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primaquine and sulfadiazine

primaquine has been researched along with sulfadiazine in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-199020 (64.52)18.7374
1990's2 (6.45)18.2507
2000's4 (12.90)29.6817
2010's5 (16.13)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Genther, CS; Smith, CS1
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Davidson, DE; Hickman, RL; Johnsen, DO; Kinnamon, KE; Tanticharoenyos, P1
Dighe, S; Gurbarg, M; Noory, A; Shah, VP; Skelly, JP1
Powell, RD1
Moxey, PC; Robles, E; Schimmel, EM; Trier, JS1
Carson, PE; Frischer, H; McNamara, JV; Powell, RD; Rieckmann, KH; Stockert, TA1
Dawkins, AT; Stahler, N; Terzian, LA1
Hall, WH; Khan, MY; Zinneman, HH1
Fink, E; Kretschmar, W1
Fink, E1
Cenedella, RJ; Saxe, LH; Van Dyke, K1
Diggens, SM1
Diggens, SM; Gregory, KG1
Gregory, KG; Peters, W1
Dann, O; Fink, E1
Clancy, CF1
Schneider, MD1
Peters, W3
Howells, RE; Judge, BM1
Holfels, E; Mack, D; McAuley, J; McLeod, R; Milhous, WK1
Lewis, BD; López-Rebollar, LM; Penzhorn, BL; Swan, GE1

Reviews

2 review(s) available for primaquine and sulfadiazine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Development of new antimalarial drugs.
    The American journal of tropical medicine and hygiene, 1972, Volume: 21, Issue:5

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance, Microbial; Folic Acid Antagonists; Humans; Malaria; Methanol; Phenanthrenes; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinolines; Research; Sulfadiazine; Sulfonamides; Sulfones; United States

1972

Other Studies

29 other study(ies) available for primaquine and sulfadiazine

ArticleYear
Antifolate studies. Activities of 40 potential antimalarial compounds against sensitive and chlorguanide triazine resistant strains of folate-requiring bacteria and Escherichia coli.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:2

    Topics: Animals; Antimalarials; Bacteria; Drug Resistance, Microbial; Escherichia coli; Folic Acid; Folic Acid Antagonists; Malaria; Mice; Plasmodium berghei; Triazines

1977
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Evaluating new antimalarial drugs against trophozoite induced Plasmodium cynomolgi malaria in rhesus monkeys.
    The American journal of tropical medicine and hygiene, 1976, Volume: 25, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Dapsone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Tolerance; Haplorhini; Macaca mulatta; Malaria; Phenanthrenes; Primaquine; Prodigiosin; Pyrimethamine; Quinine; Sulfadiazine; Sulfadimethoxine; Sulfalene; Trimethoprim

1976
Influence of higher rates of agitation on release patterns of immediate-release drug products.
    Journal of pharmaceutical sciences, 1992, Volume: 81, Issue:6

    Topics: Chloroquine; Griseofulvin; Hydroxychloroquine; Isocarboxazid; Primaquine; Quality Control; Solubility; Sulfadiazine; Tablets

1992
Chronic intestinal coccidiosis in man: intestinal morphology and response to treatment.
    Gastroenterology, 1974, Volume: 66, Issue:5

    Topics: Antiprotozoal Agents; Biopsy; Chloroquine; Chronic Disease; Coccidiosis; Diagnosis, Differential; Diarrhea; Diet Therapy; Drug Therapy, Combination; Duodenum; Follow-Up Studies; Humans; Intestinal Diseases, Parasitic; Intestine, Small; Isospora; Jejunum; Malabsorption Syndromes; Male; Metronidazole; Microscopy, Electron; Middle Aged; Nitrofurantoin; Primaquine; Pyrimethamine; Quinacrine; Sulfadiazine; Tetracycline; Time Factors

1974
Gametocytocidal and sporontocidal effects of primaquine and of sulfadiazine with pyrimethamine in a chloroquine-resistant strain of Plasmodium falciparum.
    Bulletin of the World Health Organization, 1968, Volume: 38, Issue:4

    Topics: Adult; Antimalarials; Drug Resistance, Microbial; Humans; Male; Plasmodium falciparum; Primaquine; Pyrimethamine; Sulfadiazine

1968
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones

1968
Vietnam malaria. Clinical experience with 50 patients.
    Minnesota medicine, 1970, Volume: 53, Issue:3

    Topics: Adult; Chloroquine; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Sulfadiazine; United States; Vietnam

1970
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1970, Volume: 21, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors

1970
[Causal preventive activity of standard antimalarials in rodent malaria (Plasmodium berghei yoelii)].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1972, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Mice; Mice, Inbred Strains; Plasmodium; Primaquine; Pyrimethamine; Quinine; Rodent Diseases; Sulfadiazine

1972
An automated method of mass drug testing applied to screening for antimalarial activity.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones

1970
Single step production of pyrimethamine-resistant P. berghei.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1970, Volume: 64, Issue:1

    Topics: Animals; Cricetinae; Drug Resistance, Microbial; Malaria; Male; Mice; Plasmodium; Primaquine; Pyrimethamine; Sulfadiazine

1970
Drug sensitivity of exo-erythrocytic stages in pyrimethamine-resistant Plasmodium berghei.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1970, Volume: 64, Issue:4

    Topics: Animals; Antimalarials; Drug Resistance, Microbial; Malaria; Male; Mice; Microbial Sensitivity Tests; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Sulfadiazine; Triazines

1970
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines

1970
[Further development of the Roehl test for testing antimalarial agents on Plasmodium cathemerium in the canary by intravenous administration].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1967, Volume: 18, Issue:4

    Topics: Animals; Animals, Laboratory; Antimalarials; Canaries; Chloroquine; Injections, Intravenous; Malaria, Avian; Methods; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfadiazine; Sulfanilamides; Sulfonamides

1967
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
    The American journal of tropical medicine and hygiene, 1968, Volume: 17, Issue:3

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena

1968
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine

1968
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1965
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. II. Triazine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Animals; Dapsone; In Vitro Techniques; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Sulfadiazine; Triazines

1965
Drug responses of mepacrine- and primaquine-resistant strains of Plasmodium berghei Vincke and Lips, 1948.
    Annals of tropical medicine and parasitology, 1966, Volume: 60, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinine; Sulfadiazine

1966
Sustained-release implants in the chemotherapy of experimental rodent malaria I. A comparison of the effects of some antimalarials in polydimethylsiloxane matrices.
    Annals of tropical medicine and parasitology, 1981, Volume: 75, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Dimethylpolysiloxanes; Drug Implants; Malaria; Male; Mefloquine; Mice; Mice, Inbred Strains; Naphthoquinones; Piperidines; Plasmodium berghei; Primaquine; Proguanil; Pyrimethamine; Quinolines; Silicone Elastomers; Sulfadiazine; Triazines

1981
In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:6

    Topics: Animals; Artemisinins; Female; Mefloquine; Mice; Primaquine; Proguanil; Quinine; Sesquiterpenes; Sulfadiazine; Toxoplasma; Triazines; Trifluoperazine; Uracil; Verapamil

1994
Screening of five drugs for efficacy against Babesia felis in experimentally infected cats.
    Journal of the South African Veterinary Association, 2000, Volume: 71, Issue:1

    Topics: Animals; Anti-Infective Agents; Antiprotozoal Agents; Babesiosis; Cat Diseases; Cats; Drug Combinations; Enrofloxacin; Fluoroquinolones; Hematocrit; Naphthoquinones; Parasitemia; Primaquine; Quinolones; Rifampin; Sulfadiazine; Trimethoprim

2000