Page last updated: 2024-08-16

probenecid and verlukast

probenecid has been researched along with verlukast in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's18 (66.67)29.6817
2010's8 (29.63)24.3611
2020's1 (3.70)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Elmquist, WF; Finch, RA; Johnson, DR; Miller, DW; Sartorelli, AC; Sun, H1
Taylor, EM; Yan, R1
Buesen, R; Jacob, J; Lampen, A; Mock, M; Nau, H; Seidel, A1
Lim, BG; Ng, KH; Wong, KP1
Cisternino, S; Lorico, A; Rappa, G; Rousselle, C; Scherrmann, JM1
Broxterman, HJ; de Jong, MC; Hooijberg, JH; Husain, SR; Joshi, BH; Kreitman, RJ; Meloen, RH; Puri, RK; Scheffer, GL; Scheper, RJ; Slootstra, JW1
Dogan, AL; Faussat, AM; Legrand, O; Marie, JP; Perrot, JY1
Candussio, L; Crivellato, E; Damiani, D; Decorti, G; Giraldi, T; Klugmann, FB; Michelutti, A; Rosati, A1
Capella, L; Capella, MA; Echevarria-Lima, J; Kyle-Cezar, F; P Leite, DF; Rumjanek, VM1
Chen, V; Dantzig, AH; Perry, WI; Pratt, S; Starling, JJ1
Leader, JP; O'Donnell, MJ1
Calixto, JB; Capella, MA; Echevarria-Lima, J; Leite, DF; Rumjanek, VM; Salgado, LT1
Bertelsen, KM; Greenblatt, DJ; von Moltke, LL1
Tian, X; Wang, K; Yang, X1
Chen, X; Chowbay, B; Duan, W; Li, CG; Liang, J; Lin, SG; Liu, PQ; Wen, JY; Yu, XY; Zhou, SF; Zhou, ZW1
Jani, M; Kovács, B; Krajcsi, P; Lin, G; Zhang, L; Zuo, Z1
Hakala, KE; Heikkinen, TM; Laine, KP; Rahi, MM1
Abelli, L; Adinolfi, E; Bertoni, F; Biondi, C; Cervellati, F; Ferretti, ME; Lunghi, L; Medici, S; Morano, D; Pavan, B; Vesce, F1
Jakob, I; Molinas, A; Sicard, G1
Pattabiraman, PP; Pecen, PE; Rao, PV1
Chen, Z; Han, J; Hu, T; Huang, C; Li, J; Ma, T; Zhang, L; Zhong, J1
Bai, P; Chen, M; Deng, X; Hu, J; Miao, P; Xu, Y; Yin, H; Yin, J1
Abba, M; Attorresi, AI; Carozzo, A; Davio, C; Di Siervi, N; Diez, F; Fernández, N; Gómez, N; Monczor, F; Rodríguez-González, Á; Sahores, A; Shayo, C; Yaneff, A1
Aa, JY; Deng, QQ; Han, L; Liao, XY; Pan, GY; Peng, ZL; Wang, GJ; Wu, ZT; Xie, Y1
Liang, C; Liu, M; Wang, X; Xu, F; Xu, P; Zhang, L1

Other Studies

27 other study(ies) available for probenecid and verlukast

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Transport of fluorescein in MDCKII-MRP1 transfected cells and mrp1-knockout mice.
    Biochemical and biophysical research communications, 2001, Jun-22, Volume: 284, Issue:4

    Topics: Animals; ATP-Binding Cassette Transporters; Base Pair Mismatch; Biological Transport; Blood-Brain Barrier; Brain; Dogs; Fluorescein; Kinetics; Mice; Mice, Knockout; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Recombinant Proteins; Substrate Specificity; Tissue Distribution; Transfection

2001
Neotrofin is transported out of brain by a saturable mechanism: possible involvement of multidrug resistance and monocarboxylic acid transporters.
    Drug metabolism and disposition: the biological fate of chemicals, 2002, Volume: 30, Issue:5

    Topics: Aminobenzoates; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Brain; Capillaries; Drug Resistance, Multiple; Endothelium, Vascular; Hypoxanthines; Injections, Intraventricular; Male; Mice; Monocarboxylic Acid Transporters; Nootropic Agents; Organic Anion Transporters; Probenecid; Propionates; Purines; Quinolines; Verapamil

2002
Human intestinal Caco-2 cells display active transport of benzo[a]pyrene metabolites.
    Chemico-biological interactions, 2003, Jan-06, Volume: 142, Issue:3

    Topics: Adenosine Triphosphate; Aryl Hydrocarbon Hydroxylases; ATP-Binding Cassette Transporters; Benzo(a)pyrene; Benzoflavones; Biological Transport, Active; Caco-2 Cells; Cell Polarity; Cyclosporine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1B1; Enterocytes; Gene Expression; Humans; Models, Biological; Probenecid; Propionates; Quinolines; Verapamil; Vinblastine

2003
Sulfate conjugating and transport functions of MDCK distal tubular cells.
    Kidney international, 2003, Volume: 63, Issue:3

    Topics: Animals; Biological Transport; Buthionine Sulfoximine; Carcinoma, Hepatocellular; Cell Line, Tumor; Cyclosporine; Glutathione; Harmine; Humans; Immunosuppressive Agents; Kidney Tubules, Distal; Leukotriene Antagonists; Liver; Membrane Transport Proteins; Methotrexate; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Organic Anion Transport Protein 1; Probenecid; Propionates; Quinolines; Radiation-Protective Agents; Radiation-Sensitizing Agents; Sulfates; Uricosuric Agents

2003
Apparent lack of Mrp1-mediated efflux at the luminal side of mouse blood-brain barrier endothelial cells.
    Pharmaceutical research, 2003, Volume: 20, Issue:6

    Topics: Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Blood-Brain Barrier; Chemokines, CC; Endothelial Cells; Estradiol; Etoposide; Male; Mice; Mice, Knockout; Perfusion; Probenecid; Propionates; Quinolines; Xenobiotics

2003
Multidrug-resistant tumor cells remain sensitive to a recombinant interleukin-4-Pseudomonas exotoxin, except when overexpressing the multidrug resistance protein MRP1.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2003, Oct-15, Volume: 9, Issue:13

    Topics: Antimetabolites, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bacterial Toxins; Buthionine Sulfoximine; Cell Line, Tumor; Cell Membrane; DNA, Complementary; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Exotoxins; Humans; Interleukin-4; Leukotriene Antagonists; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Recombinant Proteins; Transfection; Uricosuric Agents

2003
Evaluation and comparison of MRP1 activity with three fluorescent dyes and three modulators in leukemic cell lines.
    Leukemia research, 2004, Volume: 28, Issue:6

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Bronchodilator Agents; Cyclosporine; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; Leukemia; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Rhodamine 123; Tumor Cells, Cultured

2004
Bodipy-FL-verapamil: a fluorescent probe for the study of multidrug resistance proteins.
    Cellular oncology : the official journal of the International Society for Cellular Oncology, 2004, Volume: 26, Issue:1-2

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Assay; Cell Line, Tumor; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Dyes; Humans; Leukemia; Mice; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Predictive Value of Tests; Probenecid; Propionates; Quinolines; Sus scrofa; Up-Regulation; Verapamil; Vinblastine

2004
Expression and activity of multidrug resistance protein 1 in a murine thymoma cell line.
    Immunology, 2005, Volume: 114, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cell Differentiation; Cell Line, Tumor; Dose-Response Relationship, Drug; Fluoresceins; Fluorescent Dyes; Indomethacin; Mice; Probenecid; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; T-Lymphocytes; Thymoma

2005
Kinetic validation of the use of carboxydichlorofluorescein as a drug surrogate for MRP5-mediated transport.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2006, Volume: 27, Issue:5

    Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Antimetabolites, Antineoplastic; Cyclic Nucleotide Phosphodiesterases, Type 5; Fluoresceins; Fluorescent Dyes; Glutamates; Guanine; HeLa Cells; Humans; Kinetics; Membrane Transport Proteins; Methotrexate; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Pemetrexed; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Probenecid; Propionates; Quinolines; Reproducibility of Results; Staining and Labeling; Transfection

2006
Transepithelial transport of fluorescent p-glycoprotein and MRP2 substrates by insect Malpighian tubules: confocal microscopic analysis of secreted fluid droplets.
    The Journal of experimental biology, 2005, Volume: 208, Issue:Pt 23

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drosophila melanogaster; Epithelium; Fluorescent Dyes; Gryllidae; Malpighian Tubules; Microscopy, Confocal; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinacrine; Quinolines; Tetraethylammonium; Verapamil

2005
In vivo and in vitro modulation of MDR molecules in murine thymocytes.
    International immunopharmacology, 2006, Volume: 6, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Flow Cytometry; Fluorescent Antibody Technique; Genes, MDR; Indomethacin; Male; Mice; Mice, Inbred C3H; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Renal Agents; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; T-Lymphocytes; Thymus Gland

2006
Apparent active transport of MDMA is not mediated by P-glycoprotein: a comparison with MDCK and Caco-2 monolayers.
    Biopharmaceutics & drug disposition, 2006, Volume: 27, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line; Dogs; Humans; Indomethacin; N-Methyl-3,4-methylenedioxyamphetamine; Probenecid; Progesterone; Propionates; Quinolines; Rhodamine 123; Ritonavir; Verapamil

2006
The efflux of flavonoids morin, isorhamnetin-3-O-rutinoside and diosmetin-7-O-beta-D-xylopyranosyl-(1-6) -beta-D-glucopyranoside in the human intestinal cell line caco-2.
    Pharmaceutical research, 2006, Volume: 23, Issue:8

    Topics: Adenosine Triphosphate; Antioxidants; Biological Transport, Active; Caco-2 Cells; Chromatography, High Pressure Liquid; Disaccharides; Enzyme Inhibitors; Flavonoids; Humans; Intestinal Mucosa; Iodoacetamide; Probenecid; Propionates; Quercetin; Quinolines; Verapamil

2006
Role of P-glycoprotein in the intestinal absorption of tanshinone IIA, a major active ingredient in the root of Salvia miltiorrhiza Bunge.
    Current drug metabolism, 2007, Volume: 8, Issue:4

    Topics: Abietanes; Adenosine Triphosphate; Administration, Oral; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Availability; Caco-2 Cells; Digoxin; Dogs; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Microsomes, Liver; Multidrug Resistance-Associated Proteins; Phenanthrenes; Plant Roots; Probenecid; Propionates; Quinidine; Quinolines; Rats; Rats, Sprague-Dawley; Salvia miltiorrhiza; Temperature; Transfection; Verapamil

2007
Mechanistic study on the intestinal absorption and disposition of baicalein.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2007, Volume: 31, Issue:3-4

    Topics: Animals; ATP-Binding Cassette Transporters; Biological Transport, Active; Caco-2 Cells; Egtazic Acid; Enzyme Inhibitors; Estradiol; Flavanones; Glucuronides; Humans; Intestinal Absorption; Kinetics; Leukotriene C4; Multidrug Resistance-Associated Proteins; Permeability; Probenecid; Propionates; Quinolines; Spectrophotometry, Ultraviolet; Spodoptera; Sulfuric Acid Esters; Tandem Mass Spectrometry; Verapamil

2007
The effect of probenecid and MK-571 on the feto-maternal transfer of saquinavir in dually perfused human term placenta.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2009, Jul-12, Volume: 37, Issue:5

    Topics: Antipyrine; Biological Transport; Female; HIV Protease Inhibitors; Humans; In Vitro Techniques; Maternal-Fetal Exchange; Multidrug Resistance-Associated Proteins; Organic Anion Transporters; Perfusion; Placenta; Pregnancy; Probenecid; Propionates; Quinolines; Saquinavir; Trophoblasts

2009
cAMP efflux from human trophoblast cell lines: a role for multidrug resistance protein (MRP)1 transporter.
    Molecular human reproduction, 2010, Volume: 16, Issue:7

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cells, Cultured; Colforsin; Cyclic AMP; Estrone; Female; Fluorescent Antibody Technique; Humans; In Vitro Techniques; Interleukin-1beta; Placenta; Pregnancy; Probenecid; Progesterone; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Trophoblasts

2010
Functional evidence of multidrug resistance transporters (MDR) in rodent olfactory epithelium.
    PloS one, 2012, Volume: 7, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Sub-Family B Member 4; Biological Transport; Cyclosporine; Female; Fluoresceins; Gene Expression; Male; Mice; Mice, Inbred BALB C; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Olfactory Mucosa; Olfactory Receptor Neurons; Probenecid; Propionates; Quinolines; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Verapamil

2012
MRP4-mediated regulation of intracellular cAMP and cGMP levels in trabecular meshwork cells and homeostasis of intraocular pressure.
    Investigative ophthalmology & visual science, 2013, Mar-05, Volume: 54, Issue:3

    Topics: Actins; Adult; Aged; Animals; Aqueous Humor; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Homeostasis; Humans; Intraocular Pressure; Leukotriene Antagonists; Middle Aged; Multidrug Resistance-Associated Proteins; Myosin Light Chains; Phosphorylation; Probenecid; Propionates; Quinolines; Rabbits; RNA, Small Interfering; Signal Transduction; Trabecular Meshwork

2013
Efficiency of transcellular transport and efflux of flavonoids with different glycosidic units from flavonoids of Litsea coreana L. in a MDCK epithelial cell monolayer model.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2014, Mar-12, Volume: 53

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Dogs; Flavonoids; Glycosides; Hydrogen-Ion Concentration; Litsea; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Sodium-Glucose Transporter 1; Temperature; Verapamil

2014
ABC transporters affect the elimination and toxicity of CdTe quantum dots in liver and kidney cells.
    Toxicology and applied pharmacology, 2016, 07-15, Volume: 303

    Topics: Animals; ATP-Binding Cassette Transporters; Cadmium Compounds; Cell Line; Cell Survival; Cyclosporine; Dogs; Hep G2 Cells; Humans; Kidney; Liver; Madin Darby Canine Kidney Cells; Oligopeptides; Probenecid; Propionates; Quantum Dots; Quinolines; Rifampin; RNA, Messenger; Tellurium

2016
Identification of MRP4/ABCC4 as a Target for Reducing the Proliferation of Pancreatic Ductal Adenocarcinoma Cells by Modulating the cAMP Efflux.
    Molecular pharmacology, 2019, Volume: 96, Issue:1

    Topics: Benzothiazoles; Carcinoma, Pancreatic Ductal; Cell Differentiation; Cell Line, Tumor; Cell Proliferation; Cell Survival; Computer Simulation; Cyclic AMP; Gene Expression Regulation, Neoplastic; Gene Silencing; HEK293 Cells; Humans; Multidrug Resistance-Associated Proteins; Pancreatic Neoplasms; Probenecid; Prognosis; Propionates; Quinolines; Signal Transduction; Survival Analysis; Triazoles; Up-Regulation

2019
Leflunomide increased the renal exposure of acyclovir by inhibiting OAT1/3 and MRP2.
    Acta pharmacologica Sinica, 2020, Volume: 41, Issue:1

    Topics: Acyclovir; Administration, Intravenous; Animals; Cells, Cultured; Crotonates; Dogs; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Hydroxybutyrates; Kidney; Leflunomide; Madin Darby Canine Kidney Cells; Male; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Nitriles; Organic Anion Transport Protein 1; Organic Anion Transporters, Sodium-Independent; Probenecid; Propionates; Quinolines; Rats; Rats, Sprague-Dawley; Tissue Distribution; Toluidines

2020
Characterization of in vitro Mrp2 transporter model based on intestinal organoids.
    Regulatory toxicology and pharmacology : RTP, 2019, Volume: 108

    Topics: Animals; Fluoresceins; Intestine, Small; Male; Mice, Inbred C57BL; Models, Biological; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Organoids; Probenecid; Propionates; Quinolines

2019