Page last updated: 2024-08-16

proadifen and cimetidine

proadifen has been researched along with cimetidine in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-199012 (60.00)18.7374
1990's2 (10.00)18.2507
2000's3 (15.00)29.6817
2010's3 (15.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Dalvie, D; Hu, Q; Jones, P; Obach, RS; Pryde, DC; Tran, TD1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Nishimura, H; Yamaguchi, K1
Abernathy, CO; Bassan, H; Gillespie, J; Jacob, L; Lukacs, L; Zimmerman, HJ1
Crouch, RK; el-Hage, A; Ferrans, VJ; Herman, EH; Yang, GC1
DeMarco, GJ; Howard, PC; McCoy, GD1
Duddy, SK; Hsia, MT1
Amezcua, JL; GirĂ³n, E; Martinez-Tabche, L; Mourelle, M1
Kuroiwa, Y; Misawa, S; Tanaka, E1
Hall, ST; Houston, JB; Rhodes, JC1
Cummings, AJ; Kaelin, AC1
Christensen, JM; Parrott, KA1
Margolis, S; Schwartz, MA1
Bland, TJ; Robertson, IG1
Berger, BJ; Cerami, A; Dai, WW; Paciorkowski, A1
Doi, H; Horie, T; Iwasaki, H; Masubuchi, Y; Nishigaki, R1
Taira, Z; Ueda, Y; Yamase, D1
Choi, YH; Lee, JH; Lee, MG; Lee, U; Yang, KH1
Ishihara, Y; Ishii, S; Onishi, Y; Sakai, Y; Shimamoto, N; Yamamura, N1

Other Studies

20 other study(ies) available for proadifen and cimetidine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Aldehyde oxidase: an enzyme of emerging importance in drug discovery.
    Journal of medicinal chemistry, 2010, Dec-23, Volume: 53, Issue:24

    Topics: Aldehyde Oxidase; Animals; Drug Discovery; Humans; Models, Molecular; Organ Specificity; Oxidation-Reduction; Pharmaceutical Preparations; Pharmacokinetics; Species Specificity; Substrate Specificity

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Angiotensin II-induced relaxation of fowl aorta.
    The American journal of physiology, 1988, Volume: 255, Issue:4 Pt 2

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Angiotensin II; Animals; Aorta, Abdominal; Chickens; Cimetidine; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Indomethacin; Methysergide; Microscopy, Electron; Muscle, Smooth, Vascular; Ouabain; Proadifen; Propranolol; Pyrilamine; Vasodilation

1988
Effects of H2-blocking agents on hepatocytes in vitro: correlation with potential for causing hepatic disease in patients.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1986, Volume: 182, Issue:4

    Topics: Animals; Aspartate Aminotransferases; Chemical and Drug Induced Liver Injury; Cimetidine; Histamine H2 Antagonists; Humans; Imidazoles; Liver; Male; Proadifen; Ranitidine; Rats; Rats, Inbred Strains

1986
Mechanism of the protective activity of ICRF-187 against alloxan-induced diabetes in mice.
    Research communications in chemical pathology and pharmacology, 1986, Volume: 52, Issue:3

    Topics: Alloxan; Animals; Blood Glucose; Chelating Agents; Cimetidine; Diabetes Mellitus, Experimental; Dimethyl Sulfoxide; Hexobarbital; Hyperglycemia; Male; Mice; Mice, Inbred ICR; Piperazines; Proadifen; Razoxane; Sleep; Stereoisomerism; Superoxide Dismutase

1986
Characterization of hamster liver nicotine metabolism. I. Relative rates of microsomal C and N oxidation.
    Biochemical pharmacology, 1986, Aug-15, Volume: 35, Issue:16

    Topics: Animals; Chromatography, High Pressure Liquid; Cimetidine; Cotinine; Cricetinae; Cyanides; Cysteamine; Male; Mesocricetus; Methylation; Microsomes, Liver; Mixed Function Oxygenases; Nicotine; Oxidation-Reduction; Papain; Peptide Hydrolases; Proadifen

1986
Cytoprotective effects of modulators of oxidative xenobiotic metabolism in precocene II-induced hepatotoxicity.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1987, Volume: 9, Issue:2

    Topics: Alanine Transaminase; Animals; Aspartate Aminotransferases; Benzopyrans; Cell Survival; Chemical and Drug Induced Liver Injury; Cimetidine; Dose-Response Relationship, Drug; Insecticides; Male; Methylcholanthrene; Oxidation-Reduction; Pharmaceutical Preparations; Phenobarbital; Plants; Proadifen; Rats; Rats, Inbred Strains

1987
Cimetidine enhances and phenobarbital decreases parathion toxicity.
    Journal of applied toxicology : JAT, 1986, Volume: 6, Issue:6

    Topics: Animals; Cimetidine; Drug Synergism; Liver; Male; Parathion; Phenobarbital; Proadifen; Rats; Rats, Inbred Strains

1986
Effects of cimetidine and diethylaminoethyl 2,2-diphenylvalerate HCL (SKF 525-A) on trimethadione metabolism in the rat.
    Journal of pharmacobio-dynamics, 1985, Volume: 8, Issue:9

    Topics: Animals; Cimetidine; Cytochrome P-450 Enzyme System; Dimethadione; Kinetics; Liver; Male; Oxazoles; Proadifen; Rats; Rats, Inbred Strains; Trimethadione

1985
Inhibition of antipyrine metabolite formation in rats in vivo.
    Xenobiotica; the fate of foreign compounds in biological systems, 1984, Volume: 14, Issue:9

    Topics: Animals; Antipyrine; Benzoflavones; Cimetidine; Cytochrome P-450 Enzyme System; Male; Metyrapone; Proadifen; Rats; Rats, Inbred Strains

1984
A study of monooxygenase activity in human placental homogenates: in vitro behaviour towards a number of substrates and inhibitors.
    Biochemical pharmacology, 1983, Aug-15, Volume: 32, Issue:16

    Topics: 7-Alkoxycoumarin O-Dealkylase; Cimetidine; Female; Humans; Mixed Function Oxygenases; Oxazoles; Oxygenases; Placenta; Pregnancy; Proadifen

1983
Influence of cimetidine on the disposition of ibuprofen in the rat.
    Research communications in chemical pathology and pharmacology, 1984, Volume: 43, Issue:3

    Topics: Animals; Cimetidine; Drug Interactions; Gastric Mucosa; Hydrogen-Ion Concentration; Ibuprofen; Kinetics; Male; Models, Biological; Proadifen; Rats; Rats, Inbred Strains; Tissue Distribution

1984
Effects of drugs and sterols on cholesterol 7 alpha-hydroxylase activity in rat liver microsomes.
    Journal of lipid research, 1983, Volume: 24, Issue:1

    Topics: Aminoglutethimide; Animals; Ascorbic Acid; Bile Acids and Salts; Cholesterol 7-alpha-Hydroxylase; Cimetidine; Kinetics; Male; Metyrapone; Microsomes, Liver; Proadifen; Rats; Rats, Inbred Strains; Steroid Hydroxylases; Sterols

1983
Inhibition by SKF-525A of the aldehyde oxidase-mediated metabolism of the experimental antitumour agent acridine carboxamide.
    Biochemical pharmacology, 1993, May-25, Volume: 45, Issue:10

    Topics: Acridines; Acridones; Aldehyde Oxidase; Aldehyde Oxidoreductases; Aminoacridines; Amsacrine; Animals; Antineoplastic Agents; Cimetidine; Cytosol; Kinetics; Liver; Male; Methimazole; Metyrapone; Microsomes, Liver; NAD; Proadifen; Rats; Rats, Wistar

1993
Synergism of cimetidine with anti-malarial agents.
    The Journal of parasitology, 1997, Volume: 83, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Drug Resistance; Drug Synergism; Enzyme Inhibitors; Heme; Histamine H2 Antagonists; Plasmodium falciparum; Polymers; Proadifen; Pyrimethamine

1997
Chemiluminescence associated with the oxidative metabolism of salicylic acid in rat liver microsomes.
    Chemico-biological interactions, 2002, May-20, Volume: 140, Issue:2

    Topics: Animals; Biotransformation; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Kinetics; Luminescent Measurements; Male; Microsomes, Liver; NADP; Oxidation-Reduction; Proadifen; Rats; Rats, Wistar; Salicylic Acid; Thiobarbituric Acid Reactive Substances

2002
A new technique for assaying cytochrome P450 enzyme activity in a single cell.
    Cell biology and toxicology, 2007, Volume: 23, Issue:3

    Topics: Animals; Cimetidine; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme System; Enzyme Inhibitors; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Hepatocytes; In Vitro Techniques; Male; Microscopy, Fluorescence; Oxazines; Proadifen; Rats; Rats, Wistar; Spectrometry, Fluorescence

2007
Effects of cytochrome P450 inducers and inhibitors on the pharmacokinetics of intravenous furosemide in rats: involvement of CYP2C11, 2E1, 3A1 and 3A2 in furosemide metabolism.
    The Journal of pharmacy and pharmacology, 2009, Volume: 61, Issue:1

    Topics: Animals; Area Under Curve; Aryl Hydrocarbon Hydroxylases; Cimetidine; Cytochrome P-450 Enzyme System; Diuretics; Drug Interactions; Enzyme Activators; Enzyme Inhibitors; Furosemide; Half-Life; Infusions, Intravenous; Injections, Intravenous; Isoniazid; Male; Methylcholanthrene; Orphenadrine; Proadifen; Quinine; Rats; Rats, Sprague-Dawley; Troleandomycin; Weight Gain

2009
Crucial role of cytochrome P450 in hepatotoxicity induced by 2,3-dimethoxy-1,4-naphthoquinone in rats.
    Journal of applied toxicology : JAT, 2011, Volume: 31, Issue:2

    Topics: alpha-Tocopherol; Animals; Antioxidants; Chemical and Drug Induced Liver Injury; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Glutathione; Ketoconazole; Lipid Peroxidation; Liver; Male; Naphthoquinones; Oxidation-Reduction; Oxidative Stress; Proadifen; Rats; Rats, Wistar; Substrate Cycling

2011