Page last updated: 2024-08-16

proadifen and indomethacin

proadifen has been researched along with indomethacin in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-199011 (35.48)18.7374
1990's11 (35.48)18.2507
2000's7 (22.58)29.6817
2010's2 (6.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Barrow, SE; Hampson, AJ; Rowley, AF; Steadman, R1
Sevanian, A; Zhang, JR1
Kim, HY; Salem, N; Sawazaki, S1
Clark, JE; Harder, DR; Kauser, K; Ma, YH; Masters, BS; Ortiz de Montellano, PR; Roman, RJ1
Nishimura, H; Yamaguchi, K1
Abraham, NG; Mullane, KM; Pinto, A2
Fiera, RA; Matthews, N; Neale, ML1
Hiley, CR; Kay, AP; Randall, MD1
Berlin, T; Larsson, R; Moldéus, P; Olsson, LI; Ross, D1
Selye, H; Solymoss, B; Toth, S; Varga, S1
Gagnon, G; Regoli, D; Rioux, F1
Burke, MD; Falzon, M; Milton, AS1
Berl, T1
Brown, ML; Cohen, RA; Tesfamariam, B1
Kersting, D; Kersting, U; Spring, KR1
Huang, H; Jurima-Romet, M; Paul, CJ; Solomonraj, G; Thomas, BH1
Davis, SC; Edwards, G; Högestätt, ED; Weston, AH; Zygmunt, PM1
Abdul-Karim, RW; Holland, JA; Johnson, DK; Lemanski, LF; Meyer, JW; Patel, V; Sauro, MD; Schillinger, KJ; Schmitt, ME; Small, RF; Ziegler, LM1
Behra, A; Bode-Böger, SM; Böger, RH; Brandes, RP; Lebherz, C; Mügge, A; Phivthong-Ngam, L1
Archuleta, I; Kluger, MJ; Kozak, A; Kozak, W; Mayfield, KP; Rudolph, K1
Chiribiri, A; Gattullo, D; Pagliaro, P; Paolocci, N; Penna, C; Rastaldo, R1
Boels, PJ; Deutsch, J; Gao, B; Haworth, SG1
Bao, S; Christofi, FL; Clanton, TL; Wright, VP; Zuo, L1
Arai, K; Fujii, H; Honda, H; Kanazawa, M; Kogo, H; Moroe, H; Notoya, Y1
Cai, J; Jiang, HD; Xia, Q; Xu, JH; Zhou, XM1
Hosokawa, M; Kamata, K; Kobayashi, T; Matsumoto, T1
Castro-Chaves, P; Fontes-Carvalho, R; Leite-Moreira, AF; Soares, S1
Hayashi, H; Ikehara, O; Kaji, I; Karaki, S; Kuwahara, A; Suzuki, Y; Waguri, T1

Other Studies

31 other study(ies) available for proadifen and indomethacin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Biosynthesis of eicosanoids by blood cells of the crab, Carcinus maenas.
    Biochimica et biophysica acta, 1992, Mar-04, Volume: 1124, Issue:2

    Topics: Animals; Arachidonic Acids; Blood Cells; Brachyura; Calcimycin; Chromatography, High Pressure Liquid; Cyclooxygenase Inhibitors; Eicosanoids; Enzyme Activation; Hemolymph; Hydroxyeicosatetraenoic Acids; Indomethacin; Masoprocol; Proadifen

1992
Effect of vitamin E on arachidonic acid peroxidation and its binding to Chinese hamster V79 cell DNA.
    Biochimica et biophysica acta, 1991, Sep-11, Volume: 1085, Issue:2

    Topics: Animals; Arachidonic Acids; Cell Line; Cricetinae; DNA; Indomethacin; Kinetics; Lipid Metabolism; Lipid Peroxidation; Proadifen; Vitamin E

1991
Lipoxygenation in rat brain?
    Biochemical and biophysical research communications, 1991, Jan-31, Volume: 174, Issue:2

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Arachidonic Acid; Arachidonic Acids; Brain; Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Hydroxyeicosatetraenoic Acids; Indomethacin; Kinetics; Lipoxygenase; Male; Masoprocol; Methoxsalen; Proadifen; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Inbred Strains

1991
Inhibitors of cytochrome P-450 attenuate the myogenic response of dog renal arcuate arteries.
    Circulation research, 1991, Volume: 68, Issue:4

    Topics: Animals; Blood Pressure; Bridged Bicyclo Compounds, Heterocyclic; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Dogs; Fatty Acids, Monounsaturated; Fatty Acids, Unsaturated; Hydrazines; Indomethacin; Ketoconazole; Kinetics; Muscle, Smooth, Vascular; Phospholipases A; Phospholipases A2; Phosphorylcholine; Proadifen; Renal Artery; Triazoles

1991
Angiotensin II-induced relaxation of fowl aorta.
    The American journal of physiology, 1988, Volume: 255, Issue:4 Pt 2

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Angiotensin II; Animals; Aorta, Abdominal; Chickens; Cimetidine; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Indomethacin; Methysergide; Microscopy, Electron; Muscle, Smooth, Vascular; Ouabain; Proadifen; Propranolol; Pyrilamine; Vasodilation

1988
Cytochrome P-450-dependent monooxygenase activity and endothelial-dependent relaxations induced by arachidonic acid.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:2

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Benzoflavones; beta-Naphthoflavone; Blood Vessels; Cobalt; Cytochrome P-450 Enzyme System; Drug Synergism; Endothelium; Fatty Acids; Indomethacin; Male; Methylcholanthrene; Oxygenases; Phenylephrine; Proadifen; Pulmonary Artery; Pyrazoles; Rabbits; Vasoconstriction; Vasodilation

1986
Arachidonic acid-induced endothelial-dependent relaxations of canine coronary arteries: contribution of a cytochrome P-450-dependent pathway.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:3

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Benzoflavones; beta-Naphthoflavone; Coronary Vessels; Cytochrome P-450 Enzyme System; Dinoprost; Dogs; Endothelium; In Vitro Techniques; Indomethacin; Male; Methylcholanthrene; Muscle Contraction; Muscle Relaxation; Proadifen; Prostaglandins F

1987
Involvement of phospholipase A2 activation in tumour cell killing by tumour necrosis factor.
    Immunology, 1988, Volume: 64, Issue:1

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acids; Cell Survival; Dexamethasone; Humans; Indomethacin; Phospholipases; Phospholipases A; Phospholipases A2; Proadifen; Pyrazoles; Quinacrine; Time Factors; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha

1988
Endothelium-dependent modulation of the pressor activity of arginine vasopressin in the isolated superior mesenteric arterial bed of the rat.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arginine Vasopressin; Blood Pressure; Cholic Acids; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Masoprocol; Mesenteric Arteries; Methylene Blue; Muscle, Smooth, Vascular; Proadifen; Pyrazoles; Rats; Rats, Inbred Strains

1988
Prostaglandin synthase catalyzed metabolic activation of p-phenetidine and acetaminophen by microsomes isolated from rabbit and human kidney.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Acetaminophen; Aminophenols; Animals; Arachidonic Acid; Arachidonic Acids; Glutathione; Glutathione Disulfide; Humans; Indomethacin; Kidney; Kinetics; Linolenic Acids; Lipid Peroxides; Male; Metyrapone; Microsomes; Models, Chemical; NADP; Phenetidine; Proadifen; Prostaglandin-Endoperoxide Synthases; Protein Binding; Rabbits

1985
Protection by spironolactone and oxandrolone against chronic digitoxin or indomethacin intoxication.
    Toxicology and applied pharmacology, 1971, Volume: 18, Issue:3

    Topics: Animals; Digitoxin; Drug Antagonism; Female; Indomethacin; Intestinal Diseases; Jejunum; Microsomes, Liver; Mortality; Oxandrolone; Proadifen; Rats; Seizures; Spironolactone; Ulcer

1971
Studies on the mechanism of action of glucagon in strips of rabbit renal artery.
    British journal of pharmacology, 1980, Volume: 69, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium; Cyclic AMP; Female; Glucagon; In Vitro Techniques; Indomethacin; Male; Papaverine; Phosphodiesterase Inhibitors; Proadifen; Rabbits; Renal Artery; Theophylline; Vasodilator Agents; Verapamil

1980
Decreased hepatic microsomal cytochrome P450 due to indomethacin: protective roles of 16,16-dimethylprostaglandin F2 alpha and inducing agents.
    Biochemical pharmacology, 1983, Feb-01, Volume: 32, Issue:3

    Topics: Animals; Cytochrome P-450 Enzyme System; Dinoprost; Enzyme Induction; Indomethacin; Male; Microsomes, Liver; Mixed Function Oxygenases; Proadifen; Prostaglandins F, Synthetic; Rats; Rats, Inbred Strains

1983
Cellular calcium uptake in the action of prostaglandins on renal water excretion.
    Kidney international, 1981, Volume: 19, Issue:1

    Topics: Animals; Biological Transport; Calcium; Cell Membrane Permeability; Diuresis; Dogs; Hemodynamics; Indomethacin; Kidney; Osmolar Concentration; Proadifen; Prostaglandins; Urodynamics; Vasopressins; Verapamil

1981
15-Hydroxyeicosatetraenoic acid and diabetic endothelial dysfunction in rabbit aorta.
    Journal of cardiovascular pharmacology, 1995, Volume: 25, Issue:5

    Topics: Acetylcholine; Animals; Aorta, Abdominal; Bridged Bicyclo Compounds, Heterocyclic; Cytochrome P-450 Enzyme Inhibitors; Diabetes Mellitus, Experimental; Disease Models, Animal; Endothelium, Vascular; Fatty Acids, Unsaturated; Glucose; Hydrazines; Hydroxyeicosatetraenoic Acids; Imidazoles; Indomethacin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Proadifen; Prostaglandin H2; Prostaglandins H; Rabbits; Radioimmunoassay; Superoxide Dismutase; Thromboxane A2

1995
Ketoconazole activates Cl- conductance and blocks Cl- and fluid absorption by cultured cystic fibrosis (CFPAC-1) cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, May-01, Volume: 90, Issue:9

    Topics: Absorption; Cell Line; Cell Membrane; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelium; Humans; Hydrogen-Ion Concentration; Indomethacin; Ion Channels; Ketoconazole; Masoprocol; Membrane Potentials; Membrane Proteins; Proadifen; Thionucleotides; Transfection

1993
Metabolism of phenazopyridine by isolated rat hepatocytes.
    Biopharmaceutics & drug disposition, 1993, Volume: 14, Issue:2

    Topics: Animals; Benzoflavones; Detergents; Enzyme Induction; In Vitro Techniques; Indomethacin; Liver; Male; Metyrapone; Octoxynol; Phenazopyridine; Polyethylene Glycols; Proadifen; Rats; Rats, Wistar

1993
Effects of cytochrome P450 inhibitors on EDHF-mediated relaxation in the rat hepatic artery.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Acetylcholine; Animals; Benzopyrans; Biological Factors; Clotrimazole; Cromakalim; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fatty Acids, Unsaturated; Female; Hepatic Artery; Indomethacin; Membrane Potentials; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Nitroarginine; Potassium Channels; Proadifen; Pyrroles; Rats; Rats, Sprague-Dawley; Vasodilator Agents

1996
Low-density lipoprotein stimulated peroxide production and endocytosis in cultured human endothelial cells: mechanisms of action.
    Endothelium : journal of endothelial cell research, 1997, Volume: 5, Issue:3

    Topics: Acetophenones; Arachidonic Acid; Cells, Cultured; Cholesterol, LDL; Cyclooxygenase Inhibitors; Endocytosis; Endothelium, Vascular; Enzyme Inhibitors; Fatty Acids, Unsaturated; Humans; Hydrogen Peroxide; Indomethacin; Masoprocol; Methoxsalen; NADPH Oxidases; Phospholipases A; Phospholipases A2; Proadifen; Reactive Oxygen Species; Second Messenger Systems; Stimulation, Chemical

1997
N(G)-nitro-L-arginine- and indomethacin-resistant endothelium-dependent relaxation in the rabbit renal artery: effect of hypercholesterolemia.
    Atherosclerosis, 1997, Volume: 135, Issue:1

    Topics: Animals; Aorta, Thoracic; Cholesterol, Dietary; Dose-Response Relationship, Drug; Endothelium, Vascular; Hypercholesterolemia; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroarginine; Proadifen; Quaternary Ammonium Compounds; Rabbits; Renal Artery

1997
Inhibitors of alternative pathways of arachidonate metabolism differentially affect fever in mice.
    The American journal of physiology, 1998, Volume: 275, Issue:4

    Topics: Animals; Antioxidants; Arachidonic Acid; Body Temperature; Body Temperature Regulation; Clotrimazole; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Fever; Indomethacin; Lipopolysaccharides; Lipoxygenase Inhibitors; Male; Masoprocol; Mice; Proadifen; Pyrazoles; Time Factors; Umbelliferones

1998
Cytochrome P-450 metabolite of arachidonic acid mediates bradykinin-induced negative inotropic effect.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:6

    Topics: 8,11,14-Eicosatrienoic Acid; Animals; Arachidonic Acid; Blood Pressure; Bradykinin; Coronary Vessels; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Endothelium, Vascular; Enzyme Inhibitors; Heart; Heart Rate; In Vitro Techniques; Indomethacin; Male; Myocardium; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Octoxynol; Proadifen; Rats; Rats, Wistar; Tachyphylaxis; Triazoles; Ventricular Function, Left

2001
Perinatal development influences mechanisms of bradykinin-induced relaxations in pulmonary resistance and conduit arteries differently.
    Cardiovascular research, 2001, Volume: 51, Issue:1

    Topics: Acetylcholine; Analysis of Variance; Animals; Animals, Newborn; Bradykinin; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Indomethacin; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Proadifen; Pulmonary Artery; Substance P; Swine; Vascular Resistance; Vasodilator Agents

2001
Lipoxygenase-dependent superoxide release in skeletal muscle.
    Journal of applied physiology (Bethesda, Md. : 1985), 2004, Volume: 97, Issue:2

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Arachidonate 12-Lipoxygenase; Arachidonate 5-Lipoxygenase; Arachidonic Acid; Caffeic Acids; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Indomethacin; Lipoxygenase Inhibitors; Male; Muscle, Skeletal; Proadifen; Rats; Rats, Sprague-Dawley; Superoxides

2004
Characterization of endothelium-dependent relaxation and modulation by treatment with pioglitazone in the hypercholesterolemic rabbit renal artery.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Animals; Biological Factors; Charybdotoxin; Endothelium, Vascular; Enzyme Inhibitors; Hypercholesterolemia; Hypoglycemic Agents; Indomethacin; Male; Nitroarginine; Pioglitazone; Potassium Channel Blockers; Proadifen; Rabbits; Renal Artery; Tetraethylammonium; Thiazolidinediones; Time Factors; Vasodilation

2004
Endothelium-dependent and direct relaxation induced by ethyl acetate extract from Flos Chrysanthemi in rat thoracic aorta.
    Journal of ethnopharmacology, 2005, Oct-03, Volume: 101, Issue:1-3

    Topics: Animals; Aorta, Thoracic; Calcium; Calcium Channels; Chrysanthemum; Endothelium, Vascular; Flowers; In Vitro Techniques; Indomethacin; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Plant Extracts; Potassium Channel Blockers; Proadifen; Rats; Rats, Sprague-Dawley; Vasodilation

2005
Altered arachidonic acid-mediated responses in the perfused kidney of the streptozotocin-induced diabetic rat.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2006, Volume: 42, Issue:5

    Topics: Animals; Arachidonic Acid; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Disease Models, Animal; Disease Progression; In Vitro Techniques; Indomethacin; Kidney; Male; Muscle Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth, Vascular; Perfusion; Proadifen; Rats; Rats, Wistar; Regional Blood Flow; Streptozocin

2006
Negative inotropic effect of selective AT2 receptor stimulation and its modulation by the endocardial endothelium.
    European journal of pharmacology, 2008, Jan-14, Volume: 578, Issue:2-3

    Topics: Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Animals; Apamin; Bradykinin; Cardiovascular Agents; Charybdotoxin; Cyclooxygenase Inhibitors; Depression, Chemical; Dose-Response Relationship, Drug; Endocardium; Endothelial Cells; Enzyme Inhibitors; Hydroxocobalamin; Imidazoles; In Vitro Techniques; Indomethacin; Myocardial Contraction; Naphthyridines; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oligopeptides; Papillary Muscles; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Proadifen; Pyridines; Rabbits; Receptor, Angiotensin, Type 2; Receptor, Bradykinin B2; Time Factors

2008
Subepithelial trypsin induces enteric nerve-mediated anion secretion by activating proteinase-activated receptor 1 in the mouse cecum.
    The journal of physiological sciences : JPS, 2012, Volume: 62, Issue:3

    Topics: Animals; Anions; Cecum; Eicosanoids; Enteric Nervous System; Indomethacin; Intestinal Mucosa; Male; Masoprocol; Mice; Oligopeptides; Proadifen; Protease Inhibitors; Receptor, PAR-1; Serotonin; Trypsin

2012