Page last updated: 2024-08-23

preclamol and spiperone

preclamol has been researched along with spiperone in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19905 (50.00)18.7374
1990's3 (30.00)18.2507
2000's2 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fang, X; Hu, Z; Levant, B; Min, J; Varady, J; Wang, S; Wu, X1
Berardi, F; Daniele, E; Govoni, S; Leopoldo, M; Lograno, MD; Perrone, R; Tortorella, V1
Blier, P; de Montigny, C; Debonnel, G; Monnet, FP1
Steinfels, GF; Tam, SW1
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M1
Haubrich, DR; Martin, GE; Williams, M1
Totaro, JA; Williams, M1
Meltzer, HY; Simonovic, M1
Jeanjean, AP; Laterre, EC; Maloteaux, JM1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1

Other Studies

10 other study(ies) available for preclamol and spiperone

ArticleYear
Molecular modeling of the three-dimensional structure of dopamine 3 (D3) subtype receptor: discovery of novel and potent D3 ligands through a hybrid pharmacophore- and structure-based database searching approach.
    Journal of medicinal chemistry, 2003, Oct-09, Volume: 46, Issue:21

    Topics: Algorithms; Binding Sites; Computational Biology; Crystallography, X-Ray; Databases, Protein; Humans; Kinetics; Ligands; Lipid Bilayers; Models, Molecular; Molecular Conformation; Mutation; Receptors, Dopamine D2; Receptors, Dopamine D3; Reproducibility of Results; Solvents; Structure-Activity Relationship; Tetrahydronaphthalenes; Water

2003
Oxygen isosteric derivatives of 3-(3-hydroxyphenyl)-N-n-propylpiperidine.
    Journal of medicinal chemistry, 1992, Aug-07, Volume: 35, Issue:16

    Topics: Animals; Brain; Dopamine Agents; In Vitro Techniques; Ketanserin; Mice; Oxygen; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1992
Modulation by sigma ligands of N-methyl-D-aspartate-induced [3H]noradrenaline release in the rat hippocampus: G-protein dependency.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:1

    Topics: Animals; Calcium; Cinnamates; Cyclopropanes; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanidines; Haloperidol; Hippocampus; In Vitro Techniques; Magnesium; Male; N-Methylaspartate; Norepinephrine; Pertussis Toxin; Piperidines; Rats; Rats, Inbred Strains; Spiperone; Tritium; Virulence Factors, Bordetella

1992
Selective sigma receptor agonist and antagonist affect dopamine neuronal activity.
    European journal of pharmacology, 1989, Apr-12, Volume: 163, Issue:1

    Topics: Animals; Antipsychotic Agents; Dopamine; In Vitro Techniques; Male; Membranes; Microelectrodes; Narcotic Antagonists; Narcotics; Neurons; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Spiperone

1989
Interaction of (+)- and (-)-3-PPP with the dopamine receptor in the anterior pituitary gland.
    Life sciences, 1984, Jan-16, Volume: 34, Issue:3

    Topics: Animals; Apomorphine; Binding Sites; Cell Membrane; Depression, Chemical; In Vitro Techniques; Male; Methyltyrosines; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism

1984
A pharmacological comparison of 6,7-dihydroxy-2-dimethylaminotetralin (TL-99) and N-n-propyl-3-(3-hydroxyphenyl)piperidine with (3-PPP) selected dopamine agonists.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:2

    Topics: 4-Butyrolactone; Animals; Apomorphine; Cell Membrane; Corpus Striatum; Female; Humans; Hydroxydopamines; Naphthalenes; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes

1982
Interaction of the putative dopamine autoreceptor agonists 3-PPP and TL-99 with [3H]apomorphine binding sites in rat striatal membranes.
    European journal of pharmacology, 1982, Dec-17, Volume: 86, Issue:1

    Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Kinetics; Membranes; Naphthalenes; Piperidines; Rats; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes

1982
Effect of 3-PPP, a putative dopamine autoreceptor agonist, on rat serum prolactin levels.
    Life sciences, 1981, Jul-06, Volume: 29, Issue:1

    Topics: Animals; Apomorphine; Binding, Competitive; Humans; Male; Piperidines; Prolactin; Rats; Receptors, Dopamine; Reserpine; Spiperone; Stereotyped Behavior

1981
Neuroleptic binding to sigma receptors: possible involvement in neuroleptic-induced acute dystonia.
    Biological psychiatry, 1997, May-15, Volume: 41, Issue:10

    Topics: Animals; Antipsychotic Agents; Dopamine Agonists; Dyskinesia, Drug-Induced; Male; Piperidines; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Muscarinic; Receptors, sigma; Spiperone

1997
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001