea pig gallbladder.
Topics: Animals; Atropine; Biological Assay; Dose-Response Relationship, Drug; Eledoisin; Gallbladder; Guinea Pigs; Kassinin; Neurokinin A; Neuropeptides; Oligopeptides; Physalaemin; Proglumide; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Sincalide; Substance P; Tetrodotoxin | 1986 |
CR-1409: a potent inhibitor of cholecystokinin-stimulated amylase release and cholecystokinin binding in rat pancreatic acini.
Topics: Amylases; Animals; Dose-Response Relationship, Drug; Glutamine; Male; N-Methylscopolamine; Pancreas; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Scopolamine Derivatives; Sincalide | 1987 |
Pancreatic growth: interaction of exogenous cholecystokinin, a protease inhibitor, and a cholecystokinin receptor antagonist in mice.
Topics: Amylases; Animals; Cholecystokinin; Chymotrypsinogen; Esters; Gabexate; Glutamine; Guanidines; Male; Mice; Organ Size; Pancreas; Proglumide; Protease Inhibitors; Sincalide | 1987 |
Cholecystokinin releases [3H]GABA from the perfused subarachnoid space of the anaesthetized rat spinal cord.
Topics: Anesthesia, General; Animals; Cholecystokinin; gamma-Aminobutyric Acid; Male; Osmolar Concentration; Perfusion; Potassium; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Spinal Cord; Subarachnoid Space; Substance P; Tritium | 1987 |
Characterization of a new CCK antagonist, L364,718: in vitro and in vivo studies.
Topics: Amylases; Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; In Vitro Techniques; Kinetics; Male; Pancreas; Proglumide; Rats; Rats, Inbred Strains; Reference Values; Sincalide | 1988 |
Loxiglumide. A new proglumide analog with potent cholecystokinin antagonistic activity in the rat pancreas.
Topics: Amylases; Animals; Binding, Competitive; Cholecystokinin; Dose-Response Relationship, Drug; Glutamine; Pancreas; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide | 1989 |
[Inhibitory effect of CR 1409 (cholecystokinin antagonist) on pancreatic exocrine secretion in rats].
Topics: Amylases; Animals; Cholecystokinin; Glutamine; Male; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1989 |
[Inhibitory effect of a new proglumide derivative, loxiglumide, on CCK action in isolated rat pancreatic acini].
Topics: Amylases; Animals; Cholecystokinin; Glutamine; In Vitro Techniques; Male; Pancreas; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1989 |
Properties of receptors for gastrin and CCK on gastric smooth muscle cells.
Topics: Amylases; Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Gastrins; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Pancreas; Peptide Fragments; Proglumide; Receptors, Cholecystokinin; Sincalide; Stomach; Tetragastrin | 1989 |
Involvement of cholecystokinin receptors in the adverse effect of glucocorticoids on diet-induced necrotizing pancreatitis.
Topics: Amylases; Animals; Choline Deficiency; Diet; Dose-Response Relationship, Drug; Ethionine; Female; Glucocorticoids; Hydrocortisone; Mice; Mice, Inbred Strains; Necrosis; Pancreas; Pancreatitis; Proglumide; Receptors, Cholecystokinin; Sincalide | 1989 |
Effects of a new proglumide analogue CR 1392 on pancreatic exocrine secretion in the rat.
Topics: Amylases; Animals; Cholecystokinin; Dose-Response Relationship, Drug; Glutamine; Male; Pancreas; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide | 1989 |
Cholecystokinin receptor antagonism of stimulated pancreatic and gastric secretion.
Topics: Amylases; Animals; Food; Gastric Acid; Kinetics; Male; Pancreas; Pentagastrin; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide | 1989 |
Plasma concentrations of cholecystokinin octapeptide and food intake in male rats treated with cholecystokinin octapeptide.
Topics: Animals; Eating; Gastrins; Male; Oxytocin; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Somatostatin | 1989 |
Bombesin: an activator of specific Aeromonas antibody secretion in rat intestine.
Topics: Aeromonas; Animals; Antibodies, Anti-Idiotypic; Antibodies, Bacterial; Bacterial Infections; Bombesin; Cholecystokinin; Enzyme-Linked Immunosorbent Assay; Gastrins; Immunoglobulin A; Immunoglobulin G; Intestinal Mucosa; Intestines; Male; Pentagastrin; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1989 |
[The effect of cholecystokinin antagonists on satiety induced by cholecystokinin octapeptide in dogs].
Topics: Animals; Blood-Brain Barrier; Cholecystokinin; Dogs; Eating; Glutamine; Injections, Intravenous; Injections, Intraventricular; Proglumide; Receptors, Cholecystokinin; Sincalide | 1989 |
Age-dependent stimulation of neonatal insulin release and inositol phosphate accumulation by CCK-8 and carbachol.
Topics: Age Factors; Animals; Animals, Newborn; Carbachol; Dose-Response Relationship, Drug; Glucose; In Vitro Techniques; Inositol Phosphates; Insulin; Islets of Langerhans; Pentagastrin; Proglumide; Rats; Sincalide; Stimulation, Chemical; Vasoactive Intestinal Peptide | 1989 |
Modulation by CR-1409 (lorglumide), a cholecystokinin receptor antagonist, of trypsin inhibitor-enhanced growth of azaserine-induced putative preneoplastic lesions in rat pancreas.
Topics: Animals; Azaserine; Cholecystokinin; Esters; Gabexate; Glutamine; Guanidines; Male; Pancreatic Neoplasms; Precancerous Conditions; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide; Trypsin Inhibitors | 1989 |
Cholecystokinin-octapeptide antagonizes morphine analgesia in periaqueductal gray of the rat.
Topics: Analgesia; Animals; Dose-Response Relationship, Drug; Male; Morphine; Pain; Periaqueductal Gray; Proglumide; Rats; Rats, Inbred Strains; Sensory Thresholds; Sincalide | 1989 |
CCK receptor antagonism by loxiglumide and gall bladder contractions in response to cholecystokinin, sham feeding and ordinary feeding in man.
Topics: Adolescent; Adult; Cholecystokinin; Food; Gallbladder; Glutamine; Humans; Male; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide | 1989 |
Effect of cholecystokinin on acetylcholine turnover and dopamine release in the rat striatum and cortex.
Topics: Acetylcholine; Animals; Cerebral Cortex; Cholecystokinin; Corpus Striatum; Dopamine; Injections, Intraventricular; Male; Nerve Tissue Proteins; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1989 |
Effect of a new CCK-receptor antagonist, CR 1409, on pancreatic growth induced by caerulein, CCK-8, bombesin and gastrin-releasing peptide in the rat.
Topics: Animals; Bombesin; Ceruletide; Gastrin-Releasing Peptide; Gastrointestinal Hormones; Male; Organ Size; Pancreas; Peptides; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1989 |
Cholecystokinin modulates neurotransmission through the dentate gyrus.
Topics: Action Potentials; Animals; Benzamides; Electric Stimulation; Hippocampus; Iontophoresis; Male; Proglumide; Rats; Rats, Inbred Strains; Sciatic Nerve; Sincalide; Synaptic Transmission | 1988 |
Two proglumide analogues are equipotent antagonists of the inhibition of food intake by CCK-8.
Topics: Animals; Dose-Response Relationship, Drug; Eating; Glutamates; Male; Proglumide; Rats; Rats, Sprague-Dawley; Sincalide | 1988 |
Role of cholecystokinin in pancreatic exocrine response to intraluminal amino acids and fat.
Topics: Amino Acids; Animals; Bethanechol; Bethanechol Compounds; Bicarbonates; Cholecystokinin; Dogs; Fat Emulsions, Intravenous; Pancreas; Pancreatic Juice; Proglumide; Proteins; Receptors, Cell Surface; Receptors, Cholecystokinin; Secretin; Sincalide | 1985 |
Selective presence of opiate receptors on intestinal circular muscle cells.
Topics: Acetylcholine; Animals; Atropine; Benzomorphans; beta-Endorphin; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Methionine; Guinea Pigs; Humans; Jejunum; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Proglumide; Receptors, Opioid; Sincalide | 1985 |
Release of acetylcholine mediated by cholecystokinin receptor from the guinea pig sphincter of Oddi.
Topics: Acetylcholine; Ampulla of Vater; Angiotensin II; Animals; Atropine; Bethanechol; Bethanechol Compounds; Bradykinin; Choline; Dose-Response Relationship, Drug; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; Hydrogen; Male; Muscle Contraction; Phentolamine; Proglumide; Receptors, Cholecystokinin; Serotonin; Sincalide; Sphincter of Oddi; Tetrodotoxin | 1986 |
Cholecystokinin stimulates neuronal receptors to produce contraction of the canine colon.
Topics: Acetylcholine; Animals; Atropine; Cholecystokinin; Colon; Dibutyryl Cyclic GMP; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Injections, Intra-Arterial; Injections, Intravenous; Male; Muscle Contraction; Neurons; Pentagastrin; Peptide Fragments; Proglumide; Receptors, Cholecystokinin; Sincalide; Tetrodotoxin | 1989 |
Behavioral effects of cholecystokinin and its related peptides in rats.
Topics: Animals; beta-Endorphin; Cerebral Cortex; Cerebral Ventricles; Endorphins; Gastrins; Male; Motor Activity; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Stereotyped Behavior; Structure-Activity Relationship; Tetragastrin | 1985 |
Cholecystokinin receptor mediated hydrolysis of inositol phospholipids in guinea pig gastric glands.
Topics: Animals; Dibutyryl Cyclic GMP; Gastric Mucosa; Guinea Pigs; Hydrolysis; Inositol Phosphates; Lithium; Male; Phosphatidylinositols; Proglumide; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide | 1985 |
Structure-activity relationship of subtypes of cholecystokinin receptors in the cat lower esophageal sphincter.
Topics: Animals; Cats; Cholecystokinin; Dose-Response Relationship, Drug; Esophagogastric Junction; Female; Gastrins; Male; Muscle Contraction; Pressure; Proglumide; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide; Structure-Activity Relationship; Tetrodotoxin | 1986 |
Antagonists of central and peripheral behavioral actions of cholecystokinin octapeptide.
Topics: Animals; Behavior, Animal; Benzamides; Brain; Dopamine; Dose-Response Relationship, Drug; Eating; Exploratory Behavior; Immune Sera; Male; Mice; Motor Activity; Nucleus Accumbens; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide | 1986 |
Differentiation of central and peripheral cholecystokinin receptors by new glutaramic acid derivatives with cholecystokinin-antagonistic activity.
Topics: Animals; Benzamides; Cerebral Cortex; In Vitro Techniques; Kinetics; Male; Mice; Pancreas; Proglumide; Rats; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide; Tetragastrin | 1986 |
Proglumide (gastrin and cholecystokinin receptor antagonist) inhibits insulin secretion in vitro.
Topics: Animals; Cholecystokinin; Culture Techniques; Depression, Chemical; Female; Gastric Inhibitory Polypeptide; Glucose; Glutamine; Insulin; Insulin Secretion; Islets of Langerhans; Male; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide | 1986 |
Inhibition of synaptic transmission in the hippocampus by cholecystokinin (CCK) and its antagonism by a CCK analog (CCK27-33).
Topics: Animals; Depression, Chemical; Evoked Potentials; Hippocampus; Peptide Fragments; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Synaptic Transmission | 1987 |
The effects of cholecystokinin and cholecystokinin antagonists on synaptic function in the CA1 region of the rat hippocampal slice.
Topics: Action Potentials; Animals; Benzamides; Female; Glutamine; Hippocampus; In Vitro Techniques; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Sulfates; Synapses; Synaptic Transmission | 1987 |
Potentiation of beta-endorphin effects by proglumide in rats.
Topics: Analgesia; Animals; beta-Endorphin; Catalepsy; Dose-Response Relationship, Drug; Drug Synergism; Endorphins; Glutamine; Humans; Male; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1985 |
Cholecystokinin antagonist lorglumide reverses chronic haloperidol-induced effects on dopamine neurons.
Topics: Action Potentials; Animals; Dopamine; Glutamine; Haloperidol; Male; Nucleus Accumbens; Proglumide; Rats; Rats, Inbred Strains; Septal Nuclei; Sincalide; Substantia Nigra | 1988 |
Inhibitory effect of CR-1409, a competitive inhibitor of cholecystokinin, on pancreatic exocrine secretion in the conscious rat.
Topics: Animals; Bicarbonates; Cholecystokinin; Dose-Response Relationship, Drug; Female; Glutamine; Male; Pancreatic Juice; Proglumide; Proteins; Rats; Rats, Inbred Strains; Reference Values; Sincalide | 1988 |
Intracerebroventricular injection of cholecystokinin octapeptide elevates plasma prolactin levels through stimulation of vasoactive intestinal polypeptide.
Topics: Animals; Apomorphine; Benzamides; Dopamine Antagonists; Immunosorbent Techniques; Injections, Intraventricular; Male; Proglumide; Prolactin; Rats; Rats, Inbred Strains; Sincalide; Vasoactive Intestinal Peptide | 1987 |
Peptide YY and gallbladder contraction. Studies in vivo and in vitro.
Topics: Ampulla of Vater; Animals; Dogs; Female; Gallbladder; Gastrointestinal Hormones; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Peptide YY; Peptides; Proglumide; Sincalide; Sphincter of Oddi | 1988 |
Cholecystokinin and an evoked response in the dentate gyrus.
Topics: Animals; Cholecystokinin; Evoked Potentials; Hippocampus; Injections, Intraventricular; Male; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1988 |
Biological effects of a proglumide derivative as cholecystokinin antagonist in conscious dogs.
Topics: Animals; Cholecystokinin; Dogs; Dose-Response Relationship, Drug; Gastric Acid; Glutamine; Infusions, Intravenous; Pancreatic Juice; Pancreatic Polypeptide; Pentagastrin; Proglumide; Sincalide | 1987 |
Different peripheral and central antagonistic activity of new glutaramic acid derivatives on satiety induced by cholecystokinin in rats.
Topics: Animals; Dose-Response Relationship, Drug; Glutamine; Male; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Satiation; Sincalide | 1986 |
Proglumide has access to brain and antagonizes the central satiety effect of cholecystokinin octapeptide in the dog.
Topics: Animals; Blood-Brain Barrier; Brain; Dogs; Dose-Response Relationship, Drug; Drinking Behavior; Feeding Behavior; Glutamine; Infusions, Intravenous; Injections, Intraventricular; Proglumide; Satiation; Satiety Response; Sincalide; Time Factors | 1987 |
Receptor-mediated internalization and secretion of cholecystokinin into rat pancreatic duct fluid.
Topics: Animals; Cholecystokinin; Dose-Response Relationship, Drug; Gastrins; Male; Pancreatic Ducts; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide | 1987 |
Sexual activity increases plasma concentrations of cholecystokinin octapeptide and offsets hunger in male rats.
Topics: Animals; Gastrins; Hunger; Male; Proglumide; Rats; Rats, Inbred Strains; Sexual Behavior, Animal; Sincalide | 1987 |
Cholecystokinin octapeptide, proglumide, and conditioned taste avoidance in rats.
Topics: Animals; Avoidance Learning; Conditioning, Psychological; Female; Glutamine; Proglumide; Rats; Sincalide; Sucrose; Taste | 1987 |
Evidence for dopaminomimetic effect of intrastriatally injected cholecystokinin octapeptide in mice.
Topics: Animals; Apomorphine; Corpus Striatum; Drug Interactions; Female; Haloperidol; Injections; Mice; Proglumide; Receptors, Dopamine; Sincalide; Stereotyped Behavior | 1986 |
Intracerebroventricular injections of cholecystokinin octapeptide suppress feeding in rats--pharmacological characterization of this action.
Topics: Animals; Cerebral Ventricles; Cholecystokinin; Eating; Feeding Behavior; Food Deprivation; Injections, Intraventricular; Male; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1986 |
A new simple mouse model for the in vivo evaluation of cholecystokinin (CCK) antagonists: comparative potencies and durations of action of nonpeptide antagonists.
Topics: Administration, Oral; Animals; Benzodiazepinones; Binding, Competitive; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Female; Gastric Emptying; Mice; Proglumide; Sincalide; Time Factors | 1986 |
Regional and cellular heterogeneity of cholecystokinin receptors mediating muscle contraction in the gut.
Topics: Animals; Gallbladder; Gastric Fundus; Guinea Pigs; Ileum; Male; Muscle Contraction; Muscle, Smooth; Neurons; Proglumide; Receptors, Cholecystokinin; Receptors, Cholinergic; Sincalide | 1987 |
Residual inhibition of epidermal growth factor binding by pancreatic secretagogues and phorbol ester in rat pancreas.
Topics: Animals; Bombesin; Calcium; Carbachol; Dibutyryl Cyclic GMP; Epidermal Growth Factor; Kinetics; Male; Pancreas; Phorbol Esters; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Tetradecanoylphorbol Acetate | 1985 |
Altered responding to cholecystokinins and dopaminergic agonists following 6-hydroxydopamine treatment in rats.
Topics: Animals; Apomorphine; Brain; Dopamine; Gastrins; Hydroxydopamines; Male; Methamphetamine; Motor Activity; Oxidopamine; Proglumide; Rats; Rats, Inbred Strains; Sincalide; Tetragastrin | 1985 |
Endogenous cholecystokinin and intestinal satiety.
Topics: Analysis of Variance; Animals; Appetite; Catheters, Indwelling; Cholecystokinin; Duodenum; Food, Formulated; Male; Phenylalanine; Proglumide; Rats; Sincalide; Time Factors | 1985 |
Effects of cholecystokinin, caerulein and pentagastrin on electrical behavior of myenteric neurons.
Topics: Animals; Ceruletide; Cholecystokinin; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Myenteric Plexus; Neurons; Pentagastrin; Proglumide; Sincalide | 1985 |
Cholecystokinin-8 and proglumide modulation of electrically elicited eating.
Topics: Animals; Dose-Response Relationship, Drug; Electric Stimulation; Feeding Behavior; Glutamine; Hypothalamic Area, Lateral; Male; Proglumide; Rats; Rats, Inbred Strains; Sincalide | 1985 |
Differential antagonism by proglumide of various CCK-mediated effects in mice.
Topics: Animals; Body Temperature; Cerebral Ventricles; Glutamine; Injections, Intraventricular; Male; Mice; Motor Activity; Naloxone; Proglumide; Sincalide | 1985 |
Effect of cholecystokinin octapeptide and ceruletide on release of acetylcholine from cerebral cortex of the rat in vivo.
Topics: Acetylcholine; Animals; Blood Pressure; Cerebral Cortex; Ceruletide; Hypnotics and Sedatives; Male; Morphine; Naloxone; Nociceptors; Proglumide; Rats; Rats, Inbred Strains; Reaction Time; Sincalide | 1984 |
Interactions of cholecystokinin octapeptide and dopamine on nucleus accumbens neurons.
Topics: Animals; Antipsychotic Agents; Dopamine; Drug Interactions; Glutamates; Glutamic Acid; Humans; Male; Nucleus Accumbens; Proglumide; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Cholecystokinin; Schizophrenia; Septal Nuclei; Sincalide | 1984 |
In vitro and in vivo effect of proglumide on cholecystokinin-stimulated amylase release in mouse pancreatic acini.
Topics: Amylases; Animals; Cholecystokinin; Dose-Response Relationship, Drug; Glutamine; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Pancreas; Proglumide; Sincalide; Tetragastrin | 1984 |
Cholecystokinin-induced contraction of dispersed smooth muscle cells.
Topics: Animals; Appetite Depressants; Biological Transport, Active; Calcimycin; Carbachol; Cholecystokinin; Glucagon; Guinea Pigs; Kinetics; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Proglumide; Rubidium; Sincalide; Stomach | 1982 |
Activation of central nervous system cholecystokinin receptors stimulates respiration in the cat.
Topics: Animals; Blood Pressure; Cats; Cholecystokinin; Female; Heart Rate; Male; Pentagastrin; Peptide Fragments; Proglumide; Receptors, Cell Surface; Receptors, Cholecystokinin; Respiration; Sincalide; Tidal Volume | 1983 |
Pharmacological profile of FK480, a novel cholecystokinin type-A receptor antagonist: comparison to loxiglumide.
Topics: Amylases; Animals; Benzodiazepinones; Female; Gastric Emptying; Guinea Pigs; Indoles; Male; Mice; Mice, Inbred ICR; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide | 1994 |
Brain cholecystokinin octopeptide (CCK-8) concentrations: effect of tryptophan and other serotonergic agents.
Topics: Animals; Brain Chemistry; Corpus Striatum; Cyproheptadine; Drug Interactions; Dynorphins; Hippocampus; Hydroxyindoleacetic Acid; Hypothalamus; Imipramine; Male; Proglumide; Rats; Serotonin; Serotonin Receptor Agonists; Sincalide; Substance P; Tryptophan | 1994 |
CCK antagonists reveal that CCK-8 and JMV-180 interact with different sites on the rat pancreatic acinar cell CCKA receptor.
Topics: Amino Acid Sequence; Amylases; Animals; Benzodiazepinones; Calcium; Cholecystokinin; Devazepide; Male; Models, Biological; Molecular Sequence Data; Pancreas; Periodicity; Proglumide; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Signal Transduction; Sincalide | 1994 |
Mechanisms for pancreatic hypertrophy induced by long-term administration of bethanechol.
Topics: Amylases; Animals; Atropine; Bethanechol; Cholinergic Agonists; Cholinergic Antagonists; Drug Administration Schedule; Drug Interactions; Gastrins; Hypertrophy; Male; Organ Size; Pancreas; Pentagastrin; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1994 |
Effect of a novel cholecystokinin receptor antagonist, FK480, administered intraduodenally, on pancreatic secretion in rats.
Topics: Amylases; Animals; Benzodiazepinones; Caseins; Duodenum; Indoles; Male; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1995 |
Characterization of the receptors and mechanisms involved in the cardiovascular actions of sCCK-8 in the pithed rat.
Topics: Adrenalectomy; Adrenergic Agents; Animals; Benzodiazepinones; Blood Pressure; Bradycardia; Cholecystokinin; Decerebrate State; Devazepide; Dose-Response Relationship, Drug; Gastrins; Guanethidine; Heart Rate; Hormone Antagonists; Hormones; Hypertension; Indoles; Male; Meglumine; Pentagastrin; Phentolamine; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide; Tetragastrin | 1995 |
Effect of succinyl cholecystokinin heptapeptide on synaptosomal 45Ca uptake of mouse hippocampus.
Topics: Animals; Calcium Radioisotopes; Hippocampus; Mice; Proglumide; Sincalide; Synaptosomes | 1995 |
Receptor-evoked Ca2+ mobilization in pancreatic acinar cells: evidence for a regulatory role of protein kinase C by a mechanism involving the transition of high-affinity receptors to a low-affinity state.
Topics: Alkaloids; Animals; Brain; Calcium; Carbachol; Cholecystokinin; Fura-2; Inosine Triphosphate; Naphthalenes; Pancreas; Phosphorylation; Polycyclic Compounds; Proglumide; Protein Kinase C; Rabbits; Receptors, Cell Surface; Receptors, Cholecystokinin; Sincalide; Staurosporine; Tetradecanoylphorbol Acetate | 1993 |
PD 135158, a CCKB/gastrin receptor antagonist, stimulates rat pancreatic enzyme secretion as a CCKA receptor agonist.
Topics: Animals; Anti-Anxiety Agents; Cholecystokinin; Drug Interactions; Indoles; Lipase; Meglumine; Pancreas; Proglumide; Rats; Sincalide | 1993 |
Inhibitory action of CCK-OP on rat proximal colon.
Topics: Acetylcholine; Animals; Atropine; Colon; Fasting; Hexamethonium; Hexamethonium Compounds; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide | 1994 |
Effect of intraduodenal infusion of tocamphyl on pancreatic exocrine secretion and gastrointestinal hormone release in rats.
Topics: Analysis of Variance; Animals; Atropine; Bile; Camphor; Cholagogues and Choleretics; Cholecystokinin; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Gastrointestinal Hormones; Male; Pancreatic Juice; Proglumide; Radioimmunoassay; Rats; Rats, Wistar; Secretin; Sincalide | 1994 |
Evidence for potentiation by CCK antagonists of the effect of cholecystokinin octapeptide in the elevated plus-maze.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Cholecystokinin; Devazepide; Drug Synergism; Exploratory Behavior; Female; Mice; Motor Activity; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Sincalide | 1994 |
Treatment with cholecystokinin receptor antagonist loxiglumide enhances insulin response to intravenous glucose stimulation in postpancreatitic rats.
Topics: Acute Disease; Animals; Ceruletide; Glucose; Injections, Intravenous; Injections, Subcutaneous; Insulin; Insulin Resistance; Insulin Secretion; Islets of Langerhans; Male; Pancreatitis; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1994 |
[Effect of cholecystokinin and its antagonists lorglumide, devazepide, and L-365,260 on gastrointestinal motility in rats].
Topics: Animals; Benzodiazepinones; Devazepide; Gastric Emptying; Gastrointestinal Motility; Guinea Pigs; Ileum; Male; Muscle Contraction; Muscle, Smooth; Phenylurea Compounds; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide | 1993 |
Characterization of a new cholecystokinin receptor antagonist FK480 in in vitro isolated rat pancreatic acini.
Topics: Animals; Benzodiazepinones; Devazepide; In Vitro Techniques; Indoles; Male; Pancreas; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1994 |
The antagonistic effect of cholecystokinin octapeptide (CCK-8) on opioid effects in cardiovascular activities was mediated by CCK-B receptor.
Topics: Animals; Benzodiazepinones; Blood Pressure; Devazepide; Female; Hypotension; Muscimol; Phenylurea Compounds; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1993 |
Loxiglumide (CR1505), a cholecystokinin antagonist, specifically inhibits the growth of human pancreatic cancer lines xenografted into nude mice.
Topics: Animals; Cell Division; Chloroquine; Cholecystokinin; DNA; Esters; Gabexate; Guanidines; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Transplantation; Organ Culture Techniques; Pancreatic Neoplasms; Proglumide; Sincalide; Transplantation, Heterologous | 1993 |
Examination of the effects of cholecystokinin 26-33 and neuropeptide Y on responses of visual cortical neurons of the cat.
Topics: Animals; Baclofen; Cats; Cholecystokinin; Evoked Potentials, Visual; gamma-Aminobutyric Acid; Iontophoresis; Neural Conduction; Neurons; Neuropeptide Y; Photic Stimulation; Proglumide; Sincalide; Tachyphylaxis; Visual Cortex | 1993 |
Inhibition of growth of a transplanted rat pancreatic acinar carcinoma with CCK-8.
Topics: Animals; Carcinoma; Cell Division; Dose-Response Relationship, Drug; Neoplasm Transplantation; Pancreatic Neoplasms; Proglumide; Rats; Rats, Inbred Lew; Receptors, Cholecystokinin; Sincalide | 1993 |
Involvement of different subtypes of cholecystokinin receptors in opioid antinociception in the mouse.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Analgesics; Animals; beta-Endorphin; Drug Interactions; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Indoles; Injections, Intraventricular; Male; Meglumine; Mice; Mice, Inbred ICR; Morphine; Narcotics; Pain Measurement; Proglumide; Pyrrolidines; Receptors, Cholecystokinin; Sincalide | 1995 |
Regulation of gene expression of pancreatic secretory trypsin inhibitor-61 and -56 by bile and pancreatic juice in rats.
Topics: Animals; Base Sequence; Bile; Biliopancreatic Diversion; Ceruletide; Cholecystokinin; Gastrointestinal Agents; Gene Expression; Hormone Antagonists; Infusions, Intravenous; Male; Molecular Sequence Data; Pancreas; Pancreatic Juice; Proglumide; Rats; Rats, Wistar; RNA, Messenger; Sincalide; Trypsin Inhibitor, Kazal Pancreatic | 1995 |
Cholecystokinin [corrected] octapeptide modulates dopamine release in rat striatum.
Topics: Animals; Anti-Ulcer Agents; Apomorphine; Dopamine; Dopamine Agonists; Electric Stimulation; Hormone Antagonists; Male; Neostriatum; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Tritium | 1995 |
Cholecystokinin-GABA interactions in rat striatum.
Topics: Animals; Calcium; Cholecystokinin; Corpus Striatum; Electric Stimulation; gamma-Aminobutyric Acid; Hormone Antagonists; Indoles; Male; Meglumine; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Tetrodotoxin; Tritium | 1995 |
Luminal cholecystokinin and gastrin cause gallbladder contraction.
Topics: Animals; Bile; Cholecystokinin; Female; Gallbladder; Gastrins; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Muscle Contraction; Pentagastrin; Proglumide; Receptors, Cholecystokinin; Sincalide | 1996 |
Effects of cholecystokinin and carbachol on membrane fluidity in pancreatic acini.
Topics: Animals; Bombesin; Carbachol; Cholecystokinin; Dose-Response Relationship, Drug; Hormone Antagonists; L-Lactate Dehydrogenase; Male; Membrane Fluidity; Pancreas; Pancreatitis; Phosphatidylcholines; Proglumide; Rats; Rats, Wistar; Secretin; Sincalide | 1996 |
Pharmacological profile of TP-680, a new cholecystokininA receptor antagonist.
Topics: Amylases; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Cysteine; Devazepide; In Vitro Techniques; Intracellular Membranes; Male; Niacin; Pancreas; Proglumide; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide | 1996 |
Synergistic interactions between human transfected adenosine A1 receptors and endogenous cholecystokinin receptors in CHO cells.
Topics: Adenosine; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Benzodiazepinones; Calcium; CHO Cells; Cricetinae; Devazepide; Dose-Response Relationship, Drug; Drug Synergism; Hormone Antagonists; Humans; Inositol Phosphates; Pertussis Toxin; Proglumide; Receptors, Purinergic P1; Receptors, Serotonin; Sincalide; Virulence Factors, Bordetella | 1996 |
Effect of dexloxiglumide and spiroglumide, two new CCK-receptor antagonists, on gastric emptying and secretion in the rat: evaluation of their receptor selectivity in vivo.
Topics: Animals; Dose-Response Relationship, Drug; Gastric Acid; Gastric Emptying; Hormone Antagonists; Keto Acids; Male; Pentagastrin; Pentanoic Acids; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Spiro Compounds | 1996 |
Pharmacological profile of T-0632, a novel potent and selective CCKA receptor antagonist, in vitro.
Topics: Amylases; Animals; Benzodiazepinones; Binding, Competitive; Brain; Cell Membrane; Devazepide; Gallbladder; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Pancreas; Proglumide; Protein Binding; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide | 1996 |
Comparison of the effects of two cholecystokinin-receptor antagonists, loxiglumide and L-364,718, on the pancreatic secretory response to intraduodenal tryptophan in dogs.
Topics: Animals; Benzodiazepinones; Bicarbonates; Cholecystokinin; Devazepide; Dogs; Duodenum; Female; Male; Pancreas; Perfusion; Proglumide; Receptors, Cholecystokinin; Secretin; Sincalide; Tryptophan | 1996 |
Pharmacological profile of T-0632, a novel potent and selective CCKA receptor antagonist, in vivo.
Topics: Animals; Benzodiazepinones; Ceruletide; Devazepide; Dogs; Female; Gastric Emptying; Indoles; Male; Pancreas; Pancreatitis; Pregnancy; Proglumide; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide | 1996 |
Cholecystokinin receptor antagonist, loxiglumide, inhibits invasiveness of human pancreatic cancer cell lines.
Topics: Blotting, Western; Cell Line; Collagenases; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Gelatin; Hormone Antagonists; Humans; Kinetics; Matrix Metalloproteinase 9; Neoplasm Invasiveness; Pancreatic Neoplasms; Proglumide; Sincalide; Tumor Cells, Cultured | 1996 |
Effect of cholecystokinin and related peptides on jejunal transepithelial hexose transport in the Sprague-Dawley rat.
Topics: 3-O-Methylglucose; Animals; Biological Transport; Cholecystokinin; Glucose; Hormone Antagonists; Intestinal Absorption; Intestinal Mucosa; Jejunum; Kinetics; Leucine; Male; Perfusion; Proglumide; Rats; Rats, Sprague-Dawley; Sincalide; Tetragastrin; Tetrodotoxin | 1996 |
Effect of gastrin-releasing peptide (GRP) on guinea pig gallbladder contraction in vitro.
Topics: Acetylcholine; Animals; Atropine; Bombesin; Dose-Response Relationship, Drug; Gallbladder; Gastrin-Releasing Peptide; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Peptides; Proglumide; Sincalide | 1995 |
The effect of centrally administered CCK-receptor antagonists on food intake in rats.
Topics: Animals; Benzodiazepinones; Devazepide; Eating; Hormone Antagonists; Injections, Intraventricular; Male; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide | 1997 |
Full and partial agonist activity of C-terminal cholecystokinin peptides at the cloned human CCK-A receptor expressed in Chinese hamster ovary cells.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Devazepide; Hormone Antagonists; Humans; Hydrogen-Ion Concentration; Pentagastrin; Peptide Fragments; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Tetragastrin | 1997 |
Impairment of hepatic transport processes in perfused rat liver by the specific CCK receptor antagonist loxiglumide.
Topics: Animals; Bile; Biological Transport; Cholagogues and Choleretics; Gastrins; Hormone Antagonists; Indocyanine Green; Leukotriene D4; Liver; Male; Portal Vein; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Taurocholic Acid | 1997 |
Effects of proglumide on cholecystokinin-8-induced exocrine and endocrine pancreatic responses in conscious sheep.
Topics: Amylases; Animals; Blood Glucose; Dose-Response Relationship, Drug; Glucagon; Insulin; Insulin Secretion; Islets of Langerhans; Male; Pancreas; Pancreatic Juice; Proglumide; Receptors, Cholecystokinin; Sheep; Sincalide | 1997 |
CCK administration after CCK receptor blockade accelerates recovery from cerulein-induced acute pancreatitis in rats.
Topics: Acute Disease; Amylases; Animals; Ceruletide; Cholecystokinin; DNA; Hormone Antagonists; Lipase; Male; Organ Size; Pancreas; Pancreatitis; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Regeneration; Sincalide; Trypsin | 1998 |
Endogenous CCK inhibits colonic contractions in unrestrained conscious rats.
Topics: Animal Feed; Animals; Colon; Dose-Response Relationship, Drug; Duodenum; Eating; Fasting; Gastrointestinal Motility; Hormone Antagonists; Intubation, Gastrointestinal; Male; Muscle Contraction; Muscle, Smooth; Portal Vein; Proglumide; Radioimmunoassay; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Reference Values; Sincalide; Telemetry; Transducers | 1997 |
Endogenous cholecystokinin enhances postprandial gastroesophageal reflux in humans through extrasphincteric receptors.
Topics: Adult; Cholecystokinin; Cholestyramine Resin; Eating; Electric Stimulation; Esophagogastric Junction; Esophagus; Gallbladder; Gastroesophageal Reflux; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide | 1998 |
Cholecystokinin actions in the parabrachial nucleus: effects on thirst and salt appetite.
Topics: Animals; Appetite; Appetite Depressants; Cholecystokinin; Injections, Intraventricular; Male; Proglumide; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Rhombencephalon; Sincalide; Sodium Chloride; Water | 1998 |
Cholecystokinin stimulates ascorbic acid secretion through its specific receptor in the perfused stomach of rats.
Topics: Animals; Anti-Ulcer Agents; Ascorbic Acid; Bombesin; Dopamine Agents; Gastric Mucosa; Injections, Intravenous; Male; Neurotensin; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Stomach; Substance P | 1998 |
Involvement of endogenous cholecystokinin and somatostatin in gastroprotection induced by intraduodenal fat.
Topics: Animals; Capsaicin; Cholecystokinin; Denervation; Dinoprostone; Dopamine Agents; Enzyme Inhibitors; Gastric Acid; Gastric Mucosa; Hormone Antagonists; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oleic Acid; Pepsin A; Proglumide; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Somatostatin; Stomach Ulcer; Vagotomy | 1998 |
Pharmacologic profile of TS-941, a new benzodiazepine derivative cholecystokinin-receptor antagonist, in in vitro isolated rat pancreatic acini.
Topics: Amylases; Animals; Benzodiazepines; Binding, Competitive; Cell Membrane; Cell Survival; Cells, Cultured; Cerebral Cortex; Devazepide; Dose-Response Relationship, Drug; Hormone Antagonists; Male; Pancreas; Proglumide; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1999 |
Acceleration of ulcer healing by cholecystokinin (CCK): role of CCK-A receptors, somatostatin, nitric oxide and sensory nerves.
Topics: Animals; Cholecystokinin; DNA Replication; Dopamine Agents; Esters; Gabexate; Gastric Mucosa; Gastrins; Guanidines; Hormone Antagonists; Male; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Pancreatin; Proglumide; Protease Inhibitors; Rats; Rats, Wistar; Receptors, Cholecystokinin; Regional Blood Flow; RNA, Messenger; Sensory Receptor Cells; Sincalide; Somatostatin; Stomach; Stomach Ulcer | 1999 |
The role of brain-gut peptides in the control of sodium appetite.
Topics: Animals; Appetite; Bombesin; Brain; Captopril; Cholecystokinin; Digestive System Physiological Phenomena; Furosemide; Hormone Antagonists; Proglumide; Receptors, Cholecystokinin; Sincalide; Sodium, Dietary | 1999 |
Pharmacological and molecular characterization of muscular cholecystokinin receptors in the human lower oesophageal sphincter.
Topics: Adult; Aged; Benzodiazepines; Benzodiazepinones; Esophagogastric Junction; Female; Gastric Emptying; Gastrins; Gastrointestinal Agents; Gene Expression; Hormone Antagonists; Humans; In Vitro Techniques; Indoleacetic Acids; Male; Middle Aged; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Restriction Mapping; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sincalide; Thiazoles | 2000 |
Interaction of serotonin and cholecystokinin in the lateral parabrachial nucleus to control sodium intake.
Topics: Amphetamines; Animals; Appetite; Drug Interactions; Homeostasis; Intralaminar Thalamic Nuclei; Male; Methysergide; Microinjections; Models, Neurological; Neurons; Proglumide; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists; Sincalide; Sodium, Dietary | 2001 |
Role of cholecystokinin-8 in nerve growth factor and nerve growth factor mRNA expression in carrageenan-induced joint inflammation in adult rats.
Topics: Animals; Arthritis, Experimental; Carrageenan; Disease Models, Animal; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Female; Joints; Nerve Growth Factor; Proglumide; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sincalide | 2002 |
Role for the cholecystokinin-A receptor in fever: a study of a mutant rat strain and a pharmacological analysis.
Topics: Animals; Dose-Response Relationship, Drug; Fever; Gene Deletion; Hormone Antagonists; Lipopolysaccharides; Male; Mutagenesis; Proglumide; Rats; Rats, Inbred OLETF; Rats, Mutant Strains; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Satiety Response; Sincalide | 2003 |
Differential mechanism and site of action of CCK on the pancreatic secretion and growth in rats.
Topics: Afferent Pathways; Amylases; Animals; Capsaicin; Cholecystokinin; Duodenum; Eating; Lipase; Male; Organ Size; Pancreas; Proglumide; Rats; Rats, Wistar; Sincalide; Trypsin; Trypsinogen; Vagotomy; Vagus Nerve | 2003 |
Anxiogenic effect of cholecystokinin in the dorsal periaqueductal gray.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Appetite Depressants; Cell Count; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Hormone Antagonists; Immunohistochemistry; Indoles; Male; Maze Learning; Meglumine; Microinjections; Neurons; Periaqueductal Gray; Proglumide; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Sincalide; Superior Colliculi; Time Factors | 2004 |
Cholecystokinin octapeptide inhibits carotid sinus baroreflex in anesthetized rats.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Baroreflex; Calcium Channel Agonists; Carotid Sinus; Depression, Chemical; In Vitro Techniques; Male; NG-Nitroarginine Methyl Ester; Proglumide; Rats; Rats, Sprague-Dawley; Sincalide | 2004 |
Suppression of food intake by GI fatty acid infusions: roles of celiac vagal afferents and cholecystokinin.
Topics: Action Potentials; Animals; Cholecystokinin; Digestive System; Eating; Energy Intake; Fatty Acids; Hormone Antagonists; Infusions, Parenteral; Male; Proglumide; Rats; Rats, Sprague-Dawley; Sincalide; Time Factors; Vagotomy; Vagus Nerve | 2004 |
The effects of an essential fatty acid compound and a cholecystokinin-8 antagonist on iron deficiency induced anorexia and learning deficits.
Topics: Animal Feed; Animals; Avoidance Learning; Cholecystokinin; Energy Intake; Hormone Antagonists; Iron Deficiencies; Islets of Langerhans; Linoleic Acid; Male; Motor Activity; Peptide Fragments; Proglumide; Rats; Rats, Long-Evans; Swimming; Weight Gain | 2004 |
Pharmacological study of IQM-97,423, a potent and selective CCK1 receptor antagonist with protective effect in experimental acute pancreatitis.
Topics: Acute Disease; alpha-Amylases; Animals; Binding, Competitive; Cerebral Cortex; Cholecystokinin; Devazepide; Disease Models, Animal; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Neuromuscular Junction; Pancreatitis; Peptide Fragments; Proglumide; Pyrimidinones; Rats; Rats, Wistar; Receptor, Cholecystokinin A | 2004 |
Effect of lipopolysaccharide on expression and characterization of cholecystokinin receptors in rat pulmonary interstitial macrophages.
Topics: Animals; Benzodiazepines; Binding, Competitive; Cell Membrane; Female; Lipopolysaccharides; Macrophages, Alveolar; Proglumide; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; RNA, Messenger; Sincalide; Up-Regulation | 2004 |
Cholecystokinin octapeptide increases spontaneous glutamatergic synaptic transmission to neurons of the nucleus tractus solitarius centralis.
Topics: Anesthetics, Local; Animals; Animals, Newborn; Bicuculline; Biotin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; Glutamic Acid; Hormone Antagonists; Imaging, Three-Dimensional; Immunohistochemistry; In Vitro Techniques; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Peptides; Proglumide; Rats; Rats, Sprague-Dawley; Sincalide; Solitary Nucleus; Synaptic Transmission; Tetrodotoxin; Tyrosine 3-Monooxygenase | 2005 |
Selective CCK-A but not CCK-B receptor antagonists inhibit HT-29 cell proliferation: synergism with pharmacological levels of melatonin.
Topics: Antineoplastic Agents; Apoptosis; Cell Proliferation; Devazepide; Dose-Response Relationship, Drug; Drug Synergism; Gastrins; Growth Inhibitors; HT29 Cells; Humans; Melatonin; Proglumide; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Sincalide | 2005 |
Effects of amylin on feeding of goldfish: interactions with CCK.
Topics: Amyloid; Animals; Appetite Depressants; Cholecystokinin; Dose-Response Relationship, Drug; Drug Interactions; Eating; Goldfish; Injections, Intraperitoneal; Injections, Intraventricular; Islet Amyloid Polypeptide; Peptide Fragments; Proglumide; Receptors, Cholecystokinin; Receptors, Islet Amyloid Polypeptide; Receptors, Peptide | 2006 |
Effect of cholecystokinin octapeptide on diacylglycerol-PKC signaling pathway in rat pulmonary interstitial macrophages stimulated by lipopolysaccharide.
Topics: Animals; Benzodiazepines; Cell Membrane; Cytosol; Diglycerides; Dose-Response Relationship, Drug; Female; Isoenzymes; Lipopolysaccharides; Macrophages, Alveolar; Proglumide; Protein Kinase C; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Signal Transduction; Sincalide | 2005 |
Estrogen and CCK1 receptor modification of mu-opioid receptor binding in the cortex of female rats.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Cerebral Cortex; CHO Cells; Cricetinae; Cricetulus; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Estrogens; Female; Hormone Antagonists; Ovariectomy; Proglumide; Protein Binding; Radioligand Assay; Rats; Rats, Long-Evans; Receptors, Cholecystokinin; Receptors, Opioid, mu; Sincalide; Tritium | 2006 |
[Receptor mechanisms underlying the modulation of lipopolysaccharide-induced nuclear factor-kappaB expression in vascular endothelial cells by cholecystokinin octapeptide].
Topics: Benzodiazepines; Cells, Cultured; Endothelial Cells; Humans; Lipopolysaccharides; NF-kappa B; Proglumide; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Sincalide; Umbilical Veins | 2006 |
Anthranilic acid based CCK1 receptor antagonists and CCK-8 have a common step in their "receptor desmodynamic processes".
Topics: Animals; Binding, Competitive; Biological Assay; Humans; Indoles; Ligands; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; ortho-Aminobenzoates; Pancreas; Proglumide; Protein Conformation; Rats; Receptor, Cholecystokinin A; Sincalide; Spectrometry, Fluorescence; Structure-Activity Relationship | 2006 |
Peripheral participation of cholecystokinin in the morphine-induced peripheral antinociceptive effect in non-diabetic and diabetic rats.
Topics: Animals; Area Under Curve; Cholecystokinin; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Drug Interactions; Formaldehyde; Male; Morphine; Narcotics; Neuralgia; Pain Measurement; Pain Threshold; Peptide Fragments; Proglumide; Rats; Rats, Wistar | 2007 |
Vagally mediated, nonparacrine effects of cholecystokinin-8s on rat pancreatic exocrine secretion.
Topics: Animals; Autonomic Fibers, Preganglionic; Brain Stem; Capsaicin; Caseins; Hormone Antagonists; Microinjections; Pancreas, Exocrine; Paracrine Communication; Proglumide; Proteins; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Sincalide; Vagotomy; Vagus Nerve | 2007 |
Cholecystokinin-8s excites identified rat pancreatic-projecting vagal motoneurons.
Topics: Action Potentials; Anesthetics, Local; Animals; Animals, Newborn; Autonomic Fibers, Preganglionic; Brain Stem; Calcium; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Hormone Antagonists; Motor Neurons; Pancreas; Pancreatic Polypeptide; Patch-Clamp Techniques; Potassium; Potassium Channels, Calcium-Activated; Proglumide; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Sincalide; Tetrodotoxin; Vagus Nerve | 2007 |
Interaction of apolipoprotein AIV with cholecystokinin on the control of food intake.
Topics: Animals; Antioxidants; Apolipoproteins A; Appetite Depressants; Dose-Response Relationship, Drug; Feeding Behavior; Hormone Antagonists; Intestine, Small; Male; Proglumide; Rats; Rats, Sprague-Dawley; Sincalide; Time Factors | 2007 |
Involvement of cholecystokinin receptor in the inhibition of gastrointestinal motility by oxytocin in ovariectomized rats.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Eating; Female; Gastric Emptying; Gastrointestinal Motility; Gastrointestinal Transit; Ovariectomy; Oxytocin; Phenylurea Compounds; Proglumide; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Receptors, Oxytocin; Sincalide; Vasotocin | 2008 |
Responses of human sling and clasp fibers to cholecystokinin (CCK) and gastrin through CCK receptors.
Topics: Adult; Benzodiazepines; Dose-Response Relationship, Drug; Esophageal Sphincter, Lower; Esophagectomy; Female; Gastrins; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Myocytes, Smooth Muscle; Proglumide; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Sincalide | 2008 |
Localization of CCK-1R in the omasum and role of CCK in the regulation of omasal contractions in sheep.
Topics: Animals; Atropine; Electromyography; Hormone Antagonists; In Vitro Techniques; Indoles; Meglumine; Muscle Contraction; Omasum; Proglumide; Receptors, Cholecystokinin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sheep; Sincalide; Tetrodotoxin | 2008 |
Anti-inflammatory action of cholecystokinin and melatonin in the rat parotid gland.
Topics: Animals; Anti-Inflammatory Agents; Escherichia coli; Hormone Antagonists; Injections, Intraperitoneal; Lipopolysaccharides; Lysine; Melatonin; Neutrophil Infiltration; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Organ Size; Parasympathectomy; Parotid Gland; Parotitis; Peroxidase; Proglumide; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptor, Melatonin, MT2; Sincalide; Sympathectomy; Tryptamines | 2010 |
Additive effects of cannabinoid CB1 receptors blockade and cholecystokinin on feeding inhibition.
Topics: Animals; Anorexia; Benzoxazines; Brain; Drug Synergism; Feeding Behavior; Gene Expression; Genes, fos; Male; Morpholines; Naphthalenes; Piperidines; Proglumide; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cholecystokinin B; Rimonabant; Sincalide | 2011 |
Investigation of cholecystokinin receptors in the human lower esophageal sphincter.
Topics: Aged; Blotting, Western; Esophageal Sphincter, Lower; Esophagectomy; Esophagogastric Junction; Esophagus; Female; Gene Expression Regulation; Humans; Inhibitory Concentration 50; Isotonic Solutions; Male; Middle Aged; Proglumide; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Sincalide | 2014 |
Gut vagal afferents are necessary for the eating-suppressive effect of intraperitoneally administered ginsenoside Rb1 in rats.
Topics: Animals; Appetite Depressants; Dose-Response Relationship, Drug; Eating; Ginsenosides; Glucose; Hormone Antagonists; Injections, Intraperitoneal; Male; Neurons, Afferent; Proglumide; Rats, Long-Evans; Receptor, Cholecystokinin A; Satiation; Sincalide; Vagus Nerve | 2015 |
Effect of intracerebroventricular administration of two molecular forms of sulfated CCK octapeptide on anxiety-like behavior in the zebrafish danio rerio.
Topics: Animals; Anxiety; Behavior, Animal; Benzodiazepines; Brain; Carbolines; Injections, Intraventricular; Locomotion; Proglumide; Sincalide; Zebrafish; Zebrafish Proteins | 2020 |