primaquine has been researched along with quinine in 149 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 91 (61.07) | 18.7374 |
1990's | 15 (10.07) | 18.2507 |
2000's | 18 (12.08) | 29.6817 |
2010's | 22 (14.77) | 24.3611 |
2020's | 3 (2.01) | 2.80 |
Authors | Studies |
---|---|
Genther, CS; Smith, CS | 1 |
Topliss, JG; Yoshida, F | 1 |
Galanakis, D; Ganellin, CR | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
de L Ferreira, M; de Souza, MV; Kaiser, CR; Lourenço, MC; Pais, KC; Peralta, MA | 1 |
Masseno, V; Muriithi, S; Nzila, A | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Carvalho, L; Castanys, S; Gamarro, F; Manzano, JI; Pérez-Victoria, JM | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Fidock, DA; Flannery, EL; Winzeler, EA | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Bellman, K; Knegtel, RM; Settimo, L | 1 |
D'hooghe, M; Vandekerckhove, S | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P | 1 |
Cheong, SL; Ng, CH; Tibon, NS | 1 |
Degrémont, A | 1 |
Maier, W; Piekarski, G | 1 |
Fradkin, R; Rasco, J; Schmidt, LH; Vaughan, D | 1 |
Hall, AP | 1 |
Davidson, DE; Hickman, RL; Johnsen, DO; Kinnamon, KE; Tanticharoenyos, P | 1 |
Allison, RG; Hahn, FE | 1 |
Bradley, DJ; Lumsden, WH; Mackay, DM; Southgate, BA | 1 |
Montuori, WA; Most, H | 1 |
Mattock, NM; Peters, W | 1 |
Back, DJ; Bangchang, KN; Karbwang, J | 1 |
Trigg, PI | 1 |
Bunnag, D; Harinasuta, T; Karbwang, J; Molunto, P | 1 |
Clarke, JB; Kitteringham, NR; Neftel, K; Park, BK | 1 |
Sugioka, Y; Suzuki, M | 1 |
Pal, NL; Rastogi, M; Sen, AB | 1 |
Emerole, GO; Nashiru, TO; Thabrew, MI | 1 |
Butler, KW; Deslauriers, R; Smith, IC | 1 |
Hioki, A; Ishizaki, T; Nakabayashi, T; Ohtomo, H; Tanabe, K | 1 |
Henderson, A; McCallum, J; Melia, W; Navein, J; Simon, J | 1 |
Salako, LA | 1 |
Chou, SC; Conklin, KA; Pan, HY | 1 |
Cowan, GO; Parry, ES | 1 |
Chou, SC; Conklin, KA; Heu, P | 2 |
Bratton, JL; Cohen, M; Hanson, JP; Hunt, J; Jilek, D; Lohr, DC; Miller, MB; Reynolds, RD | 1 |
Ebihara, I; Kimura, M; Komoriya, T; Muto, T; Nakamura, S | 1 |
Peters, W | 5 |
Miller, A; Natsios, G; Smith, HC | 1 |
Alvarez Sotolongo, M; Krácmar, J; Krácmarová, J | 1 |
Olatunde, IA | 1 |
Deller, JJ | 1 |
Weinman, D | 1 |
Clyde, DF | 1 |
Charoenlarp, P; Harinasuta, T | 1 |
Poshyachinda, M; Poshyachinda, V; Siriasawakul, T; Srichaikul, T | 1 |
Briesch, PE; Coatney, GR; Collins, WE; Contacos, PG; Jeter, MH | 1 |
Saint-Yves, IF | 1 |
Charters, AD; Davis, RE | 1 |
Ansdell, VE; Boosey, CM; Geddes, AM; Morgan, HV | 1 |
Botha, D | 1 |
Chou, SC; Conklin, KA | 2 |
Collins, WE; Contacos, PG; Howard, WA; Jeffery, GM; Krotoski, WA | 1 |
Dawkins, AT; Stahler, N; Terzian, LA | 1 |
Altstatt, LB | 1 |
Blount, RE | 1 |
Martelo, OJ; Saladin, TA; Smoller, M | 1 |
Schmidt, LH | 2 |
Hall, WH; Khan, MY; Zinneman, HH | 1 |
Clyde, DF; McCarthy, VC; Sangalang, RP; Shute, GT | 1 |
Clyde, DF; McCarthy, VC; Miller, RM; Music, SI | 1 |
Fink, E; Kretschmar, W | 1 |
Richards, WH; Williams, SG | 1 |
Fink, E | 1 |
Miller, A; Smith, HC | 2 |
Waser, PG | 1 |
Ebisawa, I; Namiki, M | 1 |
Ball, EG; Markus, HB | 1 |
Wernsdorfer, G; Wernsdorfer, WH | 1 |
Cenedella, RJ; Saxe, LH; Van Dyke, K | 1 |
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K | 1 |
DeWitt Blanton, C; Hargreaves, GW; Latham, MR; Moore, EG; Talati, SM | 1 |
Polet, H | 1 |
Gregory, KG; Peters, W | 1 |
Harley, JD; Naughton, MA; Sietsma, A | 1 |
Bishop, A | 1 |
Dann, O; Fink, E | 1 |
Clancy, CF | 1 |
Schneider, MD | 1 |
Berberian, DA; Freele, HW; Slighter, RG | 1 |
Purcell, WP; Singer, JA | 1 |
Herman, R; Most, H; Schoenfeld, C | 1 |
Doberstyn, EB | 1 |
Ferrante, A; Goh, DH | 1 |
Prüfer, L; von Sonnenburg, F | 1 |
Ellis-Pegler, RB; Palmer, CW | 1 |
Cooke, RA; Shannon, J | 1 |
Ferrante, A; Secker, LK; Thong, YH | 1 |
Arnold, W; Gahl, GM; Hess, G; Meyer zum Büschenfelde, KH; Möller, B | 1 |
Chu, F; Cowman, AF; Gros, P; Karcz, S; Schurr, E; van Es, HH; Vidal, S | 1 |
Van den Abbeele, K; Van den Ende, J; Van den Enden, E | 1 |
Camargo, LM; Cardoso, MA; Ferreira, MU; Szarfarc, SC | 1 |
Holfels, E; Mack, D; McAuley, J; McLeod, R; Milhous, WK | 1 |
Corachán, M; Gascon, J; Gomez Arce, JE; Menendez, C; Valls, ME | 1 |
Babalola, CP; Bolaji, OO; Dixon, PA; Ogunbona, FA | 1 |
Davis, TM; Edwards, G; McGrath, CS; Pukrittayakamee, S; Supanaranond, W; Ward, SA; White, NJ | 1 |
Patwari, AK | 1 |
Ishizaki, T; Zhao, XJ | 1 |
Chang, HL; Chang, SC; Chen, YC; Fang, CT; Hsieh, WC; Hsueh, PR; Hung, CC | 1 |
Stephens, I; Wenk, RE | 1 |
Adjuik, M; Anto, F; Binka, F; Koram, K; Nkrumah, F; Owusu-Agyei, S; Smith, T | 1 |
Andersson, TB; Bapiro, TE; Hasler, JA; Masimirembwa, CM; Otter, C | 1 |
Nakajima, Y | 1 |
JOSEPH, N; MONTGOMERY, MM; STECK, IE; ZIVIN, S | 1 |
ALVING, AS; ARNOLD, J; BEUTLER, E; CLAYMAN, CB; DERN, RJ; FLANAGAN, CL; HOCKWALD, RS | 1 |
COLLINS, WE; JEFFERY, GM; SKINNER, JC | 2 |
SULLI, G; VARRONE, F | 1 |
ZUIDEMA, PJ | 1 |
NEELY, JM; PINSWASDI, K; SANDHINAND, U | 1 |
Katewa, SD; Katyare, SS | 2 |
Aigal, U; Chogle, AR; Dalvi, SS; Gogtay, NJ; Kamtekar, KD; Karnad, DR; Kshirsagar, NA | 1 |
Aigal, U; Chogle, AR; Dalvi, SS; Gogtay, NJ; Kamtekar, KD; Kshirsagar, NA | 1 |
Baird, JK | 1 |
Aigal, U; Chogle, AR; Dalvi, SS; Gogtay, NJ; Kamtekar, KD; Kshirsagar, NA; Mehta, SS | 1 |
Chotivanich, K; Coleman, RE; Day, NP; Looareesuwan, S; Sattabongkot, J; Udomsangpetch, R; White, NJ | 1 |
Allen, BL; Illamperuma, C | 1 |
Akida, JA; Lemnge, MM; Lugimbana, L; Malebo, HM; Malle, LN; Segeja, MD | 1 |
Baban, TA; Bouakl, I; Charafeddine, K; Haydoura, S; Kanj, SS; Mazboudi, O; Taher, AT | 1 |
Moreira-Campos, LM; Nogueira, FH; Pianetti, GA; Santos, RL | 1 |
Barnwell, JW; Collins, WE; Galland, GG; Jeffery, GM; Nace, D; Sullivan, JS; Williams, A; Williams, T | 1 |
Garner, P; Gelband, H; Graves, PM | 3 |
Bryant, PA; Burgner, D; Kiang, KM; Ladhani, S; Shingadia, D; Steer, AC | 1 |
Baird, JK; Basri, H; Ekawati, LL; Elyazar, I; Farrar, J; Meilia, RA; Nurleila, S; Putri, FA; Setiabudy, R; Sudoyo, H; Sutanto, I; Taylor, WR; Tjahjono, B | 1 |
Bala, N; Betuela, I; Davis, TM; Hetzel, MW; Lavu, EK; Page-Sharp, M; Pulford, J | 1 |
Choi, L; Garner, P; Gelband, H; Graves, PM | 1 |
Churcher, ZR; Johnson, PE; Slavkovic, S | 1 |
Cumming, BM; Goldring, JPD | 1 |
Abichabki, NLM; Abreu-Filho, PG; Baroni, L; Brochi, JCV; de Luca, G; Pereira, LM; Yatsuda, AP | 1 |
Shanks, GD | 1 |
23 review(s) available for primaquine and quinine
Article | Year |
---|---|
Using genetic methods to define the targets of compounds with antimalarial activity.
Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum | 2013 |
Quinoline-based antimalarial hybrid compounds.
Topics: Animals; Antimalarials; Drug Discovery; Humans; Malaria; Plasmodium; Quinolines | 2015 |
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Current progress in antimalarial pharmacotherapy and multi-target drug discovery.
Topics: Animals; Antimalarials; Artemisinins; Drug Discovery; Drug Resistance; Humans; Malaria; Molecular Structure; Paclitaxel; Quinolines | 2020 |
The treatment of malaria.
Topics: Anemia; Antimalarials; Blackwater Fever; Child; Child, Preschool; Chloroquine; Coma; Drug Combinations; Drug Resistance, Microbial; Hemorrhage; Humans; Kidney Failure, Chronic; Malaria; Piperidines; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pulmonary Edema; Quinine; Quinolines; Sulfadoxine | 1976 |
Pharmacokinetics of antimalarial drugs: their therapeutic and toxicological implications.
Topics: Adult; Amodiaquine; Animals; Antimalarials; Child; Chloroquine; Dapsone; Drug Combinations; Drug Resistance, Microbial; Half-Life; Humans; Kinetics; Male; Mefloquine; Mice; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Quinolines; Sulfadoxine; Sulfalene | 1985 |
Recent advances in antimalarial chemotherapy and drug resistance.
Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones | 1974 |
The present status of chloroquine in the drug treatment of malaria.
Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines | 1972 |
The problem of drug-resistant malaria.
Topics: Amodiaquine; Anopheles; Antimalarials; Asia; Chloroquine; Drug Resistance, Microbial; Humans; Insect Vectors; Malaria; Mutation; Plasmodium falciparum; Primaquine; Proguanil; Quinine; South America; Sulfonamides; Sulfones; Tetracycline; Virulence | 1972 |
Chemotherapy of the drug-resistant malarias.
Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones | 1969 |
Malaria. Chemoprophylaxis and chemotherapy.
Topics: Amodiaquine; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Drug Synergism; Humans; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Pyrimidines; Quinine; Sulfonamides; Triazines | 1971 |
Resistance of Plasmodium falciparum.
Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America | 1984 |
[Progress in immunodiagnosis and chemotherapy of protozoan infections].
Topics: Amebiasis; Animals; Antibodies; Babesiosis; Chloroquine; Drug Resistance, Microbial; Giardiasis; Humans; Leishmaniasis; Malaria; Mefloquine; Pneumocystis; Pneumonia, Pneumocystis; Primaquine; Protozoan Infections; Pyrimethamine; Quinine; Quinolines; Serologic Tests; Sulfadoxine; Tetracycline; Toxoplasmosis; Trypanosomiasis | 1983 |
New answers through chemotherapy?
Topics: Aminoquinolines; Animals; Antimalarials; Chemical Phenomena; Chemistry; Disease Models, Animal; Drug Resistance; Drug Therapy, Combination; Erythrocytes; Humans; Liver; Malaria; Mefloquine; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Quinine; Quinolines; Research; Sesquiterpenes; Species Specificity; World Health Organization | 1984 |
Antimalarial drug resistance: an increasing problem.
Topics: Aminoquinolines; Animals; Antimalarials; Aotus trivirgatus; Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Mice; Microbial Sensitivity Tests; Plasmodium; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Triazines | 1982 |
[Antiprotozoal drugs].
Topics: Animals; Antiprotozoal Agents; Drug Combinations; Emetine; Humans; Mefloquine; Metronidazole; Phenanthrenes; Primaquine; Protozoan Infections; Pyrimethamine; Quinine; Sulfadoxine; Tinidazole | 2003 |
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus | 1963 |
Effectiveness of antimalarial drugs.
Topics: Animals; Antimalarials; Chloroquine; Drug Combinations; Drug Resistance; Drug Therapy, Combination; Humans; Life Cycle Stages; Malaria; Mefloquine; Patient Compliance; Plasmodium; Primaquine; Pyrimethamine; Quinine; Secondary Prevention; Sulfadoxine; Treatment Failure | 2005 |
Primaquine for reducing Plasmodium falciparum transmission.
Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine | 2012 |
The treatment of imported malaria in children: an update.
Topics: Administration, Intravenous; Administration, Oral; Adult; Antimalarials; Artemisinins; Child; Drug Therapy, Combination; Endemic Diseases; Humans; Malaria, Falciparum; Malaria, Vivax; Plasmodium falciparum; Plasmodium vivax; Practice Guidelines as Topic; Primaquine; Quinine; United Kingdom | 2013 |
Primaquine or other 8-aminoquinoline for reducing P. falciparum transmission.
Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine | 2014 |
Primaquine or other 8-aminoquinoline for reducing Plasmodium falciparum transmission.
Topics: Antimalarials; Artemisinins; Artesunate; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine | 2015 |
Primaquine or other 8-aminoquinolines for reducing Plasmodium falciparum transmission.
Topics: Adult; Antimalarials; Artemisinins; Child; Chloroquine; Drug Combinations; Glucosephosphate Dehydrogenase Deficiency; Humans; Malaria, Falciparum; Mefloquine; Non-Randomized Controlled Trials as Topic; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Randomized Controlled Trials as Topic; Sulfadoxine; Time Factors | 2018 |
7 trial(s) available for primaquine and quinine
Article | Year |
---|---|
Characterization of a drug resistant strain of Plasmodium falciparum from the Philippines.
Topics: Adult; Anopheles; Chloroquine; Clinical Trials as Topic; Drug Resistance, Microbial; Humans; Malaria; Male; Philippines; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine | 1971 |
Prophylactic and sporontocidal treatment of chloroquine-resistant Plasmodium falciparum from Vietnam.
Topics: Adult; Antimalarials; Chloroquine; Clinical Trials as Topic; Dapsone; Humans; Malaria; Male; Methemoglobin; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfonamides; United States; Vietnam | 1971 |
Does radical cure of asymptomatic Plasmodium falciparum place adults in endemic areas at increased risk of recurrent symptomatic malaria?
Topics: Adolescent; Adult; Antimalarials; Cohort Studies; Doxycycline; Drug Administration Schedule; Drug Therapy, Combination; Female; Follow-Up Studies; Ghana; Humans; Incidence; Malaria, Falciparum; Male; Middle Aged; Primaquine; Quinine; Recurrence; Risk Assessment; Treatment Outcome | 2002 |
A prospective study evaluating the efficacy of a single, 45-mg dose of primaquine, as a gametocytocidal agent, in patients with Plasmodium falciparum malaria in Mumbai, India.
Topics: Adolescent; Adult; Aged; Antimalarials; Chloroquine; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Malaria, Falciparum; Male; Middle Aged; Parasitemia; Primaquine; Prospective Studies; Quinine | 2004 |
Preliminary report of the evaluation of the gametocytocidal action of bulaquine, in adult patients with acute, Plasmodium falciparum malaria.
Topics: Acute Disease; Adult; Animals; Antimalarials; Drug Therapy, Combination; Humans; Malaria, Falciparum; Parasitemia; Primaquine; Quinine | 2004 |
A randomized, parallel study of the safety and efficacy of 45 mg primaquine versus 75 mg bulaquine as gametocytocidal agents in adults with blood schizonticide-responsive uncomplicated falciparum malaria [ISCRTN50134587].
Topics: Adolescent; Adult; Aged; Animals; Antimalarials; Doxycycline; Drug Administration Schedule; Drug Therapy, Combination; Drug-Related Side Effects and Adverse Reactions; Humans; Malaria, Falciparum; Male; Middle Aged; Parasitemia; Plasmodium falciparum; Primaquine; Quinine; Time Factors; Treatment Outcome | 2006 |
Randomized, open-label trial of primaquine against vivax malaria relapse in Indonesia.
Topics: Adult; Antimalarials; Artemisinins; Artesunate; Drug Administration Schedule; Drug Dosage Calculations; Drug Resistance; Drug Therapy, Combination; Humans; Indonesia; Malaria; Malaria, Vivax; Male; Military Personnel; Plasmodium vivax; Primaquine; Quinine; Quinolines; Secondary Prevention | 2013 |
119 other study(ies) available for primaquine and quinine
Article | Year |
---|---|
Antifolate studies. Activities of 40 potential antimalarial compounds against sensitive and chlorguanide triazine resistant strains of folate-requiring bacteria and Escherichia coli.
Topics: Animals; Antimalarials; Bacteria; Drug Resistance, Microbial; Escherichia coli; Folic Acid; Folic Acid Antagonists; Malaria; Mice; Plasmodium berghei; Triazines | 1977 |
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated | 2004 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Synthesis and in vitro antitubercular activity of a series of quinoline derivatives.
Topics: Antitubercular Agents; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Quinolines; Structure-Activity Relationship; Tuberculosis, Multidrug-Resistant | 2009 |
In vitro chemosensitization of Plasmodium falciparum to antimalarials by verapamil and probenecid.
Topics: Adjuvants, Pharmaceutic; Animals; Antimalarials; Parasitic Sensitivity Tests; Plasmodium falciparum; Probenecid; Verapamil | 2009 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
Increased glycolytic ATP synthesis is associated with tafenoquine resistance in Leishmania major.
Topics: Adenosine Triphosphate; Aminoquinolines; Antiprotozoal Agents; Drug Resistance; Glycolysis; Leishmania major; Pyruvate Kinase | 2011 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation | 2014 |
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship | 2019 |
[Biological diagnosis of malaria and amebiasis].
Topics: Acetamides; Amebiasis; Chloroquine; Emetine; Entamoeba histolytica; Feces; Humans; Malaria; Methods; Nitroimidazoles; Primaquine; Quinine; Serologic Tests | 1977 |
[Malaria; a summary].
Topics: Chloroquine; Drug Resistance; Humans; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine | 1978 |
Radical cure of infections with Plasmodium cynomolgi: a function of total 8-aminoquinoline dose.
Topics: Aminoquinolines; Animals; Antimalarials; Blood; Chloroquine; Female; Haplorhini; Macaca mulatta; Malaria; Male; Plasmodium; Primaquine; Quinine | 1977 |
Evaluating new antimalarial drugs against trophozoite induced Plasmodium cynomolgi malaria in rhesus monkeys.
Topics: Amodiaquine; Animals; Antimalarials; Dapsone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Tolerance; Haplorhini; Macaca mulatta; Malaria; Phenanthrenes; Primaquine; Prodigiosin; Pyrimethamine; Quinine; Sulfadiazine; Sulfadimethoxine; Sulfalene; Trimethoprim | 1976 |
Changes in superhelical density of closed circular deoxyribonucleic acid by intercalation of anti-R-plasmid drugs and primaquine.
Topics: Acridines; Chemical Phenomena; Chemistry; Chloroquine; Chlorpromazine; DNA, Circular; Ethidium; Extrachromosomal Inheritance; Methylene Blue; Plasmids; Primaquine; Pseudomonas; Quinine | 1977 |
Letter: Unexplained fever.
Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine | 1975 |
Rodent systems (Plasmodium berghei-Anopheles Stephensi) for screening compounds for potential causal prophylaxis.
Topics: Animals; Anopheles; Antimalarials; Chloroquine; Drug Evaluation, Preclinical; Female; Malaria; Mice; Plasmodium berghei; Primaquine; Quinine; Quinolines; Rats | 1975 |
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin | 1975 |
Mefloquine metabolism by human liver microsomes. Effect of other antimalarial drugs.
Topics: Biotransformation; Cytochrome P-450 Enzyme Inhibitors; Humans; Ketoconazole; Kinetics; Mefloquine; Microsomes, Liver; Primaquine; Quinine | 1992 |
Drug use and design in the nineties.
Topics: Aminoquinolines; Amodiaquine; Antimalarials; Artemisinins; Calcium Channel Blockers; Chloroquine; Humans; Malaria; Mefloquine; Naphthoquinones; Phenanthrenes; Primaquine; Quinine; Sesquiterpenes; Sulfadoxine | 1991 |
Plasma quinine levels in patients with falciparum malaria when given alone or in combination with tetracycline with or without primaquine.
Topics: Adolescent; Adult; Aged; Animals; Drug Resistance; Drug Therapy, Combination; Humans; Malaria, Falciparum; Middle Aged; Plasmodium falciparum; Primaquine; Quinine; Tetracycline; Thailand | 1991 |
Detection of antidrug IgG antibodies in patients with adverse drug reactions to amodiaquine.
Topics: Adult; Aged; Amodiaquine; Antibodies, Anti-Idiotypic; Chloroquine; Dose-Response Relationship, Immunologic; Drug Hypersensitivity; Enzyme-Linked Immunosorbent Assay; Female; Humans; Immunoglobulin G; Malaria; Male; Middle Aged; Neutropenia; Primaquine; Quinine | 1991 |
The chemical basis for the ferriprotoporphyrin IX-chloroquine complex induced lipid peroxidation.
Topics: Animals; Antimalarials; Apoproteins; Benzoates; Benzoic Acid; Catalase; Chloroquine; Hemin; Hydrogen-Ion Concentration; Iron; Kinetics; Lipid Peroxidation; Liposomes; Mefloquine; Oxygen; Primaquine; Quinine; Rats; Spectrum Analysis; Superoxide Dismutase; Transferrin | 1991 |
Gametocytocidal and sporontocidal activity of some standard antimalarials on P. berghei (NK 65) infection M. natalensis.
Topics: Animals; Disease Models, Animal; Female; Malaria; Muridae; Plasmodium berghei; Primaquine; Pyrimethamine; Quinine | 1989 |
Drug induced alterations in some rat hepatic microsomal components: a comparative study of four structurally different antimalarials.
Topics: Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Antimalarials; Aryl Hydrocarbon Hydroxylases; Chloroquine; Cholesterol; Cytosol; Glutathione Transferase; Liver; Male; Microsomes, Liver; Phospholipids; Primaquine; Quinacrine; Quinine; Rats; Rats, Inbred Strains | 1985 |
Effects of antimalarial drugs on oxygen consumption by erythrocytes infected with Plasmodium berghei: an ESR study.
Topics: Animals; Antimalarials; Depression, Chemical; Electron Spin Resonance Spectroscopy; Erythrocytes; Malaria; Male; Mice; Oxygen Consumption; Plasmodium berghei; Primaquine; Quinacrine; Quinine | 1986 |
Clinical evaluation of antimalarial regimens in Japan.
Topics: Animals; Antimalarials; Chloroquine; Drug Therapy, Combination; Humans; Japan; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Prognosis; Pyrimethamine; Quinine; Recurrence; Sulfonamides; Surveys and Questionnaires | 1987 |
Polyresistant malaria in Gurkha soldiers returning from Papua New Guinea: treatment and prevention.
Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Ethnicity; Hong Kong; Humans; Malaria; Male; Military Personnel; Nepal; Oxytetracycline; Papua New Guinea; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Quinine; United Kingdom | 1986 |
Effects of antimalarial drugs and clofibrate on in vitro lipid synthesis in Tetrahymena pyriformis GL.
Topics: Acetates; Adenosine Triphosphate; Carbon Radioisotopes; Cell Division; Cell-Free System; Chloroquine; Chromatography, Thin Layer; Clofibrate; Depression, Chemical; Fatty Acids, Nonesterified; Lipids; NADH, NADPH Oxidoreductases; Phospholipids; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Tetrahymena pyriformis; Triglycerides | 1974 |
Choroquine-resistant Plasmodium falciparum malaria in the United Kingdom.
Topics: Adult; Chloroquine; England; Humans; Malaria; Malaysia; Male; Penicillin Resistance; Penicillins; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Sulfonamides | 1968 |
Drug-resistant malaria.
Topics: Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfonamides | 1969 |
The effects of antimalarial drugs on nucleic acid synthesis in vitro in Tetrahymena pyriformis.
Topics: Animals; Antimalarials; Cell Nucleus; Chloroquine; Dactinomycin; DNA; DNA Nucleotidyltransferases; DNA-Directed RNA Polymerases; Dose-Response Relationship, Drug; Guanosine Triphosphate; Primaquine; Quinine; RNA; Tetrahymena pyriformis; Tritium | 1973 |
Experience with mixed infections of Plasmodium falciparum and vivax.
Topics: Antimalarials; Chloroquine; Dapsone; Humans; Malaria; Military Medicine; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine; Sulfisoxazole; United States; Vietnam | 1973 |
[Prevention and treatment of malaria. 1. Analysis of 73 cases of malaria in Japan].
Topics: Adult; Chloroquine; Humans; Japan; Malaria; Middle Aged; Primaquine; Quinine | 1973 |
Effect of antimalarial drugs on the efflux of K+ from Streptococcus pyogenes.
Topics: Antimalarials; Biological Transport; Cell Membrane Permeability; Chloroquine; Culture Media; Potassium; Potassium Isotopes; Primaquine; Quinacrine; Quinine; Streptococcus pneumoniae; Streptococcus pyogenes | 1971 |
[UV-spectrophotometry in drug control. 14. Characterization and determination of drugs with quinoline and isoquinoline chromophores].
Topics: Amodiaquine; Chloroquine; Hydroxychloroquine; Isoquinolines; Papaverine; Primaquine; Quinidine; Quinine; Quinolines; Spectrophotometry, Ultraviolet | 1974 |
Malaria--again a diagnostic consideration.
Topics: Chloroquine; Diagnosis, Differential; Erythrocytes; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine | 1972 |
Malaria.
Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Fluorescent Antibody Technique; Humans; Immunoglobulins; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Quinine | 1972 |
Relapses of vivax malaria after a conventional course of primaquine and chloroquine: report of 2 cases.
Topics: Adult; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Glucosephosphate Dehydrogenase; Hemolysis; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Recurrence; Time Factors | 1973 |
Ferrokinetics in patients with malaria: normoblasts and iron incorporation in vitro.
Topics: Adolescent; Adult; Bone Marrow; Bone Marrow Cells; Cell Count; Cells, Cultured; Chloroquine; Erythropoiesis; Female; Humans; In Vitro Techniques; Iron; Iron Isotopes; Malaria; Male; Methods; Middle Aged; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine | 1973 |
Five day primaquine therapy--an evaluation of radical curative activity against vivax malaria infection.
Topics: Chloroquine; Evaluation Studies as Topic; Humans; India; Malaria; Male; Pakistan; Plasmodium vivax; Primaquine; Quinine; Time Factors | 1973 |
The chemotherapy and prophylaxis of malaria.
Topics: Adolescent; Adult; Amodiaquine; Child; Child, Preschool; Chloroquine; Drug Resistance, Microbial; Female; Humans; Infant; Infant, Newborn; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Pregnancy; Primaquine; Proguanil; Quinine | 1973 |
A survey of imported malaria in Western Australia including four cases of drug resistance.
Topics: Adolescent; Adult; Australia; Brain Diseases; Chloroquine; Drug Resistance, Microbial; Emigration and Immigration; Female; Humans; Malaria; Male; Middle Aged; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Quinine; Time Factors; Travel | 1974 |
Malaria in Birmingham 1968-73.
Topics: Adult; Africa; Asia; Chloroquinolinols; Disseminated Intravascular Coagulation; England; Female; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Quinine; Thrombocytopenia; Travel | 1974 |
Some pharmacological aspects of antimalarial drugs.
Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim | 1974 |
The effects of antimalarial drugs on uptake and incorporation of macromolecular precursors by Tetrahymena pyriformis.
Topics: Amino Acids; Animals; Antimalarials; Carbon Isotopes; Cell Division; Chloroquine; Cycloheximide; Dactinomycin; DNA; Kinetics; Macromolecular Substances; Nalidixic Acid; Primaquine; Quinacrine; Quinine; RNA; Tetrahymena pyriformis; Thymidine; Uridine | 1972 |
Studies on the characterization of plasmodium vivax strains from Central America.
Topics: Animals; Central America; Chloroquine; Haplorhini; Humans; Lincomycin; Malaria; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinine; Recurrence; Time Factors | 1972 |
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones | 1968 |
A clinical view of the biology of Plasmodia.
Topics: Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine | 1969 |
Acute falciparum malaria. Field experience with quinine-pyrimethamine combined therapy.
Topics: Chloroquine; Humans; Malaria; Military Medicine; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine; Vietnam | 1969 |
Malaria in American soldiers.
Topics: Anemia, Hemolytic; Blood Cell Count; Carrier State; Chloroquine; Hematocrit; Hemoglobinometry; Hepatitis; Humans; Intestinal Diseases, Parasitic; Leukopenia; Malaria; Military Medicine; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Rupture, Spontaneous; Splenic Rupture; Thrombocytopenia; United States; Vietnam | 1969 |
Vietnam malaria. Clinical experience with 50 patients.
Topics: Adult; Chloroquine; Humans; Malaria; Male; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Sulfadiazine; United States; Vietnam | 1970 |
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors | 1970 |
Action of some antimalaria compounds against Plasmodium berghei in vitro.
Topics: Animals; Antimalarials; Chloroquine; Haplorhini; Leucine; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinine; Triazines; Tritium | 1971 |
Quinine: effect of Tetrahymena pyriformis. 3. Energetics of isolated mitochondria in the presence of quinine and other antimalarial drugs.
Topics: Chloroquine; Citrates; Citric Acid Cycle; Depression, Chemical; Fumarates; Glutamates; Hydroxybutyrates; Isocitrates; Ketoglutaric Acids; Malates; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Succinates; Tetrahymena pyriformis; Uncoupling Agents | 1971 |
[Causal preventive activity of standard antimalarials in rodent malaria (Plasmodium berghei yoelii)].
Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Mice; Mice, Inbred Strains; Plasmodium; Primaquine; Pyrimethamine; Quinine; Rodent Diseases; Sulfadiazine | 1972 |
The influence of glucose and exogenous glutathione on the red cell membrane effect of the antimalarial drugs 1,4-naphthoquinone and beta-naphthol.
Topics: Cell Membrane; Erythrocytes; Glucose; Glutathione; Hemolysis; Humans; In Vitro Techniques; Methemoglobin; Naphthalenes; Naphthoquinones; Osmotic Fragility; Potassium; Primaquine; Quinacrine; Quinine | 1971 |
[Pharmacogenetics].
Topics: Anemia, Hemolytic; Antipyrine; DNA; Drug-Related Side Effects and Adverse Reactions; Europe; Glucosephosphate Dehydrogenase Deficiency; Glutathione; Humans; Isoniazid; Pharmacogenetics; Phenacetin; Polyneuropathies; Primaquine; Quinine; Racial Groups; Sulfonamides | 1967 |
Imported falciparum malaria with inadequate response to chloroquine.
Topics: Adult; Ambulatory Care; Chloroquine; Communicable Disease Control; Humans; Japan; Malaria; Male; Plasmodium falciparum; Primaquine; Quinine; Thailand | 1966 |
Inhibition of lipolytic processes in rat adipose tissue by antimalaria drugs.
Topics: Adipose Tissue; Animals; Antimalarials; Chloroquine; Epididymis; Fatty Acids; Heparin; Hydroxychloroquine; Lipid Metabolism; Male; Primaquine; Quinacrine; Quinidine; Quinine; Rats | 1969 |
[Symptomatology, diagnosis and therapy of malaria].
Topics: Chloroquine; Diagnosis, Differential; Erythrocytes; Humans; Malaria; Plasmodium; Primaquine; Quinine | 1969 |
An automated method of mass drug testing applied to screening for antimalarial activity.
Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones | 1970 |
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium | 1970 |
Synthesis of potential antimalarials: primaquine analogs.
Topics: Animals; Antimalarials; Chemical Phenomena; Chemistry; Chickens; Chloroquine; Chromatography, Thin Layer; Infrared Rays; Methods; Mice; Primaquine; Quinine; Quinolines; Spectrophotometry | 1970 |
Influence of sucrose on chloroquine-3-H3 content of mammalian cells in vitro: the possible role of lysosomes in chloroquine resistance.
Topics: Animals; Carbon Isotopes; Cell Line; Chloroquine; Cold Temperature; Cricetinae; Culture Techniques; Drug Resistance, Microbial; HeLa Cells; Hexoses; Hydrogen-Ion Concentration; Kidney; Lysosomes; Pinocytosis; Plasmodium; Primaquine; Quinacrine; Quinine; Sucrose; Tritium | 1970 |
The intracellular and membrane effects of oxidant agents on normal red cells.
Topics: Cell Membrane; Erythrocytes; Glutathione; Heinz Bodies; Hemoglobinometry; Hemolysis; Humans; Hydroquinones; Hydroxylamines; Naphthoquinones; Osmotic Fragility; Oxidation-Reduction; Phenols; Phenylhydrazines; Potassium; Primaquine; Quinacrine; Quinine | 1970 |
Antimalarials: effects on in vivo and in vitro protein synthesis.
Topics: Amino Acids; Antimalarials; Carbon Isotopes; Cell-Free System; Chloroquine; Cycloheximide; Primaquine; Protein Biosynthesis; Quinacrine; Quinine; Tetrahymena | 1970 |
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines | 1970 |
Methaemoglobin levels in soldiers receiving antimalarial drugs.
Topics: Antimalarials; Australia; Chloroquine; Dapsone; Erythrocyte Count; Humans; Methemoglobin; Military Personnel; Primaquine; Pyrimethamine; Quinine; Reticulocytes; Vietnam | 1971 |
Resistance to primaquine in Plasmodium gallinaceum, and the problem of resistance to quinoline compounds in malaria parasites.
Topics: Aedes; Animals; Chickens; Chloroquine; Drug Resistance, Microbial; Malaria, Avian; Primaquine; Quinacrine; Quinine; Quinolines | 1967 |
[Further development of the Roehl test for testing antimalarial agents on Plasmodium cathemerium in the canary by intravenous administration].
Topics: Animals; Animals, Laboratory; Antimalarials; Canaries; Chloroquine; Injections, Intravenous; Malaria, Avian; Methods; Primaquine; Proguanil; Pyrimethamine; Quinine; Sulfadiazine; Sulfanilamides; Sulfonamides | 1967 |
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena | 1968 |
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine | 1968 |
Causal prophylactic effect of Menoctone (a new hydroxynaphthoquinone) against sporozoite-induced Plasmodium berghei infection in mice.
Topics: Animals; Antimalarials; Chloroquine; Cricetinae; Malaria; Mice; Naphthoquinones; Plasmodium; Primaquine; Quinine | 1968 |
Drug responses of mepacrine- and primaquine-resistant strains of Plasmodium berghei Vincke and Lips, 1948.
Topics: Animals; Antimalarials; Chloroquine; Dapsone; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinine; Sulfadiazine | 1966 |
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA | 1967 |
Chemotherapy of sporozoite- and blood-induced Plasmodium berghei infections with selected antimalarial agents.
Topics: Animals; Chloroquine; Cricetinae; Dapsone; Malaria; Mice; Primaquine; Pyrimethamine; Quinine; Rats | 1967 |
The effect of anti-malarial drugs on human natural killer cells in vitro.
Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines | 1984 |
Imported malaria in adults in Auckland.
Topics: Adolescent; Adult; Chloroquine; Drug Resistance, Microbial; Female; Humans; Kenya; Malaria; Male; Middle Aged; New Zealand; Papua New Guinea; Plasmodium falciparum; Plasmodium vivax; Primaquine; Quinine; Splenomegaly; Time Factors; Travel | 1982 |
Malaria in southeast Queensland in 1979.
Topics: Adolescent; Adult; Australia; Child; Child, Preschool; Chloroquine; Dapsone; Female; Humans; Infant; Infant, Newborn; Malaria; Male; Middle Aged; New Guinea; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinine; Sulfadoxine; Tinnitus; Vietnam | 1980 |
Comparative efficacies of quinine and chloroquine as companions to primaquine in a curative drug regimen.
Topics: Animals; Chloroquine; Drug Administration Schedule; Drug Therapy, Combination; Macaca mulatta; Malaria; Primaquine; Quinine | 1981 |
Normal immunological responses in mice treated with chloroquine, quinine and primaquine.
Topics: Animals; Antibody Formation; Chloroquine; Drug Administration Schedule; Immunity, Cellular; Male; Mice; Mice, Inbred BALB C; Primaquine; Quinine | 1981 |
Inhibition of hepatitis B virus specific DNA polymerase by intercalating agents.
Topics: Carrier State; Chloroquine; DNA-Directed DNA Polymerase; Ethidium; Hepatitis B; Hepatitis B Antigens; Hepatitis B virus; Humans; Intercalating Agents; Magnesium; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine; Quinine | 1980 |
Expression of the plasmodial pfmdr1 gene in mammalian cells is associated with increased susceptibility to chloroquine.
Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Base Sequence; Biological Transport; Cell Survival; Chloroquine; CHO Cells; Colchicine; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; DNA, Protozoan; Doxorubicin; Drug Resistance; Female; Gene Expression; Genes, Protozoan; Membrane Proteins; Oligonucleotides, Antisense; Oocytes; Plasmodium falciparum; Primaquine; Protozoan Proteins; Quinine; Restriction Mapping; Verapamil; Vinblastine; Xenopus laevis | 1994 |
Combined chloroquine and primaquine resistant Plasmodium vivax malaria in a patient returning from India.
Topics: Adult; Chloroquine; Drug Resistance; Drug Therapy, Combination; Female; Humans; Malaria, Vivax; Primaquine; Quinine; Recurrence | 1995 |
Anaemia, iron deficiency and malaria in a rural community in Brazilian Amazon.
Topics: Adolescent; Adult; Anemia, Hemolytic, Autoimmune; Anemia, Hypochromic; Animals; Brazil; Child; Child, Preschool; Chloroquine; Cross-Sectional Studies; Female; Ferrous Compounds; Hemoglobinometry; Humans; Incidence; Infant; Intestinal Diseases, Parasitic; Malaria; Male; Mebendazole; Plasmodium falciparum; Plasmodium vivax; Population Surveillance; Pregnancy; Primaquine; Quinine; Rural Population | 1994 |
In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.
Topics: Animals; Artemisinins; Female; Mefloquine; Mice; Primaquine; Proguanil; Quinine; Sesquiterpenes; Sulfadiazine; Toxoplasma; Triazines; Trifluoperazine; Uracil; Verapamil | 1994 |
Poor response to primaquine in two cases of Plasmodium vivax malaria from Guatemala.
Topics: Chloroquine; Drug Resistance; Drug Therapy, Combination; Guatemala; Humans; Malaria, Vivax; Male; Primaquine; Quinine | 1994 |
Column liquid chromatographic analysis of quinine in human plasma, saliva and urine.
Topics: Chromatography, High Pressure Liquid; Humans; Indicators and Reagents; Primaquine; Quinidine; Quinine; Saliva; Spectrophotometry, Ultraviolet | 1993 |
Interactions among primaquine, malaria infection and other antimalarials in Thai subjects.
Topics: Acute Disease; Administration, Oral; Adult; Drug Interactions; Humans; Malaria, Falciparum; Male; Mefloquine; Primaquine; Quinine; Thailand | 1993 |
A standard regimen for treatment of plasmodium vivax malaria.
Topics: Antimalarials; Humans; Infant; Malaria, Cerebral; Malaria, Falciparum; Malaria, Vivax; Primaquine; Quinine | 1996 |
Metabolic interactions of selected antimalarial and non-antimalarial drugs with the major pathway (3-hydroxylation) of quinine in human liver microsomes.
Topics: Anti-Infective Agents; Antimalarials; Chromatography; Cytochrome P-450 Enzyme System; Doxycycline; Drug Interactions; Erythromycin; Humans; Hydroxylation; Ketoconazole; Microsomes, Liver; Nifedipine; Omeprazole; Primaquine; Quinine; Tetracycline; Troleandomycin | 1997 |
Imported malaria: successful treatment of 31 patients in the era of chloroquine resistance.
Topics: Adolescent; Adult; Antimalarials; Artemisinins; Artesunate; Child; Chloroquine; Drug Resistance; Female; Humans; Malaria; Male; Middle Aged; Primaquine; Quinine; Retrospective Studies; Sesquiterpenes; Travel | 1999 |
Erythrocyte Fy antigen phenotyping helps differentiate so-called benign tertian malarias.
Topics: Animals; Child, Preschool; Diagnosis, Differential; Drug Therapy, Combination; Duffy Blood-Group System; Erythrocytes; Humans; Immunophenotyping; Malaria; Male; Plasmodium; Primaquine; Quinine; Tetracycline | 2000 |
Cytochrome P450 1A1/2 induction by antiparasitic drugs: dose-dependent increase in ethoxyresorufin O-deethylase activity and mRNA caused by quinine, primaquine and albendazole in HepG2 cells.
Topics: Albendazole; Antiparasitic Agents; Cell Survival; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Dose-Response Relationship, Drug; Enzyme Induction; Humans; Polychlorinated Dibenzodioxins; Primaquine; Quinine; RNA, Messenger; Tumor Cells, Cultured | 2002 |
Influence of primaquine on the clinical findings and joint potentials in rheumatoid arthritis.
Topics: Arthritis; Arthritis, Rheumatoid; Humans; Joints; Primaquine; Quinine | 1952 |
Potentiation of the curative action of primaquine in vivax malaria by quinine and chloroquine.
Topics: Antimalarials; Chloroquine; Humans; Malaria; Malaria, Vivax; Primaquine; Quinine | 1955 |
ANTIMALARIAL DRUG TRIALS ON A MULTIRESISTANT STRAIN OF PLASMODIUM FALCIPARUM.
Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Thailand | 1963 |
FLUORESCENT ANTIBODY STUDIES IN HUMAN MALARIA. II. DEVELOPMENT AND PERSISTENCE OF ANTIBODIES TO PLASMODIUM FALCIPARUM.
Topics: Amodiaquine; Antibodies; Antigen-Antibody Reactions; Chloroquine; Fluorescent Antibody Technique; Humans; Immune Sera; Malaria; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinine; Vaccination | 1964 |
[A PATIENT WITH TROPICAL MALARIA].
Topics: Amodiaquine; Antimalarials; Chloroquine; Dosage Forms; Drug Resistance; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Primaquine; Quinine | 1964 |
CHLOROQUINE-RESISTANT STRAIN OF PLASMODIUM FALCIPARUM FROM KHAO MAI KHAEO, THAILAND.
Topics: Chloroquine; Drug Resistance; Drug Resistance, Microbial; Drug Therapy; Humans; Malaria; Plasmodium falciparum; Primaquine; Pyrimethamine; Quinine; Thailand | 1965 |
ARMY giving primaquine treatment to all returning servicemen.
Topics: Humans; Malaria; Primaquine; Quinine | 1952 |
PRIMAQUINE 15 mg. for 14 days cures "high percentage".
Topics: Humans; Malaria; Primaquine; Quinine | 1952 |
Treatment with antimalarials adversely affects the oxidative energy metabolism in rat liver mitochondria.
Topics: Adenosine Triphosphatases; Animals; Antimalarials; Chloroquine; Cytochromes; Energy Metabolism; Male; Mitochondria, Liver; Oxidative Phosphorylation; Primaquine; Quinine; Rats; Rats, Inbred Strains | 2004 |
Antimalarials inhibit human erythrocyte membrane acetylcholinesterase.
Topics: Acetylcholinesterase; Adult; Antimalarials; Chloroquine; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocyte Membrane; Female; Humans; Kinetics; Male; Middle Aged; Primaquine; Quinine | 2005 |
Transmission-blocking activities of quinine, primaquine, and artesunate.
Topics: Animals; Anopheles; Antimalarials; Artemisinins; Artesunate; Disease Vectors; Dose-Response Relationship, Drug; In Vitro Techniques; Life Cycle Stages; Parasite Egg Count; Plasmodium falciparum; Primaquine; Quinine; Sesquiterpenes | 2006 |
Pulmonary edema due to Plasmodium vivax malaria in an American missionary.
Topics: Animals; Antimalarials; Doxycycline; Humans; Malaria, Vivax; Male; Middle Aged; Missionaries; Plasmodium vivax; Primaquine; Pulmonary Edema; Quinine; Radiography, Thoracic; Religious Missions; Uganda | 2007 |
A simple technique for the detection of anti-malarial drug formulations and their presence in human urine.
Topics: Amodiaquine; Antimalarials; Biological Assay; Biological Availability; Chloroquine; Chromatography, Thin Layer; Fraud; Humans; Malaria; Primaquine; Product Surveillance, Postmarketing; Pyrimethamine; Quality Control; Quinine; Sulfadoxine | 2006 |
Transfusion-related Plasmodium ovale malaria complicated by acute respiratory distress syndrome (ARDS) in a non-endemic country.
Topics: Antimalarials; Doxycycline; Female; Humans; Intensive Care Units; Malaria; Middle Aged; Plasmodium ovale; Platelet Transfusion; Primaquine; Quinine; Respiratory Distress Syndrome | 2011 |
Quality of essential drugs in tropical countries: evaluation of antimalarial drugs in the Brazilian Health System.
Topics: Antimalarials; Brazil; Chloroquine; Chromatography, High Pressure Liquid; Drug Storage; Drugs, Essential; Humans; Mefloquine; Primaquine; Quality Control; Quinine | 2011 |
Mosquito infection studies with Aotus monkeys and humans infected with the Chesson strain of Plasmodiun vivax.
Topics: Animals; Anopheles; Antimalarials; Aotidae; Chloroquine; Disease Management; Disease Models, Animal; Host-Parasite Interactions; Humans; Malaria; Male; Monkey Diseases; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinine | 2012 |
Quality of antimalarial drugs and antibiotics in Papua New Guinea: a survey of the health facility supply chain.
Topics: Amodiaquine; Amoxicillin; Antimalarials; Artemether; Artemisinins; Biosimilar Pharmaceuticals; Chloroquine; Drug Resistance; Health Facilities; Humans; Malaria, Falciparum; Malaria, Vivax; Papua New Guinea; Primaquine; Quality Control; Quinine | 2014 |
Nanomolar binding affinity of quinine-based antimalarial compounds by the cocaine-binding aptamer.
Topics: Amodiaquine; Antimalarials; Aptamers, Nucleotide; Binding Sites; Chloroquine; Cocaine; Ligands; Mefloquine; Primaquine; Quinine; Thermodynamics | 2018 |
Monocyte phagocytosis of malaria β-haematin in the presence of artemisinin, amodiaquine, chloroquine, doxycycline, primaquine, pyrimethamine and quinine.
Topics: Amodiaquine; Animals; Antimalarials; Artemisinins; Cell Count; Cell Line; Chloroquine; Doxycycline; Electron Probe Microanalysis; Heme; Hemeproteins; Humans; Leukocytes, Mononuclear; Mice; Microscopy, Electron, Scanning; Microscopy, Electron, Transmission; Monocytes; Peroxidase; Phagocytosis; Primaquine; Pyrimethamine; Quinine; Spectrophotometry; Temperature; U937 Cells | 2019 |
Atovaquone, chloroquine, primaquine, quinine and tetracycline: antiproliferative effects of relevant antimalarials on Neospora caninum.
Topics: Antimalarials; Atovaquone; Chloroquine; Neospora; Primaquine; Quinine; Tetracyclines | 2021 |
Historical 8-Aminoquinoline Combinations: Not All Antimalarial Drugs Work Well Together.
Topics: Aminoquinolines; Antimalarials; Chloroquine; Hemolysis; Humans; Primaquine; Quinine | 2022 |