Page last updated: 2024-08-23

pregnanolone and chlorine

pregnanolone has been researched along with chlorine in 44 studies

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.27)18.7374
1990's24 (54.55)18.2507
2000's16 (36.36)29.6817
2010's2 (4.55)24.3611
2020's1 (2.27)2.80

Authors

AuthorsStudies
Covey, DF; Hu, Y; Isenberg, KE; Rodgers-Neame, NT; Zorumski, CF1
Gee, KW; Lan, NC1
Morrow, AL; Pace, JR; Paul, SM; Purdy, RH1
Blakeman, DP; Im, WB1
Majewska, MD1
Belelli, D; Gee, KW; McCauley, L1
Ayer, DE; Blakeman, DP; Davis, JP; Im, WB1
Blinn, JR; Morrow, AL; Paul, SM; Purdy, RH1
Costa, E; Paul, SM; Pritchett, DB; Puia, G; Purdy, RH; Santi, MR; Seeburg, PH; Vicini, S1
Belelli, D; Gee, KW1
Ticku, MK; Yu, R1
Brinton, RD1
Moore, FL; Murray, TF; Orchinik, M1
Costa, E; Ducić, I; Puia, G; Vicini, S1
Bain, CJ; Kemp, JA; McKernan, RM; Quirk, K; Wafford, KA; Whiting, PJ; Wingrove, PB1
Bitran, D; Kellogg, CK; Purdy, RH1
Akaike, N; Harata, N; Shimura, M; Tamai, M1
Biscardi, R; Wilson, MA1
Akaike, N; Imanishi, T; Xu, TL1
Akwa, Y; Baulieu, EE; El-Etr, M; Robel, P1
Kellogg, CK; Olson, VG; Pleger, GL1
Biggio, G; Concas, A; Floris, S; Follesa, P; Mostallino, MC; Tuligi, G1
Barbaccia, ML; Biggio, G; Concas, A; Follesa, P; Grisenti, P; Mostallino, MC; Porcu, P; Purdy, RH; Trabucchi, M1
de Novara, AM; Fiszer de Plazas, S; Gravielle, MC1
Chistina Grobin, A; Devaud, LL; Inglefield, JR; Morrow, AL; Schwartz-Bloom, RD1
Dekermendjian, K; Hartvig, L; Liljefors, T; Lükensmejer, B1
Fiszer de Plazas, S; Pignataro, L1
Alkana, RL; Bolger, MB; Davies, DL; McCauley, LD1
Barker, JL; Chang, YH; Liu, QY; Schaffner, AE; Smith, SV1
Druzin, M; Haage, D; Johansson, S1
Ferguson, C; Grobin, AC; Homanics, GE; Kralic, JE; Morrow, AL; O'Buckley, TK; Renzi, K; Wheeler, M1
Bäckström, T; Lundgren, P; Strömberg, J; Wang, M1
Covey, DF; Eisenman, LN; Jinadasa, D; Mennerick, S; Shu, HJ; Zorumski, CF1
Backstrom, T; Birzniece, V; Johansson, IM; Lundgren, P; Turkmen, S; Zingmark, E1
Bitran, D; Smith, SS1
Bäckström, T; Lundgren, P; Strömberg, J1
Beadles-Bohling, AS; Crabbe, JC; Douglass, AD; Finn, DA; Long, SL; Tanchuck, MA1
Babot, Z; Bujons, J; García, DA; Kasal, A; Kristofíková, Z; Matyás, L; Suñol, C1
Bäckström, T; Haage, D; Lundgren, P; Strömberg, J; Taube, M1
Lockette, W; Woodman, R1
Asiedu, MN; Kaila, K; Malan, TP; Mejia, G; Ossipov, MK; Price, TJ1
Bukanova, JV; Kondratenko, RV; Solntseva, EI1
Grobin, AC; Morrow, AL1
Chesnoy-Marchais, D1

Reviews

1 review(s) available for pregnanolone and chlorine

ArticleYear
Steroid regulation of the GABAA receptor: ligand binding, chloride transport and behaviour.
    Ciba Foundation symposium, 1990, Volume: 153

    Topics: Animals; Biological Transport; Central Nervous System; Chlorides; Desoxycorticosterone; Ligands; Mice; Pregnanolone; Rats; Receptors, GABA-A; Steroids

1990

Other Studies

43 other study(ies) available for pregnanolone and chlorine

ArticleYear
Effects of a benz[e]indene on gamma-aminobutyric acid-gated chloride currents in cultured postnatal rat hippocampal neurons.
    Molecular pharmacology, 1992, Volume: 42, Issue:6

    Topics: Animals; Cells, Cultured; Chloride Channels; Chlorides; gamma-Aminobutyric Acid; Hippocampus; Indenes; Ion Channel Gating; Ion Channels; Isomerism; Membrane Proteins; Molecular Structure; Neurons; Pregnanolone; Rats

1992
Gamma-aminobutyric acidA receptor complexes in rat frontal cortex and spinal cord show differential responses to steroid modulation.
    Molecular pharmacology, 1991, Volume: 40, Issue:6

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Desoxycorticosterone; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Pentobarbital; Pregnanediol; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Steroids; Sulfur Radioisotopes

1991
Characterization of steroid interactions with gamma-aminobutyric acid receptor-gated chloride ion channels: evidence for multiple steroid recognition sites.
    Molecular pharmacology, 1990, Volume: 37, Issue:2

    Topics: 20-alpha-Dihydroprogesterone; Animals; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; In Vitro Techniques; Ion Channel Gating; Ion Channels; Membrane Proteins; Pregnanolone; Rats; Receptors, GABA-A; Steroids; Structure-Activity Relationship; Synaptosomes

1990
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes

1991
Heterotropic cooperativity between putative recognition sites for progesterone metabolites and the atypical benzodiazepine Ro 5-4864.
    Journal of neurochemistry, 1990, Volume: 55, Issue:1

    Topics: Animals; Benzodiazepinones; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; Male; Pregnanediol; Pregnanolone; Progesterone; Rats; Rats, Inbred Strains

1990
Studies on the mechanism of interactions between anesthetic steroids and gamma-aminobutyric acidA receptors.
    Molecular pharmacology, 1990, Volume: 37, Issue:3

    Topics: Anesthetics; Animals; Chlorides; Desoxycorticosterone; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Nipecotic Acids; Pentobarbital; Pregnanolone; Progesterone; Proline; Rats; Receptors, GABA-A; Synaptic Membranes

1990
Synthesis, metabolism, and pharmacological activity of 3 alpha-hydroxy steroids which potentiate GABA-receptor-mediated chloride ion uptake in rat cerebral cortical synaptoneurosomes.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Acetates; Animals; Cerebral Cortex; Chlorides; Desoxycorticosterone; Drug Synergism; Isomerism; Male; Molecular Conformation; Muscimol; Pregnanes; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes

1990
Neurosteroids act on recombinant human GABAA receptors.
    Neuron, 1990, Volume: 4, Issue:5

    Topics: Benzodiazepines; Cell Line, Transformed; Cell Membrane Permeability; Chlorides; Desoxycorticosterone; Electric Conductivity; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Kidney; Membrane Potentials; Pentobarbital; Pregnanolone; Receptors, GABA-A; Recombinant Proteins; Transfection

1990
5 alpha-pregnan-3 alpha,20 alpha-diol behaves like a partial agonist in the modulation of GABA-stimulated chloride ion uptake by synaptoneurosomes.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Animals; Benzodiazepines; Bicuculline; Chlorides; Clonazepam; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Ionophores; Pregnanediol; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1989
Chronic neurosteroid treatment produces functional heterologous uncoupling at the gamma-aminobutyric acid type A/benzodiazepine receptor complex in mammalian cortical neurons.
    Molecular pharmacology, 1995, Volume: 47, Issue:3

    Topics: Androstanes; Animals; Azasteroids; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebral Cortex; Chlorides; Chlorine; Convulsants; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Neurons; Pregnanolone; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes; Time Factors; Tritium

1995
The neurosteroid 3 alpha-hydroxy-5 alpha-pregnan-20-one induces cytoarchitectural regression in cultured fetal hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:5 Pt 1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Cell Death; Cell Division; Cell Survival; Cells, Cultured; Chlorides; Estradiol; Fetus; Hippocampus; Isomerism; Kinetics; Neurites; Neurons; Picrotoxin; Pregnanolone; Progesterone; Rats; Time Factors

1994
Steroid modulation of GABAA receptors in an amphibian brain.
    Brain research, 1994, May-23, Volume: 646, Issue:2

    Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Convulsants; Corticosterone; Flunitrazepam; Kinetics; Male; Mammals; Neurons; Pregnanolone; Pregnenolone; Rats; Receptors, GABA-A; Salamandridae; Species Specificity; Steroids; Sulfur Radioisotopes; Synaptosomes; Tritium

1994
Does neurosteroid modulatory efficacy depend on GABAA receptor subunit composition?
    Receptors & channels, 1993, Volume: 1, Issue:2

    Topics: Allosteric Regulation; Animals; Cell Line; Cells, Cultured; Cerebral Cortex; Chlorides; Electrophysiology; Humans; Pregnanolone; Pregnenolone; Protein Conformation; Rats; Receptors, GABA-A; Recombinant Proteins

1993
A novel allosteric modulatory site on the GABAA receptor beta subunit.
    Neuron, 1994, Volume: 12, Issue:4

    Topics: Allosteric Site; Animals; Anticonvulsants; Cells, Cultured; Chlorides; Drug Synergism; Electric Conductivity; Electrophysiology; Female; gamma-Aminobutyric Acid; Gene Expression; Humans; Pentobarbital; Pregnanolone; Rats; Receptors, GABA; Transfection; Triazoles; Xenopus

1994
Anxiolytic effect of progesterone is associated with increases in cortical allopregnanolone and GABAA receptor function.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:2

    Topics: Animals; Anxiety; Cerebral Cortex; Chlorides; Female; Ovariectomy; Pregnanolone; Progesterone; Rats; Receptors, GABA-A; Synaptosomes

1993
Allosteric modulation of GABAA receptors in acutely dissociated neurons of the suprachiasmatic nucleus.
    The American journal of physiology, 1996, Volume: 270, Issue:6 Pt 1

    Topics: Allosteric Regulation; Animals; Bicuculline; Chlorides; Diazepam; Electric Conductivity; Female; GABA Antagonists; GABA-A Receptor Agonists; Intracellular Membranes; Male; Neurons; Pentobarbital; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Suprachiasmatic Nucleus

1996
Influence of gender and brain region on neurosteroid modulation of GABA responses in rats.
    Life sciences, 1997, Volume: 60, Issue:19

    Topics: Amygdala; Androgens; Androsterone; Animals; Brain; Cerebellum; Cerebral Cortex; Chlorides; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Hippocampus; Male; Pregnanolone; Rats; Sex Characteristics

1997
Modulation of the GABAA response in rat ventromedial hypothalamic neurons by pregnanolone.
    Comparative biochemistry and physiology. Part A, Physiology, 1997, Volume: 117, Issue:2

    Topics: Animals; Chloride Channels; Chlorides; Diazepam; Drug Interactions; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Transport; Pentobarbital; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship; Ventromedial Hypothalamic Nucleus

1997
Opposing effects of different steroid sulfates on GABAA receptor-mediated chloride uptake.
    Brain research, 1998, Apr-20, Volume: 790, Issue:1-2

    Topics: Animals; Biological Transport; Cerebral Cortex; Chlorides; Dehydroepiandrosterone Sulfate; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; In Vitro Techniques; Ionophores; Male; Muscimol; Pregnanolone; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptosomes

1998
Neurosteroid action at the GABAA receptor in fetal rat forebrain.
    Brain research. Developmental brain research, 1998, Jun-15, Volume: 108, Issue:1-2

    Topics: Androsterone; Animals; Chlorides; Diazepam; Female; Fetus; GABA Modulators; gamma-Aminobutyric Acid; Male; Pregnancy; Pregnanolone; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sex Factors; Synaptosomes

1998
Molecular and functional adaptation of the GABA(A) receptor complex during pregnancy and after delivery in the rat brain.
    The European journal of neuroscience, 1998, Volume: 10, Issue:9

    Topics: Allosteric Regulation; Alternative Splicing; Animals; Brain Chemistry; Cerebral Cortex; Chlorides; Diazepam; Female; Hippocampus; Isotopes; Muscimol; Postpartum Period; Pregnancy; Pregnancy, Animal; Pregnanolone; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger

1998
Role of brain allopregnanolone in the plasticity of gamma-aminobutyric acid type A receptor in rat brain during pregnancy and after delivery.
    Proceedings of the National Academy of Sciences of the United States of America, 1998, Oct-27, Volume: 95, Issue:22

    Topics: Animals; Cell Membrane; Cerebral Cortex; Chlorides; Desoxycorticosterone; Estrus; Female; Finasteride; Gene Expression Regulation; Hippocampus; Muscimol; Postpartum Period; Pregnancy; Pregnancy, Animal; Pregnanolone; Progesterone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Time Factors; Transcription, Genetic

1998
GABA-stimulated chloride uptake during avian CNS development: modulation by neurosteroids.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1998, Volume: 16, Issue:6

    Topics: Animals; Biological Transport; Brain Chemistry; Chick Embryo; Chloride Channels; Chlorides; GABA Modulators; gamma-Aminobutyric Acid; Optic Lobe, Nonmammalian; Pregnanolone; Receptors, GABA-A

1998
Fluorescence imaging of GABAA receptor-mediated intracellular [Cl-] in P19-N cells reveals unique pharmacological properties.
    Brain research, 1999, May-08, Volume: 827, Issue:1-2

    Topics: Animals; Central Nervous System Depressants; Chlorides; Diazepam; DNA Primers; Ethanol; Flunitrazepam; Fluorescent Dyes; GABA Agonists; GABA Modulators; Gene Expression; Mice; Muscimol; Neoplastic Stem Cells; Neuroglia; Pentobarbital; Pregnanolone; Quinolinium Compounds; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tritium

1999
Two conserved arginines in the extracellular N-terminal domain of the GABA(A) receptor alpha(5) subunit are crucial for receptor function.
    Journal of neurochemistry, 2000, Volume: 75, Issue:4

    Topics: Amino Acid Substitution; Animals; Arginine; Chlorides; CHO Cells; Cricetinae; Diazepam; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression; Humans; Ion Channel Gating; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Pentobarbital; Pregnanolone; Protein Structure, Tertiary; Receptors, GABA-A; Sequence Alignment; Steroids; Structure-Activity Relationship; Transfection

2000
In ovo chronic neurosteroid treatment affects the function and allosteric interactions of GABA(A) receptor modulatory sites.
    Brain research, 2001, May-25, Volume: 902, Issue:1

    Topics: Allosteric Regulation; Animals; Chick Embryo; Chloride Channels; Chlorides; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Ion Transport; Nerve Tissue Proteins; Optic Lobe, Nonmammalian; Pregnanolone; Receptors, GABA-A; Signal Transduction; Specific Pathogen-Free Organisms; Synaptic Membranes; Synaptic Transmission

2001
Pressure-sensitive and -insensitive coupling in gamma-aminobutyric acid(A) receptors.
    Psychopharmacology, 2001, Volume: 157, Issue:4

    Topics: Animals; Atmospheric Pressure; Chlorides; Chlorine; Flunitrazepam; GABA Modulators; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Pentobarbital; Pregnanolone; Radioisotopes; Receptors, GABA-A; Synaptosomes

2001
Allopregnanolone activates GABA(A) receptor/Cl(-) channels in a multiphasic manner in embryonic rat hippocampal neurons.
    Journal of neurophysiology, 2002, Volume: 88, Issue:3

    Topics: Animals; Animals, Newborn; Cell Differentiation; Cells, Cultured; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Drug Synergism; Electric Conductivity; Embryo, Mammalian; gamma-Aminobutyric Acid; Hippocampus; Neurons; Pertussis Toxin; Pregnanolone; Rats; Reaction Time; Receptors, GABA-A; Steroids; Virulence Factors, Bordetella

2002
Allopregnanolone modulates spontaneous GABA release via presynaptic Cl- permeability in rat preoptic nerve terminals.
    Brain research, 2002, Dec-27, Volume: 958, Issue:2

    Topics: Action Potentials; Animals; Chlorides; gamma-Aminobutyric Acid; Male; Permeability; Pregnanolone; Preoptic Area; Presynaptic Terminals; Rats; Rats, Sprague-Dawley

2002
Deletion of GABAA receptor alpha 1 subunit-containing receptors alters responses to ethanol and other anesthetics.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:2

    Topics: Anesthetics; Animals; Anxiety; Behavior, Animal; Bicuculline; Brain; Central Nervous System Depressants; Chlorides; Desoxycorticosterone; Drug Tolerance; Ethanol; Exploratory Behavior; Female; GABA Agonists; GABA Antagonists; Male; Mice; Mice, Knockout; Muscimol; Postural Balance; Pregnanolone; Receptors, GABA-A; Steroids

2003
Allopregnanolone-stimulated GABA-mediated chloride ion flux is inhibited by 3beta-hydroxy-5alpha-pregnan-20-one (isoallopregnanolone).
    Brain research, 2003, Aug-22, Volume: 982, Issue:1

    Topics: Animals; Cerebral Cortex; Chlorides; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Osmolar Concentration; Pentobarbital; Pregnanolone; Rats; Rats, Wistar

2003
Slow actions of neuroactive steroids at GABAA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Jul-28, Volume: 24, Issue:30

    Topics: Animals; Binding Sites; Cell Membrane; Cells, Cultured; Chlorides; GABA Agonists; GABA Antagonists; gamma-Cyclodextrins; Hippocampus; Ion Channel Gating; Ion Transport; Kinetics; Ligands; Neurons; Oocytes; Patch-Clamp Techniques; Pregnanolone; Protein Binding; Pyridazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins; RNA, Messenger; Transfection; Xenopus

2004
3beta-20beta-dihydroxy-5alpha-pregnane (UC1011) antagonism of the GABA potentiation and the learning impairment induced in rats by allopregnanolone.
    The European journal of neuroscience, 2004, Volume: 20, Issue:6

    Topics: Analysis of Variance; Animals; Behavior, Animal; Cerebral Cortex; Chlorides; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Synergism; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Learning Disabilities; Male; Maze Learning; Pregnanediol; Pregnanolone; Radioimmunoassay; Rats; Rats, Wistar; Reaction Time; Statistics, Nonparametric; Time Factors

2004
Termination of pseudopregnancy in the rat produces an anxiogenic-like response that is associated with an increase in benzodiazepine receptor binding density and a decrease in GABA-stimulated chloride influx in the hippocampus.
    Brain research bulletin, 2005, Jan-30, Volume: 64, Issue:6

    Topics: Analysis of Variance; Animals; Animals, Newborn; Anxiety; Cerebral Cortex; Chlorides; Female; gamma-Aminobutyric Acid; Gonadotropins; Gonadotropins, Equine; Hippocampus; Humans; Isotopes; Maze Learning; Ovariectomy; Pregnanolone; Pseudopregnancy; Radioimmunoassay; Radioligand Assay; Rats; Receptors, GABA-A; Steroids; Time Factors

2005
Rapid non-genomic effect of glucocorticoid metabolites and neurosteroids on the gamma-aminobutyric acid-A receptor.
    The European journal of neuroscience, 2005, Volume: 21, Issue:8

    Topics: Animals; Cerebral Cortex; Chlorides; Desoxycorticosterone; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Glucocorticoids; Male; Neurons; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Synaptosomes

2005
Selected line difference in sensitivity to a GABAergic neurosteroid during ethanol withdrawal.
    Genes, brain, and behavior, 2006, Volume: 5, Issue:1

    Topics: Alcohol Withdrawal Seizures; Animals; Anticonvulsants; Chlorides; Dose-Response Relationship, Drug; GABA Modulators; Male; Mice; Mice, Inbred Strains; Pregnanolone; Prosencephalon; Receptors, GABA-A; Species Specificity; Statistics, Nonparametric; Steroids

2006
Activity of B-nor analogues of neurosteroids on the GABA(A) receptor in primary neuronal cultures.
    Journal of medicinal chemistry, 2006, Jun-01, Volume: 49, Issue:11

    Topics: Animals; Anions; Cell Survival; Cells, Cultured; Chlorides; Computer Simulation; GABA Modulators; Male; Models, Molecular; Neocortex; Neurons; Pregnanolone; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship

2006
Neurosteroid modulation of allopregnanolone and GABA effect on the GABA-A receptor.
    Neuroscience, 2006, Nov-17, Volume: 143, Issue:1

    Topics: Analysis of Variance; Animals; Brain; Cells, Cultured; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Steroids

2006
Alpha-methyltyrosine inhibits formation of reactive oxygen species and diminishes apoptosis in PC12 cells.
    Brain research, 2009, Nov-03, Volume: 1296

    Topics: Acetazolamide; alpha-Methyltyrosine; Animals; Apoptosis; Caspases; Catecholamines; Chlorides; Chlorthalidone; Coculture Techniques; Enzyme Inhibitors; Humans; Intracellular Space; Leukocytes; Neurons; Neuroprotective Agents; PC12 Cells; Pregnanolone; Rats; Reactive Oxygen Species

2009
Modulation of spinal GABAergic analgesia by inhibition of chloride extrusion capacity in mice.
    The journal of pain, 2012, Volume: 13, Issue:6

    Topics: Analgesia; Analgesics; Animals; Benzodiazepines; Chlorides; GABA-A Receptor Agonists; Isoxazoles; K Cl- Cotransporters; Male; Mice; Mice, Inbred ICR; Muscimol; Neuralgia; Peripheral Nerve Injuries; Pregnanolone; Receptors, GABA-A; Sciatic Nerve; Symporters

2012
Positive allosteric modulators of GABA
    The Journal of steroid biochemistry and molecular biology, 2022, Volume: 224

    Topics: Animals; Chlorides; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ligands; Pregnanolone; Rats; Receptors, GABA-A

2022
3Alpha-hydroxy-5alpha-pregnan-20-one levels and GABA(A) receptor-mediated 36Cl(-) flux across development in rat cerebral cortex.
    Brain research. Developmental brain research, 2001, Nov-26, Volume: 131, Issue:1-2

    Topics: Allosteric Regulation; Animals; Animals, Newborn; Anti-Anxiety Agents; Biological Transport; Cerebral Cortex; Chlorine; Desoxycorticosterone; Female; Flunitrazepam; GABA Agonists; GABA Modulators; Labor, Obstetric; Male; Muscimol; Pregnancy; Pregnanolone; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sex Characteristics

2001
Persistent GABAA/C responses to gabazine, taurine and beta-alanine in rat hypoglossal motoneurons.
    Neuroscience, 2016, 08-25, Volume: 330

    Topics: Animals; beta-Alanine; Bicuculline; Brain Stem; Central Nervous System Agents; Chlorine; GABA Agents; Hypoglossal Nerve; Midazolam; Motor Neurons; Neuroprotective Agents; Patch-Clamp Techniques; Pentobarbital; Phosphinic Acids; Pregnanolone; Pyridazines; Pyridines; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Strychnine; Taurine; Tissue Culture Techniques

2016