Page last updated: 2024-08-16

primaquine and wr 242511

primaquine has been researched along with wr 242511 in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's6 (66.67)18.2507
2000's1 (11.11)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, EH; Nodiff, EA; Saggiomo, AJ; Tanabe, K1
Queener, SF1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Clavin, AM; Coleman, RE; Milhous, WK1
Appiah, A; Hollingdale, MR; Li, J; Long, GW; McCutchan, TF; Milhous, WK; Zhu, JD1
Fasanmade, AA; Jusko, WJ1
Brewer, TG; Marino, MT; Peggins, JO1
Bartlett, MS; Goheen, MP; Queener, SF; Shaw, MM; Smith, JW1
Armstrong, K; Baskin, S; Briscoe, C; Duniho, S; Gold, M; Kahler, D; Moran, A; Rockwood, G1

Reviews

1 review(s) available for primaquine and wr 242511

ArticleYear
New drug developments for opportunistic infections in immunosuppressed patients: Pneumocystis carinii.
    Journal of medicinal chemistry, 1995, Nov-24, Volume: 38, Issue:24

    Topics: Animals; Drug Design; Humans; Immunosuppression Therapy; Molecular Structure; Opportunistic Infections; Pneumonia, Pneumocystis; Structure-Activity Relationship

1995

Other Studies

8 other study(ies) available for primaquine and wr 242511

ArticleYear
Modifications of primaquine as antimalarials. 4. 5-Alkoxy derivatives of primaquine.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:7

    Topics: Animals; Antimalarials; Malaria; Mice; Primaquine; Structure-Activity Relationship

1987
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Gametocytocidal and sporontocidal activity of antimalarials against Plasmodium berghei ANKA in ICR Mice and Anopheles stephensi mosquitoes.
    The American journal of tropical medicine and hygiene, 1992, Volume: 46, Issue:2

    Topics: Acridines; Aminoquinolines; Analysis of Variance; Animals; Anopheles; Antimalarials; Female; Germ Cells; Guanidines; Imidazoles; Mice; Mice, Inbred ICR; Naphthoquinones; Phenanthrenes; Plasmodium berghei; Primaquine

1992
Plasmodium berghei: quantitation of in vitro effects of antimalarial drugs on exoerythrocytic development by a ribosomal RNA probe.
    Experimental parasitology, 1991, Volume: 72, Issue:4

    Topics: Aminoquinolines; Animals; Antimalarials; Base Sequence; Cells, Cultured; Liver; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Nucleic Acid Hybridization; Plasmodium berghei; Primaquine; Pyrimethamine; RNA Probes; RNA, Protozoan; RNA, Ribosomal

1991
An improved pharmacodynamic model for formation of methemoglobin by antimalarial drugs.
    Drug metabolism and disposition: the biological fate of chemicals, 1995, Volume: 23, Issue:5

    Topics: Absorption; Animals; Antimalarials; Cytochrome-B(5) Reductase; Dogs; Erythrocytes; Mathematical Computing; Methemoglobin; Models, Biological; Primaquine; Reproducibility of Results

1995
High-performance liquid chromatographic method for the determination of a candidate 8-aminoquinoline antimalarial drug (WR 242511) using oxidative electrochemical detection.
    Journal of chromatography, 1993, Jul-02, Volume: 616, Issue:2

    Topics: Animals; Antimalarials; Chromatography, High Pressure Liquid; Dogs; Electrochemistry; Humans; Injections, Intravenous; Oxidation-Reduction; Pilot Projects; Primaquine

1993
Effects of 8-aminoquinolines on the ultrastructural morphology of Pneumocystis carinii.
    International journal of experimental pathology, 1993, Volume: 74, Issue:4

    Topics: Aminoquinolines; Humans; Microscopy, Electron; Pneumocystis; Primaquine

1993
Toxicity in rhesus monkeys following administration of the 8-aminoquinoline 8-[(4-amino-l-methylbutyl)amino]- 5-(l-hexyloxy)-6-methoxy-4-methylquinoline (WR242511).
    Journal of medical toxicology : official journal of the American College of Medical Toxicology, 2008, Volume: 4, Issue:3

    Topics: Animals; Antimalarials; Female; Hemoglobinuria; Immobilization; Kidney; Liver; Lung; Macaca mulatta; Male; Methemoglobin; Myoglobinuria; Primaquine; Solvents

2008