Page last updated: 2024-08-16

primaquine and quinine

primaquine has been researched along with quinine in 149 studies

Research

Studies (149)

TimeframeStudies, this research(%)All Research%
pre-199091 (61.07)18.7374
1990's15 (10.07)18.2507
2000's18 (12.08)29.6817
2010's22 (14.77)24.3611
2020's3 (2.01)2.80

Authors

AuthorsStudies
Genther, CS; Smith, CS1
Topliss, JG; Yoshida, F1
Galanakis, D; Ganellin, CR1
Lombardo, F; Obach, RS; Waters, NJ1
de L Ferreira, M; de Souza, MV; Kaiser, CR; Lourenço, MC; Pais, KC; Peralta, MA1
Masseno, V; Muriithi, S; Nzila, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Carvalho, L; Castanys, S; Gamarro, F; Manzano, JI; Pérez-Victoria, JM1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Fidock, DA; Flannery, EL; Winzeler, EA1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bellman, K; Knegtel, RM; Settimo, L1
D'hooghe, M; Vandekerckhove, S1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P1
Cheong, SL; Ng, CH; Tibon, NS1
Degrémont, A1
Maier, W; Piekarski, G1
Fradkin, R; Rasco, J; Schmidt, LH; Vaughan, D1
Hall, AP1
Davidson, DE; Hickman, RL; Johnsen, DO; Kinnamon, KE; Tanticharoenyos, P1
Allison, RG; Hahn, FE1
Bradley, DJ; Lumsden, WH; Mackay, DM; Southgate, BA1
Montuori, WA; Most, H1
Mattock, NM; Peters, W1
Back, DJ; Bangchang, KN; Karbwang, J1
Trigg, PI1
Bunnag, D; Harinasuta, T; Karbwang, J; Molunto, P1
Clarke, JB; Kitteringham, NR; Neftel, K; Park, BK1
Sugioka, Y; Suzuki, M1
Pal, NL; Rastogi, M; Sen, AB1
Emerole, GO; Nashiru, TO; Thabrew, MI1
Butler, KW; Deslauriers, R; Smith, IC1
Hioki, A; Ishizaki, T; Nakabayashi, T; Ohtomo, H; Tanabe, K1
Henderson, A; McCallum, J; Melia, W; Navein, J; Simon, J1
Salako, LA1
Chou, SC; Conklin, KA; Pan, HY1
Cowan, GO; Parry, ES1
Chou, SC; Conklin, KA; Heu, P2
Bratton, JL; Cohen, M; Hanson, JP; Hunt, J; Jilek, D; Lohr, DC; Miller, MB; Reynolds, RD1
Ebihara, I; Kimura, M; Komoriya, T; Muto, T; Nakamura, S1
Peters, W5
Miller, A; Natsios, G; Smith, HC1
Alvarez Sotolongo, M; Krácmar, J; Krácmarová, J1
Olatunde, IA1
Deller, JJ1
Weinman, D1
Clyde, DF1
Charoenlarp, P; Harinasuta, T1
Poshyachinda, M; Poshyachinda, V; Siriasawakul, T; Srichaikul, T1
Briesch, PE; Coatney, GR; Collins, WE; Contacos, PG; Jeter, MH1
Saint-Yves, IF1
Charters, AD; Davis, RE1
Ansdell, VE; Boosey, CM; Geddes, AM; Morgan, HV1
Botha, D1
Chou, SC; Conklin, KA2
Collins, WE; Contacos, PG; Howard, WA; Jeffery, GM; Krotoski, WA1
Dawkins, AT; Stahler, N; Terzian, LA1
Altstatt, LB1
Blount, RE1
Martelo, OJ; Saladin, TA; Smoller, M1
Schmidt, LH2
Hall, WH; Khan, MY; Zinneman, HH1
Clyde, DF; McCarthy, VC; Sangalang, RP; Shute, GT1
Clyde, DF; McCarthy, VC; Miller, RM; Music, SI1
Fink, E; Kretschmar, W1
Richards, WH; Williams, SG1
Fink, E1
Miller, A; Smith, HC2
Waser, PG1
Ebisawa, I; Namiki, M1
Ball, EG; Markus, HB1
Wernsdorfer, G; Wernsdorfer, WH1
Cenedella, RJ; Saxe, LH; Van Dyke, K1
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K1
DeWitt Blanton, C; Hargreaves, GW; Latham, MR; Moore, EG; Talati, SM1
Polet, H1
Gregory, KG; Peters, W1
Harley, JD; Naughton, MA; Sietsma, A1
Bishop, A1
Dann, O; Fink, E1
Clancy, CF1
Schneider, MD1
Berberian, DA; Freele, HW; Slighter, RG1
Purcell, WP; Singer, JA1
Herman, R; Most, H; Schoenfeld, C1
Doberstyn, EB1
Ferrante, A; Goh, DH1
Prüfer, L; von Sonnenburg, F1
Ellis-Pegler, RB; Palmer, CW1
Cooke, RA; Shannon, J1
Ferrante, A; Secker, LK; Thong, YH1
Arnold, W; Gahl, GM; Hess, G; Meyer zum Büschenfelde, KH; Möller, B1
Chu, F; Cowman, AF; Gros, P; Karcz, S; Schurr, E; van Es, HH; Vidal, S1
Van den Abbeele, K; Van den Ende, J; Van den Enden, E1
Camargo, LM; Cardoso, MA; Ferreira, MU; Szarfarc, SC1
Holfels, E; Mack, D; McAuley, J; McLeod, R; Milhous, WK1
Corachán, M; Gascon, J; Gomez Arce, JE; Menendez, C; Valls, ME1
Babalola, CP; Bolaji, OO; Dixon, PA; Ogunbona, FA1
Davis, TM; Edwards, G; McGrath, CS; Pukrittayakamee, S; Supanaranond, W; Ward, SA; White, NJ1
Patwari, AK1
Ishizaki, T; Zhao, XJ1
Chang, HL; Chang, SC; Chen, YC; Fang, CT; Hsieh, WC; Hsueh, PR; Hung, CC1
Stephens, I; Wenk, RE1
Adjuik, M; Anto, F; Binka, F; Koram, K; Nkrumah, F; Owusu-Agyei, S; Smith, T1
Andersson, TB; Bapiro, TE; Hasler, JA; Masimirembwa, CM; Otter, C1
Nakajima, Y1
JOSEPH, N; MONTGOMERY, MM; STECK, IE; ZIVIN, S1
ALVING, AS; ARNOLD, J; BEUTLER, E; CLAYMAN, CB; DERN, RJ; FLANAGAN, CL; HOCKWALD, RS1
COLLINS, WE; JEFFERY, GM; SKINNER, JC2
SULLI, G; VARRONE, F1
ZUIDEMA, PJ1
NEELY, JM; PINSWASDI, K; SANDHINAND, U1
Katewa, SD; Katyare, SS2
Aigal, U; Chogle, AR; Dalvi, SS; Gogtay, NJ; Kamtekar, KD; Karnad, DR; Kshirsagar, NA1
Aigal, U; Chogle, AR; Dalvi, SS; Gogtay, NJ; Kamtekar, KD; Kshirsagar, NA1
Baird, JK1
Aigal, U; Chogle, AR; Dalvi, SS; Gogtay, NJ; Kamtekar, KD; Kshirsagar, NA; Mehta, SS1
Chotivanich, K; Coleman, RE; Day, NP; Looareesuwan, S; Sattabongkot, J; Udomsangpetch, R; White, NJ1
Allen, BL; Illamperuma, C1
Akida, JA; Lemnge, MM; Lugimbana, L; Malebo, HM; Malle, LN; Segeja, MD1
Baban, TA; Bouakl, I; Charafeddine, K; Haydoura, S; Kanj, SS; Mazboudi, O; Taher, AT1
Moreira-Campos, LM; Nogueira, FH; Pianetti, GA; Santos, RL1
Barnwell, JW; Collins, WE; Galland, GG; Jeffery, GM; Nace, D; Sullivan, JS; Williams, A; Williams, T1
Garner, P; Gelband, H; Graves, PM3
Bryant, PA; Burgner, D; Kiang, KM; Ladhani, S; Shingadia, D; Steer, AC1
Baird, JK; Basri, H; Ekawati, LL; Elyazar, I; Farrar, J; Meilia, RA; Nurleila, S; Putri, FA; Setiabudy, R; Sudoyo, H; Sutanto, I; Taylor, WR; Tjahjono, B1
Bala, N; Betuela, I; Davis, TM; Hetzel, MW; Lavu, EK; Page-Sharp, M; Pulford, J1
Choi, L; Garner, P; Gelband, H; Graves, PM1
Churcher, ZR; Johnson, PE; Slavkovic, S1
Cumming, BM; Goldring, JPD1
Abichabki, NLM; Abreu-Filho, PG; Baroni, L; Brochi, JCV; de Luca, G; Pereira, LM; Yatsuda, AP1
Shanks, GD1

Reviews

23 review(s) available for primaquine and quinine

ArticleYear
Using genetic methods to define the targets of compounds with antimalarial activity.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum

2013
Quinoline-based antimalarial hybrid compounds.
    Bioorganic & medicinal chemistry, 2015, Aug-15, Volume: 23, Issue:16

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Malaria; Plasmodium; Quinolines

2015
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Current progress in antimalarial pharmacotherapy and multi-target drug discovery.
    European journal of medicinal chemistry, 2020, Feb-15, Volume: 188

    Topics: Animals; Antimalarials; Artemisinins; Drug Discovery; Drug Resistance; Humans; Malaria; Molecular Structure; Paclitaxel; Quinolines

2020
The treatment of malaria.
    British medical journal, 1976, Feb-07, Volume: 1, Issue:6005

    Topics: Anemia; Antimalarials; Blackwater Fever; Child; Child, Preschool; Chloroquine; Coma; Drug Combinations; Drug Resistance, Microbial; Hemorrhage; Humans; Kidney Failure, Chronic; Malaria; Piperidines; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pulmonary Edema; Quinine; Quinolines; Sulfadoxine

1976
Pharmacokinetics of antimalarial drugs: their therapeutic and toxicological implications.
    Annali dell'Istituto superiore di sanita, 1985, Volume: 21, Issue:3

    Topics: Adult; Amodiaquine; Animals; Antimalarials; Child; Chloroquine; Dapsone; Drug Combinations; Drug Resistance, Microbial; Half-Life; Humans; Kinetics; Male; Mefloquine; Mice; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Quinolines; Sulfadoxine; Sulfalene

1985
Recent advances in antimalarial chemotherapy and drug resistance.
    Advances in parasitology, 1974, Volume: 12

    Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones

1974
The present status of chloroquine in the drug treatment of malaria.
    The African journal of medical sciences, 1972, Volume: 3, Issue:1

    Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines

1972
The problem of drug-resistant malaria.
    The American journal of tropical medicine and hygiene, 1972, Volume: 21, Issue:5

    Topics: Amodiaquine; Anopheles; Antimalarials; Asia; Chloroquine; Drug Resistance, Microbial; Humans; Insect Vectors; Malaria; Mutation; Plasmodium falciparum; Primaquine; Proguanil; Quinine; South America; Sulfonamides; Sulfones; Tetracycline; Virulence

1972
Chemotherapy of the drug-resistant malarias.
    Annual review of microbiology, 1969, Volume: 23

    Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones

1969
Malaria. Chemoprophylaxis and chemotherapy.
    British medical journal, 1971, Apr-10, Volume: 2, Issue:5753

    Topics: Amodiaquine; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Drug Synergism; Humans; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Pyrimidines; Quinine; Sulfonamides; Triazines

1971
Resistance of Plasmodium falciparum.
    Experientia, 1984, Dec-15, Volume: 40, Issue:12

    Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America

1984
[Progress in immunodiagnosis and chemotherapy of protozoan infections].
    Der Internist, 1983, Volume: 24, Issue:11

    Topics: Amebiasis; Animals; Antibodies; Babesiosis; Chloroquine; Drug Resistance, Microbial; Giardiasis; Humans; Leishmaniasis; Malaria; Mefloquine; Pneumocystis; Pneumonia, Pneumocystis; Primaquine; Protozoan Infections; Pyrimethamine; Quinine; Quinolines; Serologic Tests; Sulfadoxine; Tetracycline; Toxoplasmosis; Trypanosomiasis

1983
New answers through chemotherapy?
    Experientia, 1984, Dec-15, Volume: 40, Issue:12

    Topics: Aminoquinolines; Animals; Antimalarials; Chemical Phenomena; Chemistry; Disease Models, Animal; Drug Resistance; Drug Therapy, Combination; Erythrocytes; Humans; Liver; Malaria; Mefloquine; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Quinine; Quinolines; Research; Sesquiterpenes; Species Specificity; World Health Organization

1984
Antimalarial drug resistance: an increasing problem.
    British medical bulletin, 1982, Volume: 38, Issue:2

    Topics: Aminoquinolines; Animals; Antimalarials; Aotus trivirgatus; Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Mice; Microbial Sensitivity Tests; Plasmodium; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Triazines

1982
[Antiprotozoal drugs].
    Nihon rinsho. Japanese journal of clinical medicine, 2003, Volume: 61 Suppl 2

    Topics: Animals; Antiprotozoal Agents; Drug Combinations; Emetine; Humans; Mefloquine; Metronidazole; Phenanthrenes; Primaquine; Protozoan Infections; Pyrimethamine; Quinine; Sulfadoxine; Tinidazole

2003
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
    La Clinica terapeutica, 1963, Oct-31, Volume: 27

    Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus

1963
Effectiveness of antimalarial drugs.
    The New England journal of medicine, 2005, Apr-14, Volume: 352, Issue:15

    Topics: Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Life Cycle Stages; Malaria; Mefloquine; Patient Compliance; Plasmodium; Primaquine; Pyrimethamine; Quinine; Secondary Prevention; Sulfadoxine; Treatment Failure

2005
Primaquine for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2012, Sep-12, Issue:9

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2012
The treatment of imported malaria in children: an update.
    Archives of disease in childhood. Education and practice edition, 2013, Volume: 98, Issue:1

    Topics: Administration, Intravenous; Administration, Oral; Adult; Antimalarials; Artemisinins; Child; Drug Therapy, Combination; Endemic Diseases; Humans; Malaria, Falciparum; Malaria, Vivax; Plasmodium falciparum; Plasmodium vivax; Practice Guidelines as Topic; Primaquine; Quinine; United Kingdom

2013
Primaquine or other 8-aminoquinoline for reducing P. falciparum transmission.
    The Cochrane database of systematic reviews, 2014, Jun-30, Issue:6

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2014
Primaquine or other 8-aminoquinoline for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2015, Feb-19, Issue:2

    Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine

2015
Primaquine or other 8-aminoquinolines for reducing Plasmodium falciparum transmission.
    The Cochrane database of systematic reviews, 2018, 02-02, Volume: 2

    Topics: Adult; Antimalarials; Artemisinins; Child; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Non-Randomized Controlled Trials as Topic; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine; Time Factors

2018

Trials

7 trial(s) available for primaquine and quinine

ArticleYear
Characterization of a drug resistant strain of Plasmodium falciparum from the Philippines.
    The Journal of tropical medicine and hygiene, 1971, Volume: 74, Issue:5

    Topics: Adult; Anopheles; Chloroquine; Clinical Trials as Topic; Drug Resistance, Microbial; Humans; Malaria; Male; Philippines; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine

1971
Prophylactic and sporontocidal treatment of chloroquine-resistant Plasmodium falciparum from Vietnam.
    The American journal of tropical medicine and hygiene, 1971, Volume: 20, Issue:1

    Topics: Adult; Antimalarials; Chloroquine; Clinical Trials as Topic; Dapsone; Humans; Malaria; Male; Methemoglobin; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfonamides; United States; Vietnam

1971
Does radical cure of asymptomatic Plasmodium falciparum place adults in endemic areas at increased risk of recurrent symptomatic malaria?
    Tropical medicine & international health : TM & IH, 2002, Volume: 7, Issue:7

    Topics: Adolescent; Adult; Antimalarials; Cohort Studies; Doxycycline; Drug Administration Schedule; Drug Therapy, Combination; Female; Follow-Up Studies; Ghana; Humans; Incidence; Malaria, Falciparum; Male; Middle Aged; Primaquine; Quinine; Recurrence; Risk Assessment; Treatment Outcome

2002
A prospective study evaluating the efficacy of a single, 45-mg dose of primaquine, as a gametocytocidal agent, in patients with Plasmodium falciparum malaria in Mumbai, India.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:5

    Topics: Adolescent; Adult; Aged; Antimalarials; Chloroquine; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Middle Aged; Parasitemia; Primaquine; Prospective Studies; Quinine

2004
Preliminary report of the evaluation of the gametocytocidal action of bulaquine, in adult patients with acute, Plasmodium falciparum malaria.
    Annals of tropical medicine and parasitology, 2004, Volume: 98, Issue:5

    Topics: Acute Disease; Adult; Animals; Antimalarials; Drug Therapy, Combination; Humans; Malaria, Falciparum; Parasitemia; Primaquine; Quinine

2004
A randomized, parallel study of the safety and efficacy of 45 mg primaquine versus 75 mg bulaquine as gametocytocidal agents in adults with blood schizonticide-responsive uncomplicated falciparum malaria [ISCRTN50134587].
    BMC infectious diseases, 2006, Feb-01, Volume: 6

    Topics: Adolescent; Adult; Aged; Animals; Antimalarials; Doxycycline; Drug Administration Schedule; Drug Therapy, Combination; Drug-Related Side Effects and Adverse Reactions; Humans; Malaria, Falciparum; Male; Middle Aged; Parasitemia; Plasmodium falciparum; Primaquine; Quinine; Time Factors; Treatment Outcome

2006
Randomized, open-label trial of primaquine against vivax malaria relapse in Indonesia.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:3

    Topics: Adult; Antimalarials; Artemisinins; Artesunate; Drug Administration Schedule; Drug Dosage Calculations; Drug Resistance; Drug Therapy, Combination; Humans; Indonesia; Malaria; Malaria, Vivax; Male; Military Personnel; Plasmodium vivax; Primaquine; Quinine; Quinolines; Secondary Prevention

2013

Other Studies

119 other study(ies) available for primaquine and quinine

ArticleYear
Antifolate studies. Activities of 40 potential antimalarial compounds against sensitive and chlorguanide triazine resistant strains of folate-requiring bacteria and Escherichia coli.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:2

    Topics: Animals; Antimalarials; Bacteria; Drug Resistance, Microbial; Escherichia coli; Folic Acid; Folic Acid Antagonists; Malaria; Mice; Plasmodium berghei; Triazines

1977
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
    Bioorganic & medicinal chemistry letters, 2004, Aug-02, Volume: 14, Issue:15

    Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Synthesis and in vitro antitubercular activity of a series of quinoline derivatives.
    Bioorganic & medicinal chemistry, 2009, Feb-15, Volume: 17, Issue:4

    Topics: Antitubercular Agents; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Quinolines; Structure-Activity Relationship; Tuberculosis, Multidrug-Resistant

2009
In vitro chemosensitization of Plasmodium falciparum to antimalarials by verapamil and probenecid.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:7

    Topics: Adjuvants, Pharmaceutic; Animals; Antimalarials; Parasitic Sensitivity Tests; Plasmodium falciparum; Probenecid; Verapamil

2009
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Increased glycolytic ATP synthesis is associated with tafenoquine resistance in Leishmania major.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:3

    Topics: Adenosine Triphosphate; Aminoquinolines; Antiprotozoal Agents; Drug Resistance; Glycolysis; Leishmania major; Pyruvate Kinase

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
    Journal of medicinal chemistry, 2019, 04-11, Volume: 62, Issue:7

    Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship

2019
[Biological diagnosis of malaria and amebiasis].
    Schweizerische medizinische Wochenschrift, 1977, May-07, Volume: 107, Issue:18

    Topics: Acetamides; Amebiasis; Chloroquine; Emetine; Entamoeba histolytica; Feces; Humans; Malaria; Methods; Nitroimidazoles; Primaquine; Quinine; Serologic Tests

1977
[Malaria; a summary].
    Immunitat und Infektion, 1978, Volume: 6, Issue:2

    Topics: Chloroquine; Drug Resistance; Humans; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine

1978
Radical cure of infections with Plasmodium cynomolgi: a function of total 8-aminoquinoline dose.
    The American journal of tropical medicine and hygiene, 1977, Volume: 26, Issue:6 Pt 1

    Topics: Aminoquinolines; Animals; Antimalarials; Blood; Chloroquine; Female; Haplorhini; Macaca mulatta; Malaria; Male; Plasmodium; Primaquine; Quinine

1977
Evaluating new antimalarial drugs against trophozoite induced Plasmodium cynomolgi malaria in rhesus monkeys.
    The American journal of tropical medicine and hygiene, 1976, Volume: 25, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Dapsone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Tolerance; Haplorhini; Macaca mulatta; Malaria; Phenanthrenes; Primaquine; Prodigiosin; Pyrimethamine; Quinine; Sulfadiazine; Sulfadimethoxine; Sulfalene; Trimethoprim

1976
Changes in superhelical density of closed circular deoxyribonucleic acid by intercalation of anti-R-plasmid drugs and primaquine.
    Antimicrobial agents and chemotherapy, 1977, Volume: 11, Issue:2

    Topics: Acridines; Chemical Phenomena; Chemistry; Chloroquine; Chlorpromazine; DNA, Circular; Ethidium; Extrachromosomal Inheritance; Methylene Blue; Plasmids; Primaquine; Pseudomonas; Quinine

1977
Letter: Unexplained fever.
    British medical journal, 1975, Feb-15, Volume: 1, Issue:5954

    Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine

1975
Rodent systems (Plasmodium berghei-Anopheles Stephensi) for screening compounds for potential causal prophylaxis.
    The American journal of tropical medicine and hygiene, 1975, Volume: 24, Issue:2

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Drug Evaluation, Preclinical; Female; Malaria; Mice; Plasmodium berghei; Primaquine; Quinine; Quinolines; Rats

1975
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
    Annals of tropical medicine and parasitology, 1975, Volume: 69, Issue:3

    Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin

1975
Mefloquine metabolism by human liver microsomes. Effect of other antimalarial drugs.
    Biochemical pharmacology, 1992, May-08, Volume: 43, Issue:9

    Topics: Biotransformation; Cytochrome P-450 Enzyme Inhibitors; Humans; Ketoconazole; Kinetics; Mefloquine; Microsomes, Liver; Primaquine; Quinine

1992
Drug use and design in the nineties.
    Acta Leidensia, 1991, Volume: 60, Issue:1

    Topics: Aminoquinolines; Amodiaquine; Antimalarials; Artemisinins; Calcium Channel Blockers; Chloroquine; Humans; Malaria; Mefloquine; Naphthoquinones; Phenanthrenes; Primaquine; Quinine; Sesquiterpenes; Sulfadoxine

1991
Plasma quinine levels in patients with falciparum malaria when given alone or in combination with tetracycline with or without primaquine.
    The Southeast Asian journal of tropical medicine and public health, 1991, Volume: 22, Issue:1

    Topics: Adolescent; Adult; Aged; Animals; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Middle Aged; Plasmodium falciparum; Primaquine; Quinine; Tetracycline; Thailand

1991
Detection of antidrug IgG antibodies in patients with adverse drug reactions to amodiaquine.
    International archives of allergy and applied immunology, 1991, Volume: 95, Issue:4

    Topics: Adult; Aged; Amodiaquine; Antibodies, Anti-Idiotypic; Chloroquine; Dose-Response Relationship, Immunologic; Drug Hypersensitivity; Enzyme-Linked Immunosorbent Assay; Female; Humans; Immunoglobulin G; Malaria; Male; Middle Aged; Neutropenia; Primaquine; Quinine

1991
The chemical basis for the ferriprotoporphyrin IX-chloroquine complex induced lipid peroxidation.
    Biochimica et biophysica acta, 1991, May-24, Volume: 1074, Issue:1

    Topics: Animals; Antimalarials; Apoproteins; Benzoates; Benzoic Acid; Catalase; Chloroquine; Hemin; Hydrogen-Ion Concentration; Iron; Kinetics; Lipid Peroxidation; Liposomes; Mefloquine; Oxygen; Primaquine; Quinine; Rats; Spectrum Analysis; Superoxide Dismutase; Transferrin

1991
Gametocytocidal and sporontocidal activity of some standard antimalarials on P. berghei (NK 65) infection M. natalensis.
    Indian journal of malariology, 1989, Volume: 26, Issue:1

    Topics: Animals; Disease Models, Animal; Female; Malaria; Muridae; Plasmodium berghei; Primaquine; Pyrimethamine; Quinine

1989
Drug induced alterations in some rat hepatic microsomal components: a comparative study of four structurally different antimalarials.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1985, Volume: 81, Issue:1

    Topics: Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Antimalarials; Aryl Hydrocarbon Hydroxylases; Chloroquine; Cholesterol; Cytosol; Glutathione Transferase; Liver; Male; Microsomes, Liver; Phospholipids; Primaquine; Quinacrine; Quinine; Rats; Rats, Inbred Strains

1985
Effects of antimalarial drugs on oxygen consumption by erythrocytes infected with Plasmodium berghei: an ESR study.
    Magnetic resonance in medicine, 1986, Volume: 3, Issue:2

    Topics: Animals; Antimalarials; Depression, Chemical; Electron Spin Resonance Spectroscopy; Erythrocytes; Malaria; Male; Mice; Oxygen Consumption; Plasmodium berghei; Primaquine; Quinacrine; Quinine

1986
Clinical evaluation of antimalarial regimens in Japan.
    Zentralblatt fur Bakteriologie, Mikrobiologie, und Hygiene. Series A, Medical microbiology, infectious diseases, virology, parasitology, 1987, Volume: 264, Issue:3-4

    Topics: Animals; Antimalarials; Chloroquine; Drug Therapy, Combination; Humans; Japan; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Prognosis; Pyrimethamine; Quinine; Recurrence; Sulfonamides; Surveys and Questionnaires

1987
Polyresistant malaria in Gurkha soldiers returning from Papua New Guinea: treatment and prevention.
    Journal of the Royal Army Medical Corps, 1986, Volume: 132, Issue:1

    Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Ethnicity; Hong Kong; Humans; Malaria; Male; Military Personnel; Nepal; Oxytetracycline; Papua New Guinea; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Quinine; United Kingdom

1986
Effects of antimalarial drugs and clofibrate on in vitro lipid synthesis in Tetrahymena pyriformis GL.
    Pharmacology, 1974, Volume: 12, Issue:1

    Topics: Acetates; Adenosine Triphosphate; Carbon Radioisotopes; Cell Division; Cell-Free System; Chloroquine; Chromatography, Thin Layer; Clofibrate; Depression, Chemical; Fatty Acids, Nonesterified; Lipids; NADH, NADPH Oxidoreductases; Phospholipids; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Tetrahymena pyriformis; Triglycerides

1974
Choroquine-resistant Plasmodium falciparum malaria in the United Kingdom.
    Lancet (London, England), 1968, Nov-02, Volume: 2, Issue:7575

    Topics: Adult; Chloroquine; England; Humans; Malaria; Malaysia; Male; Penicillin Resistance; Penicillins; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Sulfonamides

1968
Drug-resistant malaria.
    Lancet (London, England), 1969, Jun-21, Volume: 1, Issue:7608

    Topics: Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfonamides

1969
The effects of antimalarial drugs on nucleic acid synthesis in vitro in Tetrahymena pyriformis.
    Molecular pharmacology, 1973, Volume: 9, Issue:3

    Topics: Animals; Antimalarials; Cell Nucleus; Chloroquine; Dactinomycin; DNA; DNA Nucleotidyltransferases; DNA-Directed RNA Polymerases; Dose-Response Relationship, Drug; Guanosine Triphosphate; Primaquine; Quinine; RNA; Tetrahymena pyriformis; Tritium

1973
Experience with mixed infections of Plasmodium falciparum and vivax.
    Military medicine, 1973, Volume: 138, Issue:9

    Topics: Antimalarials; Chloroquine; Dapsone; Humans; Malaria; Military Medicine; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine; Sulfisoxazole; United States; Vietnam

1973
[Prevention and treatment of malaria. 1. Analysis of 73 cases of malaria in Japan].
    Kansenshogaku zasshi. The Journal of the Japanese Association for Infectious Diseases, 1973, Volume: 47, Issue:11

    Topics: Adult; Chloroquine; Humans; Japan; Malaria; Middle Aged; Primaquine; Quinine

1973
Effect of antimalarial drugs on the efflux of K+ from Streptococcus pyogenes.
    Biochemical pharmacology, 1971, Volume: 20, Issue:11

    Topics: Antimalarials; Biological Transport; Cell Membrane Permeability; Chloroquine; Culture Media; Potassium; Potassium Isotopes; Primaquine; Quinacrine; Quinine; Streptococcus pneumoniae; Streptococcus pyogenes

1971
[UV-spectrophotometry in drug control. 14. Characterization and determination of drugs with quinoline and isoquinoline chromophores].
    Die Pharmazie, 1974, Volume: 29, Issue:12

    Topics: Amodiaquine; Chloroquine; Hydroxychloroquine; Isoquinolines; Papaverine; Primaquine; Quinidine; Quinine; Quinolines; Spectrophotometry, Ultraviolet

1974
Malaria--again a diagnostic consideration.
    American family physician, 1972, Volume: 5, Issue:2

    Topics: Chloroquine; Diagnosis, Differential; Erythrocytes; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine

1972
Malaria.
    Disease-a-month : DM, 1972

    Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Fluorescent Antibody Technique; Humans; Immunoglobulins; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Quinine

1972
Relapses of vivax malaria after a conventional course of primaquine and chloroquine: report of 2 cases.
    The Southeast Asian journal of tropical medicine and public health, 1973, Volume: 4, Issue:1

    Topics: Adult; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Glucosephosphate Dehydrogenase; Hemolysis; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Recurrence; Time Factors

1973
Ferrokinetics in patients with malaria: normoblasts and iron incorporation in vitro.
    American journal of clinical pathology, 1973, Volume: 60, Issue:2

    Topics: Adolescent; Adult; Bone Marrow; Bone Marrow Cells; Cell Count; Cells, Cultured; Chloroquine; Erythropoiesis; Female; Humans; In Vitro Techniques; Iron; Iron Isotopes; Malaria; Male; Methods; Middle Aged; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine

1973
Five day primaquine therapy--an evaluation of radical curative activity against vivax malaria infection.
    The American journal of tropical medicine and hygiene, 1973, Volume: 22, Issue:6

    Topics: Chloroquine; Evaluation Studies as Topic; Humans; India; Malaria; Male; Pakistan; Plasmodium vivax; Primaquine; Quinine; Time Factors

1973
The chemotherapy and prophylaxis of malaria.
    The Medical journal of Australia, 1973, Dec-08, Volume: 2, Issue:23

    Topics: Adolescent; Adult; Amodiaquine; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Female; Humans; Infant; Infant, Newborn; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Pregnancy; Primaquine; Proguanil; Quinine

1973
A survey of imported malaria in Western Australia including four cases of drug resistance.
    The Medical journal of Australia, 1974, Apr-06, Volume: 1, Issue:14

    Topics: Adolescent; Adult; Australia; Brain Diseases; Chloroquine; Drug Resistance, Microbial; Emigration and Immigration; Female; Humans; Malaria; Male; Middle Aged; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Quinine; Time Factors; Travel

1974
Malaria in Birmingham 1968-73.
    British medical journal, 1974, Apr-27, Volume: 2, Issue:5912

    Topics: Adult; Africa; Asia; Chloroquinolinols; Disseminated Intravascular Coagulation; England; Female; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Quinine; Thrombocytopenia; Travel

1974
Some pharmacological aspects of antimalarial drugs.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1974, Jun-15, Volume: 48, Issue:29

    Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim

1974
The effects of antimalarial drugs on uptake and incorporation of macromolecular precursors by Tetrahymena pyriformis.
    The Journal of pharmacology and experimental therapeutics, 1972, Volume: 180, Issue:1

    Topics: Amino Acids; Animals; Antimalarials; Carbon Isotopes; Cell Division; Chloroquine; Cycloheximide; Dactinomycin; DNA; Kinetics; Macromolecular Substances; Nalidixic Acid; Primaquine; Quinacrine; Quinine; RNA; Tetrahymena pyriformis; Thymidine; Uridine

1972
Studies on the characterization of plasmodium vivax strains from Central America.
    The American journal of tropical medicine and hygiene, 1972, Volume: 21, Issue:5

    Topics: Animals; Central America; Chloroquine; Haplorhini; Humans; Lincomycin; Malaria; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinine; Recurrence; Time Factors

1972
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones

1968
A clinical view of the biology of Plasmodia.
    Annals of internal medicine, 1969, Volume: 70, Issue:1

    Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine

1969
Acute falciparum malaria. Field experience with quinine-pyrimethamine combined therapy.
    Annals of internal medicine, 1969, Volume: 70, Issue:1

    Topics: Chloroquine; Humans; Malaria; Military Medicine; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine; Vietnam

1969
Malaria in American soldiers.
    Archives of internal medicine, 1969, Volume: 123, Issue:4

    Topics: Anemia, Hemolytic; Blood Cell Count; Carrier State; Chloroquine; Hematocrit; Hemoglobinometry; Hepatitis; Humans; Intestinal Diseases, Parasitic; Leukopenia; Malaria; Military Medicine; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Rupture, Spontaneous; Splenic Rupture; Thrombocytopenia; United States; Vietnam

1969
Vietnam malaria. Clinical experience with 50 patients.
    Minnesota medicine, 1970, Volume: 53, Issue:3

    Topics: Adult; Chloroquine; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Sulfadiazine; United States; Vietnam

1970
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1970, Volume: 21, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors

1970
Action of some antimalaria compounds against Plasmodium berghei in vitro.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1971, Volume: 65, Issue:4

    Topics: Animals; Antimalarials; Chloroquine; Haplorhini; Leucine; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinine; Triazines; Tritium

1971
Quinine: effect of Tetrahymena pyriformis. 3. Energetics of isolated mitochondria in the presence of quinine and other antimalarial drugs.
    Biochemical pharmacology, 1971, Volume: 20, Issue:8

    Topics: Chloroquine; Citrates; Citric Acid Cycle; Depression, Chemical; Fumarates; Glutamates; Hydroxybutyrates; Isocitrates; Ketoglutaric Acids; Malates; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Succinates; Tetrahymena pyriformis; Uncoupling Agents

1971
[Causal preventive activity of standard antimalarials in rodent malaria (Plasmodium berghei yoelii)].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1972, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Mice; Mice, Inbred Strains; Plasmodium; Primaquine; Pyrimethamine; Quinine; Rodent Diseases; Sulfadiazine

1972
The influence of glucose and exogenous glutathione on the red cell membrane effect of the antimalarial drugs 1,4-naphthoquinone and beta-naphthol.
    British journal of haematology, 1971, Volume: 20, Issue:6

    Topics: Cell Membrane; Erythrocytes; Glucose; Glutathione; Hemolysis; Humans; In Vitro Techniques; Methemoglobin; Naphthalenes; Naphthoquinones; Osmotic Fragility; Potassium; Primaquine; Quinacrine; Quinine

1971
[Pharmacogenetics].
    Helvetica medica acta. Supplementum, 1967, May-28, Volume: 47

    Topics: Anemia, Hemolytic; Antipyrine; DNA; Drug-Related Side Effects and Adverse Reactions; Europe; Glucosephosphate Dehydrogenase Deficiency; Glutathione; Humans; Isoniazid; Pharmacogenetics; Phenacetin; Polyneuropathies; Primaquine; Quinine; Racial Groups; Sulfonamides

1967
Imported falciparum malaria with inadequate response to chloroquine.
    The Japanese journal of experimental medicine, 1966, Volume: 36, Issue:6

    Topics: Adult; Ambulatory Care; Chloroquine; Communicable Disease Control; Humans; Japan; Malaria; Male; Plasmodium falciparum; Primaquine; Quinine; Thailand

1966
Inhibition of lipolytic processes in rat adipose tissue by antimalaria drugs.
    Biochimica et biophysica acta, 1969, Dec-17, Volume: 187, Issue:4

    Topics: Adipose Tissue; Animals; Antimalarials; Chloroquine; Epididymis; Fatty Acids; Heparin; Hydroxychloroquine; Lipid Metabolism; Male; Primaquine; Quinacrine; Quinidine; Quinine; Rats

1969
[Symptomatology, diagnosis and therapy of malaria].
    Munchener medizinische Wochenschrift (1950), 1969, Aug-01, Volume: 111, Issue:31

    Topics: Chloroquine; Diagnosis, Differential; Erythrocytes; Humans; Malaria; Plasmodium; Primaquine; Quinine

1969
An automated method of mass drug testing applied to screening for antimalarial activity.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones

1970
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium

1970
Synthesis of potential antimalarials: primaquine analogs.
    Journal of pharmaceutical sciences, 1970, Volume: 59, Issue:4

    Topics: Animals; Antimalarials; Chemical Phenomena; Chemistry; Chickens; Chloroquine; Chromatography, Thin Layer; Infrared Rays; Methods; Mice; Primaquine; Quinine; Quinolines; Spectrophotometry

1970
Influence of sucrose on chloroquine-3-H3 content of mammalian cells in vitro: the possible role of lysosomes in chloroquine resistance.
    The Journal of pharmacology and experimental therapeutics, 1970, Volume: 173, Issue:1

    Topics: Animals; Carbon Isotopes; Cell Line; Chloroquine; Cold Temperature; Cricetinae; Culture Techniques; Drug Resistance, Microbial; HeLa Cells; Hexoses; Hydrogen-Ion Concentration; Kidney; Lysosomes; Pinocytosis; Plasmodium; Primaquine; Quinacrine; Quinine; Sucrose; Tritium

1970
The intracellular and membrane effects of oxidant agents on normal red cells.
    British journal of haematology, 1970, Volume: 19, Issue:3

    Topics: Cell Membrane; Erythrocytes; Glutathione; Heinz Bodies; Hemoglobinometry; Hemolysis; Humans; Hydroquinones; Hydroxylamines; Naphthoquinones; Osmotic Fragility; Oxidation-Reduction; Phenols; Phenylhydrazines; Potassium; Primaquine; Quinacrine; Quinine

1970
Antimalarials: effects on in vivo and in vitro protein synthesis.
    Science (New York, N.Y.), 1970, Dec-11, Volume: 170, Issue:3963

    Topics: Amino Acids; Antimalarials; Carbon Isotopes; Cell-Free System; Chloroquine; Cycloheximide; Primaquine; Protein Biosynthesis; Quinacrine; Quinine; Tetrahymena

1970
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines

1970
Methaemoglobin levels in soldiers receiving antimalarial drugs.
    The Medical journal of Australia, 1971, Feb-27, Volume: 1, Issue:9

    Topics: Antimalarials; Australia; Chloroquine; Dapsone; Erythrocyte Count; Humans; Methemoglobin; Military Personnel; Primaquine; Pyrimethamine; Quinine; Reticulocytes; Vietnam

1971
Resistance to primaquine in Plasmodium gallinaceum, and the problem of resistance to quinoline compounds in malaria parasites.
    Parasitology, 1967, Volume: 57, Issue:4

    Topics: Aedes; Animals; Chickens; Chloroquine; Drug Resistance, Microbial; Malaria, Avian; Primaquine; Quinacrine; Quinine; Quinolines

1967
[Further development of the Roehl test for testing antimalarial agents on Plasmodium cathemerium in the canary by intravenous administration].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1967, Volume: 18, Issue:4

    Topics: Animals; Animals, Laboratory; Antimalarials; Canaries; Chloroquine; Injections, Intravenous; Malaria, Avian; Methods; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfadiazine; Sulfanilamides; Sulfonamides

1967
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
    The American journal of tropical medicine and hygiene, 1968, Volume: 17, Issue:3

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena

1968
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine

1968
Causal prophylactic effect of Menoctone (a new hydroxynaphthoquinone) against sporozoite-induced Plasmodium berghei infection in mice.
    The Journal of parasitology, 1968, Volume: 54, Issue:6

    Topics: Animals; Antimalarials; Chloroquine; Cricetinae; Malaria; Mice; Naphthoquinones; Plasmodium; Primaquine; Quinine

1968
Drug responses of mepacrine- and primaquine-resistant strains of Plasmodium berghei Vincke and Lips, 1948.
    Annals of tropical medicine and parasitology, 1966, Volume: 60, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinine; Sulfadiazine

1966
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
    Journal of medicinal chemistry, 1967, Volume: 10, Issue:5

    Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA

1967
Chemotherapy of sporozoite- and blood-induced Plasmodium berghei infections with selected antimalarial agents.
    The American journal of tropical medicine and hygiene, 1967, Volume: 16, Issue:5

    Topics: Animals; Chloroquine; Cricetinae; Dapsone; Malaria; Mice; Primaquine; Pyrimethamine; Quinine; Rats

1967
The effect of anti-malarial drugs on human natural killer cells in vitro.
    Parasite immunology, 1984, Volume: 6, Issue:6

    Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines

1984
Imported malaria in adults in Auckland.
    The New Zealand medical journal, 1982, Dec-08, Volume: 95, Issue:721

    Topics: Adolescent; Adult; Chloroquine; Drug Resistance, Microbial; Female; Humans; Kenya; Malaria; Male; Middle Aged; New Zealand; Papua New Guinea; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Splenomegaly; Time Factors; Travel

1982
Malaria in southeast Queensland in 1979.
    The Medical journal of Australia, 1980, Dec-13, Volume: 2, Issue:12

    Topics: Adolescent; Adult; Australia; Child; Child, Preschool; Chloroquine; Dapsone; Female; Humans; Infant; Infant, Newborn; Malaria; Male; Middle Aged; New Guinea; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine; Sulfadoxine; Tinnitus; Vietnam

1980
Comparative efficacies of quinine and chloroquine as companions to primaquine in a curative drug regimen.
    The American journal of tropical medicine and hygiene, 1981, Volume: 30, Issue:1

    Topics: Animals; Chloroquine; Drug Administration Schedule; Drug Therapy, Combination; Macaca mulatta; Malaria; Primaquine; Quinine

1981
Normal immunological responses in mice treated with chloroquine, quinine and primaquine.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1981, Volume: 75, Issue:1

    Topics: Animals; Antibody Formation; Chloroquine; Drug Administration Schedule; Immunity, Cellular; Male; Mice; Mice, Inbred BALB C; Primaquine; Quinine

1981
Inhibition of hepatitis B virus specific DNA polymerase by intercalating agents.
    Medical microbiology and immunology, 1980, Volume: 168, Issue:1

    Topics: Carrier State; Chloroquine; DNA-Directed DNA Polymerase; Ethidium; Hepatitis B; Hepatitis B Antigens; Hepatitis B virus; Humans; Intercalating Agents; Magnesium; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine; Quinine

1980
Expression of the plasmodial pfmdr1 gene in mammalian cells is associated with increased susceptibility to chloroquine.
    Molecular and cellular biology, 1994, Volume: 14, Issue:4

    Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Base Sequence; Biological Transport; Cell Survival; Chloroquine; CHO Cells; Colchicine; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; DNA, Protozoan; Doxorubicin; Drug Resistance; Female; Gene Expression; Genes, Protozoan; Membrane Proteins; Oligonucleotides, Antisense; Oocytes; Plasmodium falciparum; Primaquine; Protozoan Proteins; Quinine; Restriction Mapping; Verapamil; Vinblastine; Xenopus laevis

1994
Combined chloroquine and primaquine resistant Plasmodium vivax malaria in a patient returning from India.
    Annales de la Societe belge de medecine tropicale, 1995, Volume: 75, Issue:1

    Topics: Adult; Chloroquine; Drug Resistance; Drug Therapy, Combination; Female; Humans; Malaria, Vivax; Primaquine; Quinine; Recurrence

1995
Anaemia, iron deficiency and malaria in a rural community in Brazilian Amazon.
    European journal of clinical nutrition, 1994, Volume: 48, Issue:5

    Topics: Adolescent; Adult; Anemia, Hemolytic, Autoimmune; Anemia, Hypochromic; Animals; Brazil; Child; Child, Preschool; Chloroquine; Cross-Sectional Studies; Female; Ferrous Compounds; Hemoglobinometry; Humans; Incidence; Infant; Intestinal Diseases, Parasitic; Malaria; Male; Mebendazole; Plasmodium falciparum; Plasmodium vivax; Population Surveillance; Pregnancy; Primaquine; Quinine; Rural Population

1994
In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:6

    Topics: Animals; Artemisinins; Female; Mefloquine; Mice; Primaquine; Proguanil; Quinine; Sesquiterpenes; Sulfadiazine; Toxoplasma; Triazines; Trifluoperazine; Uracil; Verapamil

1994
Poor response to primaquine in two cases of Plasmodium vivax malaria from Guatemala.
    Tropical and geographical medicine, 1994, Volume: 46, Issue:1

    Topics: Chloroquine; Drug Resistance; Drug Therapy, Combination; Guatemala; Humans; Malaria, Vivax; Male; Primaquine; Quinine

1994
Column liquid chromatographic analysis of quinine in human plasma, saliva and urine.
    Journal of chromatography, 1993, Jun-23, Volume: 616, Issue:1

    Topics: Chromatography, High Pressure Liquid; Humans; Indicators and Reagents; Primaquine; Quinidine; Quinine; Saliva; Spectrophotometry, Ultraviolet

1993
Interactions among primaquine, malaria infection and other antimalarials in Thai subjects.
    British journal of clinical pharmacology, 1993, Volume: 35, Issue:2

    Topics: Acute Disease; Administration, Oral; Adult; Drug Interactions; Humans; Malaria, Falciparum; Male; Mefloquine; Primaquine; Quinine; Thailand

1993
A standard regimen for treatment of plasmodium vivax malaria.
    Indian pediatrics, 1996, Volume: 33, Issue:9

    Topics: Antimalarials; Humans; Infant; Malaria, Cerebral; Malaria, Falciparum; Malaria, Vivax; Primaquine; Quinine

1996
Metabolic interactions of selected antimalarial and non-antimalarial drugs with the major pathway (3-hydroxylation) of quinine in human liver microsomes.
    British journal of clinical pharmacology, 1997, Volume: 44, Issue:5

    Topics: Anti-Infective Agents; Antimalarials; Chromatography; Cytochrome P-450 Enzyme System; Doxycycline; Drug Interactions; Erythromycin; Humans; Hydroxylation; Ketoconazole; Microsomes, Liver; Nifedipine; Omeprazole; Primaquine; Quinine; Tetracycline; Troleandomycin

1997
Imported malaria: successful treatment of 31 patients in the era of chloroquine resistance.
    Journal of the Formosan Medical Association = Taiwan yi zhi, 1999, Volume: 98, Issue:10

    Topics: Adolescent; Adult; Antimalarials; Artemisinins; Artesunate; Child; Chloroquine; Drug Resistance; Female; Humans; Malaria; Male; Middle Aged; Primaquine; Quinine; Retrospective Studies; Sesquiterpenes; Travel

1999
Erythrocyte Fy antigen phenotyping helps differentiate so-called benign tertian malarias.
    Archives of pathology & laboratory medicine, 2000, Volume: 124, Issue:2

    Topics: Animals; Child, Preschool; Diagnosis, Differential; Drug Therapy, Combination; Duffy Blood-Group System; Erythrocytes; Humans; Immunophenotyping; Malaria; Male; Plasmodium; Primaquine; Quinine; Tetracycline

2000
Cytochrome P450 1A1/2 induction by antiparasitic drugs: dose-dependent increase in ethoxyresorufin O-deethylase activity and mRNA caused by quinine, primaquine and albendazole in HepG2 cells.
    European journal of clinical pharmacology, 2002, Volume: 58, Issue:8

    Topics: Albendazole; Antiparasitic Agents; Cell Survival; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Dose-Response Relationship, Drug; Enzyme Induction; Humans; Polychlorinated Dibenzodioxins; Primaquine; Quinine; RNA, Messenger; Tumor Cells, Cultured

2002
Influence of primaquine on the clinical findings and joint potentials in rheumatoid arthritis.
    Annals of the rheumatic diseases, 1952, Volume: 11, Issue:4

    Topics: Arthritis; Arthritis, Rheumatoid; Humans; Joints; Primaquine; Quinine

1952
Potentiation of the curative action of primaquine in vivax malaria by quinine and chloroquine.
    The Journal of laboratory and clinical medicine, 1955, Volume: 46, Issue:2

    Topics: Antimalarials; Chloroquine; Humans; Malaria; Malaria, Vivax; Primaquine; Quinine

1955
ANTIMALARIAL DRUG TRIALS ON A MULTIRESISTANT STRAIN OF PLASMODIUM FALCIPARUM.
    The American journal of tropical medicine and hygiene, 1963, Volume: 12

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Thailand

1963
FLUORESCENT ANTIBODY STUDIES IN HUMAN MALARIA. II. DEVELOPMENT AND PERSISTENCE OF ANTIBODIES TO PLASMODIUM FALCIPARUM.
    The American journal of tropical medicine and hygiene, 1964, Volume: 13

    Topics: Amodiaquine; Antibodies; Antigen-Antibody Reactions; Chloroquine; Fluorescent Antibody Technique; Humans; Immune Sera; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinine; Vaccination

1964
[A PATIENT WITH TROPICAL MALARIA].
    Nederlands tijdschrift voor geneeskunde, 1964, Jan-18, Volume: 108

    Topics: Amodiaquine; Antimalarials; Chloroquine; Dosage Forms; Drug Resistance; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Primaquine; Quinine

1964
CHLOROQUINE-RESISTANT STRAIN OF PLASMODIUM FALCIPARUM FROM KHAO MAI KHAEO, THAILAND.
    The American journal of tropical medicine and hygiene, 1965, Volume: 14

    Topics: Chloroquine; Drug Resistance; Drug Resistance, Microbial; Drug Therapy; Humans; Malaria; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Thailand

1965
ARMY giving primaquine treatment to all returning servicemen.
    Public health reports (Washington, D.C. : 1896), 1952, Volume: 67, Issue:2

    Topics: Humans; Malaria; Primaquine; Quinine

1952
PRIMAQUINE 15 mg. for 14 days cures "high percentage".
    Public health reports (Washington, D.C. : 1896), 1952, Volume: 67, Issue:2

    Topics: Humans; Malaria; Primaquine; Quinine

1952
Treatment with antimalarials adversely affects the oxidative energy metabolism in rat liver mitochondria.
    Drug and chemical toxicology, 2004, Volume: 27, Issue:1

    Topics: Adenosine Triphosphatases; Animals; Antimalarials; Chloroquine; Cytochromes; Energy Metabolism; Male; Mitochondria, Liver; Oxidative Phosphorylation; Primaquine; Quinine; Rats; Rats, Inbred Strains

2004
Antimalarials inhibit human erythrocyte membrane acetylcholinesterase.
    Drug and chemical toxicology, 2005, Volume: 28, Issue:4

    Topics: Acetylcholinesterase; Adult; Antimalarials; Chloroquine; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocyte Membrane; Female; Humans; Kinetics; Male; Middle Aged; Primaquine; Quinine

2005
Transmission-blocking activities of quinine, primaquine, and artesunate.
    Antimicrobial agents and chemotherapy, 2006, Volume: 50, Issue:6

    Topics: Animals; Anopheles; Antimalarials; Artemisinins; Artesunate; Disease Vectors; Dose-Response Relationship, Drug; In Vitro Techniques; Life Cycle Stages; Parasite Egg Count; Plasmodium falciparum; Primaquine; Quinine; Sesquiterpenes

2006
Pulmonary edema due to Plasmodium vivax malaria in an American missionary.
    Infection, 2007, Volume: 35, Issue:5

    Topics: Animals; Antimalarials; Doxycycline; Humans; Malaria, Vivax; Male; Middle Aged; Missionaries; Plasmodium vivax; Primaquine; Pulmonary Edema; Quinine; Radiography, Thoracic; Religious Missions; Uganda

2007
A simple technique for the detection of anti-malarial drug formulations and their presence in human urine.
    Tanzania health research bulletin, 2006, Volume: 8, Issue:3

    Topics: Amodiaquine; Antimalarials; Biological Assay; Biological Availability; Chloroquine; Chromatography, Thin Layer; Fraud; Humans; Malaria; Primaquine; Product Surveillance, Postmarketing; Pyrimethamine; Quality Control; Quinine; Sulfadoxine

2006
Transfusion-related Plasmodium ovale malaria complicated by acute respiratory distress syndrome (ARDS) in a non-endemic country.
    Parasitology international, 2011, Volume: 60, Issue:1

    Topics: Antimalarials; Doxycycline; Female; Humans; Intensive Care Units; Malaria; Middle Aged; Plasmodium ovale; Platelet Transfusion; Primaquine; Quinine; Respiratory Distress Syndrome

2011
Quality of essential drugs in tropical countries: evaluation of antimalarial drugs in the Brazilian Health System.
    Revista da Sociedade Brasileira de Medicina Tropical, 2011, Volume: 44, Issue:5

    Topics: Antimalarials; Brazil; Chloroquine; Chromatography, High Pressure Liquid; Drug Storage; Drugs, Essential; Humans; Mefloquine; Primaquine; Quality Control; Quinine

2011
Mosquito infection studies with Aotus monkeys and humans infected with the Chesson strain of Plasmodiun vivax.
    The American journal of tropical medicine and hygiene, 2012, Volume: 86, Issue:3

    Topics: Animals; Anopheles; Antimalarials; Aotidae; Chloroquine; Disease Management; Disease Models, Animal; Host-Parasite Interactions; Humans; Malaria; Male; Monkey Diseases; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinine

2012
Quality of antimalarial drugs and antibiotics in Papua New Guinea: a survey of the health facility supply chain.
    PloS one, 2014, Volume: 9, Issue:5

    Topics: Amodiaquine; Amoxicillin; Antimalarials; Artemether; Artemisinins; Biosimilar Pharmaceuticals; Chloroquine; Drug Resistance; Health Facilities; Humans; Malaria, Falciparum; Malaria, Vivax; Papua New Guinea; Primaquine; Quality Control; Quinine

2014
Nanomolar binding affinity of quinine-based antimalarial compounds by the cocaine-binding aptamer.
    Bioorganic & medicinal chemistry, 2018, 11-01, Volume: 26, Issue:20

    Topics: Amodiaquine; Antimalarials; Aptamers, Nucleotide; Binding Sites; Chloroquine; Cocaine; Ligands; Mefloquine; Primaquine; Quinine; Thermodynamics

2018
Monocyte phagocytosis of malaria β-haematin in the presence of artemisinin, amodiaquine, chloroquine, doxycycline, primaquine, pyrimethamine and quinine.
    Experimental parasitology, 2019, Volume: 197

    Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Cell Count; Cell Line; Chloroquine; Doxycycline; Electron Probe Microanalysis; Heme; Hemeproteins; Humans; Leukocytes, Mononuclear; Mice; Microscopy, Electron, Scanning; Microscopy, Electron, Transmission; Monocytes; Peroxidase; Phagocytosis; Primaquine; Pyrimethamine; Quinine; Spectrophotometry; Temperature; U937 Cells

2019
Atovaquone, chloroquine, primaquine, quinine and tetracycline: antiproliferative effects of relevant antimalarials on Neospora caninum.
    Revista brasileira de parasitologia veterinaria = Brazilian journal of veterinary parasitology : Orgao Oficial do Colegio Brasileiro de Parasitologia Veterinaria, 2021, Volume: 30, Issue:1

    Topics: Antimalarials; Atovaquone; Chloroquine; Neospora; Primaquine; Quinine; Tetracyclines

2021
Historical 8-Aminoquinoline Combinations: Not All Antimalarial Drugs Work Well Together.
    The American journal of tropical medicine and hygiene, 2022, 11-14, Volume: 107, Issue:5

    Topics: Aminoquinolines; Antimalarials; Chloroquine; Hemolysis; Humans; Primaquine; Quinine

2022