Page last updated: 2024-08-16

proadifen and tamoxifen

proadifen has been researched along with tamoxifen in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19902 (33.33)18.7374
1990's3 (50.00)18.2507
2000's0 (0.00)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kon, OL; Ng, SC; Sim, KY; Teo, CC1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Sutherland, RL; Watts, CK1
Ruenitz, PC; Toledo, MM1
Kupfer, D; Mani, C; Parkinson, A; Pearce, R1
Lennard, MS; Martin, IJ; Tucker, GT; Williams, ML1

Other Studies

6 other study(ies) available for proadifen and tamoxifen

ArticleYear
Synthesis of 2-(p-chlorobenzyl)-3-aryl-6-methoxybenzofurans as selective ligands for antiestrogen-binding sites. Effects on cell proliferation and cholesterol synthesis.
    Journal of medicinal chemistry, 1992, Apr-17, Volume: 35, Issue:8

    Topics: Benzofurans; Binding Sites; Binding, Competitive; Cell Division; Cell Line; Cholesterol; Estrogen Antagonists; Humans; Ligands; Receptors, Estrogen; Thymidine

1992
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Studies on the ligand specificity and potential identity of microsomal antiestrogen-binding sites.
    Molecular pharmacology, 1987, Volume: 31, Issue:5

    Topics: Animals; Breast Neoplasms; Cell Line; Cyclofenil; Estrogen Antagonists; Humans; Microsomes; Nitromifene; Phenothiazines; Proadifen; Rats; Receptors, Drug; Receptors, Estrogen; Stilbenes; Structure-Activity Relationship; Tamoxifen; Xanthines

1987
Inhibition of rabbit liver microsomal oxidative metabolism and substrate binding by tamoxifen and the geometric isomers of clomiphene.
    Biochemical pharmacology, 1980, Jun-01, Volume: 29, Issue:11

    Topics: Animals; Chemical Phenomena; Chemistry; Clomiphene; Depression, Chemical; In Vitro Techniques; Isomerism; Kinetics; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxidation-Reduction; Proadifen; Rabbits; Tamoxifen

1980
Involvement of cytochrome P4503A in catalysis of tamoxifen activation and covalent binding to rat and human liver microsomes.
    Carcinogenesis, 1994, Volume: 15, Issue:12

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Benzimidazoles; Biotransformation; Chickens; Cricetinae; Cytochrome P-450 CYP2E1; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Erythromycin; Female; Humans; Hydrocortisone; Immunoglobulin G; Male; Mesocricetus; Methylcholanthrene; Metyrapone; Mice; Microsomes, Liver; Mixed Function Oxygenases; Phenobarbital; Pregnenolone Carbonitrile; Proadifen; Protein Binding; Rats; Rats, Sprague-Dawley; Species Specificity; Tamoxifen; Troleandomycin

1994
Interindividual variation in the isomerization of 4-hydroxytamoxifen by human liver microsomes: involvement of cytochromes P450.
    Carcinogenesis, 1994, Volume: 15, Issue:12

    Topics: Adult; Biotransformation; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Resistance; Female; Genetic Variation; Humans; Isomerism; Ketoconazole; Male; Microsomes, Liver; Middle Aged; NADP; Proadifen; Tamoxifen

1994