Page last updated: 2024-08-23

progabide and gamma-aminobutyric acid

progabide has been researched along with gamma-aminobutyric acid in 159 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Research

Studies (159)

TimeframeStudies, this research(%)All Research%
pre-1990117 (73.58)18.7374
1990's21 (13.21)18.2507
2000's10 (6.29)29.6817
2010's11 (6.92)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bartholini, G; Desarmenien, M; Feltz, P; Headley, PM; Kaplan, JP; Lloyd, KG; Raizon, BM; Worms, P1
Bartholini, G4
Bachus, SE; Dale, J; Goodman, L; Kaneda, H; Shirakawa, O; Tamminga, CA1
Gautam, SK; Kulkarni, SK1
Greenshaw, AJ; McManus, DJ1
Morimoto, K; Nakamura, Y; Okamoto, M; Otsuki, S; Sato, K; Sato, M1
Mehta, AK; Ticku, MK1
Moran, M; Tamminga, CA; Thaker, GK1
Decourt, JP; Mura, P; Papet, Y; Piriou, A; Reiss, D1
Bartholini, G; Oblin, A; Zivkovic, B2
Besson, MJ; Caboche, J; Le Saux, F; Maurin, Y; Mitrovic, N; Sauter, A1
Morimoto, K1
Benoit, JP; Couvreur, P; Deverre, JR; Gayral, P; Letourneux, Y; Loiseau, P1
Porter, RJ1
Cudennec, A; Duverger, D; Lloyd, KG; MacKenzie, ET; McCulloch, J; Motohashi, N; Nishikawa, T; Scatton, B1
Blair, AJ; Crawford, IL; Feldman, M; Petty, F; Stevens, MH; Taylor, IL; Thirlby, RC; Walsh, JH1
Gale, RG; Little, HJ; Nutt, DJ; Standing, BL; Taylor, SC1
Davidoff, RA1
Bossi, L; Fournier, V; Morselli, PL; Musch, B1
Lloyd, KG; Perrault, G; Zivkovic, B1
Bathien, N; Rondot, P1
Atmadja, S; Baimbridge, KG; Fibiger, HC; Mithani, S1
Koe, BK; Kondratas, E; Russo, LL1
Bathien, N; Fournier, V; Morselli, PL; Rondot, P; Ziegler, M1
Rondot, P1
Lima, L; Sourkes, TL1
Bossi, L; Girard, M; Poulain, D1
Hilakivi, I; Hilakivi, LA; Loikas, P; Taira, T1
Chweh, AY; Kupferberg, HJ; Swinyard, EA; Wolf, HH1
Rastogi, SK; Ticku, MK2
Green, AR; Johnson, P; Mountford, JA; Nimgaonkar, VL1
Bergmann, KJ1
Di Scala, G; Fibiger, HC; Martin-Iverson, MT; Phillips, AG1
Nishikawa, T; Scatton, B1
Fadda, F; Gessa, GL; Meloni, R; Mosca, E1
Goldstein, M; Lloyd, KG; Willigens, MT1
Arbilla, S; Bartholini, G; Fage, D; Langer, SZ; Oblin, A; Scatton, B; Zivkovic, B1
Moura, D; Soares-da-Silva, P1
Löscher, W; Schwark, WS1
Lloyd, KG; Pilc, A; Thuret, F1
Bovier, P; Hilleret, H; Tissot, R1
Curet, O; Dennis, T; Nishikawa, T; Scatton, B1
Lloyd, KG1
Chweh, AY; Swinyard, EA; Ulloque, RA1
Chweh, AY; Lin-Michell, E; Swinyard, EA1
Green, AR1
Little, HJ; Nutt, DJ; Taylor, SC1
Goodwin, GM; Gray, JA; Green, AR; Metz, A1
Apud, JA; Masotto, C; Racagni, G1
Bartholini, G; Lloyd, KG; Scatton, B; Zivkovic, B1
Bartholini, G; Depoortere, H; Lloyd, KG; Sanger, D; Zivkovic, B1
Lindgren, S1
Benassi, E; Besio, G; Bo, GP; Cocito, L; Loeb, C; Maffini, M; Mainardi, P; Morselli, PL1
Graves, NM; Holmes, GB; Leppik, IE1
Chadwick, D; Crawford, P1
Comi, G; Ferini-Strambi, L; Filippi, M; Giusti, MC; Medaglini, S; Poggi, A; Smirne, S1
de Feo, MR; Mecarelli, O; Ricci, GF; Rina, MF1
Davis, SS; Farraj, NF; Parr, GD; Stevens, HN2
Benassi, E; Besio, G; Bianchetti, G; Loeb, C; Morselli, PL1
Bowman, T; Cloyd, J; Crosby, C; Dreifuss, FE; Graves, N; Jacobs, M; Leppik, IE; Porter, R; Santilli, N; Stackman, J1
Fariello, R; Maddrey, WC; Munoz, SJ1
Brundage, RC; Cloyd, JC; Graves, NM; Leppik, IE; Welty, TE1
Manev, H; Pericić, D1
Schmidt, D; Utech, K1
Barre, J; Brandebourger, M; Hamberger, C; Taiclet, A; Thenot, JP; Tillement, JP; Urien, S1
Barre, J; Essassi, D; Grimaldi, B; Hamberger, C; Taiclet, A; Thenot, JP; Tillement, JP; Urien, S1
Gupta, S; Koller, WC; Rubino, F1
Breton, D; Krall, RL; Rudick, RA1
Lheroux, A; Luquin, MR; Martinez Lage, JM; Obeso, JA; Scatton, B1
Chweh, AY; Swinyard, EA; Wolf, HH1
Ascalone, V; Dal Bo', L1
Bennett, JP; Cruz, CJ; Ferrari, MB1
Beaussart, M; Benoit, C; Broglin, D; Cambier, J; Cenraud, M; Chatel, M; Deville, MC; Fournier, V; Loiseau, P; Musch, B1
Braendgaard, H; Dupont, E; Mondrup, K1
Burke, JT; Thénot, JP1
Johns, KL; Wood, JD1
Löscher, W1
Ascalone, V; Catalani, P; Dal Bò, L1
Bartholini, G; Scatton, B; Zivkovic, B1
Arbilla, S; Bartholini, G; Beaumont, K; Briley, M; De Montis, G; Langer, SZ; Lloyd, KG; Scatton, B1
Bovier, P; Broekkamp, CL; Lloyd, KG1
Bryere, P; Kaijima, M; Naquet, R; Valin, A1
Bergmann, KJ; Limongi, JC; Lowe, YH; Mendoza, MR; Yahr, MD1
Charlier, M; Delwaide, PJ; Gonce, M; Schoenen, J1
Classen, K; Göthert, M; Schlicker, E1
Christensen, SE; Dupont, E; Mondrup, K; Olivarius, BF; Orskov, H1
Bovier, P; Broekkamp, CL; Lloyd, KG; Worms, P1
Bartholini, G; Depoortere, H; Durand, A; Lloyd, KG; Morselli, PL; Worms, P1
Bartholini, G; Constantinidis, J; Dedek, J; Lloyd, KG; Scatton, B; Tissot, R; Zivkovic, B1
Bartholini, G; Scatton, B2
Wood, PL1
Bartholini, G; Lloyd, KG; Scatton, B; Worms, P; Zivkovic, B1
Bartholini, G; Broekkamp, C; Depoortere, H; Fournier, V; Lloyd, KG; Morselli, PL; Scatton, B; Worms, P; Zivkovic, B1
Bossi, L; Guyot, M; Loiseau, P; Morselli, PL; Orofiamma, B1
Dupont, E; Mondrup, K; Pedersen, E1
Mondrup, K; Pedersen, E2
Schmidt, D1
Bossi, L; Martínez Vila, E; Martínez-Lage, JM; Morales, G; Orofiamma, B; Viteri, C1
Angelo, HR; Christensen, JM; Dam, M; Gram, L; Hansen, BS; Lyon, BB; Philbert, A1
Schwarz, M; Sontag, KH; Turski, L1
Bossi, L; Lloyd, KG; Morselli, PL; Munari, C; Worms, P1
Broekkamp, CL; Le Pichon, M; Lloyd, KG1
Bialer, M; Johno, I; Levy, RH; Nickelson, SA1
Sanger, DJ1
Marsden, CD; Sheehy, MP1
Butt, WR; Gomeni, R; London, DR; Menon, VJ; Morselli, PL; Thiercelin, JF1
Fariello, RG; Golden, GT1
Lapierre, YD; Rastogi, RB; Rastogi, SK; Singhal, RL1
Kupferberg, HJ; Lambert, T; Yonekawa, W1
Albertson, TE; Joy, RM; Stark, LG1
Bianchetti, G; Deves, C; Morselli, PL; Padovani, P; Thenot, JP1
Debeljuk, L; Díaz, MD; Maines, VM; Seilicovich, A1
Johno, I; Levy, RH; Ludwick, BT1
Dring, LG; Fraisse-André, J; Gillet, G; Lee, CR; Morselli, PL1
Cagiano, R; Cuomo, V; Mocchetti, I; Racagni, G1
Cepeda, C; Lloyd, KG; Naquet, R; Worms, P1
Georgiev, VP; Kambourova, TS; Lazarova, MB1
Berthier, M; Bonneau, D; Chevrel, J; Desbordes, JM; Jaeken, J; Laborit, H; Oriot, D1
Guyot, M; Kroetz, DL; Levy, RH; Loiseau, P1
Pierce, MW; Shu, VS1
Kubová, H; Mares, P; Polásek, R; Slamberová, R; Vorlícek, J1
Agmo, A; Garcés, I; Paredes, RG; Sierra, L1
Dey, DK; Larose, DT1
Allain, P; Cailleux, A; Lainé-Cessac, P1
Hougaard, P; Lee, ML; Whitmore, GA1
Agmo, A; Belzung, C1
Baulac, M; Lanoé, Y; Nordmann, JP1
Kozuchová, A; Mares, P; Stanková, L1
Baulac, M; Nordmann, JP; Van Egroo, C1
Louis, ED1
Gadbury, GL; Iyer, HK1
Kulkarni, SK; Naidu, PS1
Mizusawa, H1
Cook, RJ; Wei, W1
Lin, X; Zhang, D1
Rösch, T1
France, CP; McMahon, LR1
Bhandari, M; Haynes, RB1
Lin, X; Wang, YG; Zhu, M1
Jiang, Z; Park, E; Qu, A; Song, PX1
Sumi, M; Tango, T1
Hagino, T; Haro, H; Ochiai, S; Sato, E; Senga, S; Watanabe, Y1
Carey, VJ; Wang, YG1
Westgate, PM1
Moreno, E; Negrín, MA; Vázquez-Polo, FJ1
Chen, M; Li, M; Liu, LP; Liu, Y; Wang, RF; Zhang, DK1
Ara, N; Iuchi, A; Miyoshi, H; Mizuguchi, Y; Nagase, N; Oishi, Y; Oki, T1
Gargiulo, R; Lerma, EV; Suhail, F1
Kong, L; Li, Z; Wang, M; Zhang, L1
Berggren, K; Castagnoli, N; Grönberg, G; Hayes, MA; Li, XQ; Weidolf, L1
Alabed, S; Bergman, H; Latifeh, Y; Mohammad, HA1

Reviews

13 review(s) available for progabide and gamma-aminobutyric acid

ArticleYear
Antispasticity drugs: mechanisms of action.
    Annals of neurology, 1985, Volume: 17, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Baclofen; Benzodiazepines; Central Nervous System; Dantrolene; gamma-Aminobutyric Acid; Glycine; Humans; Muscle Relaxants, Central; Muscle Spasticity; Neurotransmitter Agents; Phenothiazines; Rats; Receptors, Neurotransmitter; Spinal Cord

1985
[Implications of GABAergic synapses in neuropsychiatry].
    Journal de pharmacologie, 1985, Volume: 16 Suppl 2

    Topics: 4-Aminobutyrate Transaminase; Animals; Anti-Anxiety Agents; Anticonvulsants; Antidepressive Agents; Anxiety; Brain; Cats; Cerebral Cortex; Depressive Disorder; Disease Models, Animal; Dyskinesia, Drug-Induced; Epilepsy; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haplorhini; Humans; Mental Disorders; Muscimol; Receptors, GABA-A; Seizures; Synapses; Synaptic Transmission

1985
Progabide: a new GABA-mimetic agent in clinical use.
    Clinical neuropharmacology, 1985, Volume: 8, Issue:1

    Topics: Anticonvulsants; Brain Chemistry; Chemical Phenomena; Chemistry; Epilepsy; gamma-Aminobutyric Acid; Humans; Movement Disorders; Muscle Spasticity; Receptors, GABA-A

1985
[Drug activation of GABAergic transmission in the central nervous system: benzodiazepines and GABAergic agonists].
    Acta medica portuguesa, 1985, Volume: 6, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chemical Phenomena; Chemistry; Cyclic GMP; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Receptors, GABA-A; Synaptic Transmission; Valproic Acid

1985
[GABAergic theory of epilepsy].
    La Revue du praticien, 1986, Jan-21, Volume: 36, Issue:5

    Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Dogs; Epilepsy; gamma-Aminobutyric Acid; Humans; Mice; Nerve Endings; Pentylenetetrazole; Phenobarbital; Phenytoin; Rats; Receptors, GABA-A; Synapses; Valproic Acid

1986
Changes in gamma-aminobutyric acid biochemistry and seizure threshold.
    Annals of the New York Academy of Sciences, 1986, Volume: 462

    Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Bicuculline; Brain; Cerebral Cortex; Clonidine; Corpus Striatum; Electroconvulsive Therapy; gamma-Aminobutyric Acid; Hippocampus; Hypothalamus; Male; Mice; Mice, Inbred Strains; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin

1986
Determination of antiepileptic drugs.
    Journal of chromatography, 1985, May-10, Volume: 340

    Topics: Anticonvulsants; Barbiturates; Carbamazepine; Chromatography, Gas; Chromatography, Liquid; Clonazepam; gamma-Aminobutyric Acid; Gas Chromatography-Mass Spectrometry; Humans; Mephenytoin; Monitoring, Physiologic; Phenytoin; Primidone; Succinimides; Valproic Acid

1985
GABA system, GABA receptor agonists and dyskinesia.
    Modern problems of pharmacopsychiatry, 1983, Volume: 21

    Topics: Basal Ganglia; Cholinergic Fibers; Dopamine; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Humans; Huntington Disease; Levodopa; Movement Disorders; Receptors, Cell Surface; Receptors, GABA-A

1983
Handling seizure data: special problems.
    Epilepsy research. Supplement, 1993, Volume: 10

    Topics: Anticonvulsants; Clinical Trials as Topic; Data Interpretation, Statistical; Drug Therapy, Combination; Electroencephalography; Epilepsy; Epilepsy, Complex Partial; Epilepsy, Tonic-Clonic; gamma-Aminobutyric Acid; Humans; Nipecotic Acids; Tiagabine; Valproic Acid

1993
A new twist for stopping the shakes? Revisiting GABAergic therapy for essential tremor.
    Archives of neurology, 1999, Volume: 56, Issue:7

    Topics: Acetates; Adult; Amines; Cyclohexanecarboxylic Acids; GABA Agonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Primidone; Propranolol; Tremor

1999
[Autosomal dominant hereditary distal myopathy linked to chromosome 14].
    Ryoikibetsu shokogun shirizu, 2001, Issue:35

    Topics: Chromosomes, Human, Pair 14; Diagnosis, Differential; gamma-Aminobutyric Acid; Genes, Dominant; Genetic Linkage; Humans; Muscle, Skeletal; Muscular Dystrophies

2001
Cardiovascular disease and chronic kidney disease.
    Disease-a-month : DM, 2015, Volume: 61, Issue:9

    Topics: Cardiovascular Diseases; Coronary Artery Disease; gamma-Aminobutyric Acid; Heart Diseases; Humans; Peripheral Vascular Diseases; Renal Insufficiency, Chronic

2015
Gamma-aminobutyric acid agonists for antipsychotic-induced tardive dyskinesia.
    The Cochrane database of systematic reviews, 2018, 04-17, Volume: 4

    Topics: Antipsychotic Agents; Baclofen; Dyskinesia, Drug-Induced; GABA Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Placebos; Randomized Controlled Trials as Topic; Valproic Acid

2018

Trials

22 trial(s) available for progabide and gamma-aminobutyric acid

ArticleYear
GABAmimetics: a new class of antidepressant agents?
    Archives of general psychiatry, 1990, Volume: 47, Issue:3

    Topics: Antidepressive Agents; Depressive Disorder; Female; gamma-Aminobutyric Acid; Humans; Middle Aged

1990
Clinical activity of GABA agonists in neuroleptic- and L-dopa-induced dyskinesia.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Antipsychotic Agents; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Dyskinesia, Drug-Induced; Electromyography; gamma-Aminobutyric Acid; Humans; Levodopa

1985
Movement disorders in patients with coexistent neuroleptic-induced tremor and tardive dyskinesia: EMG and pharmacological study.
    Advances in neurology, 1987, Volume: 45

    Topics: Antipsychotic Agents; Clinical Trials as Topic; Corpus Striatum; Double-Blind Method; Dyskinesia, Drug-Induced; Electromyography; gamma-Aminobutyric Acid; Humans; Parkinson Disease, Secondary; Receptors, Dopamine; Receptors, GABA-A; Tremor

1987
Therapeutic response to progabide in neuroleptic- and L-dopa-induced dyskinesias.
    Clinical neuropharmacology, 1987, Volume: 10, Issue:3

    Topics: Adult; Aged; Antipsychotic Agents; Clinical Trials as Topic; Double-Blind Method; Dyskinesia, Drug-Induced; Female; gamma-Aminobutyric Acid; Humans; Levodopa; Male; Middle Aged; Parkinson Disease, Secondary; Placebos

1987
Preliminary observations on the activity of progabide, administered as monotherapy in complex partial seizures.
    International journal of clinical pharmacology research, 1988, Volume: 8, Issue:5

    Topics: Adolescent; Adult; Clinical Trials as Topic; Drug Administration Schedule; Epilepsy, Temporal Lobe; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged

1988
Compliant populations: variability in serum concentrations.
    Epilepsy research. Supplement, 1988, Volume: 1

    Topics: Anticonvulsants; Carbamazepine; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Epilepsy; Felbamate; Female; gamma-Aminobutyric Acid; Humans; Male; Patient Compliance; Phenylcarbamates; Phenytoin; Propylene Glycols; Random Allocation

1988
A comparative study of progabide, valproate, and placebo as add-on therapy in patients with refractory epilepsy.
    Journal of neurology, neurosurgery, and psychiatry, 1986, Volume: 49, Issue:11

    Topics: Adolescent; Adult; Anticonvulsants; Chemical and Drug Induced Liver Injury; Drug Interactions; Drug Therapy, Combination; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Patient Compliance; Phenytoin; Valproic Acid

1986
A controlled study of progabide in partial seizures: methodology and results.
    Neurology, 1987, Volume: 37, Issue:6

    Topics: Adolescent; Adult; Carbamazepine; Clinical Trials as Topic; Female; gamma-Aminobutyric Acid; Humans; Male; Phenytoin; Seizures

1987
Effect of progabide on serum phenytoin and carbamazepine concentrations.
    Clinical neuropharmacology, 1987, Volume: 10, Issue:6

    Topics: Adult; Carbamazepine; Convulsants; Double-Blind Method; Drug Evaluation; Female; gamma-Aminobutyric Acid; Humans; Male; Phenytoin; Random Allocation; Seizures

1987
Progabide for refractory partial epilepsy: a controlled add-on trial.
    Neurology, 1986, Volume: 36, Issue:2

    Topics: Adolescent; Adult; Aged; Anticonvulsants; Carbamazepine; Clinical Trials as Topic; Double-Blind Method; Drug Interactions; Drug Therapy, Combination; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Phenobarbital; Phenytoin; Random Allocation

1986
Pharmacologic probe with progabide of GABA mechanisms in essential tremor.
    Archives of neurology, 1987, Volume: 44, Issue:9

    Topics: Brain; Double-Blind Method; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Random Allocation; Tremor

1987
The GABA-agonist progabide for spasticity in multiple sclerosis.
    Archives of neurology, 1987, Volume: 44, Issue:10

    Topics: Adult; Anticonvulsants; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Multiple Sclerosis; Muscle Spasticity

1987
Potentiation of the "dopa" effect in parkinsonism by a direct GABA receptor agonist.
    Lancet (London, England), 1984, Mar-10, Volume: 1, Issue:8376

    Topics: Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Drug Synergism; gamma-Aminobutyric Acid; Humans; Levodopa; Parkinson Disease; Receptors, Cell Surface; Receptors, GABA-A

1984
The potential use of GABA agonists in psychiatric disorders: evidence from studies with progabide in animal models and clinical trials.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:6

    Topics: Adjustment Disorders; Animals; Anticonvulsants; Biogenic Amines; Brain; Clinical Trials as Topic; Corpus Striatum; Depressive Disorder; Disease Models, Animal; Dopamine; gamma-Aminobutyric Acid; Humans; Imipramine; Limbic System; Neurons; Rats

1983
Double-blind crossover trial of progabide versus placebo in severe epilepsies.
    Epilepsia, 1983, Volume: 24, Issue:6

    Topics: Adolescent; Adult; Child; Clinical Trials as Topic; Double-Blind Method; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Placebos

1983
The effect of the GABA-agonist, progabide, on benign essential tremor. A controlled clinical trial.
    Acta neurologica Scandinavica, 1983, Volume: 68, Issue:4

    Topics: Adult; Aged; Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Electromyography; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Time Factors; Tremor

1983
The effect of the GABA-agonist, progabide, on stretch and flexor reflexes and on voluntary power in spastic patients.
    Acta neurologica Scandinavica, 1984, Volume: 69, Issue:4

    Topics: Achilles Tendon; Adult; Clinical Trials as Topic; Electromyography; Female; gamma-Aminobutyric Acid; H-Reflex; Hand; Humans; Isometric Contraction; Leg; Male; Middle Aged; Muscle Contraction; Muscle Spasticity; Muscles; Placebos; Reflex, Monosynaptic; Reflex, Stretch; Tibial Nerve

1984
The clinical effect of the GABA-agonist, progabide, on spasticity.
    Acta neurologica Scandinavica, 1984, Volume: 69, Issue:4

    Topics: Adult; Arm; Chemical Phenomena; Chemistry; Clinical Trials as Topic; Female; gamma-Aminobutyric Acid; Humans; Leg; Male; Middle Aged; Muscle Contraction; Muscle Hypertonia; Muscle Spasticity; Muscles; Placebos; Reflex; Reflex, Stretch; Research Design

1984
Progabide as an add-on drug for epilepsy refractory to high dose antiepileptic drug therapy.
    Neuroscience letters, 1984, Jun-29, Volume: 47, Issue:3

    Topics: Adult; Aged; Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Epilepsy; Epilepsy, Temporal Lobe; gamma-Aminobutyric Acid; Humans

1984
Progabide treatment in severe epilepsy: a double-blind cross-over trial versus placebo.
    Epilepsia, 1984, Volume: 25, Issue:5

    Topics: Adolescent; Adult; Clinical Trials as Topic; Double-Blind Method; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Placebos

1984
Progabide: a controlled trial in partial epilepsy.
    Epilepsia, 1983, Volume: 24, Issue:2

    Topics: Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Epilepsies, Partial; gamma-Aminobutyric Acid; Humans; Random Allocation

1983
GABA and movement disorders.
    Advances in biochemical psychopharmacology, 1981, Volume: 30

    Topics: Anticonvulsants; Baclofen; Clinical Trials as Topic; Double-Blind Method; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Humans; Huntington Disease; Isoniazid; Movement Disorders; Muscimol; Parkinson Disease; Valproic Acid

1981

Other Studies

124 other study(ies) available for progabide and gamma-aminobutyric acid

ArticleYear
New anticonvulsants: Schiff bases of gamma-aminobutyric acid and gamma-aminobutyramide.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:6

    Topics: Animals; Anticonvulsants; Bicuculline; Brain; Cerebellum; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Ganglia, Spinal; Humans; In Vitro Techniques; Lethal Dose 50; Male; Mice; Rats; Schiff Bases

1980
[Potential therapeutic activity of GABA-mimetic drugs in neuropsychiatry].
    Schweizer Archiv fur Neurologie, Neurochirurgie und Psychiatrie = Archives suisses de neurologie, neurochirurgie et de psychiatrie, 1979, Volume: 125, Issue:2

    Topics: 4-Aminobutyrate Transaminase; Basal Ganglia Diseases; Bicuculline; Dopamine; Dyskinesia, Drug-Induced; Epilepsy; Extrapyramidal Tracts; gamma-Aminobutyric Acid; Humans; Huntington Disease; Levodopa; Limbic System; Neural Pathways; Neurons; Neurotransmitter Agents; Parkinson Disease; Psychopharmacology

1979
Co-administration of progabide inhibits haloperidol-induced oral dyskinesias in rats.
    European journal of pharmacology, 1992, Feb-25, Volume: 212, Issue:1

    Topics: Administration, Oral; Animals; Disease Models, Animal; Drug Interactions; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Haloperidol; Male; Mastication; Rats; Rats, Inbred Strains

1992
GABA/BZ-and NMDA-receptor interaction in digoxin-induced convulsions in rats.
    Indian journal of experimental biology, 1991, Volume: 29, Issue:7

    Topics: Animals; Baclofen; Diazepam; Digoxin; Dizocilpine Maleate; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Salts; Seizures

1991
Differential effects of chronic antidepressants in behavioural tests of beta-adrenergic and GABAB receptor function.
    Psychopharmacology, 1991, Volume: 103, Issue:2

    Topics: Albuterol; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Baclofen; Behavior, Animal; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Monoamine Oxidase Inhibitors; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, GABA-A

1991
An analysis of anticonvulsant actions of GABA agonists (progabide and baclofen) in the kindling model of epilepsy.
    Epilepsy research, 1990, Volume: 5, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Dose-Response Relationship, Drug; Electroencephalography; Epilepsy; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Are GABAB receptors involved in the pharmacological effects of ethanol?
    European journal of pharmacology, 1990, Jul-17, Volume: 182, Issue:3

    Topics: Animals; Baclofen; Cells, Cultured; Chlorine; Diazepam; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; N-Methylaspartate; Picrotoxin; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Spinal Cord

1990
Simultaneous determination of progabide and its acid metabolite by reversed-phase high-performance liquid chromatography.
    Journal of chromatography, 1990, Apr-27, Volume: 527, Issue:1

    Topics: Anticonvulsants; Chromatography, High Pressure Liquid; Epilepsy; gamma-Aminobutyric Acid; Humans

1990
Progabide reverses the nigral substance P reduction induced by chronic impairment of dopaminergic transmission.
    European journal of pharmacology, 1985, Jun-07, Volume: 112, Issue:2

    Topics: Animals; gamma-Aminobutyric Acid; Haloperidol; Hydroxydopamines; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, GABA-A; Substance P; Substantia Nigra; Synaptic Transmission; Tyrosine 3-Monooxygenase

1985
Selective antagonists of dopamine receptor subtypes differentially affect substance P levels in the striatum and substantia nigra.
    Brain research, 1987, Sep-22, Volume: 421, Issue:1-2

    Topics: Animals; Benzazepines; Corpus Striatum; Dopamine Antagonists; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Substance P; Substantia Nigra; Sulpiride

1987
Postnatal evolution of the gamma-aminobutyric acid/benzodiazepine receptor complex in a model of inherited epilepsy: the quaking mouse.
    Journal of neurochemistry, 1989, Volume: 52, Issue:2

    Topics: Aging; Animals; Brain; Brain Stem; Cerebellum; Diazepam; Diencephalon; Epilepsy; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Mice, Inbred C57BL; Mice, Quaking; Muscimol; Receptors, GABA-A; Telencephalon

1989
Seizure-triggering mechanisms in the kindling model of epilepsy: collapse of GABA-mediated inhibition and activation of NMDA receptors.
    The Japanese journal of psychiatry and neurology, 1989, Volume: 43, Issue:3

    Topics: Amygdala; Animals; Anticonvulsants; Dibenzocycloheptenes; Dizocilpine Maleate; Electroencephalography; Epilepsy; Evoked Potentials; gamma-Aminobutyric Acid; Kindling, Neurologic; Neural Inhibition; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1989
In-vitro evaluation of filaricidal activity of GABA and 1,3-dipalmitoyl-2-(4-aminobutyryl)glycerol HCl: a diglyceride prodrug.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:3

    Topics: Animals; Anthelmintics; Filaricides; Filarioidea; gamma-Aminobutyric Acid; Microfilariae; Prodrugs; Triglycerides

1989
Mechanisms of action of new antiepileptic drugs.
    Epilepsia, 1989, Volume: 30 Suppl 1

    Topics: Acetamides; Acetates; Amines; Aminocaproates; Aminopyridines; Anti-Anxiety Agents; Anticonvulsants; Aspartic Acid; Benzodiazepines; Benzodiazepinones; Clobazam; Cyclohexanecarboxylic Acids; Dibenzocycloheptenes; Dizocilpine Maleate; Epilepsy; Felbamate; Flumazenil; GABA Antagonists; Gabapentin; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Imidazoles; Lamotrigine; Phenylcarbamates; Propylene Glycols; Receptors, GABA-A; Triazines; Vigabatrin

1989
Effects of the GABA receptor agonist, progabide, upon local cerebral glucose utilization.
    Brain research, 1987, Oct-13, Volume: 423, Issue:1-2

    Topics: Animals; Autoradiography; Brain; Carbon Radioisotopes; Deoxy Sugars; Deoxyglucose; gamma-Aminobutyric Acid; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Effect of GABA on basal and vagally mediated gastric acid secretion and hormone release in dogs.
    The American journal of physiology, 1988, Volume: 254, Issue:5 Pt 1

    Topics: Animals; Baclofen; Blood Glucose; Dogs; gamma-Aminobutyric Acid; Gastric Acid; Gastric Fistula; Gastrins; Gastrointestinal Hormones; Insulin; Male; Receptors, GABA-A; Vagus Nerve

1988
Changes in benzodiazepine/GABA receptor complex function in benzodiazepine-tolerant mice.
    Psychopharmacology, 1988, Volume: 95, Issue:3

    Topics: Animals; Anticonvulsants; Bicuculline; Body Temperature; Drug Tolerance; Flurazepam; gamma-Aminobutyric Acid; Infusions, Intravenous; Male; Mice; Motor Activity; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Time Factors

1988
Neuroleptic-induced oral dyskinesias: effects of progabide and lack of correlation with regional changes in glutamic acid decarboxylase and choline acetyltransferase activities.
    Psychopharmacology, 1987, Volume: 93, Issue:1

    Topics: Animals; Anticonvulsants; Antipsychotic Agents; Brain; Choline O-Acetyltransferase; Dyskinesia, Drug-Induced; Flupenthixol; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Male; Mastication; Motor Activity; Parvalbumins; Rats; Rats, Inbred Strains; S100 Calcium Binding Protein G

1987
[3H]Ro 15-1788 binding to benzodiazepine receptors in mouse brain in vivo: marked enhancement by GABA agonists and other CNS drugs.
    European journal of pharmacology, 1987, Oct-27, Volume: 142, Issue:3

    Topics: Animals; Antipsychotic Agents; Barbiturates; Brain; Buspirone; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intravenous; Male; Mice; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasodilator Agents

1987
[The electrophysiological approach to tardive dyskinesias].
    L'Encephale, 1988, Volume: 14 Spec No

    Topics: Diagnosis, Differential; Dopamine Agents; Dyskinesia, Drug-Induced; Electromyography; gamma-Aminobutyric Acid; Humans; Movement Disorders; Parasympatholytics

1988
Cholinergic and GABAergic regulation of dopamine beta-hydroxylase activity in the adrenal gland of the rat.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:1

    Topics: 5,7-Dihydroxytryptamine; Acetylcholine; Adrenal Glands; Aminocaproates; Animals; Baclofen; Bicuculline; Dopamine beta-Hydroxylase; Enzyme Induction; Fenclonine; gamma-Aminobutyric Acid; Hydroxydopamines; Male; Muscimol; Oxotremorine; Propranolol; Rats; Vigabatrin

1986
[Suicide attempted with progabide].
    Presse medicale (Paris, France : 1983), 1987, Apr-18, Volume: 16, Issue:14

    Topics: Adult; Anticonvulsants; Female; gamma-Aminobutyric Acid; Humans; Male; Suicide, Attempted

1987
Neonatal treatment with monoamine uptake inhibitors alters later response in behavioural 'despair' test to beta and GABA-B receptor agonists.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:1

    Topics: Albuterol; Animals; Animals, Newborn; Antidepressive Agents; Baclofen; Behavior, Animal; Desipramine; gamma-Aminobutyric Acid; Male; Nomifensine; Rats; Rats, Inbred Strains; Time Factors; Zimeldine

1988
Effect of GABA agonists on the neurotoxicity and anticonvulsant activity of benzodiazepines.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: Animals; Anticonvulsants; Benzodiazepines; Drug Synergism; Electroshock; Flunitrazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Muscimol; Nervous System; Receptors, GABA-A

1985
Involvement of a GABAergic mechanism in the anticonvulsant effect of pentobarbital against maximal electroshock-induced seizures in rats.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Bicuculline; Drug Interactions; Electroshock; Ethanol; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Sleep

1985
Some anticonvulsant drugs alter monoamine-mediated behaviour in mice in ways similar to electroconvulsive shock; implications for antidepressant therapy.
    British journal of pharmacology, 1985, Volume: 84, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Anticonvulsants; Antidepressive Agents; Apomorphine; Behavior, Animal; Biogenic Amines; Clonidine; Diazepam; Electroshock; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Motor Activity; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Serotonin; Valproic Acid

1985
The effects of progabide (SL 76002) on locomotor activity and conditioned place preference induced by d-amphetamine.
    European journal of pharmacology, 1985, Jan-02, Volume: 107, Issue:2

    Topics: Animals; Anticonvulsants; Conditioning, Psychological; Dextroamphetamine; gamma-Aminobutyric Acid; Male; Motor Activity; Rats; Receptors, GABA-A

1985
Inhibitory influence of GABA on central serotonergic transmission. Raphé nuclei as the neuroanatomical site of the GABAergic inhibition of cerebral serotonergic neurons.
    Brain research, 1985, Apr-01, Volume: 331, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Brain; gamma-Aminobutyric Acid; Male; Neural Inhibition; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission

1985
Suppression by progabide of ethanol withdrawal syndrome in rats.
    European journal of pharmacology, 1985, Mar-12, Volume: 109, Issue:3

    Topics: Acoustic Stimulation; Animals; Ethanol; gamma-Aminobutyric Acid; Humans; Male; Rats; Rats, Inbred Strains; Seizures; Substance Withdrawal Syndrome; Synaptic Transmission; Tremor

1985
Induction and reversal of dopamine dyskinesia in rat, cat, and monkey.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Animals; Apomorphine; Brain; Cats; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Haplorhini; Humans; Levodopa; Motor Activity; Muscimol; Nomifensine; Piribedil; Rats; Receptors, Dopamine; Receptors, GABA-A; Stereotyped Behavior

1985
Influence of GABA mimetics and lithium on biochemical manifestations of striatal dopamine target cell hypersensitivity.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Animals; Corpus Striatum; gamma-Aminobutyric Acid; Haloperidol; Kinetics; Lithium; Rats; Receptors, Dopamine; Spiperone; Synapses; Synaptic Transmission

1985
Evaluation of different GABA receptor agonists in the kindled amygdala seizure model in rats.
    Experimental neurology, 1985, Volume: 89, Issue:2

    Topics: Amygdala; Animals; Female; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Isoxazoles; Kindling, Neurologic; Muscimol; Muscle Relaxation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1985
Upregulation of gamma-aminobutyric acid (GABA) B binding sites in rat frontal cortex: a common action of repeated administration of different classes of antidepressants and electroshock.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:1

    Topics: Animals; Antidepressive Agents; Cerebral Cortex; Desipramine; Dose-Response Relationship, Drug; Electroshock; Fluoxetine; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Male; Monoamine Oxidase Inhibitors; Nomifensine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin Antagonists; Time Factors; Viloxazine

1985
[Progabide treatment of a case of the syndrome of painful legs and moving toes].
    Revue neurologique, 1985, Volume: 141, Issue:5

    Topics: Adult; Female; gamma-Aminobutyric Acid; Humans; Leg; Middle Aged; Movement Disorders; Pain; Receptors, GABA-A; Syndrome; Toes

1985
Further evidence for, and nature of, the facilitatory GABAergic influence on central noradrenergic transmission.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:2-3

    Topics: Afferent Pathways; Animals; Central Nervous System; Cerebral Cortex; Clonidine; gamma-Aminobutyric Acid; Hypothalamus; Ibotenic Acid; Methoxyhydroxyphenylglycol; Muscimol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Spinal Cord; Synaptic Transmission; Yohimbine

1985
Effects of gamma-aminobutyric acid (GABA) receptor agonists on the neurotoxicity and anticonvulsant activity of barbiturates in mice.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; Dose-Response Relationship, Drug; Drug Synergism; Electroshock; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Nervous System; Oxazoles; Receptors, GABA-A; Seizures

1986
Effect of ethosuximide alone and in combination with gamma-aminobutyric acid receptor agonists on brain gamma-aminobutyric acid concentration, anticonvulsant activity and neurotoxicity in mice.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Brain Chemistry; Ethosuximide; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Mice, Inbred Strains; Nervous System; Pentylenetetrazole; Receptors, GABA-A; Seizures

1986
Anticonvulsant profile of drugs which facilitate GABAergic transmission on convulsions mediated by a GABAergic mechanism.
    Neuropharmacology, 1986, Volume: 25, Issue:2

    Topics: Animals; Anticonvulsants; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; gamma-Aminobutyric Acid; Male; Pentobarbital; Rats; Rats, Inbred Strains; Seizures; Synaptic Transmission

1986
The effects of drugs acting at the GABAA-receptor/ionophore after chemical kindling with the benzodiazepine receptor ligand FG 7142.
    British journal of pharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Bicuculline; Body Temperature; Carbolines; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Mice; Muscimol; Pentobarbital; Pentylenetetrazole; Picrotoxin; Receptors, GABA-A; Seizures; Time Factors

1986
The effects of the GABA-mimetic drugs, progabide and baclofen, on the biochemistry and function of 5-hydroxytryptamine and noradrenaline.
    Neuropharmacology, 1986, Volume: 25, Issue:7

    Topics: Animals; Baclofen; Brain; Brain Chemistry; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Norepinephrine; Receptors, Adrenergic, beta; Receptors, GABA-A; Receptors, Serotonin; Serotonin; Stereoisomerism

1986
Effect of THIP and SL 76002, two clinically experimented GABA-mimetic compounds, on anterior pituitary GABA receptors and prolactin secretion in the rat.
    Life sciences, 1987, Mar-02, Volume: 40, Issue:9

    Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Female; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Kinetics; Male; Muscimol; Ovariectomy; Oxazoles; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
GABA receptor agonists and extrapyramidal motor function: therapeutic implications for Parkinson's disease.
    Advances in neurology, 1987, Volume: 45

    Topics: Acetylcholine; Animals; Antiparkinson Agents; Cholinergic Fibers; Corpus Striatum; Dopamine; Extrapyramidal Tracts; gamma-Aminobutyric Acid; Humans; Motor Skills; Parkinson Disease; Receptors, Dopamine; Receptors, GABA-A; Synapses; Synaptic Transmission

1987
Fengabine, a novel antidepressant GABAergic agent. I. Activity in models for antidepressant drugs and psychopharmacological profile.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Animals; Antidepressive Agents; Avoidance Learning; Behavior, Animal; Bicuculline; Chlorophenols; Clomipramine; Depressive Disorder; Disease Models, Animal; gamma-Aminobutyric Acid; Imipramine; Male; Olfactory Bulb; Rats; Receptors, GABA-A; Seizures; Sleep

1987
Effects of GABAergic drugs on the GABA turnover in the substantia nigra and the corpus striatum of the rat.
    Journal of neural transmission, 1987, Volume: 69, Issue:1-2

    Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1987
Effects of long-lasting antiepileptic therapy on brainstem auditory evoked potentials.
    Neuropsychobiology, 1988, Volume: 19, Issue:2

    Topics: Adolescent; Adult; Anticonvulsants; Brain Stem; Carbamazepine; Child; Epilepsies, Partial; Evoked Potentials, Auditory; Female; gamma-Aminobutyric Acid; Humans; Long-Term Care; Male; Middle Aged; Phenobarbital; Reaction Time; Valproic Acid

1988
Effects of progabide on bicuculline-induced epileptic seizures in developing rats.
    Clinical neuropharmacology, 1988, Volume: 11, Issue:5

    Topics: Aging; Animals; Anticonvulsants; Bicuculline; Female; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Seizures; Status Epilepticus

1988
The stability and solubility of progabide and its related metabolic derivatives.
    Pharmaceutical research, 1988, Volume: 5, Issue:4

    Topics: Anticonvulsants; Drug Stability; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Prodrugs; Solubility; Spectrophotometry; Temperature

1988
Blood levels of progabide and its active metabolite in epileptic patients: relationships to the therapeutic outcome.
    International journal of clinical pharmacology research, 1988, Volume: 8, Issue:6

    Topics: Adult; Dose-Response Relationship, Drug; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Monitoring, Physiologic

1988
Submassive hepatic necrosis associated with the use of progabide: a GABA receptor agonist.
    Digestive diseases and sciences, 1988, Volume: 33, Issue:3

    Topics: Adult; Anticonvulsants; Chemical and Drug Induced Liver Injury; Female; gamma-Aminobutyric Acid; Humans; Liver; Liver Function Tests; Necrosis; Seizures

1988
Progabide, a GABA mimetic drug, stimulates the secretion of plasma corticosterone in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:4

    Topics: Animals; Anticonvulsants; Clonidine; Corticosterone; Dexamethasone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Picrotoxin; Rats; Rats, Inbred Strains; Stimulation, Chemical

1987
A reversed-phase high-performance liquid chromatography assay procedure for progabide and its related metabolic derivatives.
    Pharmaceutical research, 1987, Volume: 4, Issue:1

    Topics: Calibration; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Solutions

1987
Progabide and SL 75102 binding to plasma proteins and red blood cells in humans.
    International journal of clinical pharmacology, therapy, and toxicology, 1987, Volume: 25, Issue:4

    Topics: Anticonvulsants; Blood Proteins; Dialysis; Erythrocytes; gamma-Aminobutyric Acid; Hematocrit; Humans; Protein Binding

1987
Effect of erythrocytes and plasma protein binding on the transport of progabide and SL 75102 through the rat blood-brain barrier.
    Biochemical pharmacology, 1987, Aug-15, Volume: 36, Issue:16

    Topics: Biological Transport, Active; Blood Proteins; Blood-Brain Barrier; Erythrocytes; gamma-Aminobutyric Acid; Humans; Lipoproteins; Mathematics

1987
Progabide in Parkinson's disease.
    Annals of neurology, 1987, Volume: 22, Issue:2

    Topics: gamma-Aminobutyric Acid; Humans; Parkinson Disease

1987
Involvement of a GABAergic mechanism in the pharmacologic action of phenytoin.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:5

    Topics: Animals; Anticonvulsants; Baclofen; Electroshock; gamma-Aminobutyric Acid; Male; Mice; Phenytoin; Postural Balance; Seizures

1986
Chromatographic selectivity and maintenance of column efficiency during the high-performance liquid chromatographic analysis of progabide and its acid metabolite.
    Journal of chromatography, 1986, Oct-31, Volume: 382

    Topics: Anticonvulsants; Carbamazepine; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Humans; Spectrophotometry, Ultraviolet

1986
GABA-mimetic drugs enhance apomorphine-induced contralateral turning in rats with unilateral nigrostriatal dopamine denervation: implications for the therapy of Parkinson's disease.
    Annals of neurology, 1987, Volume: 21, Issue:1

    Topics: Alkynes; Aminocaproates; Animals; Antiparkinson Agents; Apomorphine; Drug Synergism; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Parkinson Disease; Rats; Rats, Inbred Strains

1987
Long-term treatment of epilepsy: open multicenter trial with progabide in epileptic patients.
    European neurology, 1987, Volume: 26, Issue:2

    Topics: Adolescent; Adult; Anticonvulsants; Child; Child, Preschool; Dose-Response Relationship, Drug; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Infant; Male; Middle Aged

1987
Progabide in the treatment of hyperkinetic extrapyramidal movement disorders.
    Acta neurologica Scandinavica, 1985, Volume: 72, Issue:3

    Topics: Adolescent; Adult; Aged; Athetosis; Basal Ganglia Diseases; Child; Chorea; Female; gamma-Aminobutyric Acid; Humans; Hyperkinesis; Male; Middle Aged; Myoclonus; Tourette Syndrome

1985
Stability of the amino acid content of nerve endings after administration of gamma-aminobutyrate agonists and antagonists.
    Neuropharmacology, 1985, Volume: 24, Issue:7

    Topics: Amino Acids; Animals; Anticonvulsants; Aspartic Acid; Baclofen; Bicuculline; Brain Chemistry; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Mice; Muscimol; Nerve Endings; Picrotoxin; Synaptosomes

1985
Anticonvulsant action of GABA agonists and prodrugs on minor and major seizures in epileptic gerbils. Comparison with mouse models of seizure states.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 276, Issue:2

    Topics: Animals; Anticonvulsants; Disease Models, Animal; Electroshock; Female; gamma-Aminobutyric Acid; Gerbillinae; In Vitro Techniques; Isoxazoles; Mice; Pentylenetetrazole; Seizures; Species Specificity

1985
Determination of progabide and its acid metabolite in biological fluids by high-performance liquid chromatography on silica column with ultraviolet detection.
    Journal of chromatography, 1985, Nov-08, Volume: 344

    Topics: Biotransformation; Body Fluids; Chromatography, High Pressure Liquid; Drug Stability; Electrochemistry; gamma-Aminobutyric Acid; Humans; Kinetics; Solvents; Spectrophotometry, Ultraviolet

1985
Experimental basis for the antidepressant action of the GABA receptor agonist progabide.
    Neuroscience letters, 1984, Jun-29, Volume: 47, Issue:3

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Brain; Depressive Disorder; gamma-Aminobutyric Acid; Humans; Mice; Norepinephrine; Receptors, Cell Surface; Receptors, GABA-A; Serotonin; Synaptic Transmission

1984
Pharmacology of the GABAergic system: effects of progabide, a GABA receptor agonist.
    Psychoneuroendocrinology, 1984, Volume: 9, Issue:2

    Topics: Animals; Brain; Dopamine; gamma-Aminobutyric Acid; Humans; Norepinephrine; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Serotonin; Synaptic Transmission

1984
Effect of the new gamma-aminobutyric acid agonist SL 76 002 on striatal acetylcholine: relation to neuroleptic-induced extrapyramidal alterations.
    Advances in biochemical psychopharmacology, 1980, Volume: 24

    Topics: Acetylcholine; Animals; Antipsychotic Agents; Corpus Striatum; Dopamine; Extrapyramidal Tracts; gamma-Aminobutyric Acid; Haloperidol; Humans; Neurons; Parasympathetic Nervous System

1980
gamma-Aminobutyric acid (GABA) receptor stimulation. II. Specificity of progabide (SL 76002) and SL 75102 for the GABA receptor.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 220, Issue:3

    Topics: Animals; Brain; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Muscimol; Neurotransmitter Agents; Rabbits; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1982
Enhancing GABAergic transmission reverses the aversive state in rats induced by electrical stimulation of the periaqueductal grey region.
    Brain research, 1982, Sep-30, Volume: 248, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Disease Models, Animal; Drug Interactions; Electric Stimulation; Escape Reaction; gamma-Aminobutyric Acid; Humans; Male; Periaqueductal Gray; Rats; Synaptic Transmission

1982
Differential effects of the benzodiazepine antagonist Ro 15-1788 on two types of myoclonus in baboon Papio papio.
    Neuroscience letters, 1983, Jul-15, Volume: 38, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Flumazenil; gamma-Aminobutyric Acid; Light; Lorazepam; Myoclonus; Papio; Seizures

1983
Successful treatment of hemiballismus with progabide, a new GABA-mimetic agent.
    Journal of neurology, 1983, Volume: 229, Issue:2

    Topics: Aged; Brain; Female; gamma-Aminobutyric Acid; Humans; Movement Disorders; Thalamic Nuclei; Tomography, X-Ray Computed

1983
GABAB receptor-mediated inhibition of serotonin release in the rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 326, Issue:2

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Brain Chemistry; Cerebral Cortex; Diazepam; Electric Stimulation; gamma-Aminobutyric Acid; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Nipecotic Acids; Phentolamine; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin

1984
Parkinson's disease and benign essential tremor: somatostatin-like immunoreactivity in the cerebrospinal fluid.
    Advances in neurology, 1984, Volume: 40

    Topics: Adult; Aged; Alzheimer Disease; Atrophy; Brain Diseases; Female; gamma-Aminobutyric Acid; Humans; Huntington Disease; Male; Middle Aged; Multiple Sclerosis; Parkinson Disease; Peptides; Tremor

1984
Reversal of the antiaversive and anticonvulsant actions of diazepam, but not of progabide, by a selective antagonist of benzodiazepine receptors.
    European journal of pharmacology, 1981, Oct-15, Volume: 75, Issue:1

    Topics: Animals; Anxiety; Benzodiazepinones; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures

1981
gamma-Aminobutyric acid (GABA) receptor stimulation. I. Neuropharmacological profiles of progabide (SL 76002) and SL 75102, with emphasis on their anticonvulsant spectra.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 220, Issue:3

    Topics: Animals; Anticonvulsants; Apomorphine; Behavior, Animal; Catalepsy; Drug Interactions; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Mice; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stereotyped Behavior

1982
gamma-Aminobutyric acid (GABA) receptor stimulation. III. Effect of progabide (SL 76002) on norepinephrine, dopamine and 5-hydroxytryptamine turnover in rat brain areas.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 220, Issue:3

    Topics: Animals; Brain; Dopamine; gamma-Aminobutyric Acid; Male; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin; Synaptic Transmission; Tryptamines

1982
gamma-Aminobutyric acid (GABA) receptor stimulation. IV. Effect of progabide (SL 76002) and other GABAergic agents on acetylcholine turnover in rat brain areas.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 220, Issue:3

    Topics: Acetylcholine; Animals; Brain; Corpus Striatum; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission

1982
Actions of GABAergic agents on dopamine metabolism in the nigrostriatal pathway of the rat.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:3

    Topics: 4-Aminobutyrate Transaminase; Aminooxyacetic Acid; Animals; Corpus Striatum; Diazepam; Dopamine; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Neural Pathways; Pyrones; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra

1982
Pharmacological and therapeutic actions of GABA receptor agonists.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Bipolar Disorder; Emotions; gamma-Aminobutyric Acid; Humans; Movement Disorders; Norepinephrine; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Serotonin

1983
Reversal of the muscle relaxant effect of diazepam but not of progabide by a specific benzodiazepine antagonist: Ro 15-1788.
    European journal of pharmacology, 1983, May-20, Volume: 90, Issue:1

    Topics: Animals; Benzodiazepinones; Diazepam; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscle Contraction; Muscle Relaxants, Central; Rats; Rats, Inbred Strains; Time Factors

1983
Indications for the use of gamma-aminobutyric acid (GABA)-agonists in convulsant disorders.
    Progress in clinical and biological research, 1983, Volume: 124

    Topics: Animals; Anticonvulsants; Disease Models, Animal; Epilepsies, Partial; Epilepsy; gamma-Aminobutyric Acid; Humans; Nervous System; Papio; Seizures; Synapses

1983
The comparative effects of benzodiazepines, progabide and PK 9084 on acquisition of passive avoidance in mice.
    Psychopharmacology, 1984, Volume: 83, Issue:1

    Topics: Animals; Avoidance Learning; Benzodiazepines; gamma-Aminobutyric Acid; Male; Mice; Motor Activity; Quinolines

1984
Disposition of progabide and valproic acid following intraperitoneal administration in rhesus monkey.
    Epilepsia, 1984, Volume: 25, Issue:5

    Topics: Absorption; Administration, Oral; Animals; Biological Availability; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Injections, Intravenous; Kinetics; Macaca mulatta; Male; Peritoneum; Valproic Acid

1984
Chlordiazepoxide-induced hyperphagia in rats: lack of effect of GABA agonists and antagonists.
    Psychopharmacology, 1984, Volume: 84, Issue:3

    Topics: Animals; Chlordiazepoxide; Eating; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains

1984
Effects in man of progabide on prolactin release induced by haloperidol or domperidone.
    Psychoneuroendocrinology, 1984, Volume: 9, Issue:2

    Topics: Adult; Domperidone; gamma-Aminobutyric Acid; Haloperidol; Humans; Male; Premedication; Prolactin

1984
Penicillin spikes in rats. Limitations of a simple model for the study of anticonvulsants.
    Neuropharmacology, 1984, Volume: 23, Issue:9

    Topics: Action Potentials; Animals; Anticonvulsants; Dimethyl Sulfoxide; Disease Models, Animal; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Isoxazoles; Male; Penicillins; Phenytoin; Rats; Rats, Inbred Strains; Seizures; Taurine; Time Factors

1984
SL76002 - effect on gamma-aminobutyric acid and dopamine in animals treated chronically with haloperidol.
    Neuropsychobiology, 1983, Volume: 9, Issue:4

    Topics: Animals; Brain Chemistry; Corpus Striatum; Dopamine; Dyskinesia, Drug-Induced; Frontal Lobe; gamma-Aminobutyric Acid; Haloperidol; Male; Mesencephalon; Rats; Rats, Inbred Strains

1983
Measurement of progabide and its deaminated metabolite in plasma by high-performance liquid chromatography and electrochemical detection.
    Journal of chromatography, 1983, Aug-12, Volume: 276, Issue:1

    Topics: Chromatography, High Pressure Liquid; Electrochemistry; gamma-Aminobutyric Acid; Half-Life; Humans; Kinetics; Spectrophotometry, Ultraviolet

1983
An analysis of the actions of progabide, a specific GABA receptor agonist, on kindling and kindled seizures.
    Experimental neurology, 1984, Volume: 83, Issue:1

    Topics: Amygdala; Animals; Anticonvulsants; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains; Seizures

1984
Determination of progabide and its main acid metabolite in biological fluids using high-performance liquid chromatography and electrochemical detection. Application to the measurement of blood/plasma partition ratio.
    Journal of chromatography, 1984, Jun-08, Volume: 308

    Topics: Anticonvulsants; Chromatography, Gas; Chromatography, High Pressure Liquid; Drug Stability; Electrochemistry; gamma-Aminobutyric Acid; Humans; Hydrogen-Ion Concentration; Kinetics; Oxidation-Reduction; Solubility; Temperature

1984
Increase in striatal acetylcholine levels by GABAergic agents: dependence on corticostriatal neurons.
    Brain research, 1980, Oct-27, Volume: 200, Issue:1

    Topics: Acetylcholine; Animals; Cerebral Cortex; Corpus Striatum; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Muscimol; Neurons; Rats; Valproic Acid

1980
Prolonged treatment with gamma-aminobutyric acid (GABA)-mimetic substances in prepubertal male rats.
    Archives of andrology, 1983, Volume: 10, Issue:3

    Topics: 4-Butyrolactone; Alkynes; Aminocaproates; Animals; Body Weight; gamma-Aminobutyric Acid; Male; Organ Size; Prolactin; Rats; Rats, Inbred Strains; Seminal Vesicles; Sexual Maturation; Testis; Time Factors

1983
Pharmacokinetic profile of progabide, a new gamma-aminobutyric acid-mimetic drug, in rhesus monkey.
    Journal of pharmaceutical sciences, 1982, Volume: 71, Issue:6

    Topics: Administration, Oral; Animals; Anticonvulsants; gamma-Aminobutyric Acid; Injections, Intravenous; Kinetics; Macaca mulatta; Male; Protein Binding; Time Factors

1982
Gas chromatographic method for the determination of progabide (SL 76.002) in biological fluids.
    Journal of chromatography, 1982, Jun-11, Volume: 230, Issue:1

    Topics: Animals; Chromatography, Gas; Dogs; gamma-Aminobutyric Acid; Humans; Rats; Reference Values; Time Factors

1982
Effects of GABA analogues and their interactions with morphine on locomotor activity in two inbred strains of mice.
    Pharmacological research communications, 1982, Volume: 14, Issue:5

    Topics: Animals; Drug Interactions; gamma-Aminobutyric Acid; Isoxazoles; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Morphine; Motor Activity; Muscimol; Piracetam

1982
Action of progabide in the photosensitive baboon, Papio papio.
    Epilepsia, 1982, Volume: 23, Issue:5

    Topics: Allylglycine; Animals; Anticonvulsants; Blood-Brain Barrier; Brain; Dose-Response Relationship, Drug; Drug Synergism; Electroencephalography; Epilepsy; gamma-Aminobutyric Acid; Papio; Photosensitivity Disorders; Sleep Stages

1982
Further evidence for the interactions between angiotensin II and GABAergic transmission in pentylenetetrazol kindling seizures in mice.
    Neuropeptides, 1995, Volume: 28, Issue:1

    Topics: Angiotensin II; Animals; Baclofen; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Mice; Nipecotic Acids; Pentylenetetrazole; Phenylurea Compounds; Receptors, GABA; Seizures

1995
Possible involvement of a gamma-hydroxybutyric acid receptor in startle disease.
    Acta paediatrica (Oslo, Norway : 1992), 1994, Volume: 83, Issue:6

    Topics: Anesthetics; Anticonvulsants; GABA Agonists; gamma-Aminobutyric Acid; Humans; Infant, Newborn; Male; Neuromuscular Diseases; Receptors, Cell Surface; Reflex, Abnormal; Reflex, Startle; Sodium Oxybate

1994
In vivo and in vitro correlation of microsomal epoxide hydrolase inhibition by progabide.
    Clinical pharmacology and therapeutics, 1993, Volume: 54, Issue:5

    Topics: Adult; Anticonvulsants; Carbamazepine; Drug Interactions; Epoxide Hydrolases; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Least-Squares Analysis; Male; Microsomes, Liver; Reference Values

1993
Suppression of cortical epileptic afterdischarges in developing rats by anticonvulsants increasing GABAergic inhibition.
    Epilepsy research, 1996, Volume: 25, Issue:3

    Topics: Animals; Anticonvulsants; Cerebral Cortex; Depression, Chemical; Drug Evaluation, Preclinical; Electric Stimulation; Electroencephalography; Enzyme Inhibitors; Epilepsy; GABA Agents; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Neural Inhibition; Phenobarbital; Rats; Valproic Acid

1996
The inhibitory effects on sexual behavior and ambulatory activity of the mixed GABAA/GABAB agonist progabide are differentially blocked by GABA receptor antagonists.
    Psychopharmacology, 1997, Volume: 129, Issue:1

    Topics: Animals; Bicuculline; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Motor Activity; Organophosphorus Compounds; Psychomotor Performance; Rats; Rats, Wistar; Sexual Behavior, Animal

1997
Grouped random effects models for Bayesian meta-analysis.
    Statistics in medicine, 1997, Aug-30, Volume: 16, Issue:16

    Topics: Algorithms; Anticonvulsants; Bayes Theorem; gamma-Aminobutyric Acid; Humans; Markov Chains; Meta-Analysis as Topic; Models, Statistical; Monte Carlo Method; Research Design

1997
Mechanisms of the inhibition of human erythrocyte pyridoxal kinase by drugs.
    Biochemical pharmacology, 1997, Oct-15, Volume: 54, Issue:8

    Topics: Drug Interactions; Enzyme Inhibitors; Erythrocytes; gamma-Aminobutyric Acid; Humans; Kinetics; Muzolimine; Pyridoxal; Pyridoxal Kinase; Spectrophotometry, Ultraviolet; Thiamphenicol

1997
Analysis of overdispersed count data by mixtures of Poisson variables and Poisson processes.
    Biometrics, 1997, Volume: 53, Issue:4

    Topics: Anticonvulsants; Biometry; Epilepsy; gamma-Aminobutyric Acid; Humans; Likelihood Functions; Normal Distribution; Poisson Distribution; Probability; Seizures; Statistical Distributions

1997
Interactions between dopamine and GABA in the control of ambulatory activity and neophobia in the mouse.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 59, Issue:1

    Topics: Amphetamine; Animals; Chi-Square Distribution; Dopamine; Dopamine Agents; Exploratory Behavior; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Phobic Disorders

1998
Severe visual-field constriction and side-effects of GABA-mimetic antiepileptic agents.
    Lancet (London, England), 1998, Aug-15, Volume: 352, Issue:9127

    Topics: Anticonvulsants; Epilepsies, Myoclonic; Epilepsy, Tonic-Clonic; Female; Follow-Up Studies; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Humans; Middle Aged; Phenobarbital; Vision Disorders; Visual Fields

1998
Anticonvulsant effect of progabide in rats during ontogenesis.
    Physiological research, 1997, Volume: 46, Issue:1

    Topics: Aging; Animals; Anticonvulsants; Behavior, Animal; Convulsants; gamma-Aminobutyric Acid; Male; Pentylenetetrazole; Rats; Rats, Wistar; Seizures

1997
[Concentric changes in the visual field associated with GABA-mimetic antiepileptic agents].
    Journal francais d'ophtalmologie, 1999, Volume: 22, Issue:4

    Topics: Adult; Anticonvulsants; Female; GABA Modulators; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Phenobarbital; Vigabatrin; Visual Field Tests; Visual Fields

1999
Unit-treatment interaction and its practical consequences.
    Biometrics, 2000, Volume: 56, Issue:3

    Topics: Analysis of Variance; Anticonvulsants; Clinical Trials as Topic; Epilepsy; gamma-Aminobutyric Acid; Humans; Likelihood Functions; Models, Statistical; Randomized Controlled Trials as Topic; Seizures

2000
Differential role of dopamine D1 and D2 receptors in isoniazid-induced vacuous chewing movements.
    Methods and findings in experimental and clinical pharmacology, 2000, Volume: 22, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anticonvulsants; Antipsychotic Agents; Antitubercular Agents; Behavior, Animal; Diazepam; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Isoniazid; Male; Mastication; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Time Factors

2000
Selection effects in randomized trials with count data.
    Statistics in medicine, 2002, Feb-28, Volume: 21, Issue:4

    Topics: Anticonvulsants; Computer Simulation; Electrocardiography, Ambulatory; Epilepsy; gamma-Aminobutyric Acid; Humans; Models, Biological; Myocardial Ischemia; Randomized Controlled Trials as Topic; Seizures; Selection Bias

2002
Hypothesis testing in semiparametric additive mixed models.
    Biostatistics (Oxford, England), 2003, Volume: 4, Issue:1

    Topics: Anticonvulsants; Child; Computer Simulation; Data Interpretation, Statistical; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Indonesia; Likelihood Functions; Longitudinal Studies; Male; Models, Statistical; Placebos; Randomized Controlled Trials as Topic; Respiratory Tract Infections; Statistics, Nonparametric; Xerophthalmia

2003
[Endoscopic mucosal resection in the upper and lower GI tract].
    Deutsche medizinische Wochenschrift (1946), 2004, Sep-03, Volume: 129 Suppl 2

    Topics: Carcinoma in Situ; Contraindications; Endoscopy, Gastrointestinal; gamma-Aminobutyric Acid; Gastric Mucosa; Gastrointestinal Neoplasms; Intestinal Mucosa; Lymphatic Metastasis; Neoplasm Staging; Precancerous Conditions; Surgical Instruments

2004
Combined discriminative stimulus effects of midazolam with other positive GABAA modulators and GABAA receptor agonists in rhesus monkeys.
    Psychopharmacology, 2005, Volume: 178, Issue:4

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Ethanol; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Injections, Subcutaneous; Isoxazoles; Macaca mulatta; Male; Midazolam; Pentobarbital; Pregnanolone; Receptors, GABA-A; Time Factors; Triazolam; Women

2005
How to appraise the effectiveness of treatment.
    World journal of surgery, 2005, Volume: 29, Issue:5

    Topics: Evaluation Studies as Topic; Evidence-Based Medicine; gamma-Aminobutyric Acid; Guidelines as Topic; Humans; Outcome Assessment, Health Care; Randomized Controlled Trials as Topic; Research Design

2005
Robust estimating functions and bias correction for longitudinal data analysis.
    Biometrics, 2005, Volume: 61, Issue:3

    Topics: Age Factors; Anticonvulsants; Bias; Data Interpretation, Statistical; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Randomized Controlled Trials as Topic; Seizures

2005
Quadratic inference functions in marginal models for longitudinal data.
    Statistics in medicine, 2009, Dec-20, Volume: 28, Issue:29

    Topics: Anticonvulsants; Computer Simulation; Data Interpretation, Statistical; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Models, Statistical; Seizures; Software

2009
Inference on the rate ratio of recurrent events for the matched pairs design.
    Statistics in medicine, 2010, Dec-30, Volume: 29, Issue:30

    Topics: Anticonvulsants; Data Interpretation, Statistical; Epilepsy; gamma-Aminobutyric Acid; Humans; Incidence; Product Surveillance, Postmarketing; Randomized Controlled Trials as Topic; Recurrence; Sample Size; Seizures

2010
Prognostic prediction in patients with hip fracture: risk factors predicting difficulties with discharge to own home.
    Journal of orthopaedics and traumatology : official journal of the Italian Society of Orthopaedics and Traumatology, 2011, Volume: 12, Issue:2

    Topics: Age Distribution; Aged; Aged, 80 and over; Comorbidity; Dementia; Disability Evaluation; Female; Femoral Neck Fractures; gamma-Aminobutyric Acid; Hospital Mortality; Humans; Male; Middle Aged; Multivariate Analysis; Patient Discharge; Predictive Value of Tests; Risk Factors; Walking

2011
Working covariance model selection for generalized estimating equations.
    Statistics in medicine, 2011, Nov-20, Volume: 30, Issue:26

    Topics: Anticonvulsants; Computer Simulation; Data Interpretation, Statistical; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Models, Statistical; Normal Distribution; Randomized Controlled Trials as Topic; Software

2011
A bias correction for covariance estimators to improve inference with generalized estimating equations that use an unstructured correlation matrix.
    Statistics in medicine, 2013, Jul-20, Volume: 32, Issue:16

    Topics: Anticonvulsants; Bias; Computer Simulation; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Models, Statistical; Seizures

2013
Objective Bayesian meta-analysis for sparse discrete data.
    Statistics in medicine, 2014, Sep-20, Volume: 33, Issue:21

    Topics: Bayes Theorem; Cardiovascular Diseases; Diabetes Mellitus, Type 2; Diabetes, Gestational; Epilepsy; Female; gamma-Aminobutyric Acid; Hormone Replacement Therapy; Humans; Meta-Analysis as Topic; Models, Statistical; Multicenter Studies as Topic; Pregnancy; Rosiglitazone; Thiazolidinediones; Treatment Outcome

2014
Acoustic radiation force impulse elastography for non-invasive assessment of disease stage in patients with primary biliary cirrhosis: A preliminary study.
    Clinical radiology, 2014, Volume: 69, Issue:8

    Topics: Biopsy; Elasticity Imaging Techniques; Female; gamma-Aminobutyric Acid; Humans; Liver; Liver Cirrhosis, Biliary; Male; Middle Aged; Reproducibility of Results; ROC Curve; Sensitivity and Specificity

2014
Association of left atrial reservoir function with left atrial structural remodeling related to left ventricular dysfunction in asymptomatic patients with hypertension: evaluation by two-dimensional speckle-tracking echocardiography.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2015, Volume: 37, Issue:2

    Topics: Atrial Function, Left; Echocardiography; Female; Follow-Up Studies; gamma-Aminobutyric Acid; Heart Atria; Heart Ventricles; Humans; Hypertension; Male; Middle Aged; Retrospective Studies; Ventricular Dysfunction, Left; Ventricular Function, Left; Ventricular Remodeling

2015
Covariance estimators for generalized estimating equations (GEE) in longitudinal analysis with small samples.
    Statistics in medicine, 2016, May-10, Volume: 35, Issue:10

    Topics: Adolescent; Anticonvulsants; Bias; Child; Computer Simulation; Epilepsy; Female; gamma-Aminobutyric Acid; Head; Humans; Longitudinal Studies; Male; Models, Statistical; Randomized Controlled Trials as Topic; Sample Size; Software

2016
Discovery of a Novel Microsomal Epoxide Hydrolase-Catalyzed Hydration of a Spiro Oxetane.
    Drug metabolism and disposition: the biological fate of chemicals, 2016, Volume: 44, Issue:8

    Topics: Azetidines; Biotransformation; Catalysis; Enzyme Inhibitors; Epoxide Hydrolases; gamma-Aminobutyric Acid; Humans; Kinetics; Microsomes, Liver; Molecular Structure; Oxadiazoles; Substrate Specificity

2016