progabide has been researched along with gamma-aminobutyric acid in 159 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 117 (73.58) | 18.7374 |
1990's | 21 (13.21) | 18.2507 |
2000's | 10 (6.29) | 29.6817 |
2010's | 11 (6.92) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bartholini, G; Desarmenien, M; Feltz, P; Headley, PM; Kaplan, JP; Lloyd, KG; Raizon, BM; Worms, P | 1 |
Bartholini, G | 4 |
Bachus, SE; Dale, J; Goodman, L; Kaneda, H; Shirakawa, O; Tamminga, CA | 1 |
Gautam, SK; Kulkarni, SK | 1 |
Greenshaw, AJ; McManus, DJ | 1 |
Morimoto, K; Nakamura, Y; Okamoto, M; Otsuki, S; Sato, K; Sato, M | 1 |
Mehta, AK; Ticku, MK | 1 |
Moran, M; Tamminga, CA; Thaker, GK | 1 |
Decourt, JP; Mura, P; Papet, Y; Piriou, A; Reiss, D | 1 |
Bartholini, G; Oblin, A; Zivkovic, B | 2 |
Besson, MJ; Caboche, J; Le Saux, F; Maurin, Y; Mitrovic, N; Sauter, A | 1 |
Morimoto, K | 1 |
Benoit, JP; Couvreur, P; Deverre, JR; Gayral, P; Letourneux, Y; Loiseau, P | 1 |
Porter, RJ | 1 |
Cudennec, A; Duverger, D; Lloyd, KG; MacKenzie, ET; McCulloch, J; Motohashi, N; Nishikawa, T; Scatton, B | 1 |
Blair, AJ; Crawford, IL; Feldman, M; Petty, F; Stevens, MH; Taylor, IL; Thirlby, RC; Walsh, JH | 1 |
Gale, RG; Little, HJ; Nutt, DJ; Standing, BL; Taylor, SC | 1 |
Davidoff, RA | 1 |
Bossi, L; Fournier, V; Morselli, PL; Musch, B | 1 |
Lloyd, KG; Perrault, G; Zivkovic, B | 1 |
Bathien, N; Rondot, P | 1 |
Atmadja, S; Baimbridge, KG; Fibiger, HC; Mithani, S | 1 |
Koe, BK; Kondratas, E; Russo, LL | 1 |
Bathien, N; Fournier, V; Morselli, PL; Rondot, P; Ziegler, M | 1 |
Rondot, P | 1 |
Lima, L; Sourkes, TL | 1 |
Bossi, L; Girard, M; Poulain, D | 1 |
Hilakivi, I; Hilakivi, LA; Loikas, P; Taira, T | 1 |
Chweh, AY; Kupferberg, HJ; Swinyard, EA; Wolf, HH | 1 |
Rastogi, SK; Ticku, MK | 2 |
Green, AR; Johnson, P; Mountford, JA; Nimgaonkar, VL | 1 |
Bergmann, KJ | 1 |
Di Scala, G; Fibiger, HC; Martin-Iverson, MT; Phillips, AG | 1 |
Nishikawa, T; Scatton, B | 1 |
Fadda, F; Gessa, GL; Meloni, R; Mosca, E | 1 |
Goldstein, M; Lloyd, KG; Willigens, MT | 1 |
Arbilla, S; Bartholini, G; Fage, D; Langer, SZ; Oblin, A; Scatton, B; Zivkovic, B | 1 |
Moura, D; Soares-da-Silva, P | 1 |
Löscher, W; Schwark, WS | 1 |
Lloyd, KG; Pilc, A; Thuret, F | 1 |
Bovier, P; Hilleret, H; Tissot, R | 1 |
Curet, O; Dennis, T; Nishikawa, T; Scatton, B | 1 |
Lloyd, KG | 1 |
Chweh, AY; Swinyard, EA; Ulloque, RA | 1 |
Chweh, AY; Lin-Michell, E; Swinyard, EA | 1 |
Green, AR | 1 |
Little, HJ; Nutt, DJ; Taylor, SC | 1 |
Goodwin, GM; Gray, JA; Green, AR; Metz, A | 1 |
Apud, JA; Masotto, C; Racagni, G | 1 |
Bartholini, G; Lloyd, KG; Scatton, B; Zivkovic, B | 1 |
Bartholini, G; Depoortere, H; Lloyd, KG; Sanger, D; Zivkovic, B | 1 |
Lindgren, S | 1 |
Benassi, E; Besio, G; Bo, GP; Cocito, L; Loeb, C; Maffini, M; Mainardi, P; Morselli, PL | 1 |
Graves, NM; Holmes, GB; Leppik, IE | 1 |
Chadwick, D; Crawford, P | 1 |
Comi, G; Ferini-Strambi, L; Filippi, M; Giusti, MC; Medaglini, S; Poggi, A; Smirne, S | 1 |
de Feo, MR; Mecarelli, O; Ricci, GF; Rina, MF | 1 |
Davis, SS; Farraj, NF; Parr, GD; Stevens, HN | 2 |
Benassi, E; Besio, G; Bianchetti, G; Loeb, C; Morselli, PL | 1 |
Bowman, T; Cloyd, J; Crosby, C; Dreifuss, FE; Graves, N; Jacobs, M; Leppik, IE; Porter, R; Santilli, N; Stackman, J | 1 |
Fariello, R; Maddrey, WC; Munoz, SJ | 1 |
Brundage, RC; Cloyd, JC; Graves, NM; Leppik, IE; Welty, TE | 1 |
Manev, H; Pericić, D | 1 |
Schmidt, D; Utech, K | 1 |
Barre, J; Brandebourger, M; Hamberger, C; Taiclet, A; Thenot, JP; Tillement, JP; Urien, S | 1 |
Barre, J; Essassi, D; Grimaldi, B; Hamberger, C; Taiclet, A; Thenot, JP; Tillement, JP; Urien, S | 1 |
Gupta, S; Koller, WC; Rubino, F | 1 |
Breton, D; Krall, RL; Rudick, RA | 1 |
Lheroux, A; Luquin, MR; Martinez Lage, JM; Obeso, JA; Scatton, B | 1 |
Chweh, AY; Swinyard, EA; Wolf, HH | 1 |
Ascalone, V; Dal Bo', L | 1 |
Bennett, JP; Cruz, CJ; Ferrari, MB | 1 |
Beaussart, M; Benoit, C; Broglin, D; Cambier, J; Cenraud, M; Chatel, M; Deville, MC; Fournier, V; Loiseau, P; Musch, B | 1 |
Braendgaard, H; Dupont, E; Mondrup, K | 1 |
Burke, JT; Thénot, JP | 1 |
Johns, KL; Wood, JD | 1 |
Löscher, W | 1 |
Ascalone, V; Catalani, P; Dal Bò, L | 1 |
Bartholini, G; Scatton, B; Zivkovic, B | 1 |
Arbilla, S; Bartholini, G; Beaumont, K; Briley, M; De Montis, G; Langer, SZ; Lloyd, KG; Scatton, B | 1 |
Bovier, P; Broekkamp, CL; Lloyd, KG | 1 |
Bryere, P; Kaijima, M; Naquet, R; Valin, A | 1 |
Bergmann, KJ; Limongi, JC; Lowe, YH; Mendoza, MR; Yahr, MD | 1 |
Charlier, M; Delwaide, PJ; Gonce, M; Schoenen, J | 1 |
Classen, K; Göthert, M; Schlicker, E | 1 |
Christensen, SE; Dupont, E; Mondrup, K; Olivarius, BF; Orskov, H | 1 |
Bovier, P; Broekkamp, CL; Lloyd, KG; Worms, P | 1 |
Bartholini, G; Depoortere, H; Durand, A; Lloyd, KG; Morselli, PL; Worms, P | 1 |
Bartholini, G; Constantinidis, J; Dedek, J; Lloyd, KG; Scatton, B; Tissot, R; Zivkovic, B | 1 |
Bartholini, G; Scatton, B | 2 |
Wood, PL | 1 |
Bartholini, G; Lloyd, KG; Scatton, B; Worms, P; Zivkovic, B | 1 |
Bartholini, G; Broekkamp, C; Depoortere, H; Fournier, V; Lloyd, KG; Morselli, PL; Scatton, B; Worms, P; Zivkovic, B | 1 |
Bossi, L; Guyot, M; Loiseau, P; Morselli, PL; Orofiamma, B | 1 |
Dupont, E; Mondrup, K; Pedersen, E | 1 |
Mondrup, K; Pedersen, E | 2 |
Schmidt, D | 1 |
Bossi, L; Martínez Vila, E; Martínez-Lage, JM; Morales, G; Orofiamma, B; Viteri, C | 1 |
Angelo, HR; Christensen, JM; Dam, M; Gram, L; Hansen, BS; Lyon, BB; Philbert, A | 1 |
Schwarz, M; Sontag, KH; Turski, L | 1 |
Bossi, L; Lloyd, KG; Morselli, PL; Munari, C; Worms, P | 1 |
Broekkamp, CL; Le Pichon, M; Lloyd, KG | 1 |
Bialer, M; Johno, I; Levy, RH; Nickelson, SA | 1 |
Sanger, DJ | 1 |
Marsden, CD; Sheehy, MP | 1 |
Butt, WR; Gomeni, R; London, DR; Menon, VJ; Morselli, PL; Thiercelin, JF | 1 |
Fariello, RG; Golden, GT | 1 |
Lapierre, YD; Rastogi, RB; Rastogi, SK; Singhal, RL | 1 |
Kupferberg, HJ; Lambert, T; Yonekawa, W | 1 |
Albertson, TE; Joy, RM; Stark, LG | 1 |
Bianchetti, G; Deves, C; Morselli, PL; Padovani, P; Thenot, JP | 1 |
Debeljuk, L; Díaz, MD; Maines, VM; Seilicovich, A | 1 |
Johno, I; Levy, RH; Ludwick, BT | 1 |
Dring, LG; Fraisse-André, J; Gillet, G; Lee, CR; Morselli, PL | 1 |
Cagiano, R; Cuomo, V; Mocchetti, I; Racagni, G | 1 |
Cepeda, C; Lloyd, KG; Naquet, R; Worms, P | 1 |
Georgiev, VP; Kambourova, TS; Lazarova, MB | 1 |
Berthier, M; Bonneau, D; Chevrel, J; Desbordes, JM; Jaeken, J; Laborit, H; Oriot, D | 1 |
Guyot, M; Kroetz, DL; Levy, RH; Loiseau, P | 1 |
Pierce, MW; Shu, VS | 1 |
Kubová, H; Mares, P; Polásek, R; Slamberová, R; Vorlícek, J | 1 |
Agmo, A; Garcés, I; Paredes, RG; Sierra, L | 1 |
Dey, DK; Larose, DT | 1 |
Allain, P; Cailleux, A; Lainé-Cessac, P | 1 |
Hougaard, P; Lee, ML; Whitmore, GA | 1 |
Agmo, A; Belzung, C | 1 |
Baulac, M; Lanoé, Y; Nordmann, JP | 1 |
Kozuchová, A; Mares, P; Stanková, L | 1 |
Baulac, M; Nordmann, JP; Van Egroo, C | 1 |
Louis, ED | 1 |
Gadbury, GL; Iyer, HK | 1 |
Kulkarni, SK; Naidu, PS | 1 |
Mizusawa, H | 1 |
Cook, RJ; Wei, W | 1 |
Lin, X; Zhang, D | 1 |
Rösch, T | 1 |
France, CP; McMahon, LR | 1 |
Bhandari, M; Haynes, RB | 1 |
Lin, X; Wang, YG; Zhu, M | 1 |
Jiang, Z; Park, E; Qu, A; Song, PX | 1 |
Sumi, M; Tango, T | 1 |
Hagino, T; Haro, H; Ochiai, S; Sato, E; Senga, S; Watanabe, Y | 1 |
Carey, VJ; Wang, YG | 1 |
Westgate, PM | 1 |
Moreno, E; Negrín, MA; Vázquez-Polo, FJ | 1 |
Chen, M; Li, M; Liu, LP; Liu, Y; Wang, RF; Zhang, DK | 1 |
Ara, N; Iuchi, A; Miyoshi, H; Mizuguchi, Y; Nagase, N; Oishi, Y; Oki, T | 1 |
Gargiulo, R; Lerma, EV; Suhail, F | 1 |
Kong, L; Li, Z; Wang, M; Zhang, L | 1 |
Berggren, K; Castagnoli, N; Grönberg, G; Hayes, MA; Li, XQ; Weidolf, L | 1 |
Alabed, S; Bergman, H; Latifeh, Y; Mohammad, HA | 1 |
13 review(s) available for progabide and gamma-aminobutyric acid
Article | Year |
---|---|
Antispasticity drugs: mechanisms of action.
Topics: Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Baclofen; Benzodiazepines; Central Nervous System; Dantrolene; gamma-Aminobutyric Acid; Glycine; Humans; Muscle Relaxants, Central; Muscle Spasticity; Neurotransmitter Agents; Phenothiazines; Rats; Receptors, Neurotransmitter; Spinal Cord | 1985 |
[Implications of GABAergic synapses in neuropsychiatry].
Topics: 4-Aminobutyrate Transaminase; Animals; Anti-Anxiety Agents; Anticonvulsants; Antidepressive Agents; Anxiety; Brain; Cats; Cerebral Cortex; Depressive Disorder; Disease Models, Animal; Dyskinesia, Drug-Induced; Epilepsy; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haplorhini; Humans; Mental Disorders; Muscimol; Receptors, GABA-A; Seizures; Synapses; Synaptic Transmission | 1985 |
Progabide: a new GABA-mimetic agent in clinical use.
Topics: Anticonvulsants; Brain Chemistry; Chemical Phenomena; Chemistry; Epilepsy; gamma-Aminobutyric Acid; Humans; Movement Disorders; Muscle Spasticity; Receptors, GABA-A | 1985 |
[Drug activation of GABAergic transmission in the central nervous system: benzodiazepines and GABAergic agonists].
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chemical Phenomena; Chemistry; Cyclic GMP; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Receptors, GABA-A; Synaptic Transmission; Valproic Acid | 1985 |
[GABAergic theory of epilepsy].
Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Dogs; Epilepsy; gamma-Aminobutyric Acid; Humans; Mice; Nerve Endings; Pentylenetetrazole; Phenobarbital; Phenytoin; Rats; Receptors, GABA-A; Synapses; Valproic Acid | 1986 |
Changes in gamma-aminobutyric acid biochemistry and seizure threshold.
Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Bicuculline; Brain; Cerebral Cortex; Clonidine; Corpus Striatum; Electroconvulsive Therapy; gamma-Aminobutyric Acid; Hippocampus; Hypothalamus; Male; Mice; Mice, Inbred Strains; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin | 1986 |
Determination of antiepileptic drugs.
Topics: Anticonvulsants; Barbiturates; Carbamazepine; Chromatography, Gas; Chromatography, Liquid; Clonazepam; gamma-Aminobutyric Acid; Gas Chromatography-Mass Spectrometry; Humans; Mephenytoin; Monitoring, Physiologic; Phenytoin; Primidone; Succinimides; Valproic Acid | 1985 |
GABA system, GABA receptor agonists and dyskinesia.
Topics: Basal Ganglia; Cholinergic Fibers; Dopamine; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Humans; Huntington Disease; Levodopa; Movement Disorders; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Handling seizure data: special problems.
Topics: Anticonvulsants; Clinical Trials as Topic; Data Interpretation, Statistical; Drug Therapy, Combination; Electroencephalography; Epilepsy; Epilepsy, Complex Partial; Epilepsy, Tonic-Clonic; gamma-Aminobutyric Acid; Humans; Nipecotic Acids; Tiagabine; Valproic Acid | 1993 |
A new twist for stopping the shakes? Revisiting GABAergic therapy for essential tremor.
Topics: Acetates; Adult; Amines; Cyclohexanecarboxylic Acids; GABA Agonists; Gabapentin; gamma-Aminobutyric Acid; Humans; Primidone; Propranolol; Tremor | 1999 |
[Autosomal dominant hereditary distal myopathy linked to chromosome 14].
Topics: Chromosomes, Human, Pair 14; Diagnosis, Differential; gamma-Aminobutyric Acid; Genes, Dominant; Genetic Linkage; Humans; Muscle, Skeletal; Muscular Dystrophies | 2001 |
Cardiovascular disease and chronic kidney disease.
Topics: Cardiovascular Diseases; Coronary Artery Disease; gamma-Aminobutyric Acid; Heart Diseases; Humans; Peripheral Vascular Diseases; Renal Insufficiency, Chronic | 2015 |
Gamma-aminobutyric acid agonists for antipsychotic-induced tardive dyskinesia.
Topics: Antipsychotic Agents; Baclofen; Dyskinesia, Drug-Induced; GABA Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Placebos; Randomized Controlled Trials as Topic; Valproic Acid | 2018 |
22 trial(s) available for progabide and gamma-aminobutyric acid
Article | Year |
---|---|
GABAmimetics: a new class of antidepressant agents?
Topics: Antidepressive Agents; Depressive Disorder; Female; gamma-Aminobutyric Acid; Humans; Middle Aged | 1990 |
Clinical activity of GABA agonists in neuroleptic- and L-dopa-induced dyskinesia.
Topics: Antipsychotic Agents; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Dyskinesia, Drug-Induced; Electromyography; gamma-Aminobutyric Acid; Humans; Levodopa | 1985 |
Movement disorders in patients with coexistent neuroleptic-induced tremor and tardive dyskinesia: EMG and pharmacological study.
Topics: Antipsychotic Agents; Clinical Trials as Topic; Corpus Striatum; Double-Blind Method; Dyskinesia, Drug-Induced; Electromyography; gamma-Aminobutyric Acid; Humans; Parkinson Disease, Secondary; Receptors, Dopamine; Receptors, GABA-A; Tremor | 1987 |
Therapeutic response to progabide in neuroleptic- and L-dopa-induced dyskinesias.
Topics: Adult; Aged; Antipsychotic Agents; Clinical Trials as Topic; Double-Blind Method; Dyskinesia, Drug-Induced; Female; gamma-Aminobutyric Acid; Humans; Levodopa; Male; Middle Aged; Parkinson Disease, Secondary; Placebos | 1987 |
Preliminary observations on the activity of progabide, administered as monotherapy in complex partial seizures.
Topics: Adolescent; Adult; Clinical Trials as Topic; Drug Administration Schedule; Epilepsy, Temporal Lobe; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged | 1988 |
Compliant populations: variability in serum concentrations.
Topics: Anticonvulsants; Carbamazepine; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Epilepsy; Felbamate; Female; gamma-Aminobutyric Acid; Humans; Male; Patient Compliance; Phenylcarbamates; Phenytoin; Propylene Glycols; Random Allocation | 1988 |
A comparative study of progabide, valproate, and placebo as add-on therapy in patients with refractory epilepsy.
Topics: Adolescent; Adult; Anticonvulsants; Chemical and Drug Induced Liver Injury; Drug Interactions; Drug Therapy, Combination; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Patient Compliance; Phenytoin; Valproic Acid | 1986 |
A controlled study of progabide in partial seizures: methodology and results.
Topics: Adolescent; Adult; Carbamazepine; Clinical Trials as Topic; Female; gamma-Aminobutyric Acid; Humans; Male; Phenytoin; Seizures | 1987 |
Effect of progabide on serum phenytoin and carbamazepine concentrations.
Topics: Adult; Carbamazepine; Convulsants; Double-Blind Method; Drug Evaluation; Female; gamma-Aminobutyric Acid; Humans; Male; Phenytoin; Random Allocation; Seizures | 1987 |
Progabide for refractory partial epilepsy: a controlled add-on trial.
Topics: Adolescent; Adult; Aged; Anticonvulsants; Carbamazepine; Clinical Trials as Topic; Double-Blind Method; Drug Interactions; Drug Therapy, Combination; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Phenobarbital; Phenytoin; Random Allocation | 1986 |
Pharmacologic probe with progabide of GABA mechanisms in essential tremor.
Topics: Brain; Double-Blind Method; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Random Allocation; Tremor | 1987 |
The GABA-agonist progabide for spasticity in multiple sclerosis.
Topics: Adult; Anticonvulsants; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Multiple Sclerosis; Muscle Spasticity | 1987 |
Potentiation of the "dopa" effect in parkinsonism by a direct GABA receptor agonist.
Topics: Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Drug Synergism; gamma-Aminobutyric Acid; Humans; Levodopa; Parkinson Disease; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
The potential use of GABA agonists in psychiatric disorders: evidence from studies with progabide in animal models and clinical trials.
Topics: Adjustment Disorders; Animals; Anticonvulsants; Biogenic Amines; Brain; Clinical Trials as Topic; Corpus Striatum; Depressive Disorder; Disease Models, Animal; Dopamine; gamma-Aminobutyric Acid; Humans; Imipramine; Limbic System; Neurons; Rats | 1983 |
Double-blind crossover trial of progabide versus placebo in severe epilepsies.
Topics: Adolescent; Adult; Child; Clinical Trials as Topic; Double-Blind Method; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Placebos | 1983 |
The effect of the GABA-agonist, progabide, on benign essential tremor. A controlled clinical trial.
Topics: Adult; Aged; Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Electromyography; Female; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Time Factors; Tremor | 1983 |
The effect of the GABA-agonist, progabide, on stretch and flexor reflexes and on voluntary power in spastic patients.
Topics: Achilles Tendon; Adult; Clinical Trials as Topic; Electromyography; Female; gamma-Aminobutyric Acid; H-Reflex; Hand; Humans; Isometric Contraction; Leg; Male; Middle Aged; Muscle Contraction; Muscle Spasticity; Muscles; Placebos; Reflex, Monosynaptic; Reflex, Stretch; Tibial Nerve | 1984 |
The clinical effect of the GABA-agonist, progabide, on spasticity.
Topics: Adult; Arm; Chemical Phenomena; Chemistry; Clinical Trials as Topic; Female; gamma-Aminobutyric Acid; Humans; Leg; Male; Middle Aged; Muscle Contraction; Muscle Hypertonia; Muscle Spasticity; Muscles; Placebos; Reflex; Reflex, Stretch; Research Design | 1984 |
Progabide as an add-on drug for epilepsy refractory to high dose antiepileptic drug therapy.
Topics: Adult; Aged; Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Epilepsy; Epilepsy, Temporal Lobe; gamma-Aminobutyric Acid; Humans | 1984 |
Progabide treatment in severe epilepsy: a double-blind cross-over trial versus placebo.
Topics: Adolescent; Adult; Clinical Trials as Topic; Double-Blind Method; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Male; Placebos | 1984 |
Progabide: a controlled trial in partial epilepsy.
Topics: Anticonvulsants; Clinical Trials as Topic; Double-Blind Method; Epilepsies, Partial; gamma-Aminobutyric Acid; Humans; Random Allocation | 1983 |
GABA and movement disorders.
Topics: Anticonvulsants; Baclofen; Clinical Trials as Topic; Double-Blind Method; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Humans; Huntington Disease; Isoniazid; Movement Disorders; Muscimol; Parkinson Disease; Valproic Acid | 1981 |
124 other study(ies) available for progabide and gamma-aminobutyric acid
Article | Year |
---|---|
New anticonvulsants: Schiff bases of gamma-aminobutyric acid and gamma-aminobutyramide.
Topics: Animals; Anticonvulsants; Bicuculline; Brain; Cerebellum; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Ganglia, Spinal; Humans; In Vitro Techniques; Lethal Dose 50; Male; Mice; Rats; Schiff Bases | 1980 |
[Potential therapeutic activity of GABA-mimetic drugs in neuropsychiatry].
Topics: 4-Aminobutyrate Transaminase; Basal Ganglia Diseases; Bicuculline; Dopamine; Dyskinesia, Drug-Induced; Epilepsy; Extrapyramidal Tracts; gamma-Aminobutyric Acid; Humans; Huntington Disease; Levodopa; Limbic System; Neural Pathways; Neurons; Neurotransmitter Agents; Parkinson Disease; Psychopharmacology | 1979 |
Co-administration of progabide inhibits haloperidol-induced oral dyskinesias in rats.
Topics: Administration, Oral; Animals; Disease Models, Animal; Drug Interactions; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Haloperidol; Male; Mastication; Rats; Rats, Inbred Strains | 1992 |
GABA/BZ-and NMDA-receptor interaction in digoxin-induced convulsions in rats.
Topics: Animals; Baclofen; Diazepam; Digoxin; Dizocilpine Maleate; Female; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Salts; Seizures | 1991 |
Differential effects of chronic antidepressants in behavioural tests of beta-adrenergic and GABAB receptor function.
Topics: Albuterol; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Baclofen; Behavior, Animal; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Monoamine Oxidase Inhibitors; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, GABA-A | 1991 |
An analysis of anticonvulsant actions of GABA agonists (progabide and baclofen) in the kindling model of epilepsy.
Topics: Animals; Anticonvulsants; Baclofen; Dose-Response Relationship, Drug; Electroencephalography; Epilepsy; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Are GABAB receptors involved in the pharmacological effects of ethanol?
Topics: Animals; Baclofen; Cells, Cultured; Chlorine; Diazepam; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; N-Methylaspartate; Picrotoxin; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Spinal Cord | 1990 |
Simultaneous determination of progabide and its acid metabolite by reversed-phase high-performance liquid chromatography.
Topics: Anticonvulsants; Chromatography, High Pressure Liquid; Epilepsy; gamma-Aminobutyric Acid; Humans | 1990 |
Progabide reverses the nigral substance P reduction induced by chronic impairment of dopaminergic transmission.
Topics: Animals; gamma-Aminobutyric Acid; Haloperidol; Hydroxydopamines; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, GABA-A; Substance P; Substantia Nigra; Synaptic Transmission; Tyrosine 3-Monooxygenase | 1985 |
Selective antagonists of dopamine receptor subtypes differentially affect substance P levels in the striatum and substantia nigra.
Topics: Animals; Benzazepines; Corpus Striatum; Dopamine Antagonists; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Substance P; Substantia Nigra; Sulpiride | 1987 |
Postnatal evolution of the gamma-aminobutyric acid/benzodiazepine receptor complex in a model of inherited epilepsy: the quaking mouse.
Topics: Aging; Animals; Brain; Brain Stem; Cerebellum; Diazepam; Diencephalon; Epilepsy; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Mice, Inbred C57BL; Mice, Quaking; Muscimol; Receptors, GABA-A; Telencephalon | 1989 |
Seizure-triggering mechanisms in the kindling model of epilepsy: collapse of GABA-mediated inhibition and activation of NMDA receptors.
Topics: Amygdala; Animals; Anticonvulsants; Dibenzocycloheptenes; Dizocilpine Maleate; Electroencephalography; Epilepsy; Evoked Potentials; gamma-Aminobutyric Acid; Kindling, Neurologic; Neural Inhibition; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter | 1989 |
In-vitro evaluation of filaricidal activity of GABA and 1,3-dipalmitoyl-2-(4-aminobutyryl)glycerol HCl: a diglyceride prodrug.
Topics: Animals; Anthelmintics; Filaricides; Filarioidea; gamma-Aminobutyric Acid; Microfilariae; Prodrugs; Triglycerides | 1989 |
Mechanisms of action of new antiepileptic drugs.
Topics: Acetamides; Acetates; Amines; Aminocaproates; Aminopyridines; Anti-Anxiety Agents; Anticonvulsants; Aspartic Acid; Benzodiazepines; Benzodiazepinones; Clobazam; Cyclohexanecarboxylic Acids; Dibenzocycloheptenes; Dizocilpine Maleate; Epilepsy; Felbamate; Flumazenil; GABA Antagonists; Gabapentin; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Imidazoles; Lamotrigine; Phenylcarbamates; Propylene Glycols; Receptors, GABA-A; Triazines; Vigabatrin | 1989 |
Effects of the GABA receptor agonist, progabide, upon local cerebral glucose utilization.
Topics: Animals; Autoradiography; Brain; Carbon Radioisotopes; Deoxy Sugars; Deoxyglucose; gamma-Aminobutyric Acid; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Effect of GABA on basal and vagally mediated gastric acid secretion and hormone release in dogs.
Topics: Animals; Baclofen; Blood Glucose; Dogs; gamma-Aminobutyric Acid; Gastric Acid; Gastric Fistula; Gastrins; Gastrointestinal Hormones; Insulin; Male; Receptors, GABA-A; Vagus Nerve | 1988 |
Changes in benzodiazepine/GABA receptor complex function in benzodiazepine-tolerant mice.
Topics: Animals; Anticonvulsants; Bicuculline; Body Temperature; Drug Tolerance; Flurazepam; gamma-Aminobutyric Acid; Infusions, Intravenous; Male; Mice; Motor Activity; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Time Factors | 1988 |
Neuroleptic-induced oral dyskinesias: effects of progabide and lack of correlation with regional changes in glutamic acid decarboxylase and choline acetyltransferase activities.
Topics: Animals; Anticonvulsants; Antipsychotic Agents; Brain; Choline O-Acetyltransferase; Dyskinesia, Drug-Induced; Flupenthixol; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Haloperidol; Male; Mastication; Motor Activity; Parvalbumins; Rats; Rats, Inbred Strains; S100 Calcium Binding Protein G | 1987 |
[3H]Ro 15-1788 binding to benzodiazepine receptors in mouse brain in vivo: marked enhancement by GABA agonists and other CNS drugs.
Topics: Animals; Antipsychotic Agents; Barbiturates; Brain; Buspirone; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Injections, Intravenous; Male; Mice; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Vasodilator Agents | 1987 |
[The electrophysiological approach to tardive dyskinesias].
Topics: Diagnosis, Differential; Dopamine Agents; Dyskinesia, Drug-Induced; Electromyography; gamma-Aminobutyric Acid; Humans; Movement Disorders; Parasympatholytics | 1988 |
Cholinergic and GABAergic regulation of dopamine beta-hydroxylase activity in the adrenal gland of the rat.
Topics: 5,7-Dihydroxytryptamine; Acetylcholine; Adrenal Glands; Aminocaproates; Animals; Baclofen; Bicuculline; Dopamine beta-Hydroxylase; Enzyme Induction; Fenclonine; gamma-Aminobutyric Acid; Hydroxydopamines; Male; Muscimol; Oxotremorine; Propranolol; Rats; Vigabatrin | 1986 |
[Suicide attempted with progabide].
Topics: Adult; Anticonvulsants; Female; gamma-Aminobutyric Acid; Humans; Male; Suicide, Attempted | 1987 |
Neonatal treatment with monoamine uptake inhibitors alters later response in behavioural 'despair' test to beta and GABA-B receptor agonists.
Topics: Albuterol; Animals; Animals, Newborn; Antidepressive Agents; Baclofen; Behavior, Animal; Desipramine; gamma-Aminobutyric Acid; Male; Nomifensine; Rats; Rats, Inbred Strains; Time Factors; Zimeldine | 1988 |
Effect of GABA agonists on the neurotoxicity and anticonvulsant activity of benzodiazepines.
Topics: Animals; Anticonvulsants; Benzodiazepines; Drug Synergism; Electroshock; Flunitrazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Muscimol; Nervous System; Receptors, GABA-A | 1985 |
Involvement of a GABAergic mechanism in the anticonvulsant effect of pentobarbital against maximal electroshock-induced seizures in rats.
Topics: Animals; Anticonvulsants; Benzodiazepinones; Bicuculline; Drug Interactions; Electroshock; Ethanol; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Sleep | 1985 |
Some anticonvulsant drugs alter monoamine-mediated behaviour in mice in ways similar to electroconvulsive shock; implications for antidepressant therapy.
Topics: 5-Hydroxytryptophan; Animals; Anticonvulsants; Antidepressive Agents; Apomorphine; Behavior, Animal; Biogenic Amines; Clonidine; Diazepam; Electroshock; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Motor Activity; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Serotonin; Valproic Acid | 1985 |
The effects of progabide (SL 76002) on locomotor activity and conditioned place preference induced by d-amphetamine.
Topics: Animals; Anticonvulsants; Conditioning, Psychological; Dextroamphetamine; gamma-Aminobutyric Acid; Male; Motor Activity; Rats; Receptors, GABA-A | 1985 |
Inhibitory influence of GABA on central serotonergic transmission. Raphé nuclei as the neuroanatomical site of the GABAergic inhibition of cerebral serotonergic neurons.
Topics: 5-Hydroxytryptophan; Animals; Brain; gamma-Aminobutyric Acid; Male; Neural Inhibition; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission | 1985 |
Suppression by progabide of ethanol withdrawal syndrome in rats.
Topics: Acoustic Stimulation; Animals; Ethanol; gamma-Aminobutyric Acid; Humans; Male; Rats; Rats, Inbred Strains; Seizures; Substance Withdrawal Syndrome; Synaptic Transmission; Tremor | 1985 |
Induction and reversal of dopamine dyskinesia in rat, cat, and monkey.
Topics: Animals; Apomorphine; Brain; Cats; Dextroamphetamine; Dopamine; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Haplorhini; Humans; Levodopa; Motor Activity; Muscimol; Nomifensine; Piribedil; Rats; Receptors, Dopamine; Receptors, GABA-A; Stereotyped Behavior | 1985 |
Influence of GABA mimetics and lithium on biochemical manifestations of striatal dopamine target cell hypersensitivity.
Topics: Animals; Corpus Striatum; gamma-Aminobutyric Acid; Haloperidol; Kinetics; Lithium; Rats; Receptors, Dopamine; Spiperone; Synapses; Synaptic Transmission | 1985 |
Evaluation of different GABA receptor agonists in the kindled amygdala seizure model in rats.
Topics: Amygdala; Animals; Female; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Isoxazoles; Kindling, Neurologic; Muscimol; Muscle Relaxation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures | 1985 |
Upregulation of gamma-aminobutyric acid (GABA) B binding sites in rat frontal cortex: a common action of repeated administration of different classes of antidepressants and electroshock.
Topics: Animals; Antidepressive Agents; Cerebral Cortex; Desipramine; Dose-Response Relationship, Drug; Electroshock; Fluoxetine; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Male; Monoamine Oxidase Inhibitors; Nomifensine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin Antagonists; Time Factors; Viloxazine | 1985 |
[Progabide treatment of a case of the syndrome of painful legs and moving toes].
Topics: Adult; Female; gamma-Aminobutyric Acid; Humans; Leg; Middle Aged; Movement Disorders; Pain; Receptors, GABA-A; Syndrome; Toes | 1985 |
Further evidence for, and nature of, the facilitatory GABAergic influence on central noradrenergic transmission.
Topics: Afferent Pathways; Animals; Central Nervous System; Cerebral Cortex; Clonidine; gamma-Aminobutyric Acid; Hypothalamus; Ibotenic Acid; Methoxyhydroxyphenylglycol; Muscimol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Spinal Cord; Synaptic Transmission; Yohimbine | 1985 |
Effects of gamma-aminobutyric acid (GABA) receptor agonists on the neurotoxicity and anticonvulsant activity of barbiturates in mice.
Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; Dose-Response Relationship, Drug; Drug Synergism; Electroshock; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Nervous System; Oxazoles; Receptors, GABA-A; Seizures | 1986 |
Effect of ethosuximide alone and in combination with gamma-aminobutyric acid receptor agonists on brain gamma-aminobutyric acid concentration, anticonvulsant activity and neurotoxicity in mice.
Topics: Animals; Brain Chemistry; Ethosuximide; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Mice, Inbred Strains; Nervous System; Pentylenetetrazole; Receptors, GABA-A; Seizures | 1986 |
Anticonvulsant profile of drugs which facilitate GABAergic transmission on convulsions mediated by a GABAergic mechanism.
Topics: Animals; Anticonvulsants; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; gamma-Aminobutyric Acid; Male; Pentobarbital; Rats; Rats, Inbred Strains; Seizures; Synaptic Transmission | 1986 |
The effects of drugs acting at the GABAA-receptor/ionophore after chemical kindling with the benzodiazepine receptor ligand FG 7142.
Topics: Animals; Bicuculline; Body Temperature; Carbolines; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Mice; Muscimol; Pentobarbital; Pentylenetetrazole; Picrotoxin; Receptors, GABA-A; Seizures; Time Factors | 1986 |
The effects of the GABA-mimetic drugs, progabide and baclofen, on the biochemistry and function of 5-hydroxytryptamine and noradrenaline.
Topics: Animals; Baclofen; Brain; Brain Chemistry; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Norepinephrine; Receptors, Adrenergic, beta; Receptors, GABA-A; Receptors, Serotonin; Serotonin; Stereoisomerism | 1986 |
Effect of THIP and SL 76002, two clinically experimented GABA-mimetic compounds, on anterior pituitary GABA receptors and prolactin secretion in the rat.
Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Female; gamma-Aminobutyric Acid; Haloperidol; Isoxazoles; Kinetics; Male; Muscimol; Ovariectomy; Oxazoles; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
GABA receptor agonists and extrapyramidal motor function: therapeutic implications for Parkinson's disease.
Topics: Acetylcholine; Animals; Antiparkinson Agents; Cholinergic Fibers; Corpus Striatum; Dopamine; Extrapyramidal Tracts; gamma-Aminobutyric Acid; Humans; Motor Skills; Parkinson Disease; Receptors, Dopamine; Receptors, GABA-A; Synapses; Synaptic Transmission | 1987 |
Fengabine, a novel antidepressant GABAergic agent. I. Activity in models for antidepressant drugs and psychopharmacological profile.
Topics: Animals; Antidepressive Agents; Avoidance Learning; Behavior, Animal; Bicuculline; Chlorophenols; Clomipramine; Depressive Disorder; Disease Models, Animal; gamma-Aminobutyric Acid; Imipramine; Male; Olfactory Bulb; Rats; Receptors, GABA-A; Seizures; Sleep | 1987 |
Effects of GABAergic drugs on the GABA turnover in the substantia nigra and the corpus striatum of the rat.
Topics: Alkynes; Aminocaproates; Animals; Baclofen; Bicuculline; Corpus Striatum; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1987 |
Effects of long-lasting antiepileptic therapy on brainstem auditory evoked potentials.
Topics: Adolescent; Adult; Anticonvulsants; Brain Stem; Carbamazepine; Child; Epilepsies, Partial; Evoked Potentials, Auditory; Female; gamma-Aminobutyric Acid; Humans; Long-Term Care; Male; Middle Aged; Phenobarbital; Reaction Time; Valproic Acid | 1988 |
Effects of progabide on bicuculline-induced epileptic seizures in developing rats.
Topics: Aging; Animals; Anticonvulsants; Bicuculline; Female; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Seizures; Status Epilepticus | 1988 |
The stability and solubility of progabide and its related metabolic derivatives.
Topics: Anticonvulsants; Drug Stability; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Prodrugs; Solubility; Spectrophotometry; Temperature | 1988 |
Blood levels of progabide and its active metabolite in epileptic patients: relationships to the therapeutic outcome.
Topics: Adult; Dose-Response Relationship, Drug; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Monitoring, Physiologic | 1988 |
Submassive hepatic necrosis associated with the use of progabide: a GABA receptor agonist.
Topics: Adult; Anticonvulsants; Chemical and Drug Induced Liver Injury; Female; gamma-Aminobutyric Acid; Humans; Liver; Liver Function Tests; Necrosis; Seizures | 1988 |
Progabide, a GABA mimetic drug, stimulates the secretion of plasma corticosterone in rats.
Topics: Animals; Anticonvulsants; Clonidine; Corticosterone; Dexamethasone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Picrotoxin; Rats; Rats, Inbred Strains; Stimulation, Chemical | 1987 |
A reversed-phase high-performance liquid chromatography assay procedure for progabide and its related metabolic derivatives.
Topics: Calibration; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Solutions | 1987 |
Progabide and SL 75102 binding to plasma proteins and red blood cells in humans.
Topics: Anticonvulsants; Blood Proteins; Dialysis; Erythrocytes; gamma-Aminobutyric Acid; Hematocrit; Humans; Protein Binding | 1987 |
Effect of erythrocytes and plasma protein binding on the transport of progabide and SL 75102 through the rat blood-brain barrier.
Topics: Biological Transport, Active; Blood Proteins; Blood-Brain Barrier; Erythrocytes; gamma-Aminobutyric Acid; Humans; Lipoproteins; Mathematics | 1987 |
Progabide in Parkinson's disease.
Topics: gamma-Aminobutyric Acid; Humans; Parkinson Disease | 1987 |
Involvement of a GABAergic mechanism in the pharmacologic action of phenytoin.
Topics: Animals; Anticonvulsants; Baclofen; Electroshock; gamma-Aminobutyric Acid; Male; Mice; Phenytoin; Postural Balance; Seizures | 1986 |
Chromatographic selectivity and maintenance of column efficiency during the high-performance liquid chromatographic analysis of progabide and its acid metabolite.
Topics: Anticonvulsants; Carbamazepine; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Humans; Spectrophotometry, Ultraviolet | 1986 |
GABA-mimetic drugs enhance apomorphine-induced contralateral turning in rats with unilateral nigrostriatal dopamine denervation: implications for the therapy of Parkinson's disease.
Topics: Alkynes; Aminocaproates; Animals; Antiparkinson Agents; Apomorphine; Drug Synergism; gamma-Aminobutyric Acid; Isoxazoles; Male; Motor Activity; Nicotinic Acids; Parkinson Disease; Rats; Rats, Inbred Strains | 1987 |
Long-term treatment of epilepsy: open multicenter trial with progabide in epileptic patients.
Topics: Adolescent; Adult; Anticonvulsants; Child; Child, Preschool; Dose-Response Relationship, Drug; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Infant; Male; Middle Aged | 1987 |
Progabide in the treatment of hyperkinetic extrapyramidal movement disorders.
Topics: Adolescent; Adult; Aged; Athetosis; Basal Ganglia Diseases; Child; Chorea; Female; gamma-Aminobutyric Acid; Humans; Hyperkinesis; Male; Middle Aged; Myoclonus; Tourette Syndrome | 1985 |
Stability of the amino acid content of nerve endings after administration of gamma-aminobutyrate agonists and antagonists.
Topics: Amino Acids; Animals; Anticonvulsants; Aspartic Acid; Baclofen; Bicuculline; Brain Chemistry; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Mice; Muscimol; Nerve Endings; Picrotoxin; Synaptosomes | 1985 |
Anticonvulsant action of GABA agonists and prodrugs on minor and major seizures in epileptic gerbils. Comparison with mouse models of seizure states.
Topics: Animals; Anticonvulsants; Disease Models, Animal; Electroshock; Female; gamma-Aminobutyric Acid; Gerbillinae; In Vitro Techniques; Isoxazoles; Mice; Pentylenetetrazole; Seizures; Species Specificity | 1985 |
Determination of progabide and its acid metabolite in biological fluids by high-performance liquid chromatography on silica column with ultraviolet detection.
Topics: Biotransformation; Body Fluids; Chromatography, High Pressure Liquid; Drug Stability; Electrochemistry; gamma-Aminobutyric Acid; Humans; Kinetics; Solvents; Spectrophotometry, Ultraviolet | 1985 |
Experimental basis for the antidepressant action of the GABA receptor agonist progabide.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Brain; Depressive Disorder; gamma-Aminobutyric Acid; Humans; Mice; Norepinephrine; Receptors, Cell Surface; Receptors, GABA-A; Serotonin; Synaptic Transmission | 1984 |
Pharmacology of the GABAergic system: effects of progabide, a GABA receptor agonist.
Topics: Animals; Brain; Dopamine; gamma-Aminobutyric Acid; Humans; Norepinephrine; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Serotonin; Synaptic Transmission | 1984 |
Effect of the new gamma-aminobutyric acid agonist SL 76 002 on striatal acetylcholine: relation to neuroleptic-induced extrapyramidal alterations.
Topics: Acetylcholine; Animals; Antipsychotic Agents; Corpus Striatum; Dopamine; Extrapyramidal Tracts; gamma-Aminobutyric Acid; Haloperidol; Humans; Neurons; Parasympathetic Nervous System | 1980 |
gamma-Aminobutyric acid (GABA) receptor stimulation. II. Specificity of progabide (SL 76002) and SL 75102 for the GABA receptor.
Topics: Animals; Brain; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Muscimol; Neurotransmitter Agents; Rabbits; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1982 |
Enhancing GABAergic transmission reverses the aversive state in rats induced by electrical stimulation of the periaqueductal grey region.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Disease Models, Animal; Drug Interactions; Electric Stimulation; Escape Reaction; gamma-Aminobutyric Acid; Humans; Male; Periaqueductal Gray; Rats; Synaptic Transmission | 1982 |
Differential effects of the benzodiazepine antagonist Ro 15-1788 on two types of myoclonus in baboon Papio papio.
Topics: 5-Hydroxytryptophan; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Flumazenil; gamma-Aminobutyric Acid; Light; Lorazepam; Myoclonus; Papio; Seizures | 1983 |
Successful treatment of hemiballismus with progabide, a new GABA-mimetic agent.
Topics: Aged; Brain; Female; gamma-Aminobutyric Acid; Humans; Movement Disorders; Thalamic Nuclei; Tomography, X-Ray Computed | 1983 |
GABAB receptor-mediated inhibition of serotonin release in the rat brain.
Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Brain Chemistry; Cerebral Cortex; Diazepam; Electric Stimulation; gamma-Aminobutyric Acid; Hydroxyindoleacetic Acid; In Vitro Techniques; Male; Nipecotic Acids; Phentolamine; Picrotoxin; Proline; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin | 1984 |
Parkinson's disease and benign essential tremor: somatostatin-like immunoreactivity in the cerebrospinal fluid.
Topics: Adult; Aged; Alzheimer Disease; Atrophy; Brain Diseases; Female; gamma-Aminobutyric Acid; Humans; Huntington Disease; Male; Middle Aged; Multiple Sclerosis; Parkinson Disease; Peptides; Tremor | 1984 |
Reversal of the antiaversive and anticonvulsant actions of diazepam, but not of progabide, by a selective antagonist of benzodiazepine receptors.
Topics: Animals; Anxiety; Benzodiazepinones; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures | 1981 |
gamma-Aminobutyric acid (GABA) receptor stimulation. I. Neuropharmacological profiles of progabide (SL 76002) and SL 75102, with emphasis on their anticonvulsant spectra.
Topics: Animals; Anticonvulsants; Apomorphine; Behavior, Animal; Catalepsy; Drug Interactions; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Mice; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stereotyped Behavior | 1982 |
gamma-Aminobutyric acid (GABA) receptor stimulation. III. Effect of progabide (SL 76002) on norepinephrine, dopamine and 5-hydroxytryptamine turnover in rat brain areas.
Topics: Animals; Brain; Dopamine; gamma-Aminobutyric Acid; Male; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin; Synaptic Transmission; Tryptamines | 1982 |
gamma-Aminobutyric acid (GABA) receptor stimulation. IV. Effect of progabide (SL 76002) and other GABAergic agents on acetylcholine turnover in rat brain areas.
Topics: Acetylcholine; Animals; Brain; Corpus Striatum; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission | 1982 |
Actions of GABAergic agents on dopamine metabolism in the nigrostriatal pathway of the rat.
Topics: 4-Aminobutyrate Transaminase; Aminooxyacetic Acid; Animals; Corpus Striatum; Diazepam; Dopamine; GABA Antagonists; gamma-Aminobutyric Acid; Isoxazoles; Male; Muscimol; Neural Pathways; Pyrones; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra | 1982 |
Pharmacological and therapeutic actions of GABA receptor agonists.
Topics: Bipolar Disorder; Emotions; gamma-Aminobutyric Acid; Humans; Movement Disorders; Norepinephrine; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Serotonin | 1983 |
Reversal of the muscle relaxant effect of diazepam but not of progabide by a specific benzodiazepine antagonist: Ro 15-1788.
Topics: Animals; Benzodiazepinones; Diazepam; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscle Contraction; Muscle Relaxants, Central; Rats; Rats, Inbred Strains; Time Factors | 1983 |
Indications for the use of gamma-aminobutyric acid (GABA)-agonists in convulsant disorders.
Topics: Animals; Anticonvulsants; Disease Models, Animal; Epilepsies, Partial; Epilepsy; gamma-Aminobutyric Acid; Humans; Nervous System; Papio; Seizures; Synapses | 1983 |
The comparative effects of benzodiazepines, progabide and PK 9084 on acquisition of passive avoidance in mice.
Topics: Animals; Avoidance Learning; Benzodiazepines; gamma-Aminobutyric Acid; Male; Mice; Motor Activity; Quinolines | 1984 |
Disposition of progabide and valproic acid following intraperitoneal administration in rhesus monkey.
Topics: Absorption; Administration, Oral; Animals; Biological Availability; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Injections, Intravenous; Kinetics; Macaca mulatta; Male; Peritoneum; Valproic Acid | 1984 |
Chlordiazepoxide-induced hyperphagia in rats: lack of effect of GABA agonists and antagonists.
Topics: Animals; Chlordiazepoxide; Eating; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains | 1984 |
Effects in man of progabide on prolactin release induced by haloperidol or domperidone.
Topics: Adult; Domperidone; gamma-Aminobutyric Acid; Haloperidol; Humans; Male; Premedication; Prolactin | 1984 |
Penicillin spikes in rats. Limitations of a simple model for the study of anticonvulsants.
Topics: Action Potentials; Animals; Anticonvulsants; Dimethyl Sulfoxide; Disease Models, Animal; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Isoxazoles; Male; Penicillins; Phenytoin; Rats; Rats, Inbred Strains; Seizures; Taurine; Time Factors | 1984 |
SL76002 - effect on gamma-aminobutyric acid and dopamine in animals treated chronically with haloperidol.
Topics: Animals; Brain Chemistry; Corpus Striatum; Dopamine; Dyskinesia, Drug-Induced; Frontal Lobe; gamma-Aminobutyric Acid; Haloperidol; Male; Mesencephalon; Rats; Rats, Inbred Strains | 1983 |
Measurement of progabide and its deaminated metabolite in plasma by high-performance liquid chromatography and electrochemical detection.
Topics: Chromatography, High Pressure Liquid; Electrochemistry; gamma-Aminobutyric Acid; Half-Life; Humans; Kinetics; Spectrophotometry, Ultraviolet | 1983 |
An analysis of the actions of progabide, a specific GABA receptor agonist, on kindling and kindled seizures.
Topics: Amygdala; Animals; Anticonvulsants; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains; Seizures | 1984 |
Determination of progabide and its main acid metabolite in biological fluids using high-performance liquid chromatography and electrochemical detection. Application to the measurement of blood/plasma partition ratio.
Topics: Anticonvulsants; Chromatography, Gas; Chromatography, High Pressure Liquid; Drug Stability; Electrochemistry; gamma-Aminobutyric Acid; Humans; Hydrogen-Ion Concentration; Kinetics; Oxidation-Reduction; Solubility; Temperature | 1984 |
Increase in striatal acetylcholine levels by GABAergic agents: dependence on corticostriatal neurons.
Topics: Acetylcholine; Animals; Cerebral Cortex; Corpus Striatum; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Muscimol; Neurons; Rats; Valproic Acid | 1980 |
Prolonged treatment with gamma-aminobutyric acid (GABA)-mimetic substances in prepubertal male rats.
Topics: 4-Butyrolactone; Alkynes; Aminocaproates; Animals; Body Weight; gamma-Aminobutyric Acid; Male; Organ Size; Prolactin; Rats; Rats, Inbred Strains; Seminal Vesicles; Sexual Maturation; Testis; Time Factors | 1983 |
Pharmacokinetic profile of progabide, a new gamma-aminobutyric acid-mimetic drug, in rhesus monkey.
Topics: Administration, Oral; Animals; Anticonvulsants; gamma-Aminobutyric Acid; Injections, Intravenous; Kinetics; Macaca mulatta; Male; Protein Binding; Time Factors | 1982 |
Gas chromatographic method for the determination of progabide (SL 76.002) in biological fluids.
Topics: Animals; Chromatography, Gas; Dogs; gamma-Aminobutyric Acid; Humans; Rats; Reference Values; Time Factors | 1982 |
Effects of GABA analogues and their interactions with morphine on locomotor activity in two inbred strains of mice.
Topics: Animals; Drug Interactions; gamma-Aminobutyric Acid; Isoxazoles; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Morphine; Motor Activity; Muscimol; Piracetam | 1982 |
Action of progabide in the photosensitive baboon, Papio papio.
Topics: Allylglycine; Animals; Anticonvulsants; Blood-Brain Barrier; Brain; Dose-Response Relationship, Drug; Drug Synergism; Electroencephalography; Epilepsy; gamma-Aminobutyric Acid; Papio; Photosensitivity Disorders; Sleep Stages | 1982 |
Further evidence for the interactions between angiotensin II and GABAergic transmission in pentylenetetrazol kindling seizures in mice.
Topics: Angiotensin II; Animals; Baclofen; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Mice; Nipecotic Acids; Pentylenetetrazole; Phenylurea Compounds; Receptors, GABA; Seizures | 1995 |
Possible involvement of a gamma-hydroxybutyric acid receptor in startle disease.
Topics: Anesthetics; Anticonvulsants; GABA Agonists; gamma-Aminobutyric Acid; Humans; Infant, Newborn; Male; Neuromuscular Diseases; Receptors, Cell Surface; Reflex, Abnormal; Reflex, Startle; Sodium Oxybate | 1994 |
In vivo and in vitro correlation of microsomal epoxide hydrolase inhibition by progabide.
Topics: Adult; Anticonvulsants; Carbamazepine; Drug Interactions; Epoxide Hydrolases; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Least-Squares Analysis; Male; Microsomes, Liver; Reference Values | 1993 |
Suppression of cortical epileptic afterdischarges in developing rats by anticonvulsants increasing GABAergic inhibition.
Topics: Animals; Anticonvulsants; Cerebral Cortex; Depression, Chemical; Drug Evaluation, Preclinical; Electric Stimulation; Electroencephalography; Enzyme Inhibitors; Epilepsy; GABA Agents; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Neural Inhibition; Phenobarbital; Rats; Valproic Acid | 1996 |
The inhibitory effects on sexual behavior and ambulatory activity of the mixed GABAA/GABAB agonist progabide are differentially blocked by GABA receptor antagonists.
Topics: Animals; Bicuculline; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Motor Activity; Organophosphorus Compounds; Psychomotor Performance; Rats; Rats, Wistar; Sexual Behavior, Animal | 1997 |
Grouped random effects models for Bayesian meta-analysis.
Topics: Algorithms; Anticonvulsants; Bayes Theorem; gamma-Aminobutyric Acid; Humans; Markov Chains; Meta-Analysis as Topic; Models, Statistical; Monte Carlo Method; Research Design | 1997 |
Mechanisms of the inhibition of human erythrocyte pyridoxal kinase by drugs.
Topics: Drug Interactions; Enzyme Inhibitors; Erythrocytes; gamma-Aminobutyric Acid; Humans; Kinetics; Muzolimine; Pyridoxal; Pyridoxal Kinase; Spectrophotometry, Ultraviolet; Thiamphenicol | 1997 |
Analysis of overdispersed count data by mixtures of Poisson variables and Poisson processes.
Topics: Anticonvulsants; Biometry; Epilepsy; gamma-Aminobutyric Acid; Humans; Likelihood Functions; Normal Distribution; Poisson Distribution; Probability; Seizures; Statistical Distributions | 1997 |
Interactions between dopamine and GABA in the control of ambulatory activity and neophobia in the mouse.
Topics: Amphetamine; Animals; Chi-Square Distribution; Dopamine; Dopamine Agents; Exploratory Behavior; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Phobic Disorders | 1998 |
Severe visual-field constriction and side-effects of GABA-mimetic antiepileptic agents.
Topics: Anticonvulsants; Epilepsies, Myoclonic; Epilepsy, Tonic-Clonic; Female; Follow-Up Studies; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Humans; Middle Aged; Phenobarbital; Vision Disorders; Visual Fields | 1998 |
Anticonvulsant effect of progabide in rats during ontogenesis.
Topics: Aging; Animals; Anticonvulsants; Behavior, Animal; Convulsants; gamma-Aminobutyric Acid; Male; Pentylenetetrazole; Rats; Rats, Wistar; Seizures | 1997 |
[Concentric changes in the visual field associated with GABA-mimetic antiepileptic agents].
Topics: Adult; Anticonvulsants; Female; GABA Modulators; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Phenobarbital; Vigabatrin; Visual Field Tests; Visual Fields | 1999 |
Unit-treatment interaction and its practical consequences.
Topics: Analysis of Variance; Anticonvulsants; Clinical Trials as Topic; Epilepsy; gamma-Aminobutyric Acid; Humans; Likelihood Functions; Models, Statistical; Randomized Controlled Trials as Topic; Seizures | 2000 |
Differential role of dopamine D1 and D2 receptors in isoniazid-induced vacuous chewing movements.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Anticonvulsants; Antipsychotic Agents; Antitubercular Agents; Behavior, Animal; Diazepam; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; gamma-Aminobutyric Acid; Isoniazid; Male; Mastication; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Stereotyped Behavior; Time Factors | 2000 |
Selection effects in randomized trials with count data.
Topics: Anticonvulsants; Computer Simulation; Electrocardiography, Ambulatory; Epilepsy; gamma-Aminobutyric Acid; Humans; Models, Biological; Myocardial Ischemia; Randomized Controlled Trials as Topic; Seizures; Selection Bias | 2002 |
Hypothesis testing in semiparametric additive mixed models.
Topics: Anticonvulsants; Child; Computer Simulation; Data Interpretation, Statistical; Epilepsy; Female; gamma-Aminobutyric Acid; Humans; Indonesia; Likelihood Functions; Longitudinal Studies; Male; Models, Statistical; Placebos; Randomized Controlled Trials as Topic; Respiratory Tract Infections; Statistics, Nonparametric; Xerophthalmia | 2003 |
[Endoscopic mucosal resection in the upper and lower GI tract].
Topics: Carcinoma in Situ; Contraindications; Endoscopy, Gastrointestinal; gamma-Aminobutyric Acid; Gastric Mucosa; Gastrointestinal Neoplasms; Intestinal Mucosa; Lymphatic Metastasis; Neoplasm Staging; Precancerous Conditions; Surgical Instruments | 2004 |
Combined discriminative stimulus effects of midazolam with other positive GABAA modulators and GABAA receptor agonists in rhesus monkeys.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Ethanol; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Injections, Subcutaneous; Isoxazoles; Macaca mulatta; Male; Midazolam; Pentobarbital; Pregnanolone; Receptors, GABA-A; Time Factors; Triazolam; Women | 2005 |
How to appraise the effectiveness of treatment.
Topics: Evaluation Studies as Topic; Evidence-Based Medicine; gamma-Aminobutyric Acid; Guidelines as Topic; Humans; Outcome Assessment, Health Care; Randomized Controlled Trials as Topic; Research Design | 2005 |
Robust estimating functions and bias correction for longitudinal data analysis.
Topics: Age Factors; Anticonvulsants; Bias; Data Interpretation, Statistical; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Randomized Controlled Trials as Topic; Seizures | 2005 |
Quadratic inference functions in marginal models for longitudinal data.
Topics: Anticonvulsants; Computer Simulation; Data Interpretation, Statistical; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Models, Statistical; Seizures; Software | 2009 |
Inference on the rate ratio of recurrent events for the matched pairs design.
Topics: Anticonvulsants; Data Interpretation, Statistical; Epilepsy; gamma-Aminobutyric Acid; Humans; Incidence; Product Surveillance, Postmarketing; Randomized Controlled Trials as Topic; Recurrence; Sample Size; Seizures | 2010 |
Prognostic prediction in patients with hip fracture: risk factors predicting difficulties with discharge to own home.
Topics: Age Distribution; Aged; Aged, 80 and over; Comorbidity; Dementia; Disability Evaluation; Female; Femoral Neck Fractures; gamma-Aminobutyric Acid; Hospital Mortality; Humans; Male; Middle Aged; Multivariate Analysis; Patient Discharge; Predictive Value of Tests; Risk Factors; Walking | 2011 |
Working covariance model selection for generalized estimating equations.
Topics: Anticonvulsants; Computer Simulation; Data Interpretation, Statistical; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Models, Statistical; Normal Distribution; Randomized Controlled Trials as Topic; Software | 2011 |
A bias correction for covariance estimators to improve inference with generalized estimating equations that use an unstructured correlation matrix.
Topics: Anticonvulsants; Bias; Computer Simulation; Epilepsy; gamma-Aminobutyric Acid; Humans; Longitudinal Studies; Models, Statistical; Seizures | 2013 |
Objective Bayesian meta-analysis for sparse discrete data.
Topics: Bayes Theorem; Cardiovascular Diseases; Diabetes Mellitus, Type 2; Diabetes, Gestational; Epilepsy; Female; gamma-Aminobutyric Acid; Hormone Replacement Therapy; Humans; Meta-Analysis as Topic; Models, Statistical; Multicenter Studies as Topic; Pregnancy; Rosiglitazone; Thiazolidinediones; Treatment Outcome | 2014 |
Acoustic radiation force impulse elastography for non-invasive assessment of disease stage in patients with primary biliary cirrhosis: A preliminary study.
Topics: Biopsy; Elasticity Imaging Techniques; Female; gamma-Aminobutyric Acid; Humans; Liver; Liver Cirrhosis, Biliary; Male; Middle Aged; Reproducibility of Results; ROC Curve; Sensitivity and Specificity | 2014 |
Association of left atrial reservoir function with left atrial structural remodeling related to left ventricular dysfunction in asymptomatic patients with hypertension: evaluation by two-dimensional speckle-tracking echocardiography.
Topics: Atrial Function, Left; Echocardiography; Female; Follow-Up Studies; gamma-Aminobutyric Acid; Heart Atria; Heart Ventricles; Humans; Hypertension; Male; Middle Aged; Retrospective Studies; Ventricular Dysfunction, Left; Ventricular Function, Left; Ventricular Remodeling | 2015 |
Covariance estimators for generalized estimating equations (GEE) in longitudinal analysis with small samples.
Topics: Adolescent; Anticonvulsants; Bias; Child; Computer Simulation; Epilepsy; Female; gamma-Aminobutyric Acid; Head; Humans; Longitudinal Studies; Male; Models, Statistical; Randomized Controlled Trials as Topic; Sample Size; Software | 2016 |
Discovery of a Novel Microsomal Epoxide Hydrolase-Catalyzed Hydration of a Spiro Oxetane.
Topics: Azetidines; Biotransformation; Catalysis; Enzyme Inhibitors; Epoxide Hydrolases; gamma-Aminobutyric Acid; Humans; Kinetics; Microsomes, Liver; Molecular Structure; Oxadiazoles; Substrate Specificity | 2016 |