Page last updated: 2024-08-16

probenecid and amiloride

probenecid has been researched along with amiloride in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19905 (31.25)18.7374
1990's2 (12.50)18.2507
2000's5 (31.25)29.6817
2010's4 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Boyd, CA; Gerard, EM; Hollander, D1
Hugentobler, G; Meier, PJ; Rahm, I; Valantinas, J1
Hugentobler, G; Meier, PJ1
Pace, CS; Smith, JS; Tarvin, JT1
Beigelman, PM; Eddlestone, GT1
Azoui, R; Cuche, JL; Dagher, G; Renaud, JF; Safar, M1
Deschepper, CF; Picard, S; Schiffrin, EL; Touyz, RM1
Ortiz, A; Said, HM; Vaziri, ND1
Cragoe, EJ; Edwards, AM; Lee, CH1

Reviews

3 review(s) available for probenecid and amiloride

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Stimulus-secretion coupling in beta-cells: modulation by pH.
    The American journal of physiology, 1983, Volume: 244, Issue:1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Action Potentials; Amiloride; Ammonium Chloride; Animals; Antiporters; Bicarbonates; Carrier Proteins; Cell Membrane; Cell Membrane Permeability; Chlorides; Electrophysiology; Glucose; Hydrogen-Ion Concentration; Imidazoles; Insulin; Insulin Secretion; Ion Exchange; Islets of Langerhans; Models, Biological; Probenecid; Protons; Radioisotopes; Rubidium; Sodium; Trialkyltin Compounds

1983

Other Studies

13 other study(ies) available for probenecid and amiloride

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Transport of butyric acid in vascularly perfused anuran small intestine: importance of pH and anion transport.
    The American journal of physiology, 1986, Volume: 250, Issue:4 Pt 1

    Topics: 3-O-Methylglucose; 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetazolamide; Amiloride; Animals; Anions; Biological Transport; Butyrates; Butyric Acid; Hydrogen-Ion Concentration; Intestine, Small; Kinetics; Methylglucosides; Perfusion; Probenecid; Rana esculenta

1986
Bicarbonate sulfate exchange in canalicular rat liver plasma membrane vesicles.
    The American journal of physiology, 1987, Volume: 253, Issue:4 Pt 1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetazolamide; Amiloride; Animals; Bicarbonates; Biological Transport, Active; Cell Membrane; Furosemide; Hydrogen-Ion Concentration; Kinetics; Liver; Male; Membrane Potentials; Probenecid; Rats; Rats, Inbred Strains; Substrate Specificity; Sulfates; Taurine

1987
Multispecific anion exchange in basolateral (sinusoidal) rat liver plasma membrane vesicles.
    The American journal of physiology, 1986, Volume: 251, Issue:5 Pt 1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Anions; Binding, Competitive; Biological Transport; Cell Membrane; Cholic Acid; Cholic Acids; Hydrogen-Ion Concentration; Kinetics; Liver; Male; Nigericin; Probenecid; Rats; Rats, Inbred Strains; Sodium; Sulfates; Sulfobromophthalein

1986
Pancreatic beta-cell electrical activity: the role of anions and the control of pH.
    The American journal of physiology, 1983, Volume: 244, Issue:3

    Topics: Amiloride; Animals; Anions; Chlorides; Electric Conductivity; Electric Stimulation; Glucose; Hydrogen-Ion Concentration; Islets of Langerhans; Membrane Potentials; Mice; Microelectrodes; Probenecid

1983
A dopamine transporter in human erythrocytes: modulation by insulin.
    Experimental physiology, 1996, Volume: 81, Issue:3

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Biological Transport; Carrier Proteins; Catecholamines; Choline; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Epinephrine; Erythrocytes; Humans; Hydrogen-Ion Concentration; Insulin; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Piperazines; Probenecid; Reserpine; Time Factors

1996
Cyclic GMP inhibits a pharmacologically distinct Na+/H+ exchanger variant in cultured rat astrocytes via an extracellular site of action.
    Journal of neurochemistry, 1997, Volume: 68, Issue:4

    Topics: Amiloride; Animals; Anti-Inflammatory Agents, Non-Steroidal; Astrocytes; Atrial Natriuretic Factor; Cells, Cultured; Choline; Cyclic GMP; Diuretics; Extracellular Space; Hydrogen-Ion Concentration; Natriuretic Peptide, C-Type; Niflumic Acid; Nootropic Agents; Probenecid; Proteins; Rats; Renal Agents; Sodium; Sodium-Hydrogen Exchangers

1997
Mechanism and regulation of vitamin B(6) uptake by renal tubular epithelia: studies with cultured OK cells.
    American journal of physiology. Renal physiology, 2002, Volume: 282, Issue:3

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Biological Transport; Calcium; Calmodulin; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dinitrophenols; Diuretics; Enzyme Inhibitors; Epithelial Cells; Extracellular Matrix; Furosemide; Imidazoles; Iodoacetates; Kidney Tubules; Opossums; Probenecid; Pyridoxine; Sodium Azide; Tritium; Uncoupling Agents; Uricosuric Agents

2002
Control of hepatocyte DNA synthesis by intracellular pH and its role in the action of tumor promoters.
    Journal of cellular physiology, 2003, Volume: 195, Issue:1

    Topics: Amiloride; Ammonium Chloride; Animals; Bicarbonates; Carcinogens; Cell Division; Cells, Cultured; DNA; Dose-Response Relationship, Drug; Fluoresceins; Fluorescent Dyes; Hepatocytes; HEPES; Hydrogen-Ion Concentration; Insulin; Intracellular Fluid; Ionophores; Male; Monensin; Probenecid; Rats; Rats, Wistar; Sodium-Hydrogen Exchangers

2003