Page last updated: 2024-08-20

pregnenolone and piperidines

pregnenolone has been researched along with piperidines in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19902 (16.67)18.7374
1990's0 (0.00)18.2507
2000's6 (50.00)29.6817
2010's3 (25.00)24.3611
2020's1 (8.33)2.80

Authors

AuthorsStudies
Veldhuis, JD1
Furlanetto, RW; Rodgers, RJ; Veldhuis, JD1
Akk, G; Bracamontes, J; Steinbach, JH1
Carta, M; Mameli, M; Partridge, LD; Valenzuela, CF1
Frändberg, PA; Johansson, T; Le Grevès, P; Nyberg, F1
Birgner, C; Elfverson, M; Frändberg, PA; Johansson, T; Le Grevès, P; Nyberg, F1
Elfverson, M; Johansson, T; Le Grevès, P; Linde, AM; Nyberg, F; Zhou, Q1
Akk, G; Bracamontes, J; Covey, DF; Li, P; Reichert, DE; Steinbach, JH1
Bose, HS; Marriott, KS; Prasad, M; Thapliyal, V1
Hermann, GE; Rogers, RC; Vance, KM1
Farquhar, CE; Gamage, TF; Lefever, TW; Nguyen, T; Thomas, BF; Wiley, JL; Zhang, Y1
Abood, ME; Leo, LM1

Reviews

1 review(s) available for pregnenolone and piperidines

ArticleYear
CB1 Cannabinoid Receptor Signaling and Biased Signaling.
    Molecules (Basel, Switzerland), 2021, Sep-06, Volume: 26, Issue:17

    Topics: Allosteric Site; Cannabinoid Receptor Agonists; Central Nervous System; Humans; Indoles; Ligands; Models, Molecular; Piperidines; Pregnenolone; Protein Binding; Protein Conformation; Receptor, Cannabinoid, CB1; Signal Transduction

2021

Other Studies

11 other study(ies) available for pregnenolone and piperidines

ArticleYear
Mechanisms subserving the bipotential actions of estrogen on ovarian cells: studies with a selective anti-estrogen, LY156758, and the sparingly metabolizable estrogen agonist, moxestrol.
    Journal of steroid biochemistry, 1986, Volume: 24, Issue:5

    Topics: 3-Hydroxysteroid Dehydrogenases; Animals; Dose-Response Relationship, Drug; Estradiol; Ethinyl Estradiol; Female; Ovary; Piperidines; Pregnenolone; Progesterone; Raloxifene Hydrochloride; Receptors, Estradiol; Swine

1986
Synergistic actions of estradiol and the insulin-like growth factor somatomedin-C on swine ovarian (granulosa) cells.
    Endocrinology, 1986, Volume: 119, Issue:2

    Topics: Animals; Cells, Cultured; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Synergism; Estradiol; Female; Granulosa Cells; Hydroxycholesterols; Insulin-Like Growth Factor I; Kinetics; Piperidines; Pregnenolone; Progesterone; Raloxifene Hydrochloride; Somatomedins; Swine

1986
Pregnenolone sulfate block of GABA(A) receptors: mechanism and involvement of a residue in the M2 region of the alpha subunit.
    The Journal of physiology, 2001, May-01, Volume: 532, Issue:Pt 3

    Topics: Binding Sites; Cell Line; Estranes; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Kidney; Ligands; Membrane Potentials; Mutagenesis; Nitriles; Patch-Clamp Techniques; Pentobarbital; Piperidines; Pregnenolone; Receptors, GABA-A; Transfection

2001
Neurosteroid-induced plasticity of immature synapses via retrograde modulation of presynaptic NMDA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Mar-02, Volume: 25, Issue:9

    Topics: Age Factors; Animals; Animals, Newborn; Antibodies; Calcium; Calcium Channel Blockers; Chelating Agents; Dizocilpine Maleate; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Membrane Potentials; Neuronal Plasticity; Patch-Clamp Techniques; Piperidines; Pregnenolone; Presynaptic Terminals; Quinolinic Acids; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Sodium Channel Blockers; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors

2005
Low concentrations of neuroactive steroids alter kinetics of [3H]ifenprodil binding to the NMDA receptor in rat frontal cortex.
    British journal of pharmacology, 2005, Volume: 146, Issue:6

    Topics: Animals; Binding, Competitive; Dose-Response Relationship, Drug; Frontal Lobe; Male; Piperidines; Pregnanolone; Pregnenolone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Tritium

2005
Neurosteroids alter glutamate-induced changes in neurite morphology of NG108-15 cells.
    The Journal of steroid biochemistry and molecular biology, 2007, Volume: 104, Issue:3-5

    Topics: 2-Amino-5-phosphonovalerate; Cell Adhesion; Cell Line, Tumor; Excitatory Amino Acid Agonists; Glioma; Glutamic Acid; Humans; Hybrid Cells; Neurites; Neuroblastoma; Piperidines; Pregnenolone; Receptors, N-Methyl-D-Aspartate; Steroids

2007
Neurosteroids allosterically modulate the ion pore of the NMDA receptor consisting of NR1/NR2B but not NR1/NR2A.
    Biochemical and biophysical research communications, 2008, Jul-25, Volume: 372, Issue:2

    Topics: Allosteric Regulation; Animals; CHO Cells; Cricetinae; Cricetulus; Hippocampus; Ion Channels; Male; Piperidines; Pregnanolone; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins

2008
Mutations of the GABA-A receptor alpha1 subunit M1 domain reveal unexpected complexity for modulation by neuroactive steroids.
    Molecular pharmacology, 2008, Volume: 74, Issue:3

    Topics: Amino Acid Substitution; Animals; Cell Line; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Mutant Proteins; Mutation; Piperidines; Pregnanetriol; Pregnanolone; Pregnenolone; Protein Structure, Secondary; Protein Structure, Tertiary; Protein Subunits; Rats; Receptors, GABA-A; Serine; Steroids; Tryptophan

2008
σ-1 receptor at the mitochondrial-associated endoplasmic reticulum membrane is responsible for mitochondrial metabolic regulation.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 343, Issue:3

    Topics: Animals; Benzofurans; Blotting, Western; Cell Line; Cholesterol; Dose-Response Relationship, Drug; Endoplasmic Reticulum; Gene Knockdown Techniques; Leydig Cells; Ligands; Male; Mice; Mitochondrial Membranes; Molecular Structure; Piperidines; Pregnenolone; Protein Binding; Receptors, sigma; Sigma-1 Receptor

2012
NMDA receptors control vagal afferent excitability in the nucleus of the solitary tract.
    Brain research, 2015, Jan-21, Volume: 1595

    Topics: 2-Amino-5-phosphonovalerate; Adenosine Triphosphate; Afferent Pathways; Animals; Aspartic Acid; Benzimidazoles; Calcium; Excitatory Amino Acid Antagonists; In Vitro Techniques; Piperidines; Pregnenolone; Rats; Rats, Long-Evans; Receptors, N-Methyl-D-Aspartate; Solitary Nucleus; Sulfonamides; Vagus Nerve

2015
The great divide: Separation between in vitro and in vivo effects of PSNCBAM-based CB
    Neuropharmacology, 2017, Volume: 125

    Topics: Allosteric Regulation; Animals; Cannabinoid Receptor Modulators; Cerebellum; Cyclohexanols; Discrimination, Psychological; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Guanosine 5'-O-(3-Thiotriphosphate); Male; Mice, Inbred C57BL; Mice, Inbred ICR; Motor Activity; Phenylurea Compounds; Piperidines; Pregnenolone; Pyrazoles; Pyridines; Receptor, Cannabinoid, CB1; Rimonabant

2017