Page last updated: 2024-08-23

preclamol and piperidines

preclamol has been researched along with piperidines in 332 studies

Research

Studies (332)

TimeframeStudies, this research(%)All Research%
pre-1990160 (48.19)18.7374
1990's149 (44.88)18.2507
2000's12 (3.61)29.6817
2010's11 (3.31)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Klein, M; Musacchio, JM2
Lemaire, S; Rogers, C1
DeHaven-Hudkins, DL; Fleissner, LC1
Hudzik, TJ1
Akiyama, K; Okumura, K; Otsuki, S; Ujike, H; Zushi, Y1
Ahlenius, S; Hillegaart, V; Lindgren, JE; Lundström, J1
Araki, H; Hasegawa, Y; Kaku, S; Otomo, S1
Akiyama, K; Otsuki, S; Tsuchida, K; Ujike, H1
Ericson, H; Ross, SB1
Berardi, F; Daniele, E; Govoni, S; Leopoldo, M; Lograno, MD; Perrone, R; Tortorella, V1
Ahlenius, S1
Bohmaker, K; Bordi, F; Meller, E1
Carlsson, A; Cascella, NG; Lahti, RA; Lindberg, M; Tamminga, CA1
Hariton, C2
Bohmaker, K; Diamond, J; Lieu, HD; Meller, E; Puza, T1
DeHaven-Hudkins, DL; Fleissner, LC; Ford-Rice, FY1
Ekman, A; Eriksson, E2
Fukamauchi, F; Shibuya, H; Yoshikawa, T1
Akiyama, K; Kanzaki, A; Okumura, K; Otsuki, S; Tsuchida, K; Ujike, H1
Cook, L; Gilligan, PJ; Schmidt, WK; Steinfels, GF; Tam, SW1
Culp, SG; De Souza, EB; Rominger, D; Tam, SW1
Connick, JH; Fox, PK; France, L; Hanlon, G; Nicholson, CD; Roberts, J1
Chavkin, C; Connor, MA2
Blier, P; de Montigny, C; Debonnel, G; Monnet, FP1
Codd, EE; Shank, RP1
Mash, DC; Zabetian, CP1
Ross, SB1
Musacchio, JM; Zhou, GZ1
Bem, WT; Coscia, CJ; Homan, SM; Johnson, FE; Levy, BK; Mamone, JY; Thomas, GE1
Itzhak, Y; Stein, I1
Ekman, A; Eriksson, E; Quiding, M1
Kruk, ZL; Millar, J; Stamford, JA2
Karbon, EW; Naper, K; Pontecorvo, MJ1
Burke, M; Earley, B; Gouret, CJ; Junien, JL; Leonard, BE1
Carlsson, A; Kujacic, M; Löfberg, L; Svensson, K1
Clark, D; Furmidge, L; Petry, N; Tong, ZY1
Gillard, J; Knight, AR; Middlemiss, DN; Wong, EH1
Cler, JA; Contreras, PC; Dilworth, VM; Emmett, MR; Gray, NM; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL1
Engberg, G; Wikström, H1
Code, RA; Tang, AH1
Clark, D; Ericsson, M; Furmidge, LJ; Johnson, D; Petry, N; Tong, ZY1
Blazynski, C; Cohen, AI1
Contreras, PC; Dilworth, VM; Farah, JM; Gray, NM; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL1
Duckles, SP; Massamiri, T3
Itzhak, Y; Mash, D; Stein, I; Zhang, SH1
Cristante, D; Itzhak, Y; Kassim, CO; Stein, I; Zhang, SH1
Bell, JA; London, ED; Spivak, CE; Su, TP; Wu, XZ1
Clark, D; Galloway, MP; Salah, RS1
Cler, JA; Contreras, PC; Dilworth, VM; Iyengar, S; Mick, SJ; Rao, TS; Wood, PL1
Battaglia, G; Glennon, RA; Smith, JD1
Fiorica-Howells, E; Spector, S1
Bøgesø, KP; Carlsson, A; Hyttel, J; Liljefors, T; Svensson, K; Wikström, H1
Svensson, L1
Church, J; Lodge, D1
Itzhak, Y; Krähling, H; Ruhland, M1
Henderson, G; Kennedy, C2
Henderson, G; Jarvis, GE; Kennedy, C1
Kuypers, G; Paul, IA; Skolnick, P; Youdim, M1
Chaki, S; Muramatsu, M; Otomo, S; Usuki-Ito, C1
Bremer, ME; Contreras, PC; Gray, NM1
Al'perina, EL; Cheĭdo, MA; Idova, GV1
Bremer, ME; Contreras, PC; Rao, TS1
Feuerstein, G; Lysko, PG1
Dubrovina, NI; Il'iuchenok, RIu; Parkhomenko, RI1
Bowen, WD; DeCosta, B; Hellewell, SB; Rice, KC; Thurkauf, A; Walker, JM1
Klein, M; Musacchio, J; Paturzo, JJ; Zhou, GZ1
Lemaire, S; Rogers, CA1
Ferkany, JW; Karbon, EW; Patch, RJ; Pontecorvo, MJ1
Bowen, WD; Moses, EL; Tolentino, PJ; Walker, JM1
Byrd, JC; Paleos, GA; Yang, ZW2
Bowen, WD; De Costa, BR; Hellewell, SB; Hemstreet, MK; Lai, NL; Matsumoto, RR; Rice, KC; Thurkauf, A; Walker, JM1
Bauerle, LM; DeNoble, VJ; Jones, KW1
Canoll, PD; Gottesman, S; Musacchio, JM; Smith, PR1
Carlsson, A; Clark, D; Hjorth, S5
Klein, M; Musacchio, JM; Paturzo, JJ1
Culp, SG; De Souza, EB; Wolfe, SA1
Bluth, LS; Bowen, WD; Jacobson, AE; Rice, KC1
Bowen, WD; Hellewell, SB; McGarry, KA1
Emori, T; Hirata, Y; Marumo, F; Ohta, K; Shichiri, M1
Aanonsen, LM; Seybold, VS1
Heym, J; Koe, BK; Lebel, L; Schmidt, A; Seeger, T1
Denavit-Saubié, M; Foutz, AS1
Itzhak, Y2
Canoll, PD; Klein, M; Musacchio, JM1
Burkhart, CA; Koe, BK; Lebel, LA1
Steinfels, GF; Tam, SW1
Bowen, WD; de Costa, BR; Hellewell, SB; Jacobson, AE; Rice, KC; Thurkauf, A; Walker, JM1
Carlsson, M; Eriksson, E3
Ahlenius, S; Hillegaart, V; Wijkström, A1
Cook, L; Steinfels, GF; Tam, SW2
Domae, M; Furukawa, T; Matsumoto, S; Nagashima, M; Shirakawa, K; Yamada, K1
Fico, TA; Spoerlein, MT; Vanderwende, C; Wilmot, CA1
Martínez, JA; Milanés, MV; Vargas, ML1
Bobker, DH; Shen, KZ; Surprenant, A; Williams, JT1
Bagetta, G; de Sarro, GB; Marra, R; Nisticò, G; Priolo, E1
Gundlach, AL; Largent, BL; Snyder, SH; Wikström, H1
Hiltunen, AJ; Järbe, TU2
Itzhak, Y; Khouri, M1
Chavkin, C; Malouf, AT; Swearengen, E1
Beart, PM; Manallack, DT1
Tam, SW; Zhang, AZ1
Claustre, Y; Fage, D; Scatton, B; Zivkovic, B1
Sethy, VH; Wenger, D1
Horn, AS; Mastebroek, D; Rollema, H; Wikström, H1
Andersson, M; Fowler, CJ; Magnusson, O; Thorell, G1
Carnoy, P; Puech, AJ; Simon, P; Soubrie, P1
Magistretti, PJ; Ofori, S; Schorderet, M1
Goiny, M; Uvnäs-Moberg, K1
Nichols, NF; Schreur, PJ1
Keana, JF; McLean, S; Pou, S; Quarum, M; Sonders, M; Weber, E1
Di Chiara, G; Longoni, R; Spina, L1
Jenner, P; Kelly, E; Marsden, CD2
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Namba, Y1
Aihara, H; Hashimoto, S; Okuyama, S1
Bagetta, G; Corasaniti, MT; Nisticò, G; Sakurada, S; Strongoli, MC1
Bagetta, G; Nistico, G; Priolo, E1
George, SR; Seeman, P; Watanabe, M1
Bagetta, G; De Sarro, G; Nisticò, G; Priolo, E1
Gundlach, AL; Largent, BL; Snyder, SH5
Balster, RL1
Fowler, CJ; Thorell, G1
Bobker, DH; Campbell, BG; Leslie, FM; Mefford, IN; Weber, E1
Jenner, P; Marsden, CD; Nomoto, M1
Carlsson, A; Engel, JA; Hjorth, S1
Hiyama, T; Kikuchi, T; Suzuki, S; Tsutsui, M; Yamada, K; Yasuda, Y1
Altar, CA; Gerber, R; Hall, NR; Liebman, JM1
Christoffersen, CL; Meltzer, LT1
Clark, D; Kovacic, B; Le Witt, P1
Di Chiara, G; Frau, R; Imperato, A; Tanda, G1
Baldessarini, RJ; Campbell, A; Froimowitz, M; Gao, YG; Neumeyer, JL1
Ahlénius, S; Johansson, L; Lennmark, M; Lundström, J; Säfholm, C; Teiling, A; Thorberg, SO1
Argiolas, A; Gessa, GL; Melis, MR1
Carlsson, M; Clark, D; Eriksson, E; Nilsson, C; Svensson, K1
Ahlenius, S; Hillegaart, V1
Ahlenius, S; Criborn, CO; Henriksson, C; Hillegaart, V1
Berg, S; Lindberg, P; Lundström, J; Nilsson, JL; Pettersson, B; Sanchez, D; Thorberg, SO; Wijkström, A1
Ståhle, L; Ungerstedt, U2
Carlsson, A; Carlsson, M; Eriksson, E1
Bergstrom, DA; Bromley, SD; Carlson, JH; Jackson, DM; Walters, JR1
Bonsall, RW; Michael, RP; Schaefer, GJ1
Baldessarini, RJ; Froimowitz, M; Neumeyer, JL1
Andersson, B; Eriksson, E; Hjorth, S1
Carlsson, A; Mastebroek, D; Rollema, H; Sundell, S; Svensson, K; Wikström, H1
Liljefors, T; Wikström, H1
Andersson, B; Carlsson, A; Hjorth, S; Svensson, K; Wikström, H1
Carlsson, A; Carlsson, M; Eriksson, E; Nilsson, C1
Clark, D; Elam, M; Svensson, TH1
Arnt, J; Bøgesø, KP; Lundmark, M; Sundell, S1
Carlsson, A2
Broekkamp, CL; Gower, AJ1
Hedner, T; Lundborg, P1
Howard, HR; Kelly, TR; Koe, BK; Sarges, R1
Carlsson, A; Clark, D; Hjorth, S; Svensson, K; Thorberg, O1
Collu, M; Gessa, GL; Serra, G1
Draper, R; Mulder, AH; Schoffelmeer, AN; Sminia, P; Stoof, JC1
Carlsson, A; Clark, D; Hjorth, S; Sanchez, D; Svensson, K1
Brown, F; Campbell, W; Mitchell, PJ; Randall, K1
Gaillard, JM; Hjorth, S; Kafi-de St Hilaire, S; Sovilla, JY1
Bunney, BS; Carlsson, A; Clark, D; Engberg, G; Freeman, AS; Pileblad, E; Svensson, TH1
Bhaird, NN; Fowler, CJ; Thorberg, O; Tipton, KF1
Glock, D; Goldberg, LI; Kohli, JD1
Carlsson, A; Löfberg, L1
Arvidsson, LE; Hacksell, U; Hjorth, S; Johansson, AM; Lindberg, P; Nilsson, JL; Sanchez, D; Svensson, K; Thorberg, SO; Wikström, H1
Arbilla, S; Langer, SZ1
Arvidsson, LE; Carlsson, A; Hacksell, U; Hjorth, S; Lindberg, P; Nilsson, JL; Sanchez, D; Svensson, U; Wikström, H1
Carlsson, A; Clark, D; Engel, J; Hjorth, S; Sanchez, D; Svensson, K1
Bymaster, FP; Wong, DT1
Bendesky, RJ; Jones, JH; Martin, GE1
Bacopoulos, NG; Koch, SW; Koe, BK1
Carlsson, A; Clark, D; Engel, J; Hjorth, S; Lindberg, P1
Hjorth, S1
Arnt, J; Bøgesø, KP; Christensen, AV; Hyttel, J; Larsen, JJ; Svendsen, O1
Gudelsky, GA; Meltzer, HY; Simonovic, M1
Boissard, CG; Delini-Stula, A; Mogilnicka, E1
Arnt, J; Bøgesø, KP; Hyttel, J; Larsen, JJ; Svendsen, O1
Palacios, JM; Wiederhold, KH1
Billingsley, ML; Roth, RH1
Daus, FJ; Hansen, HA; Plantjé, JF; Stoof, JC1
Watling, KJ; Williams, M1
Carlsson, A; Hjorth, S; Jackson, D; Lindberg, P2
Jones, JH; Watling, KJ; Williams, M1
Fallon, S; Liebman, JM; Pastor, G; Welch, JJ1
Mulder, AH; Plantjé, JF; Stoof, JC1
Lahaye, D; Markstein, R1
Hacksell, U; Hjorth, S; Schorderet, M1
Dijkstra, D; Horn, AS; Houwing, HA; Van Oene, JC1
Arvidsson, LE; Carlsson, A; Clark, D; Hacksell, U; Hjorth, S; Johansson, A; Lindberg, P; Sanchez, D; Svensson, K; Wikström, H1
Arnt, J; Hyttel, J1
Ahlenius, S; Archer, T; Hillegaart, V; Tandberg, B1
Fenton, HM; Gerhardt, S; Leszczak, E; Liebman, JM1
Ahlenius, S; Hillegaart, V; Svensson, L; Thorberg, O1
Berendsen, HG; Broekkamp, CL; Gower, AJ; Princen, MM1
Ahlenius, S; Hillegaart, V; Lundström, J; Magnusson, O1
Ahlenius, S; Larsson, K1
Arvidsson, LE; Carlsson, A; Clark, D; Hacksell, U; Hjorth, S; Johansson, A; Lindberg, P; Nilsson, JL; Sanchez, D; Svensson, K; Wikström, H1
Adelung, C; Lang, JD; Späth, L; Starke, K1
Robinson, JL; Watling, KJ; Williams, M1
Arnt, J1
Fenton, HM; Gerhardt, S; Hall, NR; Liebman, JM; Neale, R; Noreika, L1
Geyer, MA; Lee, EH1
Carlsson, A; Eriksson, E; Modigh, K; Wikström, H1
Carlsson, A; Gunne, LM; Häggström, JE; Wikström, H1
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M1
Fratta, W; Gessa, GL; Napoli-Farris, L1
Pinnock, RD1
Haubrich, DR; Martin, GE; Williams, M2
Ahlenius, S; Svensson, L1
Mulder, AH; Sminia, P1
Waldmeier, PC1
Gudelsky, GA; Meltzer, HY; Passaro, E1
Totaro, JA; Williams, M1
Meltzer, HY; Simonovic, M1
Carlsson, A; Hjorth, S; Lindberg, P1
Bergstrom, DA; Gonzalez, AM; Huang, KX; Kreiss, DS; Sibley, DR; Walters, JR1
Sonsalla, PK; Terleckyj, I1
Dubrovina, NI2
Bowen, WD; Carr, DJ; DeCosta, BR; Garza, HH; Mayo, S1
Appleyard, SM; Chavkin, C; Connor, M; Patterson, TA1
See, RE1
Arnold, FJ; Murphy, RB; Schuster, DI1
DeCoster, MA; Klette, KL; Knight, ES; Tortella, FC1
Matsunaga, KH; Matsuno, K; Mita, S1
Di Giannuario, A; Pieretti, S; Sagratella, S1
Leander, JD; Wolff, MC1
Lin, MY; Walters, DE1
Carlsson, A; Huff, RM; Kling-Petersen, T; Svensson, K; Waters, N1
De Costa, BR; Martin, WJ; Walker, JM1
Beart, PM; Jarrott, B; Mercer, LD; Ryan, MC; Wong, MG1
Jeanjean, AP; Laduron, PM; Maloteaux, JM; Mestre, M1
Eguíbar, JR; Holmgren, B; Santos, A; Urbá-Holmgren, R1
Bailey, MA; Karbon, EW1
Chaki, S; Muramatsu, M; Otomo, S; Tanaka, M1
Hashimoto, K; London, ED; Mantione, CR; Neumeyer, JL; Spada, MR1
Chiodo, LA; Freeman, AS; Zhang, J1
Hirotsu, I; Honbo, N; Koyama, M; Ohno, T1
Bonhaus, DW; Eglen, RM; Hsu, SA; Jakeman, LB; Leung, E; Loury, DN; To, ZP; Wong, EH; Zeitung, KD1
Bravi, D; Chase, TN; Hoff, JI; Metman, LV; Mouradian, MM; Roberts, JR; Sethy, VH1
Davies, JA; Ellis, Y1
Matsunaga, K; Matsuno, K; Mita, S; Senda, T1
Cooper, TB; Klein, M; Musacchio, JM1
Barg, J; Eilam, Y; Ela, C; Hasin, Y; Vogel, Z1
Amoo, VE; Cannon, JG; Johnson, AK; Kirschbaum, KS; Long, JP1
Gerlach, J; Peacock, L1
Kaku, S; Muramatsu, M; Otomo, S; Tanaka, M1
Bonhaus, DW; DeSouza, A; Eglen, RM; Jakeman, LB; Loury, DN; To, Z; Wong, EH1
Dwoskin, L; Jewell, A; Wedlund, P1
Enomoto, R; Ogita, K; Yoneda, Y1
Callahan, PM; Cunningham, KA1
Bailey, MA; Kaiser, C; Karbon, EW; Mathew, RM; Mewshaw, RE; Sherrill, RG1
Järbe, TU1
Matsuno, K; Mita, S; Senda, T1
Allen, JT; DeHaven-Hudkins, DL; Ford-Rice, FY; Hudkins, RL1
Barg, J; Eilam, Y; Ela, C; Hasin, Y; Novakova, M; Vogel, Z1
Gudelsky, GA1
Brum, JM; Estafanous, FG; Murray, PA; Schubert, A; Tsuchida, H1
Carlsson, A; Merello, M; Pirtosek, Z; Stern, G2
Kling-Petersen, T; Ljung, E; Svensson, K; Wollter, L1
Kobayashi, T; Matsuno, K; Mita, S1
Ahtee, L; Kivastik, T; Piepponen, TP; Vuorikallas, K; Zharkovsky, A1
Barrett, TW; Chang, S; Ha, BK; Liu, Y; Saini, P; Whitlock, BB; Wolfe, SA1
Cochrane, EV; Dijkstra, D; Lahti, RA; Mutin, A; Tamminga, CA; Tepper, PG; Wikström, H1
Kling-Petersen, T; Ljung, E; Svensson, K1
Fujikawa, M; Furukawa, T; Inoue, T; Nagashima, M; Yamada, K1
Brent, PJ1
Ha, BK; Saini, P; Whitlock, BB; Wolfe, SA1
Akiyama, K; Kuroda, S; Okumura, K; Ujike, H1
Furukawa, H; Hasegawa, T; Kitaichi, K; Nabeshima, T; Noda, Y1
Kobayashi, T; Matsuno, K; Mita, S; Senda, T1
Earley, B; Faherty, CJ; Leonard, BE1
Jeanjean, AP; Laterre, EC; Maloteaux, JM1
Fang, H; Helmeste, DM; Li, M; Tang, SW1
Carlsson, A; Corey, PK; Lahti, AC; Lahti, RA; Tamminga, CA; Weiler, MA1
Curzon, P; Decker, MW1
Ekman, A; Eriksson, E; Hellstrand, M; Nilsson, CL2
Chan, SL; Morgan, NG1
Carey, JE; Frey, KA; Kilbourn, MR; Kuhl, DE; Mulholland, GK; Sherman, PS; Wieland, DM1
Camarasa, J; Camins, A; Canudas, AM; Escubedo, E; Pallas, M; Pubill, D; Sureda, FX1
Kobayashi, T; Matsuno, K; Mita, S; Murai, M; Senda, T1
Borowicz, KK; Czuczwar, SJ; Kleinrok, Z1
Garrone, B; Magnani, M; Pinza, M; Polenzani, L1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1
Tamminga, CA1
Takigawa, M; Wang, H1
Akaike, A; Hashino, A; Kaneko, S; Katsuki, H; Kume, T; Minami, M; Nishikawa, H; Satoh, M; Taguchi, R1
Carlsson, A; Carlsson, ML; Nilsson, M1
Brown-Borg, HM; Ebadi, M; Muralikrishnan, D1
Baeyens, JM; Cobos, EJ; Del Pozo, E1
Burris, KD; Kikuchi, T; Miwa, T; Mori, T; Stark, A; Tadori, Y; Tottori, K1
Galineau, L; Garcia, A; Houle, S; McCormick, P; Natesan, S; Seeman, P; Stableford, WT; Vasdev, N; Wilson, AA1
Chen, R; Johnson, JL; Jordan, S; Kambayashi, J; Kikuchi, T; Kitagawa, H; McQuade, R; Regardie, K; Tadori, Y1
Corsini, GU; Maggio, R; Millan, MJ; Novi, F1
Calas, AG; Goursaud, S; Hermans, E; Jeanjean, AP; Koener, B; Maloteaux, JM; Van De Stadt, M1
Carlsson, A; Carlsson, ML; Johansson, AM; Rung, E; Rung, JP; Svensson, K1
Edmunds, AJ; Gao, GL; Morris, JA; Worthington, PA; Ye, M; Yu, JQ1
Lowry, JP; O'Connor, JJ1
Anwar-Ul Azim, M; Kitamura, Y; Kozaka, T; Miwa, D; Ogawa, K; Shiba, K; Uno, I1
Azim, MA; Kitamura, Y; Kiyono, Y; Kozaka, T; Makino, A; Miwa, D; Ogawa, K; Shiba, K; Uno, I1
Ma, GF; Ortiz, J; Raivio, N; Sabrià, J1
Cao, P; Jia, T; Liao, J; Lou, Y; Wang, B; Wang, M; Yin, X1
Canals, M; Capuano, B; Charlton, SJ; Christopoulos, A; Coudrat, T; Donthamsetti, P; Javitch, JA; Klein Herenbrink, C; Lane, JR; Scammells, PJ; Sexton, PM; Shonberg, J; Sykes, DA1
Bezprozvanny, I; Geva, M; Grossman, I; Hayden, M; Kusko, R; Ryskamp, D; Wu, J1
Bezprozvanny, IB; Bol'shakova, AV; Gainullina, AN; Kraskovskaya, NA; Kukanova, EO; Vlasova, OL1

Reviews

7 review(s) available for preclamol and piperidines

ArticleYear
Dextromethorphan and sigma ligands: common sites but diverse effects.
    Life sciences, 1989, Volume: 45, Issue:19

    Topics: Animals; Dextromethorphan; Endorphins; Hallucinogens; Humans; Levorphanol; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism

1989
Dopamine receptor agonists: mechanisms underlying autoreceptor selectivity. II. Theoretical considerations.
    Journal of neural transmission, 1985, Volume: 62, Issue:3-4

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Corpus Striatum; Cyclic AMP; Dextroamphetamine; Dopamine; Humans; Isomerism; Lisuride; Models, Neurological; Molecular Conformation; Motor Activity; Nucleus Accumbens; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Substantia Nigra; Synaptosomes

1985
Dopamine-receptor agonists: mechanisms underlying autoreceptor selectivity. I. Review of the evidence.
    Journal of neural transmission, 1985, Volume: 62, Issue:1-2

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Behavior, Animal; Brain; Caudate Nucleus; Deoxyglucose; Dopamine; Humans; Lisuride; Models, Biological; Nerve Tissue Proteins; Phenanthrenes; Piperidines; Rats; Receptors, Dopamine; Stereoisomerism; Substantia Nigra; Synaptosomes; Tegmentum Mesencephali

1985
Dopaminergic and serotonergic control of neuroendocrine function.
    Monographs in neural sciences, 1984, Volume: 10

    Topics: alpha-Methyltyrosine; Animals; Antipsychotic Agents; Benzamides; Cattle; Dopamine; Hallucinogens; Hypothalamo-Hypophyseal System; Indoles; Methyltyrosines; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Serotonin; Tetrahydronaphthalenes

1984
Preclamol. A "designer drug" in the treatment of advanced Parkinson's disease.
    Advances in neurology, 1996, Volume: 69

    Topics: Antiparkinson Agents; Dopamine Agonists; Humans; Parkinson Disease; Piperidines

1996
Partial dopamine agonists in the treatment of psychosis.
    Journal of neural transmission (Vienna, Austria : 1996), 2002, Volume: 109, Issue:3

    Topics: Animals; Apomorphine; Autoreceptors; Brain; Dopamine Agonists; Humans; Piperidines; Psychotic Disorders; Receptors, Dopamine

2002
Schizophrenia: from dopamine to glutamate and back.
    Current medicinal chemistry, 2004, Volume: 11, Issue:3

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Disease Models, Animal; Dopamine; Dopamine Agonists; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Mice; Piperazines; Piperidines; Quinolones; Schizophrenia

2004

Trials

5 trial(s) available for preclamol and piperidines

ArticleYear
Pharmacologic properties of (-)-3PPP (preclamol) in man.
    Journal of neural transmission. General section, 1992, Volume: 88, Issue:3

    Topics: Administration, Oral; Adult; Chromatography, Gas; Dopamine Agents; Double-Blind Method; Half-Life; Humans; Injections, Intramuscular; Male; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology

1992
Motor effects of the partial dopamine agonist (-)-3-(3-hydroxyphenyl)-N-n-propylpiperidine (preclamol) in Parkinson's disease.
    Movement disorders : official journal of the Movement Disorder Society, 1994, Volume: 9, Issue:5

    Topics: Aged; Antiparkinson Agents; Dose-Response Relationship, Drug; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Infusions, Intravenous; Injections, Intramuscular; Levodopa; Male; Middle Aged; Neurologic Examination; Parkinson Disease; Piperidines

1994
Morphine- and cocaine-induced conditioned place preference: effects of quinpirole and preclamol.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 54, Issue:2

    Topics: Animals; Cocaine; Conditioning, Operant; Dopamine Agonists; Male; Morphine; Narcotics; Piperidines; Rats; Rats, Wistar; Synaptic Transmission

1996
Preclamol and parkinsonian fluctuations.
    Clinical neuropharmacology, 1993, Volume: 16, Issue:6

    Topics: Antiparkinson Agents; Apomorphine; Blood Pressure; Dopamine Agonists; Female; Humans; Injections, Subcutaneous; Male; Middle Aged; Movement; Parkinson Disease; Piperidines; Receptors, Dopamine D1; Receptors, Dopamine D2

1993
Antipsychotic properties of the partial dopamine agonist (-)-3-(3-hydroxyphenyl)-N-n-propylpiperidine(preclamol) in schizophrenia.
    Biological psychiatry, 1998, Jan-01, Volume: 43, Issue:1

    Topics: Adult; Antiparkinson Agents; Antipsychotic Agents; Cross-Over Studies; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Female; Humans; Male; Middle Aged; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenic Psychology

1998

Other Studies

320 other study(ies) available for preclamol and piperidines

ArticleYear
High-affinity dextromethorphan and (+)-3-(-3-hydroxyphenyl)-N-(1-propyl)piperidine binding sites in rat brain. Allosteric effects of ropizine.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:3

    Topics: Allosteric Regulation; Animals; Antitussive Agents; Binding Sites; Brain; Computer Simulation; Dextromethorphan; Guinea Pigs; Hydrogen-Ion Concentration; Male; Pentazocine; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1992
Characterization of [3H]desmethylimipramine binding in bovine adrenal medulla: interactions with sigma- and (or) phencyclidine-receptor ligands.
    Canadian journal of physiology and pharmacology, 1992, Volume: 70, Issue:11

    Topics: Adrenal Medulla; Animals; Binding Sites; Cattle; Desipramine; Dextromethorphan; Dizocilpine Maleate; Phenazocine; Phencyclidine; Piperidines; Potassium Chloride; Receptors, Opioid, delta; Receptors, Phencyclidine; Tranquilizing Agents

1992
Competitive interactions at [3H]1,3-di(2-tolyl)guanidine (DTG)-defined sigma recognition sites in guinea pig brain.
    Life sciences, 1992, Volume: 50, Issue:9

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Carbazoles; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Male; Pentazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma

1992
Sigma ligand-induced emesis in the pigeon.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1

    Topics: Animals; Apomorphine; Columbidae; Dextromethorphan; Dizocilpine Maleate; Dopamine Agents; Guanidines; Haloperidol; Male; Pentobarbital; Phenazocine; Piperidines; Propranolol; Psychotropic Drugs; Pyrimidines; Receptors, Opioid; Receptors, sigma; Vomiting

1992
Persistent supersensitivity of sigma receptors develops during repeated methamphetamine treatment.
    European journal of pharmacology, 1992, Feb-18, Volume: 211, Issue:3

    Topics: Animals; Behavior, Animal; Dopamine Agents; Dose-Response Relationship, Drug; Drug Tolerance; Male; Methamphetamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1992
Relationship between brain levels of 3-(3-hydroxyphenyl)-N-n-propylpiperidine HCl enantiomers and effects on locomotor activity in rats.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Animals; Brain; Dopamine Agents; Dose-Response Relationship, Drug; Half-Life; Injections, Subcutaneous; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Stereoisomerism; Tissue Distribution

1992
Sigma receptor modulation of the muscle relaxant action of eperisone.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1992, Volume: 2, Issue:2

    Topics: Animals; Behavior, Animal; Dopamine Agents; Dose-Response Relationship, Drug; Haloperidol; In Vitro Techniques; Mice; Mice, Inbred ICR; Muscle Relaxants, Central; Piperidines; Propiophenones; Receptors, Opioid; Receptors, sigma

1992
Supersensitivity of sigma receptors after repeated administration of cocaine.
    Life sciences, 1992, Volume: 51, Issue:6

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Agents; Drug Administration Schedule; Injections, Intraperitoneal; Male; Narcotic Antagonists; Piperidines; Psychotropic Drugs; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1992
Subchronic treatment of rats with remoxipride fails to modify sigma binding sites in the brain.
    European journal of pharmacology, 1992, Jun-05, Volume: 226, Issue:2

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Corpus Striatum; Dopamine Agents; Dopamine Antagonists; Haloperidol; In Vitro Techniques; Liver; Male; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Opioid; Receptors, sigma; Remoxipride; Salicylamides

1992
Oxygen isosteric derivatives of 3-(3-hydroxyphenyl)-N-n-propylpiperidine.
    Journal of medicinal chemistry, 1992, Aug-07, Volume: 35, Issue:16

    Topics: Animals; Brain; Dopamine Agents; In Vitro Techniques; Ketanserin; Mice; Oxygen; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone

1992
Effects of the local application of 3-PPP and sulpiride enantiomers into the nucleus accumbens or into the ventral tegmental area on rat locomotor activity: evidence for the functional importance of somatodendritic autoreceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:5

    Topics: Animals; Dopamine Agents; Male; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sulpiride; Tegmentum Mesencephali

1992
The effects of pertussis toxin on dopamine D2 and serotonin 5-HT1A autoreceptor-mediated inhibition of neurotransmitter synthesis: relationship to receptor reserve.
    Neuropharmacology, 1992, Volume: 31, Issue:5

    Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Brain; Dopamine Agents; GTP-Binding Proteins; Levodopa; Male; Neurotransmitter Agents; Pertussis Toxin; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Ribose; Virulence Factors, Bordetella

1992
Biphasic dose-dependent effects of dopamine and involvement of dopamine autoreceptors on intra-ocular pressure in the rabbit.
    Journal of autonomic pharmacology, 1992, Volume: 12, Issue:5

    Topics: Animals; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Intraocular Pressure; Male; N-Methylaspartate; Ocular Hypertension; Piperidines; Rabbits; Receptors, Dopamine; Thiothixene

1992
Comparative effects of receptor inactivation, 17 beta-estradiol and pertussis toxin on dopaminergic inhibition of prolactin secretion in vitro.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Estradiol; GTP-Binding Proteins; Male; Pertussis Toxin; Phenoxybenzamine; Piperidines; Pituitary Gland, Anterior; Prolactin; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Drug; Virulence Factors, Bordetella

1992
Characterization of the binding of [3H](+)-pentazocine to sigma recognition sites in guinea pig brain.
    European journal of pharmacology, 1992, Dec-01, Volume: 227, Issue:4

    Topics: Animals; Antipsychotic Agents; Binding Sites; Binding, Competitive; Brain; Carbazoles; Dopamine Agents; Guinea Pigs; Haloperidol; Kinetics; Male; Pentazocine; Piperidines; Receptors, sigma

1992
Effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline on the prolactin suppression induced by a series of full and partial dopamine D2 receptor agonists in male rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:2

    Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Dopamine Agents; Ergolines; Levodopa; Male; Piperidines; Prolactin; Quinolines; Rats; Rats, Sprague-Dawley

1992
Pre-synaptic dopaminergic control mechanisms for CCK-8 like immunoreactivity in the rat medial frontal cortex.
    Neuropeptides, 1992, Volume: 23, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Cholecystokinin; Dopamine; Dopamine Agents; In Vitro Techniques; Male; Microinjections; N-Methylaspartate; Nerve Degeneration; Neurons; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Dopamine

1992
BMY-14802 reverses the reduction of striatal dopamine release induced by (+)-3-[3-hydroxyphenyl]-N-(1-propyl)piperidine.
    Journal of neural transmission. General section, 1992, Volume: 90, Issue:2

    Topics: Animals; Corpus Striatum; Dialysis; Dopamine; Dopamine Agents; Male; Piperidines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stereoisomerism

1992
DuP 734 [1-(cyclopropylmethyl)-4-(2'(4''-fluorophenyl)-2'-oxoethyl)- piperidine HBr], a sigma and 5-hydroxytryptamine2 receptor antagonist: receptor-binding, electrophysiological and neuropharmacological profiles.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Biogenic Amines; Guinea Pigs; Male; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Serotonin; Receptors, sigma; Rotation; Serotonin Antagonists

1992
[3H]DuP 734 [1-(cyclopropylmethyl)-4-(2'-(4''-fluorophenyl)-2'- oxoethyl)-piperidine HBr]: a receptor binding profile of a high-affinity novel sigma receptor ligand in guinea pig brain.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:3

    Topics: Animals; Antipsychotic Agents; Brain; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Male; Mice; Phenazocine; Phenytoin; Piperidines; Receptors, sigma; Structure-Activity Relationship; Temperature

1992
Multiple sigma binding sites in guinea-pig and rat brain membranes: G-protein interactions.
    British journal of pharmacology, 1992, Volume: 107, Issue:3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Dextromethorphan; Dopamine Agents; GTP-Binding Proteins; Guanidines; Guinea Pigs; In Vitro Techniques; Male; Membranes; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Opioid, delta

1992
Ionic zinc may function as an endogenous ligand for the haloperidol-sensitive sigma 2 receptor in rat brain.
    Molecular pharmacology, 1992, Volume: 42, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Cations, Divalent; Copper; Electric Stimulation; Guanidines; Haloperidol; Hippocampus; Hydrogen-Ion Concentration; Kinetics; Male; Membranes; Pentazocine; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sensitivity and Specificity; Tritium; Zinc

1992
Modulation by sigma ligands of N-methyl-D-aspartate-induced [3H]noradrenaline release in the rat hippocampus: G-protein dependency.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:1

    Topics: Animals; Calcium; Cinnamates; Cyclopropanes; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanidines; Haloperidol; Hippocampus; In Vitro Techniques; Magnesium; Male; N-Methylaspartate; Norepinephrine; Pertussis Toxin; Piperidines; Rats; Rats, Inbred Strains; Spiperone; Tritium; Virulence Factors, Bordetella

1992
1,3-Di(2-[5-3H]tolyl)guanidine labels more than one site in rat forebrain.
    European journal of pharmacology, 1992, Jul-07, Volume: 217, Issue:2-3

    Topics: Animals; Binding Sites; Binding, Competitive; Carbamazepine; Guanidines; Haloperidol; Male; Pentazocine; Phenytoin; Piperidines; Prosencephalon; Rats; Rats, Wistar; Receptors, sigma; Stereoisomerism

1992
Sigma receptors are associated with cortical limbic areas in the primate brain.
    Synapse (New York, N.Y.), 1992, Volume: 12, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Brain; Cerebral Cortex; Image Processing, Computer-Assisted; Limbic System; Macaca mulatta; Male; Piperidines; Radioligand Assay; Receptors, sigma; Tissue Distribution

1992
Heterogeneous binding of sigma radioligands in the rat brain and liver: possible relationship to subforms of cytochrome P-450.
    Pharmacology & toxicology, 1991, Volume: 68, Issue:4

    Topics: Animals; Brain; Cytochrome P-450 Enzyme System; Guanidines; Haloperidol; Kinetics; Ligands; Liver; Male; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Subcellular Fractions

1991
Computer-assisted modeling of multiple dextromethorphan and sigma binding sites in guinea pig brain.
    European journal of pharmacology, 1991, Apr-25, Volume: 206, Issue:4

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Computer Simulation; Dextromethorphan; Guanidines; Guinea Pigs; Haloperidol; Kinetics; Male; Models, Biological; Piperidines; Receptors, Opioid; Receptors, sigma; Tritium

1991
Overexpression of sigma receptors in nonneural human tumors.
    Cancer research, 1991, Dec-15, Volume: 51, Issue:24

    Topics: Binding, Competitive; Carcinoma; Colonic Neoplasms; Guanidines; Humans; In Vitro Techniques; Kidney Neoplasms; Neoplasms; Piperidines; Receptors, Opioid; Receptors, sigma; Sarcoma

1991
Regulation of sigma receptors and responsiveness to guanine nucleotides following repeated exposure of rats to haloperidol: further evidence for multiple sigma binding sites.
    Brain research, 1991, Dec-06, Volume: 566, Issue:1-2

    Topics: Adenosine Triphosphate; Animals; Brain; Cell Membrane; Down-Regulation; Guanidines; Guanine Nucleotides; Guanylyl Imidodiphosphate; Haloperidol; Kinetics; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Reference Values

1991
Effects of the two partial D2 agonists (+)- and (-)-3-PPP on prolactin release in EEDQ treated male rats.
    Life sciences, 1991, Volume: 48, Issue:4

    Topics: 4-Butyrolactone; Animals; Brain; Dopamine Agents; Male; Piperidines; Prolactin; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Reference Values

1991
Differential effects of dopamine agonists upon stimulated limbic and striatal dopamine release: in vivo voltammetric data.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Bromocriptine; Corpus Striatum; Dopamine; Dopamine Agents; Electrochemistry; Electrophysiology; Ergolines; In Vitro Techniques; Limbic System; Male; Microelectrodes; Nucleus Accumbens; Pergolide; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Stereotaxic Techniques

1991
[3H]DTG and [3H](+)-3-PPP label pharmacologically distinct sigma binding sites in guinea pig brain membranes.
    European journal of pharmacology, 1991, Jan-25, Volume: 193, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dopamine Agents; Guanidines; Guinea Pigs; Haloperidol; In Vitro Techniques; Kinetics; Membranes; Phenazocine; Phenytoin; Piperidines; Receptors, Opioid; Receptors, sigma

1991
Evidence for an anti-amnesic effect of JO 1784 in the rat: a potent and selective ligand for the sigma receptor.
    Brain research, 1991, Apr-19, Volume: 546, Issue:2

    Topics: Amnesia; Animals; Antipsychotic Agents; Avoidance Learning; Behavior, Animal; Carbazoles; Cinnamates; Cyclopropanes; Dopamine Agents; Dose-Response Relationship, Drug; Guanidines; Ligands; Male; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Scopolamine

1991
Dopamine receptors, controlling dopamine levels in rat adrenal glands-comparison with central dopaminergic autoreceptors.
    Journal of neural transmission. General section, 1991, Volume: 84, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenal Medulla; Animals; Apomorphine; Azepines; Diencephalon; Domperidone; Dopamine; Dopamine Agents; Epinephrine; Ergolines; Lisuride; Male; Norepinephrine; Phenanthrenes; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Telencephalon

1991
Focal stimulation of specific pathways in the rat hippocampus causes a reduction in radioligand binding to the haloperidol-sensitive sigma receptor.
    Experimental brain research, 1991, Volume: 85, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Electric Stimulation; Guanidines; Haloperidol; Hippocampus; Male; Piperidines; Quinoxalines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1991
Effects of low, autoreceptor selective doses of dopamine agonists on the discriminative cue and locomotor hyperactivity produced by d-amphetamine.
    Journal of neural transmission. General section, 1991, Volume: 86, Issue:1

    Topics: Animals; Conditioning, Operant; Cues; Dextroamphetamine; Discrimination, Psychological; Dopamine Agents; Ergolines; Male; Motor Activity; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine

1991
The human sigma site, which resembles that in NCB20 cells, may correspond to a low-affinity site in guinea pig brain.
    Neuroscience letters, 1991, Oct-14, Volume: 131, Issue:2

    Topics: Animals; Brain Chemistry; Cells, Cultured; Cerebral Cortex; Cricetinae; Cricetulus; Dopamine Agents; Guanidines; Guinea Pigs; Humans; Kinetics; Male; Mice; Neuroblastoma; Pentazocine; Phenazocine; Piperidines; Radioligand Assay; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Tumor Cells, Cultured

1991
Effects of sigma ligands on mouse cerebellar cyclic guanosine monophosphate (cGMP) levels in vivo: further evidence for a functional modulation of N-methyl-D-aspartate (NMDA) receptor complex-mediated events by sigma ligands.
    Brain research, 1991, Oct-04, Volume: 561, Issue:1

    Topics: Animals; Cerebellum; Cyclic GMP; Dopamine Agents; Harmaline; Ligands; Male; Methamphetamine; Mice; Pentylenetetrazole; Piperidines; Quisqualic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma; Serine

1991
Sigma-receptors: implication for the control of neuronal activity of nigral dopamine-containing neurons.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: Animals; Apomorphine; Binding, Competitive; Dizocilpine Maleate; Dopamine; Dopamine Agents; Male; Neurons; Piperidines; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereotaxic Techniques; Substantia Nigra

1991
Yawning produced by dopamine agonists in rhesus monkeys.
    European journal of pharmacology, 1991, Aug-29, Volume: 201, Issue:2-3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Macaca mulatta; Male; Physostigmine; Piperidines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Yawning

1991
Behavioural profile of partial D2 dopamine receptor agonists. 1. Atypical inhibition of d-amphetamine-induced locomotor hyperactivity and stereotypy.
    Psychopharmacology, 1991, Volume: 105, Issue:3

    Topics: Animals; Dextroamphetamine; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Lisuride; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Stereotyped Behavior

1991
Dopamine and its agonists reduce a light-sensitive pool of cyclic AMP in mouse photoreceptors.
    Visual neuroscience, 1990, Volume: 4, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Benzazepines; Cyclic AMP; Dark Adaptation; Dopamine; Dopamine Agents; Ergolines; Ligands; Light; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Photoreceptor Cells; Piperidines; Quinpirole; Receptors, Dopamine

1990
(+) 3-[3-hydroxyphenyl-N-(1-propyl) piperidine] selectively differentiates effects of sigma ligands on neurochemical pathways modulated by sigma receptors: evidence for subtypes, in vivo.
    Neuropharmacology, 1991, Volume: 30, Issue:8

    Topics: Adrenocorticotropic Hormone; Animals; Brain; Butaclamol; Cerebellum; Corpus Striatum; Cyclic GMP; Dopamine; Dopamine Agents; Male; Mice; Pentazocine; Phenazocine; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid; Receptors, sigma

1991
Interactions of sigma and phencyclidine receptor ligands with the norepinephrine uptake carrier in both rat brain and rat tail artery.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Animals; Biological Transport; Brain; Desipramine; Dizocilpine Maleate; Male; Norepinephrine; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tail; Vasoconstriction

1991
Characterization of N-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP) binding sites in C57BL/6 mouse brain: mutual effects of monoamine oxidase inhibitors and sigma ligands on MPTP and sigma binding sites.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Brain; Cell Membrane; Clorgyline; Kinetics; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Piperidines; Receptors, Opioid; Receptors, sigma; Selegiline

1991
Binding of sigma-ligands to C57BL/6 mouse brain membranes: effects of monoamine oxidase inhibitors and subcellular distribution studies suggest the existence of sigma-receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Binding Sites; Brain; Guanidines; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase Inhibitors; Phenazocine; Piperidines; Receptors, Opioid; Receptors, sigma

1991
Electrophysiological and binding studies on intact NCB-20 cells suggest presence of a low affinity sigma receptor.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Animals; Cricetinae; Cricetulus; Hybrid Cells; Ligands; Mice; Neuroblastoma; Phenazocine; Piperidines; Potassium Channels; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Tumor Cells, Cultured

1991
Differential agonist profile of the enantiomers of 3-PPP at striatal dopamine autoreceptors: dependence on extracellular dopamine.
    Synapse (New York, N.Y.), 1991, Volume: 8, Issue:3

    Topics: Animals; Biogenic Monoamines; Cerebral Cortex; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Electrochemistry; Ergolines; In Vitro Techniques; Lisuride; Male; Nerve Tissue Proteins; Nucleus Accumbens; Piperidines; Potassium; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1991
Neurochemical characterization of dopaminergic effects of opipramol, a potent sigma receptor ligand, in vivo.
    Neuropharmacology, 1990, Volume: 29, Issue:12

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Corpus Striatum; Dopamine; Haloperidol; Homovanillic Acid; Ligands; Male; Mice; Opipramol; Organ Specificity; Phencyclidine; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
(-)PPAP: a new and selective ligand for sigma binding sites.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Animals; Catalysis; Dextroamphetamine; Discrimination, Psychological; Guinea Pigs; Haloperidol; In Vitro Techniques; Male; Piperidines; Propylamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
Selectivity of some "specific" opioid ligands?
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Benzomorphans; Binding, Competitive; Brain; Dynorphins; Female; Haloperidol; In Vitro Techniques; Mice; Morphinans; Peptide Fragments; Phencyclidine; Piperidines; Receptors, Opioid

1990
Pre- and postsynaptic dopaminergic activities of indolizidine and quinolizidine derivatives of 3-(3-hydroxyphenyl)-N-(n-propyl)piperidine (3-PPP). Further developments of a dopamine receptor model.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; 5-Hydroxytryptophan; Animals; Dopamine Agents; Dopamine Antagonists; Male; Models, Structural; Molecular Conformation; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Structure-Activity Relationship

1990
No mediolateral differences in striatal autoreceptor-mediated modulation of dopamine release: in vivo voltammetric data.
    Neuroscience letters, 1990, Feb-05, Volume: 109, Issue:1-2

    Topics: Animals; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Antagonists; Electrochemistry; Male; Metoclopramide; Piperidines; Rats; Rats, Inbred Strains

1990
The role of the dopaminergic system in the modulation of the acoustic startle response in the rat.
    European journal of pharmacology, 1990, Jan-03, Volume: 175, Issue:1

    Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Reflex, Startle; Stereoisomerism

1990
Failure of sigma-receptor ligands to reduce the excitatory actions of N-methyl-DL-aspartate on rat spinal neurons in-vivo.
    The Journal of pharmacy and pharmacology, 1990, Volume: 42, Issue:1

    Topics: Animals; Aspartic Acid; Haloperidol; In Vitro Techniques; Kainic Acid; Ligands; N-Methylaspartate; Neurons; Oxadiazoles; Piperidines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Spinal Cord; Stereoisomerism

1990
Binding of umespirone to the sigma receptor: evidence for multiple affinity states.
    Neuropharmacology, 1990, Volume: 29, Issue:2

    Topics: Animals; Antipsychotic Agents; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorpromazine; Guanylyl Imidodiphosphate; Haloperidol; In Vitro Techniques; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine

1990
Inhibition of potassium currents by the sigma receptor ligand (+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine in sympathetic neurons of the mouse isolated hypogastric ganglion.
    Neuroscience, 1990, Volume: 35, Issue:3

    Topics: Animals; Atropine; Carbazoles; Dopamine Agents; Evoked Potentials; Ganglia, Sympathetic; In Vitro Techniques; Male; Membrane Potentials; Mice; Mice, Inbred DBA; Neurons; Piperidines; Potassium Channels; Receptors, Opioid; Receptors, sigma; Sulpiride; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin

1990
The sigma [corrected] ligand rimcazole antagonises (+)SKF 10,047, but not (+)3-PPP, in the mouse isolated vas deferens.
    European journal of pharmacology, 1990, Jun-08, Volume: 181, Issue:3

    Topics: Animals; Antipsychotic Agents; Carbazoles; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Muscle, Smooth; Phenazocine; Piperidines; Stereoisomerism; Vas Deferens

1990
Polyamines non-competitively inhibit [3H]3-PPP binding to sigma receptors.
    European journal of pharmacology, 1990, Aug-02, Volume: 184, Issue:1

    Topics: Adrenal Medulla; Animals; Biogenic Polyamines; Brain Chemistry; Cattle; Dopamine Agents; Guinea Pigs; In Vitro Techniques; Kinetics; Piperidines; Rats; Receptors, Opioid; Receptors, sigma

1990
Differentiation of the active site of minaprine from that of phencyclidine in rat hippocampus.
    Research communications in chemical pathology and pharmacology, 1990, Volume: 69, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Binding Sites; Hippocampus; Ketamine; Male; Membranes; N-Methylaspartate; Phencyclidine; Piperazines; Piperidines; Potassium Channels; Pyridazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1990
Ifenprodil and SL 82.0715 potently inhibit binding of [3H](+)-3-PPP to sigma binding sites in rat brain.
    Neuroscience letters, 1990, Aug-14, Volume: 116, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain; Dopamine Agents; Kinetics; Male; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Tritium

1990
[Increase of the number of bone marrow T-suppressor cells under inhibition of immunogenesis during changes of the activity of the neuromediator system].
    Biulleten' eksperimental'noi biologii i meditsiny, 1990, Volume: 110, Issue:9

    Topics: 1-Naphthylamine; Animals; Bone Marrow; Bone Marrow Cells; Dopamine Agents; Leukocyte Count; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Neuroimmunomodulation; Neurotransmitter Agents; Piperidines; Serotonin Antagonists; Sertraline; T-Lymphocytes, Regulatory

1990
GBR-12909 and fluspirilene potently inhibited binding of [3H] (+)3-PPP to sigma receptors in rat brain.
    Life sciences, 1990, Volume: 47, Issue:22

    Topics: Animals; Antipsychotic Agents; Brain; Dopamine Agents; Fluspirilene; Male; Neurotransmitter Uptake Inhibitors; Piperazines; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1990
Excitatory amino acid neurotoxicity at the N-methyl-D-aspartate receptor in cultured neurons: protection by SKF 10,047.
    Neuroscience letters, 1990, Dec-11, Volume: 120, Issue:2

    Topics: Animals; Cell Survival; Cells, Cultured; Cerebellum; Dopamine Agents; Glutamates; Glutamic Acid; Neurons; Neurotoxins; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine

1990
[GABAergic modulation of amnesic trace reproduction by activation of the dopaminergic system].
    Biulleten' eksperimental'noi biologii i meditsiny, 1990, Volume: 110, Issue:12

    Topics: Animals; Avoidance Learning; Bupropion; Diazepam; Dopamine Agents; Ergolines; Male; Mice; Mice, Inbred BALB C; Piperidines; Propiophenones; Quinpirole; Receptors, GABA-A

1990
Characterization of [3H] (+)-pentazocine, a highly selective sigma ligand.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Binding, Competitive; Brain; Guinea Pigs; In Vitro Techniques; Kinetics; Pentazocine; Phenazocine; Piperidines; Receptors, Opioid; Receptors, sigma

1990
The effect of sigma ligands on dextromethorphan binding sites in the guinea pig.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Binding Sites; Dextromethorphan; Guinea Pigs; Hallucinogens; Haloperidol; In Vitro Techniques; Kinetics; Levorphanol; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
Characterization of (+)-[3H]3-PPP and [3H]TCP binding sites in membrane preparations of bovine adrenal medulla.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Adrenal Medulla; Animals; Binding Sites; Binding, Competitive; Cattle; In Vitro Techniques; Membranes; Phencyclidine; Piperidines; Receptors, Opioid; Receptors, sigma

1990
Ifenprodil potently interacts with [3H](+)-3-PPP-labeled sigma binding sites in guinea pig brain membranes.
    European journal of pharmacology, 1990, Feb-06, Volume: 176, Issue:2

    Topics: Animals; Brain; Guinea Pigs; In Vitro Techniques; Kinetics; Piperidines; Receptors, Opioid; Receptors, Opioid, delta

1990
Metabolites of haloperidol display preferential activity at sigma receptors compared to dopamine D-2 receptors.
    European journal of pharmacology, 1990, Feb-27, Volume: 177, Issue:3

    Topics: Animals; Brain; Haloperidol; In Vitro Techniques; Male; Motor Activity; Parasympathetic Nervous System; Pentazocine; Phosphatidylinositols; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Opioid; Receptors, sigma

1990
Ontogeny of PCP and sigma receptors in rat brain.
    Brain research. Developmental brain research, 1990, Feb-01, Volume: 51, Issue:2

    Topics: Aging; Animals; Brain; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
Multiple vascular effects of sigma and PCP ligands: inhibition of amine uptake and contractile responses.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:1

    Topics: Animals; Cocaine; Desoxycorticosterone; Haloperidol; Male; Norepinephrine; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Serotonin; Vasoconstriction

1990
Drug specificity of pharmacological dystonia.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:1

    Topics: Animals; Benzomorphans; Drug Interactions; Dystonia; Male; Microinjections; Morphinans; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Red Nucleus

1990
Differential effects of sigma and phencyclidine receptor ligands on learning.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Avoidance Learning; Dibenzocycloheptenes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Ligands; Male; Memory; Pentazocine; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Retention, Psychology

1990
Computer-assisted analysis of dextromethorphan and (+)-3-(-3-hydroxyphenyl)-N-(1-propyl)piperidine binding sites in rat brain. Allosteric effects of ropizine.
    Life sciences, 1990, Volume: 47, Issue:18

    Topics: Allosteric Site; Animals; Binding, Competitive; Brain; Dextromethorphan; Electronic Data Processing; In Vitro Techniques; Kinetics; Models, Biological; Pentazocine; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Tritium

1990
Multiple sites of action of (+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine ((+)-3PPP) in blood vessels.
    European journal of pharmacology, 1990, Nov-13, Volume: 190, Issue:3

    Topics: Animals; Arteries; Cocaine; Desoxycorticosterone; Ear; Male; Muscle Contraction; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Stimulation, Chemical; Sulpiride; Tail

1990
Autoradiographic localization of [3H]dextromethorphan (DM) in guinea pig brain: allosteric enhancement by ropizine.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Allosteric Regulation; Animals; Autoradiography; Binding Sites; Brain; Dextromethorphan; Guinea Pigs; In Vitro Techniques; Levorphanol; Piperazines; Piperidines; Tissue Distribution

1990
Lack of functional evidence for the involvement of sigma opiate receptors in the actions of the 3-PPP enantiomers on central dopaminergic systems: discrepancies between in vitro and in vivo observations.
    Life sciences, 1985, Aug-19, Volume: 37, Issue:7

    Topics: Animals; Butaclamol; Corpus Striatum; Dopamine; Limbic System; Male; Motor Activity; Pentazocine; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Reserpine; Stereoisomerism

1985
Effects of dextromethorphan site ligands and allosteric modifiers on the binding of (+)-[3H]3-(-3-hydroxyphenyl)-N-(1-propyl)piperidine.
    Molecular pharmacology, 1989, Volume: 35, Issue:1

    Topics: Allosteric Regulation; Animals; Binding Sites; Binding, Competitive; Dextromethorphan; Guinea Pigs; In Vitro Techniques; Levorphanol; Phenytoin; Piperazines; Piperidines; Receptors, Opioid; Receptors, sigma

1989
Sigma-receptors in endocrine organs: identification, characterization, and autoradiographic localization in rat pituitary, adrenal, testis, and ovary.
    Endocrinology, 1989, Volume: 124, Issue:3

    Topics: Adrenal Glands; Animals; Autoradiography; Brain Chemistry; Cell Membrane; Dibenzocycloheptenes; Dizocilpine Maleate; Female; Haloperidol; Hypophysectomy; Male; Ovary; Phencyclidine; Piperidines; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Testis; Tissue Distribution

1989
Acylation of sigma receptors by Metaphit, an isothiocyanate derivative of phencyclidine.
    European journal of pharmacology, 1989, Feb-28, Volume: 161, Issue:2-3

    Topics: Acylation; Animals; Behavior, Animal; Brain Chemistry; Electrophysiology; Guinea Pigs; In Vitro Techniques; Membranes; Phencyclidine; Piperidines; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine

1989
Evidence for a multi-site model of the rat brain sigma receptor.
    European journal of pharmacology, 1989, Apr-25, Volume: 163, Issue:2-3

    Topics: Animals; Brain; In Vitro Techniques; Male; Membranes; Models, Biological; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Synaptosomes; Ultraviolet Rays

1989
Vasoconstrictor-induced heterologous down-regulation of vascular atrial natriuretic peptide receptor.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: Angiotensin II; Animals; Arginine Vasopressin; Cyclic GMP; Humans; In Vitro Techniques; Iodine Radioisotopes; Muscle, Smooth, Vascular; Piperidines; Rats; Receptors, Atrial Natriuretic Factor; Receptors, Cell Surface; Tetradecanoylphorbol Acetate; Vasoconstrictor Agents

1989
Phencyclidine and sigma receptors in rat spinal cord: binding characterization and quantitative autoradiography.
    Synapse (New York, N.Y.), 1989, Volume: 4, Issue:1

    Topics: Animals; Autoradiography; Binding, Competitive; Ganglia, Spinal; Male; Narcotic Antagonists; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Spinal Cord

1989
Sertraline potently displaces (+)-[3H]3-PPP binding to sigma sites in rat brain.
    European journal of pharmacology, 1989, Jun-20, Volume: 165, Issue:2-3

    Topics: 1-Naphthylamine; Animals; Binding, Competitive; Brain Chemistry; In Vitro Techniques; Naphthalenes; Piperidines; Rats; Receptors, Opioid; Receptors, Opioid, delta; Serotonin Antagonists; Sertraline

1989
Differentiation of phencyclidine and sigma receptor types affecting the central inspiratory termination mechanism in cat.
    Life sciences, 1989, Volume: 45, Issue:14

    Topics: Animals; Brain Stem; Cats; Decerebrate State; Dextrorphan; Dibenzocycloheptenes; Dizocilpine Maleate; Guanidines; Phencyclidine; Phrenic Nerve; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Respiration

1989
Multiple affinity binding states of the sigma receptor: effect of GTP-binding protein-modifying agents.
    Molecular pharmacology, 1989, Volume: 36, Issue:4

    Topics: Animals; Binding, Competitive; Chlorpromazine; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Pentazocine; Pertussis Toxin; Piperidines; Rats; Receptors, Opioid; Receptors, sigma; Virulence Factors, Bordetella

1989
An examination of the putative sigma-receptor in the mouse isolated vas deferens.
    British journal of pharmacology, 1989, Volume: 98, Issue:2

    Topics: Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Muscle Contraction; Muscle, Smooth; Naloxone; Piperidines; Receptors, Opioid; Receptors, sigma; Vas Deferens

1989
(+)-[3H]3-(3-hydroxyphenyl)-N-(1-propyl)-piperidine binding to sigma receptors in mouse brain in vivo.
    European journal of pharmacology, 1989, Feb-28, Volume: 161, Issue:2-3

    Topics: Animals; Brain Chemistry; Dopamine Agents; Dose-Response Relationship, Drug; Mice; Piperidines; Rats; Receptors, Opioid; Receptors, Opioid, delta; Time Factors

1989
Selective sigma receptor agonist and antagonist affect dopamine neuronal activity.
    European journal of pharmacology, 1989, Apr-12, Volume: 163, Issue:1

    Topics: Animals; Antipsychotic Agents; Dopamine; In Vitro Techniques; Male; Membranes; Microelectrodes; Narcotic Antagonists; Narcotics; Neurons; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Spiperone

1989
Synthesis and evaluation of optically pure [3H]-(+)-pentazocine, a highly potent and selective radioligand for sigma receptors.
    FEBS letters, 1989, Jul-17, Volume: 251, Issue:1-2

    Topics: Animals; Apomorphine; Binding, Competitive; Brain; Cell Membrane; Chemical Phenomena; Chemistry; Dopamine Agents; Guanidines; Guinea Pigs; Hydroxides; Molecular Structure; Pentazocine; Phencyclidine; Piperidines; Potassium; Potassium Compounds; Receptors, Dopamine; Receptors, Opioid; Receptors, sigma; Tritium

1989
The partial dopamine receptor agonists (--)-3-PPP and transdihydrolisuride enhance prolactin secretion in female but not in male rats.
    Journal of neural transmission, 1989, Volume: 77, Issue:2-3

    Topics: Animals; Dopamine Agents; Dose-Response Relationship, Drug; Female; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Sex Factors

1989
Expression of (+)-3-PPP binding sites in the PC12 pheochromocytoma cell line.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: Adrenal Gland Neoplasms; Animals; Cell Line; Cell Membrane; Dopamine Agents; Humans; Pheochromocytoma; Piperidines; Radioligand Assay; Receptors, Drug

1989
Evidence for selective inhibition of limbic forebrain dopamine synthesis by 8-OH-DPAT in the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:5

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Corpus Striatum; Depression, Chemical; Dihydroxyphenylalanine; Dopamine; Ergolines; Hydrazines; Limbic System; Male; Naphthalenes; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Reserpine; Serotonin; Tetrahydronaphthalenes; Tryptophan Hydroxylase; Tyrosine 3-Monooxygenase

1989
Electrophysiological effects of selective sigma-receptor agonists, antagonists, and the selective phencyclidine receptor agonist MK-801 on midbrain dopamine neurons.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1989, Volume: 2, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Antipsychotic Agents; Carbazoles; Cell Membrane; Dibenzocycloheptenes; Dizocilpine Maleate; Dopamine; Dopamine Agents; Male; Neurons; Pentazocine; Phencyclidine; Piperidines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Substantia Nigra

1989
Occurrence of yawning and decrease of prolactin levels via stimulation of dopamine D2-receptors after administration of SND 919 in rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Azepines; Behavior, Animal; Benzothiazoles; Dopamine Agents; Male; Methyltyrosines; Piperidines; Pramipexole; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Thiazoles; Yawning

1989
Dopamine autoreceptor agonists attenuate spontaneous motor activity but not spontaneous fighting in individually-housed mice.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:2

    Topics: Aggression; Agonistic Behavior; Animals; Apomorphine; Catalepsy; Dopamine Agents; Dose-Response Relationship, Drug; Housing, Animal; Male; Mice; Motor Activity; Piperidines; Social Isolation; Stereoisomerism

1989
Influence of dopaminergic and noradrenergic systems on the release of opioid peptides in guinea-pig ileum.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Domperidone; Dopamine; Endorphins; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Myenteric Plexus; Naloxone; Norepinephrine; Piperidines; Prazosin; Receptors, Dopamine; Yohimbine

1989
DTG and (+)-3-PPP inhibit a ligand-activated hyperpolarization in mammalian neurons.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:3

    Topics: Animals; Brimonidine Tartrate; Dopamine Agents; Enkephalin, Methionine; Guanidines; Haloperidol; Male; Membrane Potentials; Neurons; Norepinephrine; Piperidines; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Serotonin

1989
Inhibition by pertussis toxin of the soporific effects induced by stimulation of dopamine D2 autoreceptors in the ventral tegmental area in rats.
    Neuropharmacology, 1989, Volume: 28, Issue:9

    Topics: Adenylate Cyclase Toxin; Animals; Apomorphine; Electrocardiography; Male; Pertussis Toxin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tegmentum Mesencephali; Time Factors; Virulence Factors, Bordetella

1989
The enhanced responsiveness of hypophyseal DA receptors in female rats induced by repeated reserpine treatment is not due to decreased oestrogen secretion.
    Pharmacology & toxicology, 1989, Volume: 65, Issue:3

    Topics: Animals; Estradiol; Estrogens; Female; Lisuride; Ovariectomy; Piperidines; Pituitary Gland, Posterior; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine

1989
Structural determinants of sigma receptor affinity.
    Molecular pharmacology, 1987, Volume: 32, Issue:6

    Topics: Animals; Brain; Hydrogen-Ion Concentration; Male; Molecular Conformation; Narcotics; Phenothiazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship; Tritium

1987
Limited stimulus generalization between delta 9-THC and diazepam in pigeons and gerbils.
    Psychopharmacology, 1988, Volume: 94, Issue:3

    Topics: Animals; Benzodiazepinones; Columbidae; Diazepam; Discrimination, Psychological; Dronabinol; Generalization, Stimulus; Gerbillinae; Male; Piperidines; Receptors, GABA-A

1988
Regulation of the binding of sigma- and phencyclidine (PCP)-receptor ligands in rat brain membranes by guanine nucleotides and ions.
    Neuroscience letters, 1988, Feb-15, Volume: 85, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Cations; Guanine Nucleotides; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Receptors, Neurotransmitter; Receptors, Phencyclidine; Subcellular Fractions

1988
Comparison of the actions of phencyclidine and sigma ligands on CA1 hippocampal pyramidal neurons in the rat.
    Neuropharmacology, 1988, Volume: 27, Issue:11

    Topics: Action Potentials; Animals; Aspartic Acid; Guanidines; Hippocampus; Male; N-Methylaspartate; Neurons; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1988
Up-regulation of rat cortical sigma receptors after subchronic administration of rimcazole and 1,3-di(2-tolyl)guanidine.
    Neuropharmacology, 1988, Volume: 27, Issue:11

    Topics: Animals; Carbazoles; Guanidines; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma

1988
Sigma and PCP receptors in human frontal cortex membranes.
    European journal of pharmacology, 1988, Sep-23, Volume: 154, Issue:3

    Topics: Brain; Dibenzocycloheptenes; Dizocilpine Maleate; Humans; In Vitro Techniques; Membranes; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1988
Relative selectivity of 6,7-dihydroxy-2-dimethylaminotetralin, N-n-propyl-3-(3-hydroxyphenyl)piperidine, N-n-propylnorapomorphine and pergolide as agonists at striatal dopamine autoreceptors and postsynaptic dopamine receptors.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:2

    Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Haloperidol; Homovanillic Acid; Male; Naphthalenes; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sodium Oxybate; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase

1985
Effect of dopaminergic drugs on striatal acetylcholine concentration.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:1

    Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1985
In-vitro and in-vivo metabolism of the presynaptic dopamine agonist 3-PPP to a catecholic analogue in rats.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:5

    Topics: Animals; Biotransformation; Catecholamines; Female; Hydrogen-Ion Concentration; Hydroxylation; In Vitro Techniques; Kinetics; Methylation; Microsomes, Liver; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Stereoisomerism

1985
Is inhibition of striatal synaptosomal tyrosine hydroxylation by dopamine agonists a measure of dopamine autoreceptor function?
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Azepines; Corpus Striatum; Depression, Chemical; Dopamine; Ergolines; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Synaptosomes; Tyrosine 3-Monooxygenase

1985
Performance deficit induced by low doses of dopamine agonists in rats. Toward a model for approaching the neurobiology of negative schizophrenic symptomatology?
    Biological psychiatry, 1986, Volume: 21, Issue:1

    Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Disease Models, Animal; Male; Phenothiazines; Pimozide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reinforcement Schedule; Reinforcement, Psychology; Schizophrenia; Schizophrenic Psychology; Sulpiride

1986
Investigation of dopamine content, synthesis, and release in the rabbit retina in vitro: II. Effects of high potassium, adenylate cyclase activators, and N-n-propyl-3-(3-hydroxyphenyl) piperidine.
    Journal of neurochemistry, 1986, Volume: 47, Issue:4

    Topics: 2-Chloroadenosine; Adenosine; Adenylyl Cyclases; Animals; Calcium; Colforsin; Dopamine; Enzyme Activation; Female; Male; Piperidines; Potassium; Rabbits; Retina; Tyrosine 3-Monooxygenase; Vasoactive Intestinal Peptide

1986
Effects of dopaminomimetics on the secretion of VIP-like immunoreactivity in conscious dogs.
    Peptides, 1986, Volume: 7 Suppl 1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Apomorphine; Benzazepines; Dogs; Ergolines; Nitroglycerin; Pergolide; Piperidines; Prazosin; Receptors, Dopamine; Somatostatin; Vasoactive Intestinal Peptide

1986
Two automated locomotor activity tests for dopamine autoreceptor agonists.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Drug Evaluation, Preclinical; Exploratory Behavior; Indoles; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1986
1,3-Di(2-[5-3H]tolyl)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:22

    Topics: Animals; Antipsychotic Agents; Benzomorphans; Binding Sites; Brain; Guanidines; Guinea Pigs; Hallucinogens; In Vitro Techniques; Ligands; Male; Morphinans; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Tritium

1986
Permissive role of D-1 receptor stimulation by endogenous dopamine for the expression of postsynaptic D-2-mediated behavioural responses. Yawning in rats.
    European journal of pharmacology, 1987, Feb-10, Volume: 134, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Azepines; Benzazepines; Brain Chemistry; Dopamine; Ergolines; Kainic Acid; Ketanserin; Male; Metergoline; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sulpiride; Yawning

1987
Comparison of changes in locomotor activity with striatal homovanillic acid and 3,4-dihydroxyphenylacetic acid concentrations following the bilateral intranigral injection of dopamine agonist drugs in rats.
    The Journal of pharmacy and pharmacology, 1987, Volume: 39, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Female; Homovanillic Acid; Motor Activity; Phenylacetates; Piperidines; Rats; Rats, Inbred Strains; Substantia Nigra; Sucrose

1987
Relationship between receptor occupancy and response at striatal dopamine autoreceptors.
    Molecular pharmacology, 1987, Volume: 31, Issue:6

    Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Homeostasis; Hydrazines; Levodopa; Male; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1987
Effects of apomorphine and (+/-)-3-(3-hydroxyphenyl)-N-n-propylpiperidine, injected into the striatum, on the caudate spindle in the rat.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dopamine; Electric Stimulation; Electrophysiology; Injections; Male; Piperidines; Rats; Rats, Inbred Strains

1987
Behavioural and ECoG spectrum power effects after intraventricular injection of drugs altering dopaminergic transmission in rats.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Benzazepines; Brain; Catheters, Indwelling; Dopamine; Dose-Response Relationship, Drug; Electroencephalography; Electrophysiology; Injections, Intraventricular; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Synaptic Transmission

1987
Pharmacological specificity of some psychotomimetic and antipsychotic agents for the sigma and PCP binding sites.
    Life sciences, 1988, Volume: 42, Issue:7

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Haloperidol; In Vitro Techniques; Male; Phenazocine; Phencyclidine; Piperidines; Psychotropic Drugs; Rats; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1988
Dopamine D-2 receptors in the ventral tegmental area mediate behavioural and electrocortical sleep of dopaminergic drugs in rats.
    Pharmacological research communications, 1988, Volume: 20, Issue:12

    Topics: Animals; Apomorphine; Behavior, Animal; Cerebral Cortex; Dopamine Agents; Electric Stimulation; Electroencephalography; Piperidines; Rats; Receptors, Dopamine; Sleep; Tegmentum Mesencephali

1988
Dopamine D2 receptors in brain and anterior pituitary recognize agonist and antagonist actions of (-)-3-PPP.
    Journal of neural transmission, 1985, Volume: 64, Issue:1

    Topics: Animals; Brain; Cattle; Caudate Nucleus; Cell Membrane; Corpus Striatum; Dopamine Antagonists; Guanine Nucleotides; Male; Piperidines; Pituitary Gland, Anterior; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Sodium Chloride; Swine

1985
Ventral tegmental area: site through which dopamine D2-receptor agonists evoke behavioural and electrocortical sleep in rats.
    British journal of pharmacology, 1988, Volume: 95, Issue:3

    Topics: Animals; Apomorphine; Cerebral Cortex; Electroencephalography; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sleep; Sulpiride; Tegmentum Mesencephali

1988
Phencyclidine and sigma opiate receptors in brain: biochemical and autoradiographical differentiation.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Autoradiography; Brain; Humans; In Vitro Techniques; Membranes; Phenazocine; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine

1985
Interactions between delta 9-tetrahydrocannabinol and cannabidiol as evaluated by drug discrimination procedures in rats and pigeons.
    Neuropharmacology, 1986, Volume: 25, Issue:2

    Topics: Animals; Cannabidiol; Cannabinoids; Columbidae; Discrimination Learning; Discrimination, Psychological; Dronabinol; Male; Piperidines; Rats; Rats, Inbred Strains; Species Specificity; Time Factors

1986
Autoradiographic localization of sigma receptor binding sites in guinea pig and rat central nervous system with (+)3H-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:6

    Topics: Animals; Autoradiography; Binding Sites; Brain Chemistry; Guinea Pigs; Male; Piperidines; Rats; Receptors, Opioid; Spinal Cord; Tritium

1986
Sigma receptors on NCB-20 hybrid neurotumor cells labeled with (+)[3H]SKF 10,047 and (+)[3H]3-PPP.
    European journal of pharmacology, 1986, May-13, Volume: 124, Issue:1-2

    Topics: Animals; Brain; Cells, Cultured; Cricetinae; Cricetulus; Hybrid Cells; Kinetics; Neuroblastoma; Phenazocine; Phencyclidine; Piperidines; Receptors, Opioid; Receptors, Opioid, delta; Stereoisomerism

1986
Pharmacological and autoradiographic discrimination of sigma and phencyclidine receptor binding sites in brain with (+)-[3H]SKF 10,047, (+)-[3H]-3-[3-hydroxyphenyl]-N-(1-propyl)piperidine and [3H]-1-[1-(2-thienyl)cyclohexyl]piperidine.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; In Vitro Techniques; Kinetics; Male; Phenazocine; Phencyclidine; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism

1986
(+)-3-PPP antagonizes the discriminative stimulus effects of (+)-N-allylnormetazocine.
    European journal of pharmacology, 1986, Aug-15, Volume: 127, Issue:3

    Topics: Animals; Binding Sites; Conditioning, Operant; Discrimination, Psychological; Generalization, Stimulus; Phenazocine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta

1986
Antagonist effects of the enantiomers of 3-PPP towards alpha 1-adrenoceptors coupled to inositol phospholipid breakdown in the rat cerebral cortex.
    Pharmacology & toxicology, 1987, Volume: 60, Issue:5

    Topics: Animals; Antiparkinson Agents; Atropine; Carbachol; Cerebral Cortex; Haloperidol; In Vitro Techniques; Inositol Phosphates; Male; Norepinephrine; Phenoxybenzamine; Piperidines; Prazosin; Raclopride; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Salicylamides; Stereoisomerism; Sugar Phosphates

1987
Both the sigma receptor-specific ligand (+)3-PPP and the PCP receptor-specific ligand TCP act in the mouse vas deferens via augmentation of electrically evoked norepinephrine release.
    European journal of pharmacology, 1987, Jun-26, Volume: 138, Issue:3

    Topics: Animals; Electric Stimulation; In Vitro Techniques; Male; Mice; Muscle Contraction; Norepinephrine; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Vas Deferens

1987
Alterations in motor behaviour produced by the isomers of 3-PPP in the MPTP-treated marmoset.
    European journal of pharmacology, 1986, Feb-11, Volume: 121, Issue:1

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Callitrichinae; Female; Isomerism; Levodopa; Male; Motor Activity; Piperidines; Pyridines; Receptors, Dopamine; Time Factors

1986
Anxiolytic-like action of the 3-PPP enantiomers in the Vogel conflict paradigm.
    Psychopharmacology, 1987, Volume: 92, Issue:3

    Topics: Animals; Arousal; Avoidance Learning; Conflict, Psychological; Dose-Response Relationship, Drug; Drinking; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1987
7-[3-(4-[2,3-Dimethylphenyl]piperazinyl)propoxy]-2(1H)-quinolinone (OPC-4392), a presynaptic dopamine autoreceptor agonist and postsynaptic D2 receptor antagonist.
    Life sciences, 1988, Volume: 42, Issue:20

    Topics: Animals; Apomorphine; Brain; Corpus Striatum; Diencephalon; Dihydroxyphenylalanine; Frontal Lobe; Hydroxydopamines; Kainic Acid; Kinetics; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxidopamine; Piperazines; Piperidines; Quinolines; Quinolones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Telencephalon

1988
Dopamine (DA) autoreceptor efficacy of 3-PPP enantiomers after short-term synaptic DA deprivation.
    European journal of pharmacology, 1988, Aug-02, Volume: 152, Issue:3

    Topics: Animals; Antiparkinson Agents; Behavior, Animal; Brain; Brain Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Limbic System; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism; Synapses

1988
Heterogeneous rotational responsiveness in 6-hydroxydopamine-denervated rats: pharmacological and neurochemical characterization.
    Psychopharmacology, 1988, Volume: 96, Issue:4

    Topics: Animals; Apomorphine; Benzopyrans; Brain Chemistry; Corpus Striatum; Dopamine; Ergolines; Hydroxydopamines; Male; Oxidopamine; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Rotation; Stereotyped Behavior; Sympathectomy, Chemical

1988
Effects of intraperitoneal administration of apomorphine and the isomers of 3-(1-propyl-3-piperidinyl)phenol on the firing activity of substantia nigra dopamine neurons: comparison of agonist efficacies and development of acute tolerance.
    Neuropharmacology, 1988, Volume: 27, Issue:9

    Topics: Action Potentials; Animals; Apomorphine; Drug Tolerance; Injections, Intraperitoneal; Injections, Intravenous; Male; Neurons; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Substantia Nigra

1988
Suppression of neuroleptic-induced persistent abnormal movements in Cebus apella monkeys by enantiomers of 3-PPP.
    Journal of neural transmission, 1988, Volume: 74, Issue:2

    Topics: Animals; Cebus; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Female; Fluphenazine; Piperidines; Stereoisomerism; Time Factors

1988
Pharmacological profile of dopamine receptor agonists as studied by brain dialysis in behaving rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Azepines; Behavior, Animal; Benzazepines; Brain; Dialysis; Dopamine; Ergolines; Homovanillic Acid; Isomerism; Male; Motor Activity; Neurons; Pergolide; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors

1988
The intrinsic activity of (-)-3-PPP (preclamol) on pituitary DA receptors in female rats is enhanced following chronic DA depletion.
    Life sciences, 1988, Volume: 42, Issue:5

    Topics: Animals; Dopamine; Female; Hyperprolactinemia; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine

1988
Neuropharmacology and stereochemistry of dopamine receptor agonist and antagonist enantiomeric pairs.
    Journal of receptor research, 1988, Volume: 8, Issue:1-4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aporphines; Dopamine; Molecular Conformation; Naphthalenes; Piperidines; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes

1988
O-methylated catechol metabolites of 3-(3-hydroxy-phenyl)-N-propyl piperidine (3-PPP): synthesis, pharmacological and acute toxicological evaluation.
    Acta pharmaceutica Suecica, 1987, Volume: 24, Issue:4

    Topics: Animals; Antiparkinson Agents; Chemical Phenomena; Chemistry; Female; Male; Piperidines; Rats; Rats, Inbred Strains

1987
Apomorphine-induced penile erection and yawning: site of action in brain.
    Brain research, 1987, Jul-07, Volume: 415, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Brain; Dopamine; Dopamine Antagonists; Ergolines; Male; Microinjections; Paraventricular Hypothalamic Nucleus; Penile Erection; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Yawning

1987
Compounds with selectivity for dopamine autoreceptors: effects on prolactin secretion in male and female rats.
    Clinical neuropharmacology, 1986, Volume: 9 Suppl 4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Azepines; Female; Male; Phenanthrenes; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tetrahydronaphthalenes

1986
Effects of raclopride on exploratory locomotor activity, treadmill locomotion, conditioned avoidance behaviour and catalepsy in rats: behavioural profile comparisons between raclopride, haloperidol and preclamol.
    Pharmacology & toxicology, 1987, Volume: 60, Issue:5

    Topics: Animals; Avoidance Learning; Behavior, Animal; Catalepsy; Exploratory Behavior; Haloperidol; Male; Motor Activity; Piperidines; Raclopride; Rats; Rats, Inbred Strains; Salicylamides; Scopolamine

1987
Partial protection against hyperbaric oxygen induced convulsions by dopaminergic agents in mice: possible involvement of autoreceptors?
    Journal of neural transmission, 1987, Volume: 69, Issue:3-4

    Topics: Animals; Antiparkinson Agents; Apomorphine; Body Temperature; Dose-Response Relationship, Drug; Haloperidol; Hyperbaric Oxygenation; Levodopa; Male; Mice; Mice, Inbred CBA; Piperidines; Reaction Time; Receptors, Dopamine; Respiration; Seizures

1987
Carbamate ester derivatives as potential prodrugs of the presynaptic dopamine autoreceptor agonist (-)-3-(3-hydroxyphenyl)-N-propylpiperidine.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:11

    Topics: Animals; Carbamates; Pharmaceutical Preparations; Piperidines; Prodrugs; Rats; Rats, Inbred Strains; Receptors, Dopamine; Structure-Activity Relationship

1987
On the mode of action of six putative dopamine receptor agonists on suppression of exploratory behaviour in rats.
    Psychopharmacology, 1987, Volume: 91, Issue:2

    Topics: Animals; Bromocriptine; Ergolines; Exploratory Behavior; Habituation, Psychophysiologic; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1987
The intrinsic activities of the partial dopamine receptor agonists (-)-3-PPP and TDHL on pituitary dopamine receptors are lower in female than in male rats.
    European journal of pharmacology, 1987, Oct-06, Volume: 142, Issue:1

    Topics: Animals; Antiparkinson Agents; Ergolines; Female; In Vitro Techniques; Lisuride; Male; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sex Factors; Stereoisomerism

1987
Differential electrophysiological effects of 3-PPP and its enantiomers on dopamine autoreceptors and postsynaptic receptors.
    European journal of pharmacology, 1986, May-13, Volume: 124, Issue:1-2

    Topics: Action Potentials; Animals; Apomorphine; Electrodes, Implanted; Globus Pallidus; Male; Neurons; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Substantia Nigra; Synapses

1986
An automatic device for measuring speed of movement and time spent at rest: its application to testing dopaminergic drugs.
    Physiology & behavior, 1986, Volume: 37, Issue:1

    Topics: Animals; Dextroamphetamine; Dose-Response Relationship, Drug; Female; Haloperidol; Motor Activity; Neurophysiology; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1986
A stereochemical explanation of the dopamine agonist and antagonist activity of stereoisomeric pairs.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Apomorphine; Chemical Phenomena; Chemistry; Dopamine; Dopamine Antagonists; Molecular Conformation; Naphthalenes; Piperidines; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes; Thermodynamics

1986
Stereoselective inhibition of prolactin secretion by (-)-HW-165, a novel 3-PPP congener; further support for similarities between central DA autoreceptors and pituitary lactotroph DA receptors.
    European journal of pharmacology, 1986, Jun-24, Volume: 125, Issue:3

    Topics: 4-Butyrolactone; Animals; Apomorphine; Depression, Chemical; Male; Phenanthrenes; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism

1986
Enantiomers of 3-(3,4-dihydroxyphenyl)- and 3-(3-hydroxyphenyl)-N-n-propylpiperidine: central pre- and postsynaptic dopaminergic effects and pharmacokinetics.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:10

    Topics: Animals; Brain; Kinetics; Male; Methylation; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1986
A molecular mechanics approach to the understanding of presynaptic selectivity for centrally acting dopamine receptor agonists of the phenylpiperidine series.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:10

    Topics: Brain; Models, Molecular; Molecular Conformation; Piperidines; Receptors, Dopamine; Structure-Activity Relationship

1986
Central dopaminergic properties of HW-165 and its enantiomers; trans-octahydrobenzo(f)quinoline congeners of 3-PPP.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:3

    Topics: 4-Butyrolactone; Animals; Behavior, Animal; Catecholamines; Corpus Striatum; Limbic System; Male; Motor Activity; Phenanthrenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism

1986
Sexually differentiated actions of 3-PPP enantiomers on prolactin secretion.
    Neuropharmacology, 1986, Volume: 25, Issue:8

    Topics: 4-Butyrolactone; Animals; Female; Furans; Male; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sex Factors; Stereoisomerism

1986
Electrophysiological effects of the enantiomers of 3-PPP on neurons in the locus coeruleus of the rat.
    Neuropharmacology, 1986, Volume: 25, Issue:9

    Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Haloperidol; Injections, Intravenous; Iontophoresis; Locus Coeruleus; Male; Neurons; Piperidines; Prazosin; Rats; Rats, Inbred Strains; Stereoisomerism; Yohimbine

1986
(+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine [(+)-3-PPP] but not (-)-3-PPP produces (+)-N-allylnormetazocine-like (SKF 10,047) discriminative stimuli.
    Life sciences, 1986, Dec-29, Volume: 39, Issue:26

    Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Isomerism; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred F344

1986
Indolizidine and quinolizidine derivatives of the dopamine autoreceptor agonist 3-(3-hydroxyphenyl)-N-n-propylpiperidine (3-PPP).
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Methyltyrosines; Molecular Conformation; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Structure-Activity Relationship

1987
Pharmacological properties of presynaptic dopamine receptor agonists.
    Psychopharmacology. Supplementum, 1985, Volume: 2

    Topics: Animals; Binding, Competitive; Brain; Corpus Striatum; Dogs; Dopamine; Piperidines; Prolactin; Rats; Receptors, Dopamine; Stereoisomerism; Substantia Nigra; Synapses; Vomiting

1985
Dopaminergic agents including 3-PPP and its enantiomers on medial septal self-stimulation.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Appetite Depressants; Benzazepines; Dextroamphetamine; Drug Interactions; Haloperidol; Male; Nomifensine; Piperidines; Rats; Receptors, Dopamine; Self Stimulation; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes

1985
Development of dopamine autoreceptors in the postnatal rat brain.
    Journal of neural transmission, 1985, Volume: 62, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Age Factors; Animals; Brain; Brain Chemistry; Dihydroxyphenylalanine; Motor Activity; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1985
Synthesis and dopamine autoreceptor activity of a 5-(methylmercapto)methyl-substituted derivative of (+/-)-3-PPP (3-(3-hydroxyphenyl)-1-n-propylpiperidine).
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: 4-Butyrolactone; Animals; Chemical Phenomena; Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Mice; Piperidines; Rats; Receptors, Dopamine; Structure-Activity Relationship

1985
Sub-chronic administration of (-)-3-PPP and central dopamine receptor sensitivity changes.
    Journal of neural transmission, 1985, Volume: 64, Issue:3-4

    Topics: Animals; Body Weight; Brain; Corpus Striatum; Dihydroxyphenylalanine; Limbic System; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1985
Dopamine receptors mediating yawning: are they autoreceptors?
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: Animals; Domperidone; Drug Synergism; Haloperidol; Male; Methyltyrosines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reflex; Reserpine; Stereoisomerism; Sulpiride

1986
Agonist and antagonist effects of 3-PPP enantiomers on functional dopamine autoreceptors and postsynaptic dopamine receptors in vitro.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Acetylcholine; Animals; Cholera Toxin; Corpus Striatum; Dopamine; In Vitro Techniques; Male; Melanocyte-Stimulating Hormones; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride

1985
Dopamine receptor-mediated hypothermia induced in rats by (+)-, but not by (-)-3-PPP.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Animals; Apomorphine; Biogenic Amines; Body Temperature; Brain Chemistry; Dose-Response Relationship, Drug; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1985
Dopamine autoreceptors and the effects of drugs on locomotion and dopamine synthesis.
    British journal of pharmacology, 1985, Volume: 84, Issue:4

    Topics: alpha-Methyltyrosine; Animals; Dopamine; Levodopa; Locomotion; Male; Methyltyrosines; Mice; Mice, Inbred Strains; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1985
Lack of effect of intranigral administration of a dopamine analogue, (+/-)-3-(3-hydroxyphenyl)-N,n-propylpiperidine [(+/-)-3-PPP], on nigrostriatal dopamine neurones.
    Neuroscience letters, 1985, May-01, Volume: 56, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Female; Homovanillic Acid; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra

1985
Modifications of sleep parameters in the rat by (+)- and (-)-3-PPP.
    Journal of neural transmission, 1985, Volume: 62, Issue:3-4

    Topics: Animals; Isomerism; Male; Piperidines; Rats; Rats, Inbred Strains; Reaction Time; Sleep; Sleep Stages

1985
An electrophysiological analysis of the actions of the 3-PPP enantiomers on the nigrostriatal dopamine system.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Caudate Nucleus; Chloral Hydrate; Dopamine; Dose-Response Relationship, Drug; Electrophysiology; Iontophoresis; Male; Piperidines; Rats; Rats, Inbred Strains; Stereoisomerism; Substantia Nigra

1985
Involvement of catechol-O-methyl transferase in the metabolism of the putative dopamine autoreceptor agonist 3-PPP(3-(3-hydroxyphenyl)-N-n-propylpiperidine).
    Biochemical pharmacology, 1985, Oct-01, Volume: 34, Issue:19

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Catechol O-Methyltransferase; Cattle; Dopamine; Kinetics; Liver; Methylation; Piperidines; Pyrogallol

1985
Effects of the enantiomers of 3-PPP on DA1 and DA2 dopamine receptors in the dog.
    European journal of pharmacology, 1985, Aug-27, Volume: 114, Issue:3

    Topics: Animals; Dogs; Femoral Artery; Models, Biological; Piperidines; Receptors, Dopamine; Regional Blood Flow; Renal Artery; Stereoisomerism

1985
In vivo displacement by 3-PPP enantiomers of N,N-dipropyl-5,6-ADTN from dopamine receptor-binding sites in rat striatum.
    Journal of neural transmission, 1985, Volume: 64, Issue:3-4

    Topics: Animals; Binding, Competitive; Brain; Cerebellum; Corpus Striatum; Haloperidol; Isomerism; Male; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tetrahydronaphthalenes

1985
Resolved 3-(3-hydroxyphenyl)-N-n-propylpiperidine and its analogues: central dopamine receptor activity.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:8

    Topics: Animals; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Male; Motor Activity; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Reserpine; Serotonin; X-Ray Diffraction

1984
Psychotomimetic opiate receptors labeled and visualized with (+)-[3H]3-(3-hydroxyphenyl)-N-(1-propyl)piperidine.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:15

    Topics: Animals; Brain Mapping; Brain Stem; Cerebellum; Guinea Pigs; Haloperidol; Hypothalamus; Limbic System; Mesencephalon; Piperidines; Rats; Receptors, Dopamine; Receptors, Opioid; Stereoisomerism

1984
Differential effects of the stereoisomers of 3PPP on dopaminergic and cholinergic neurotransmission in superfused slices of the corpus striatum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 327, Issue:1

    Topics: Acetylcholine; Animals; Corpus Striatum; Dextroamphetamine; Dopamine; Electric Stimulation; In Vitro Techniques; Male; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Synaptic Transmission; Tritium

1984
(+)- and (-)-3-PPP exhibit different intrinsic activity at striatal dopamine autoreceptors controlling dopamine synthesis.
    European journal of pharmacology, 1984, Oct-30, Volume: 106, Issue:1

    Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine; Isomerism; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter

1984
3-PPP, a new centrally acting DA-receptor agonist with selectivity for autoreceptors.
    Life sciences, 1981, Mar-16, Volume: 28, Issue:11

    Topics: Animals; Behavior, Animal; Brain; Dopamine; Drug Interactions; Humans; Kinetics; Male; Motor Activity; Piperidines; Rats; Receptors, Dopamine; Stereotyped Behavior; Tyrosine 3-Monooxygenase

1981
Is 3-PPP a potential antipsychotic agent? Evidence from animal behavioral studies.
    European journal of pharmacology, 1982, Sep-10, Volume: 83, Issue:1-2

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Behavior, Animal; Dextroamphetamine; Humans; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Stereotyped Behavior; Time Factors

1982
LY141865, a D2-dopamine agonist, increases acetylcholine concentration in rat corpus striatum.
    The Journal of pharmacy and pharmacology, 1983, Volume: 35, Issue:5

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Corpus Striatum; Ergolines; Male; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine

1983
Different actions of TL-99 and 3-PPP in producing contraversive turning in the 6-OHDA-lesioned rat.
    European journal of pharmacology, 1983, Sep-02, Volume: 92, Issue:3-4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apomorphine; Female; Hydroxydopamines; Motor Activity; Naphthalenes; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Tetrahydronaphthalenes; Yohimbine

1983
Differential effects of the enantiomers of 3-(3-hydroxyphenyl)-N-n-propylpiperidine (3-PPP) at dopamine receptor sites.
    European journal of pharmacology, 1983, Sep-02, Volume: 92, Issue:3-4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Homovanillic Acid; Male; Mice; Molecular Conformation; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Synaptosomes; Tyrosine 3-Monooxygenase

1983
The effect of the enantiomers of 3-PPP on conditioned avoidance responding in the rat.
    Psychopharmacology, 1983, Volume: 81, Issue:1

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Catalepsy; Humans; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Stereoisomerism; Time Factors

1983
On the mode of action of 3-(3-hydroxyphenyl)-N-n-propylpiperidine, 3-PPP, and its enantiomers. With particular reference to dopaminergic mechanisms in the central nervous system.
    Acta physiologica Scandinavica. Supplementum, 1983, Volume: 517

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Behavior, Animal; Brain; Cyclic AMP; Escape Reaction; Humans; Locomotion; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Stereotyped Behavior

1983
Dopamine receptor agonistic and antagonistic effects of 3-PPP enantiomers.
    Psychopharmacology, 1983, Volume: 81, Issue:3

    Topics: Adenylyl Cyclases; Animals; Antiemetics; Antipsychotic Agents; Catalepsy; Dogs; Dopamine; Female; Guinea Pigs; Humans; Male; Mice; Motor Activity; Norepinephrine; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Serotonin; Stereoisomerism; Stereotyped Behavior; Synaptosomes

1983
Effects of apomorphine, TL-99 and 3-PPP on yawning in rats.
    Neuropharmacology, 1984, Volume: 23, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apomorphine; Behavior, Animal; Haloperidol; Male; Naphthalenes; Piperidines; Rats; Tetrahydronaphthalenes

1984
Effects of S (+)-3-phenethyl-PP, a putative dopamine autoreceptors agonist with greater autoreceptor selectivity than 3-PPP enantiomers.
    European journal of pharmacology, 1984, Jun-15, Volume: 102, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antiemetics; Catalepsy; Dogs; Dopamine; Female; Guinea Pigs; Histamine Antagonists; Humans; Male; Mice; Motor Activity; Norepinephrine; Parasympatholytics; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Stereotyped Behavior; Synaptosomes

1984
Presynaptic dopaminergic agonists modify brain glucose metabolism in a way similar to the neuroleptics.
    Neuroscience letters, 1984, Sep-07, Volume: 50, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Catecholamines; Ergolines; Glucose; Naphthalenes; Piperidines; Rats; Reserpine; Tetrahydronaphthalenes

1984
Dopamine agonists stimulate protein carboxylmethylation in striatal synaptosomes.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:3

    Topics: Animals; Apomorphine; Butaclamol; Corpus Striatum; Dopamine; Hydroxydopamines; In Vitro Techniques; Male; Nerve Tissue Proteins; Piperidines; Potassium; Protein Methyltransferases; Protein O-Methyltransferase; Rats; Rats, Inbred Strains; S-Adenosylhomocysteine; S-Adenosylmethionine; Synaptosomes

1982
The effects of SCH 23390, YM 09151-2, (+)- and (-)-3-PPP and some classical neuroleptics on D-1 and D-2 receptors in rat neostriatum in vitro.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Antipsychotic Agents; Aporphines; Benzamides; Benzazepines; Caudate Nucleus; Chlorpromazine; Clozapine; Flupenthixol; Haloperidol; In Vitro Techniques; Male; Piperidines; Potassium; Putamen; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1984
Interaction of the putative dopamine autoreceptor agonists, 3-PPP and TL-99, with the dopamine-sensitive adenylate cyclase of carp retina.
    European journal of pharmacology, 1982, Feb-05, Volume: 77, Issue:4

    Topics: Adenylyl Cyclases; Animals; Carps; Cyclic AMP; Enzyme Activation; Naphthalenes; Piperidines; Receptors, Dopamine; Retina; Tetrahydronaphthalenes

1982
A behavioural study of the changes in the central nervous system of mice after subchronic treatment with the selective dopamine autoreceptor agonist 3-PPP (dl-3-[3-hydroxyphenyl]-N-n-propylpiperidine).
    Journal of neural transmission, 1982, Volume: 53, Issue:4

    Topics: Animals; Apomorphine; Behavior, Animal; Dextroamphetamine; Dose-Response Relationship, Drug; Male; Motor Activity; Muridae; Piperidines; Receptors, Dopamine; Synaptic Transmission

1982
Inhibition of postsynaptic dopamine-sensitive adenylate cyclase in carp retina by the putative dopamine autoreceptor agonist, 3-PPP.
    European journal of pharmacology, 1982, Aug-13, Volume: 82, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Carps; Cyclic AMP; Cyprinidae; In Vitro Techniques; Piperidines; Receptors, Dopamine; Retina; Synapses

1982
Postsynaptic dopamine agonist properties of TL-99 are revealed by yohimbine co-treatment.
    European journal of pharmacology, 1983, Mar-04, Volume: 87, Issue:4

    Topics: Animals; Male; Motor Activity; Naphthalenes; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Rotation; Tetrahydronaphthalenes; Yohimbine

1983
3-PPP antagonizes the in vitro effects of D-1 and D-2 dopamine receptor agonists in rat neostriatum.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Acetylcholine; Animals; Corpus Striatum; Cyclic AMP; In Vitro Techniques; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1983
In vitro effect of the racemic mixture and the (-)enantiomer of N-n-propyl-3-(3-hydroxyphenyl)-piperidine (3-PPP) on postsynaptic dopamine receptors and on a presynaptic dopamine autoreceptor.
    Journal of neural transmission, 1983, Volume: 58, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Cyclic AMP; Male; Models, Neurological; Piperidines; Rats; Receptors, Dopamine; Stereoisomerism

1983
Differential effects of the enantiomers of 3-PPP on dopamine D1-receptors of isolated rabbit retina.
    Journal of neural transmission, 1984, Volume: 59, Issue:1

    Topics: Animals; Cyclic AMP; Dopamine; In Vitro Techniques; Isomerism; Piperidines; Rabbits; Receptors, Dopamine; Receptors, Dopamine D1; Retina

1984
trans-N-n-Propyl-7-hydroxy-octahydrobenzo(f)quinoline, a rigid 3-PPP analogue with greater potency but lack of selectivity for dopamine autoreceptors.
    European journal of pharmacology, 1983, Mar-04, Volume: 87, Issue:4

    Topics: 4-Butyrolactone; Animals; Corpus Striatum; Dihydroxyphenylalanine; Female; Hydroxyquinolines; Male; Mice; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine

1983
Central dopamine receptor agonist and antagonist actions of the enantiomers of 3-PPP.
    Psychopharmacology, 1983, Volume: 81, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Biogenic Amines; Brain Chemistry; Dextroamphetamine; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism

1983
Dopamine receptor agonists: intrinsic activity vs. state of receptor.
    Journal of neural transmission, 1983, Volume: 57, Issue:4

    Topics: Animals; Apomorphine; Brain; Denervation; Exploratory Behavior; Hydroxydopamines; Oxidopamine; Piperidines; Prolactin; Rats; Receptors, Dopamine; Stereoisomerism; Sympathectomy, Chemical

1983
Postsynaptic dopamine agonistic effects of 3-PPP enantiomers revealed by bilateral 6-hydroxy-dopamine lesions and by chronic reserpine treatment in rats.
    Journal of neural transmission, 1984, Volume: 60, Issue:3-4

    Topics: Animals; Antiparkinson Agents; Apomorphine; Behavior, Animal; Drug Interactions; Hydroxydopamines; Male; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism; Stimulation, Chemical

1984
Effects of (-)3-PPP on acquisition and retention of a conditioned avoidance response in the rat.
    Psychopharmacology, 1984, Volume: 84, Issue:4

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Discrimination Learning; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains

1984
Evidence for heterogeneous rotational responsiveness to apomorphine, 3-PPP and SKF 38393 in 6-hydroxydopamine-denervated rats.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Clozapine; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Piperidines; Postural Balance; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sympathectomy, Chemical

1984
Antagonism by haloperidol of the suppression of exploratory locomotor activity induced by the local application of (-)3-(3-hydroxyphenyl)-N-n-propylpiperidine into the nucleus accumbens of the rat.
    Experientia, 1984, Aug-15, Volume: 40, Issue:8

    Topics: Animals; Exploratory Behavior; Haloperidol; Male; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Septal Nuclei

1984
The yawning-penile erection syndrome as a model for putative dopamine autoreceptor activity.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Apomorphine; Drug Interactions; Haloperidol; Inhalation; Isomerism; Male; Models, Psychological; Penis; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Respiration; Sexual Behavior, Animal; Syndrome

1984
Behavioral and biochemical effects of subchronic treatment with (-)3-(3-hydroxyphenyl)-N-n-propylpiperidine in the rat: dopamine receptor sensitivity and tolerance.
    Journal of neural transmission, 1984, Volume: 60, Issue:2

    Topics: Animals; Body Weight; Corpus Striatum; Dopamine; Kinetics; Male; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1984
Apomorphine and haloperidol-induced effects on male rat sexual behavior: no evidence for actions due to stimulation of central dopamine autoreceptors.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:3

    Topics: Animals; Apomorphine; Brain; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal

1984
The search for selective dopaminergic autoreceptor agonists.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Animals; Apomorphine; Dextroamphetamine; Dose-Response Relationship, Drug; Motor Activity; Optical Rotation; Piperidines; Rats; Receptors, Dopamine; Reserpine

1983
Further functional in vitro comparison of pre- and postsynaptic dopamine receptors in the rabbit caudate nucleus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 323, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Apomorphine; Benzazepines; Caudate Nucleus; Choline; Clonidine; Female; Male; Piperidines; Rabbits; Receptors, Dopamine

1983
Assessment of the chloroethyl analog of 3-PPP (N-n-propyl-3-(3-hydroxyphenyl)-piperidine), 3-PPP-C1 as an irreversible ligand for central dopaminergic recognition sites.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Animals; Aporphines; Brain; In Vitro Techniques; Ligands; Piperidines; Rats; Receptors, Dopamine

1983
Differential behavioural effects of dopamine agonists in developing rats: a study of 3-PPP enantiomers.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Age Factors; Animals; Dextroamphetamine; Female; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism

1983
Avoidance and ICSS behavioral models dissociate TL-99 and 3-PPP from dopamine receptor antagonists.
    European journal of pharmacology, 1983, Aug-05, Volume: 91, Issue:4

    Topics: Animals; Avoidance Learning; Haloperidol; Male; Models, Psychological; Naphthalenes; Piperidines; Rats; Rats, Inbred F344; Receptors, Dopamine; Saimiri; Self Stimulation; Tetrahydronaphthalenes

1983
Similarities of the effects of apomorphine and 3-PPP on serotonin neurons.
    European journal of pharmacology, 1983, Oct-28, Volume: 94, Issue:3-4

    Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Corpus Striatum; Haloperidol; Hippocampus; Male; Neurons; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spectrometry, Fluorescence

1983
Dopamine receptors involved in prolactin secretion pharmacologically characterized by means of 3-PPP enantiomers.
    European journal of pharmacology, 1983, Dec-09, Volume: 96, Issue:1-2

    Topics: Animals; Isomerism; Male; Piperidines; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Tranquilizing Agents

1983
Antidyskinetic action of 3-PPP, a selective dopaminergic autoreceptor agonist, in Cebus monkeys with persistent neuroleptic-induced dyskinesias.
    Journal of neural transmission, 1983, Volume: 58, Issue:3-4

    Topics: Animals; Cebus; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Female; Fluphenazine; Haloperidol; Male; Piperidines; Stereoisomerism

1983
Interaction of (+)- and (-)-3-PPP with the dopamine receptor in the anterior pituitary gland.
    Life sciences, 1984, Jan-16, Volume: 34, Issue:3

    Topics: Animals; Apomorphine; Binding Sites; Cell Membrane; Depression, Chemical; In Vitro Techniques; Male; Methyltyrosines; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism

1984
Stimulation of dopamine autoreceptors elicits "premature ejaculation" in rats.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 20, Issue:1

    Topics: Animals; Apomorphine; Copulation; Domperidone; Dopamine Antagonists; Ejaculation; Female; Haloperidol; Lisuride; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal

1984
Action of putative dopamine receptor agonists, TL-99, 3-PPP and RDS-127 on substantia nigra neurons.
    Brain research, 1984, Jan-30, Volume: 292, Issue:1

    Topics: Action Potentials; Animals; Depression, Chemical; Dopamine Antagonists; Indans; Indenes; Male; Naphthalenes; Piperidines; Rats; Substantia Nigra; Tetrahydronaphthalenes

1984
Assessment of dopamine autoreceptor agonist properties of apomorphine, (+)-3-PPP and (-)-3-PPP by recording of yawning behaviour in rats.
    European journal of pharmacology, 1984, Feb-17, Volume: 98, Issue:2

    Topics: Animals; Apomorphine; Behavior, Animal; Domperidone; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride

1984
A pharmacological comparison of 6,7-dihydroxy-2-dimethylaminotetralin (TL-99) and N-n-propyl-3-(3-hydroxyphenyl)piperidine with (3-PPP) selected dopamine agonists.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:2

    Topics: 4-Butyrolactone; Animals; Apomorphine; Cell Membrane; Corpus Striatum; Female; Humans; Hydroxydopamines; Naphthalenes; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes

1982
Suppression of exploratory locomotor activity in the rat by the local application of 3-PPP enantiomers into the nucleus accumbens.
    European journal of pharmacology, 1983, Apr-08, Volume: 88, Issue:4

    Topics: Animals; Exploratory Behavior; Male; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Stereoisomerism

1983
Failure of 3-PPP to activate dopamine autoreceptors in vitro.
    European journal of pharmacology, 1983, Apr-22, Volume: 89, Issue:1-2

    Topics: Acetylcholine; Animals; In Vitro Techniques; Naphthalenes; Piperidines; Potassium; Rats; Receptors, Dopamine; Tetrahydronaphthalenes

1983
Biphasic effects of some dopamine agonists on striatal acetylcholine concentrations.
    European journal of pharmacology, 1983, May-20, Volume: 90, Issue:1

    Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dopamine; Male; Piperidines; Piribedil; Rats; Tetrahydronaphthalenes; Time Factors

1983
Effect of two dopamine agonists, TL-99 and 3-PPP, on prolactin secretion in the rat.
    European journal of pharmacology, 1983, Jun-17, Volume: 90, Issue:4

    Topics: Animals; Male; Naphthalenes; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tetrahydronaphthalenes

1983
A behavioral study of the changes in the CNS of mice after subchronic treatment with the dopamine autoreceptor agonist 3-PPP.
    Psychopharmacology bulletin, 1982, Volume: 18, Issue:4

    Topics: Animals; Behavior, Animal; Male; Mice; Piperidines; Receptors, Dopamine

1982
Interaction of the putative dopamine autoreceptor agonists 3-PPP and TL-99 with [3H]apomorphine binding sites in rat striatal membranes.
    European journal of pharmacology, 1982, Dec-17, Volume: 86, Issue:1

    Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Kinetics; Membranes; Naphthalenes; Piperidines; Rats; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes

1982
Effect of 3-PPP, a putative dopamine autoreceptor agonist, on rat serum prolactin levels.
    Life sciences, 1981, Jul-06, Volume: 29, Issue:1

    Topics: Animals; Apomorphine; Binding, Competitive; Humans; Male; Piperidines; Prolactin; Rats; Receptors, Dopamine; Reserpine; Spiperone; Stereotyped Behavior

1981
Pharmacological profiles of the putative dopamine autoreceptor agonists 3-PPP and TL-99.
    European journal of pharmacology, 1981, Nov-19, Volume: 76, Issue:1

    Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Dogs; Dopamine; Female; Male; Mice; Motor Activity; Naphthalenes; Piperidines; Rats; Receptors, Dopamine; Tetrahydronaphthalenes

1981
A new centrally acting DA-receptor agonist with selectivity for autoreceptors.
    Psychopharmacology bulletin, 1980, Volume: 16, Issue:3

    Topics: Animals; Behavior, Animal; Brain; Dopamine; Piperidines; Rats; Receptors, Dopamine

1980
Dopamine receptor agonist potencies for inhibition of cell firing correlate with dopamine D3 receptor binding affinities.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Aminoquinolines; Animals; Apomorphine; Azepines; Benzothiazoles; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Male; Neurons; Phenethylamines; Piperidines; Pramipexole; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Substantia Nigra; Tetrahydronaphthalenes; Thiazoles; Thiophenes; Transfection

1995
The sigma receptor ligand (+/-)-BMY 14802 prevents methamphetamine-induced dopaminergic neurotoxicity via interactions at dopamine receptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:1

    Topics: Animals; Anticonvulsants; Antipsychotic Agents; Brain Diseases; Butaclamol; Carbazoles; Dizocilpine Maleate; Dopamine; Dopamine Agents; Drug Interactions; Drug Synergism; Guanidines; Ligands; Male; Methamphetamine; Mice; MPTP Poisoning; Neostriatum; Piperidines; Psychotropic Drugs; Pyrimidines; Receptors, Dopamine; Receptors, sigma; Stereoisomerism; Tyrosine 3-Monooxygenase

1994
[Contribution of dopamine autoreceptors in the reactive effect of opioid antagonists].
    Biulleten' eksperimental'noi biologii i meditsiny, 1995, Volume: 119, Issue:2

    Topics: Animals; Avoidance Learning; Dopamine Agonists; Enkephalin, Leucine; Male; Mice; Mice, Inbred BALB C; Naloxone; Narcotic Antagonists; Piperidines; Receptors, Dopamine; Receptors, Opioid, delta; Receptors, Opioid, mu

1995
Characterization of a (+)-azidophenazocine-sensitive sigma receptor on splenic lymphocytes.
    Journal of immunology (Baltimore, Md. : 1950), 1993, Nov-01, Volume: 151, Issue:9

    Topics: Affinity Labels; Animals; Binding Sites; Binding, Competitive; Female; Haloperidol; Interferons; Lymphocytes; Mice; Mice, Inbred C57BL; Phenazocine; Piperidines; Receptors, sigma; Spleen

1993
Oocytes from Xenopus laevis contain an intrinsic sigma 2-like binding site.
    Neuroscience letters, 1994, Oct-24, Volume: 180, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carbazoles; Dextromethorphan; Female; Guanidines; Haloperidol; Liver; Mazindol; Oocytes; Pentazocine; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Rats; Receptors, sigma; Xenopus laevis; Zinc

1994
Differential effects of 3-PPP enantiomers on extracellular dopamine concentration in the caudate-putamen and nucleus accumbens of rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 350, Issue:6

    Topics: Animals; Caudate Nucleus; Dopamine; Dopamine Agonists; Extracellular Space; Female; Nomifensine; Nucleus Accumbens; Piperidines; Putamen; Rats; Rats, Sprague-Dawley

1994
Purification, pharmacological characterization and photoaffinity labeling of sigma receptors from rat and bovine brain.
    Brain research, 1995, Jan-23, Volume: 670, Issue:1

    Topics: Animals; Binding Sites; Cattle; Cerebellum; Dopamine Agonists; Haloperidol; Male; Phenazocine; Piperidines; Rats; Receptors, sigma

1995
Sigma receptor-mediated neuroprotection against glutamate toxicity in primary rat neuronal cultures.
    Brain research, 1995, Feb-06, Volume: 671, Issue:1

    Topics: Animals; Calcium; Cells, Cultured; Cyclazocine; Cyclopentanes; Dextromethorphan; Glutamic Acid; Guanidines; Haloperidol; L-Lactate Dehydrogenase; Neurons; Neuroprotective Agents; Pentazocine; Phenazocine; Piperidines; Rats; Receptors, sigma

1995
Acute effects of sigma ligands on the extracellular DOPAC level in rat frontal cortex and striatum.
    Neurochemical research, 1995, Volume: 20, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Corpus Striatum; Extracellular Space; Frontal Lobe; Guanidines; Kinetics; Ligands; Male; Microdialysis; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Time Factors

1995
3-(3-Hydroxyphenyl)-N-(1-propyl)piperidine elicits convulsant effects in mice.
    General pharmacology, 1995, Volume: 26, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Convulsants; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; Electroencephalography; Male; Mice; Piperidines; Receptors, sigma; Seizures; Stereoisomerism

1995
Antiemetic effects of 5-HT1A agonists in the pigeon.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:2

    Topics: Animals; Anticonvulsants; Antiemetics; Columbidae; Conditioning, Classical; Dopamine Agonists; Dose-Response Relationship, Drug; Emetics; Guanidines; Male; Pentobarbital; Piperidines; Serotonin Receptor Agonists

1994
Dopamine D2 autoreceptors in rats are behaviorally functional at 21 but not 10 days of age.
    Psychopharmacology, 1994, Volume: 114, Issue:2

    Topics: Aging; Aminoquinolines; Animals; Apomorphine; Azepines; Behavior, Animal; Benzothiazoles; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Motor Activity; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Thiazoles

1994
Behavioral and neurochemical data suggest functional differences between dopamine D2 and D3 receptors.
    European journal of pharmacology, 1994, Oct-03, Volume: 263, Issue:3

    Topics: Analysis of Variance; Animals; Apomorphine; Benzothiazoles; CHO Cells; Cricetinae; Cricetulus; Dihydroxyphenylalanine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Microdialysis; Mitogens; Motor Activity; Piperidines; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Thiazoles; Transfection

1994
Effects of sigma ligands on rat cerebellar Purkinje neuron firing: an iontophoretic study.
    Brain research bulletin, 1994, Volume: 35, Issue:4

    Topics: Animals; Ethylamines; Guanidines; Iontophoresis; Levallorphan; Male; Pentazocine; Piperidines; Purkinje Cells; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, sigma

1994
Heterocyclic amino alcohols related to ifenprodil as sigma receptor ligands: binding and conformational analyses.
    European journal of pharmacology, 1994, Oct-14, Volume: 269, Issue:2

    Topics: Adrenergic alpha-Antagonists; Amino Alcohols; Animals; Binding, Competitive; Cerebral Cortex; Crystallization; Dopamine Agonists; Heterocyclic Compounds; In Vitro Techniques; Ligands; Models, Molecular; Molecular Conformation; Piperidines; Propanolamines; Rats; Receptors, Adrenergic, alpha-1; Receptors, sigma

1994
Is the sigma 2 receptor in rat brain related to the K+ channel of class III antiarrhythmic drugs?
    European journal of pharmacology, 1993, Sep-07, Volume: 241, Issue:1

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Cerebral Cortex; Dopamine Agents; Electrophysiology; Glioma; Guinea Pigs; In Vitro Techniques; Male; Piperidines; Potassium Channels; Purkinje Fibers; Rats; Rats, Wistar; Receptors, sigma; Tumor Cells, Cultured

1993
Two inbred rat sublines that differ in spontaneous yawning behavior also differ in their responses to cholinergic and dopaminergic drugs.
    Behavioural brain research, 1993, Sep-30, Volume: 56, Issue:2

    Topics: Animals; Apomorphine; Dopamine Agents; Dose-Response Relationship, Drug; Male; Parasympathomimetics; Physostigmine; Pilocarpine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Receptors, Dopamine; Species Specificity; Yawning

1993
Haloperidol treatment differentially regulates [3H]DTG and [3H](+)-3-PPP labeled sigma binding sites.
    European journal of pharmacology, 1993, Aug-24, Volume: 240, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Binding Sites; Brain; Dopamine Agents; Drug Administration Schedule; Guanidines; Guinea Pigs; Haloperidol; Male; Phenytoin; Piperidines; Receptors, sigma

1993
A high dose of EEDQ reduces pituitary dopamine D2 receptor density and the prolactin suppressive potency of agonists.
    European journal of pharmacology, 1993, Oct-26, Volume: 243, Issue:3

    Topics: Animals; Azepines; Dopamine Agents; Male; Piperidines; Pituitary Gland; Prolactin; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

1993
Discrimination of (+)-3-PPP sites from DTG sites by FH-510, a novel potent sigma ligand, in rat brain.
    European journal of pharmacology, 1993, Nov-30, Volume: 250, Issue:1

    Topics: Animals; Anticonvulsants; Binding Sites; Brain; Carbazoles; Dopamine Agents; Guanidines; In Vitro Techniques; Male; Piperidines; Propylamines; Radioligand Assay; Rats; Rats, Wistar

1993
Further characterization of [3H]ifenprodil binding in rat brain.
    European journal of pharmacology, 1994, Jan-01, Volume: 266, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brain; Dizocilpine Maleate; Dopamine Agents; Dose-Response Relationship, Drug; Guanidines; In Vitro Techniques; Male; Neurotransmitter Uptake Inhibitors; Piperazines; Piperidines; Rats; Rats, Inbred F344; Receptors, sigma

1994
Further characterization of the effects of BMY 14802 on dopamine neuronal activity.
    Synapse (New York, N.Y.), 1993, Volume: 15, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Dopamine; Dopamine Agents; Ergolines; Injections, Intravenous; Iontophoresis; Male; Neurons; Piperidines; Pyrimidines; Quinpirole; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Stereoisomerism; Sulpiride

1993
Pharmacological characteristics of hyperambulation induced by the sigma ligand (+)-3-PPP in rats.
    Japanese journal of pharmacology, 1994, Volume: 65, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ligands; Male; Motor Activity; Piperidines; Rats; Rats, Wistar; Receptors, sigma; Serotonin Receptor Agonists; Stereoisomerism; Tryptophan Hydroxylase; Tyrosine 3-Monooxygenase

1994
Ocular hypotension induced by topical dopaminergic drugs and phosphodiesterase inhibitors.
    European journal of pharmacology, 1994, Jun-02, Volume: 258, Issue:1-2

    Topics: Administration, Topical; Animals; Dopamine Agents; Glucose; Male; Ocular Hypotension; Ophthalmic Solutions; Pentoxifylline; Phosphodiesterase Inhibitors; Piperidines; Rabbits; Stereoisomerism; Trifluperidol; Xanthines

1994
[3H]RS-23597-190, a potent 5-hydroxytryptamine4 antagonist labels sigma-1 but not sigma-2 binding sites in guinea pig brain.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:1

    Topics: Aminobenzoates; Animals; Binding Sites; Brain; Guinea Pigs; Male; para-Aminobenzoates; Piperidines; Receptors, Serotonin; Receptors, sigma; Serotonin Antagonists

1994
The effects of sigma ligands on the release of glutamate from rat striatal slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 350, Issue:2

    Topics: Animals; Corpus Striatum; Female; Glutamic Acid; Haloperidol; In Vitro Techniques; Ligands; Neuropeptide Y; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, sigma

1994
Ameliorating effects of sigma receptor ligands on the impairment of passive avoidance tasks in mice: involvement in the central acetylcholinergic system.
    European journal of pharmacology, 1994, Aug-11, Volume: 261, Issue:1-2

    Topics: Acetylcholine; Amnesia; Animals; Anticonvulsants; Avoidance Learning; Brain; Cholinesterase Inhibitors; Dopamine Agonists; Electroshock; Guanidines; Ligands; Male; Memory; Mice; Mice, Inbred Strains; p-Chloroamphetamine; Phenazocine; Piperidines; Receptors, sigma; Serotonin Antagonists

1994
Effects of haloperidol and reduced haloperidol on binding to sigma sites.
    European journal of pharmacology, 1994, Mar-21, Volume: 254, Issue:3

    Topics: Animals; Binding Sites; Brain; Dextromethorphan; Guinea Pigs; Haloperidol; Male; Oxidation-Reduction; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma

1994
Sigma receptor ligands modulate contractility, Ca++ influx and beating rate in cultured cardiac myocytes.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:3

    Topics: Animals; Calcium; Cells, Cultured; GTP-Binding Proteins; Guanidines; Haloperidol; Heart Rate; Myocardial Contraction; Pentazocine; Piperidines; Rats; Receptors, sigma; Sarcoplasmic Reticulum

1994
2,5-Dimethoxy congeners of (+)-and (-)-3-(3-hydroxyphenyl)-N-n- propylpiperidine.
    Journal of medicinal chemistry, 1993, Aug-06, Volume: 36, Issue:16

    Topics: Animals; Bradycardia; Dopamine Agents; Hypotension; Piperidines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

1993
Effects of several partial dopamine D2 receptor agonists in Cebus apella monkeys previously treated with haloperidol.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: Administration, Oral; Amphetamine; Animals; Antipsychotic Agents; Behavior, Animal; Benzothiazoles; Cebus; Disease Models, Animal; Dopamine Agents; Dopamine D2 Receptor Antagonists; Dyskinesia, Drug-Induced; Dystonia; Ergolines; Female; Haloperidol; Lisuride; Male; Piperidines; Pramipexole; Quinpirole; Raclopride; Salicylamides; Thiazoles

1993
Binding of [3H]FH-510 to sigma ligand recognition sites in guinea-pig brain membranes.
    European journal of pharmacology, 1993, Jul-06, Volume: 238, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Binding, Competitive; Brain; Carbazoles; Dopamine Agents; Guinea Pigs; Histamine; In Vitro Techniques; Kinetics; Male; Microsomes; Phenazocine; Piperidines; Propylamines; Pyrimidines; Radioligand Assay; Receptors, sigma; Serotonin

1993
[3H]BIMU-1, a 5-hydroxytryptamine3 receptor ligand in NG-108 cells, selectively labels sigma-2 binding sites in guinea pig hippocampus.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Animals; Autoradiography; Benzimidazoles; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Guinea Pigs; Hippocampus; Male; Membranes; Mice; Neuroblastoma; Piperidines; Rats; Receptors, Serotonin; Receptors, sigma; Sensitivity and Specificity; Tritium; Tumor Cells, Cultured

1993
Strain differences in rat brain and liver sigma binding: lack of cytochrome P450-2D1 involvement.
    European journal of pharmacology, 1993, Oct-26, Volume: 243, Issue:3

    Topics: Analysis of Variance; Animals; Binding Sites; Brain; Cytochrome P-450 CYP2D6; Cytochrome P-450 Enzyme System; Liver; Mixed Function Oxygenases; Piperidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, sigma; Sex Factors; Species Specificity

1993
Multiplicity of [3H]1,3-di-o-tolylguanidine binding sites with low affinity for haloperidol in rat brain.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:10

    Topics: Animals; Binding Sites; Brain; Guanidines; Haloperidol; Male; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma

1993
Discriminative stimulus properties of cocaine in relation to dopamine D2 receptor function in rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Animals; Bromocriptine; Cocaine; Discrimination Learning; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Male; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

1993
Synthesis and in vitro evaluation of 5,6,7,8,9,10-hexahydro-7,10-iminocyclohept[b]indoles: high-affinity ligands for the N,N'-di-o-tolylguanidine-labeled sigma binding site.
    Journal of medicinal chemistry, 1993, Feb-05, Volume: 36, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Guanidines; Guinea Pigs; In Vitro Techniques; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship; Sulpiride; X-Ray Diffraction

1993
Repeated testing within drug discrimination learning: time course studies with cocaine, amphetamine, and 3-PPP.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:2

    Topics: Amphetamine; Animals; Cocaine; Columbidae; Discrimination Learning; Dopamine Antagonists; Male; Piperidines; Time Factors

1993
Correlation between potentiation of neurogenic twitch contraction and benzomorphan sigma receptor binding potency in the mouse vas deferens.
    European journal of pharmacology, 1993, Feb-16, Volume: 231, Issue:3

    Topics: Animals; Antiparkinson Agents; Brain; Drug Synergism; Guinea Pigs; Haloperidol; Ligands; Male; Mice; Phenazocine; Piperidines; Receptors, sigma; Spasm; Vas Deferens

1993
Allosteric modulation of ligand binding to [3H](+)pentazocine-defined sigma recognition sites by phenytoin.
    Life sciences, 1993, Volume: 53, Issue:1

    Topics: Allosteric Regulation; Animals; Binding Sites; Cyclopentanes; Dextromethorphan; Dextrorphan; Guinea Pigs; Ligands; Male; Pentazocine; Phenazocine; Phenytoin; Piperidines; Radioligand Assay; Receptors, sigma; Tritium

1993
Inotropic action of sigma receptor ligands in isolated cardiac myocytes from adult rats.
    European journal of pharmacology, 1995, Nov-03, Volume: 286, Issue:1

    Topics: Animals; Binding Sites; Calcium; Guanidines; In Vitro Techniques; Ligands; Myocardial Contraction; Myocardium; Pentazocine; Piperidines; Rats; Receptors, sigma; Stimulation, Chemical

1995
Effects of sigma receptor ligands on the extracellular concentration of dopamine in the striatum and prefrontal cortex of the rat.
    European journal of pharmacology, 1995, Nov-24, Volume: 286, Issue:3

    Topics: Animals; Benzomorphans; Corpus Striatum; Dopamine; Guanidines; Ligands; Male; Pentazocine; Piperazines; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, sigma; Stereoisomerism

1995
Sigma receptor activation does not mediate fentanyl-induced attenuation of muscarinic coronary contraction.
    Anesthesia and analgesia, 1996, Volume: 82, Issue:5

    Topics: Acetylcholine; Anesthetics, Intravenous; Animals; Coronary Vessels; Cyclazocine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fentanyl; Guanidines; Haloperidol; Muscarine; Muscarinic Agonists; Narcotic Antagonists; Narcotics; Pentazocine; Phencyclidine; Piperidines; Potassium Channel Blockers; Receptors, Dopamine; Receptors, sigma; Signal Transduction; Swine; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

1996
Effects of dopamine D3 preferring compounds on conditioned place preference and intracranial self-stimulation in the rat.
    Journal of neural transmission. General section, 1995, Volume: 101, Issue:1-3

    Topics: Animals; Brain; Conditioning, Operant; Dextroamphetamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Indans; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Stimulation; Tetrahydronaphthalenes

1995
Involvement of sigma-receptors in the increase in contraction of mouse vas deferens induced by exogenous ATP.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:1

    Topics: Adenosine Triphosphate; Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Carbazoles; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guanidines; Haloperidol; Ligands; Male; Mice; Muscle Contraction; Muscle, Smooth; Pentazocine; Phenazocine; Piperidines; Receptors, sigma; Regression Analysis; Structure-Activity Relationship; Vas Deferens

1996
Initial characterization and autoradiographic localization of a novel sigma/opioid binding site in immune tissues.
    Journal of neuroimmunology, 1996, Volume: 67, Issue:2

    Topics: Animals; Anticonvulsants; Autoradiography; Binding Sites; Binding, Competitive; Brain Chemistry; Cytochrome P-450 Enzyme System; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Hydrogen-Ion Concentration; Kinetics; Leukocytes; Monoamine Oxidase; Naltrexone; Narcotic Antagonists; Narcotics; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Spleen; Tritium

1996
Affinities and intrinsic activities of dopamine receptor agonists for the hD21 and hD4.4 receptors.
    European journal of pharmacology, 1996, Apr-22, Volume: 301, Issue:1-3

    Topics: Aminoquinolines; Animals; Cell Membrane; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Humans; Piperidines; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides

1996
Effects on locomotor activity after local application of D3 preferring compounds in discrete areas of the rat brain.
    Journal of neural transmission. General section, 1995, Volume: 102, Issue:3

    Topics: Animals; Brain; Cortical Spreading Depression; Dextroamphetamine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Indans; Injections, Intraventricular; Male; Microinjections; Motor Activity; Nucleus Accumbens; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Ventral Tegmental Area

1995
Partial agonistic effects of OPC-14597, a potential antipsychotic agent, on yawning behavior in rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:4

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Azepines; Dopamine Agonists; Drug Synergism; Male; Oxidopamine; Piperazines; Piperidines; Quinolones; Rats; Rats, Wistar; Receptors, Dopamine; Stereotyped Behavior; Sympathectomy, Chemical; Yawning

1996
Kappa opioid receptor agonists inhibit sigma-1 (sigma 1) receptor binding in guinea-pig brain, liver and spleen: autoradiographical evidence.
    Brain research, 1996, Jul-01, Volume: 725, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Autoradiography; Benzomorphans; Binding Sites; Brain; Guinea Pigs; Liver; Piperidines; Pyrrolidines; Receptors, Opioid, kappa; Receptors, sigma; Spinal Cord; Spleen

1996
Dopamine and opioid regulation of the memory retrieval recovery in mice.
    Behavioural brain research, 1996, Volume: 79, Issue:1-2

    Topics: Animals; Avoidance Learning; Dopamine Agonists; Enkephalin, Leucine; Male; Memory; Mice; Mice, Inbred BALB C; Narcotic Antagonists; Piperidines; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta

1996
Differential localization of three distinct binding sites for sigma receptor ligands in rat spleen.
    Journal of neuroimmunology, 1997, Volume: 72, Issue:1

    Topics: Analgesics, Opioid; Animals; Anticonvulsants; Antipsychotic Agents; Autoradiography; Binding Sites; Dopamine Agonists; Dopamine Antagonists; Female; Guanidines; Haloperidol; Image Processing, Computer-Assisted; Ligands; Male; Naltrexone; Narcotic Antagonists; Pentazocine; Phenazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Spleen; Tritium

1997
BMY-14802 reversed the sigma receptor agonist-induced neck dystonia in rats.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:10

    Topics: Animals; Antipsychotic Agents; Dibenzothiepins; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dystonia; Guanidines; Haloperidol; Male; Microinjections; Nerve Tissue Proteins; Perphenazine; Piperidines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, sigma; Red Nucleus; Sulpiride; Torticollis

1996
In vivo functional interaction between phencyclidine binding sites and sigma receptors to produce head-weaving behavior in rats.
    European journal of pharmacology, 1996, Dec-30, Volume: 318, Issue:2-3

    Topics: Animals; Anisoles; Behavior, Animal; Binding Sites; Dizocilpine Maleate; Guanidines; Male; Phenazocine; Piperidines; Propylamines; Pyrimidines; Rats; Rats, Wistar; Receptors, Phencyclidine; Receptors, sigma

1996
Reduction of the scopolamine-induced impairment of passive-avoidance performance by sigma receptor agonist in mice.
    Physiology & behavior, 1997, Volume: 61, Issue:2

    Topics: Acetylcholinesterase; Animals; Antipsychotic Agents; Avoidance Learning; Brain; Dose-Response Relationship, Drug; Guanidines; Male; Mental Recall; Mice; Mice, Inbred Strains; Phenazocine; Piperidines; Receptors, sigma; Scopolamine

1997
Behavioural effects of selective serotonin reuptake inhibitors following direct micro injection into the left red nucleus of the rat.
    Journal of psychopharmacology (Oxford, England), 1997, Volume: 11, Issue:1

    Topics: 1-Naphthylamine; Animals; Behavior, Animal; Chlorpromazine; Citalopram; Fluoxetine; Fluvoxamine; Guanidines; Haloperidol; Male; Microinjections; Motor Activity; Paroxetine; Piperidines; Posture; Rats; Rats, Sprague-Dawley; Receptors, sigma; Red Nucleus; Selective Serotonin Reuptake Inhibitors; Sertraline

1997
Neuroleptic binding to sigma receptors: possible involvement in neuroleptic-induced acute dystonia.
    Biological psychiatry, 1997, May-15, Volume: 41, Issue:10

    Topics: Animals; Antipsychotic Agents; Dopamine Agonists; Dyskinesia, Drug-Induced; Male; Piperidines; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Muscarinic; Receptors, sigma; Spiperone

1997
Multiple [3H]-nemonapride binding sites in calf brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Antagonists; Animals; Anticonvulsants; Benzamides; Binding, Competitive; Brain; Cattle; Cerebellum; Cerebral Cortex; Corpus Striatum; Dioxanes; Dopamine Agonists; Dopamine Antagonists; Guanidines; Haloperidol; In Vitro Techniques; Isotope Labeling; Narcotic Antagonists; Pentazocine; Piperidines; Propylamines; Pyrrolidines; Receptors, Dopamine D2; Receptors, sigma; Sulpiride; Tritium

1997
Effects of phencyclidine (PCP) and (+)MK-801 on sensorimotor gating in CD-1 mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 1998, Volume: 22, Issue:1

    Topics: Acoustic Stimulation; Animals; Apomorphine; Clozapine; Dextroamphetamine; Dizocilpine Maleate; Dopamine Agonists; Dose-Response Relationship, Drug; Haloperidol; Male; Mice; Mice, Inbred Strains; Phencyclidine; Piperidines; Rats; Receptors, sigma; Reflex, Startle; Species Specificity

1998
The intrinsic activity of (-)-3-PPP vis-à-vis prolactin-suppressing dopamine D2 receptors in transfected GH4C1 cells is dependent on which secretagogue that is used to provoke prolactin release.
    Neuropharmacology, 1998, Volume: 37, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cell Line; Dopamine; Dopamine Agonists; Humans; Piperidines; Potassium; Prolactin; Receptors, Dopamine D2; Tetraethylammonium; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide

1998
Sigma receptor ligands and imidazoline secretagogues mediate their insulin secretory effects by activating distinct receptor systems in isolated islets.
    European journal of pharmacology, 1998, Jun-05, Volume: 350, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Animals; Azides; Benzofurans; Dopamine Agonists; Dose-Response Relationship, Drug; Guanidines; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Ligands; Male; Piperidines; Rats; Rats, Wistar; Receptors, Drug; Receptors, sigma

1998
Direct dopamine D2-receptor-mediated modulation of arachidonic acid release in transfected CHO cells without the concomitant administration of a Ca2+-mobilizing agent.
    British journal of pharmacology, 1998, Volume: 124, Issue:8

    Topics: Adenosine Triphosphate; Animals; Arachidonic Acid; Calcium; Calcium Channel Blockers; CHO Cells; Cricetinae; Cyclooxygenase Inhibitors; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gallic Acid; Pertussis Toxin; Piperidines; Receptors, Dopamine D2; Transfection; Virulence Factors, Bordetella

1998
[18F]fluoroethoxy-benzovesamicol, a PET radiotracer for the vesicular acetylcholine transporter and cholinergic synapses.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:3

    Topics: Acetylcholine; Animals; Autoradiography; Brain; Calibration; Carrier Proteins; Cholinesterase Inhibitors; Donepezil; Dopamine Agonists; Female; Fluorine Radioisotopes; Haloperidol; Humans; Indans; Kinetics; Male; Membrane Transport Proteins; Mice; Organ Specificity; Piperidines; Rats; Rats, Sprague-Dawley; Stereoisomerism; Synapses; Tissue Distribution; Tomography, Emission-Computed; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

1998
Effect of PCP and sigma ligands on both noradrenaline- and electrically-induced contractions and on [3H]-noradrenaline uptake in rat vas deferens.
    Journal of autonomic pharmacology, 1998, Volume: 18, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Dextromethorphan; Dizocilpine Maleate; Dopamine Agonists; Electric Stimulation; Excitatory Amino Acid Antagonists; Ligands; Male; Muscle Contraction; Neuroprotective Agents; Norepinephrine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Phencyclidine; Receptors, sigma; Tritium; Vas Deferens

1998
Reduction of 4-cyclohexyl-1-[(1R)-1,2-diphenylethyl]-piperazine-induced memory impairment of passive avoidance performance by sigma 1 receptor agonists in mice.
    Methods and findings in experimental and clinical pharmacology, 1998, Volume: 20, Issue:7

    Topics: Animals; Antipsychotic Agents; Avoidance Learning; Binding, Competitive; Brain Chemistry; Dopamine Agonists; Guinea Pigs; Male; Membranes; Memory Disorders; Mice; Phenazocine; Piperazines; Piperidines; Radioligand Assay; Receptors, sigma

1998
Influence of 3-PPP, a sigma receptor ligand, on the anticonvulsive action of conventional antiepileptic drugs.
    Pharmacological research, 1999, Volume: 40, Issue:6

    Topics: Animals; Anticonvulsants; Avoidance Learning; Dizocilpine Maleate; Female; Guanidines; Mice; Phenobarbital; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Valproic Acid

1999
Effects of trazodone on neurotransmitter release from rat mossy fibre cerebellar synaptosomes.
    European journal of pharmacology, 2000, Jul-14, Volume: 400, Issue:1

    Topics: Animals; Antidepressive Agents, Second-Generation; Cerebellum; Ethylenediamines; gamma-Aminobutyric Acid; Glutamic Acid; Male; Nerve Fibers; Phenazocine; Piperidines; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, sigma; Serotonin; Synaptosomes; Trazodone

2000
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001
The selective sigma ligand MS-377 attenuates the blockade by phencyclidine of NMDA-induced intracellular calcium.
    The international journal of neuropsychopharmacology, 2002, Volume: 5, Issue:3

    Topics: Algorithms; Animals; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Image Processing, Computer-Assisted; Ligands; Microscopy, Confocal; Neocortex; Phencyclidine; Piperidines; Pyrrolidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Tartrates

2002
Antagonism of NMDA receptors by sigma receptor ligands attenuates chemical ischemia-induced neuronal death in vitro.
    European journal of pharmacology, 2002, Nov-29, Volume: 455, Issue:2-3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Calcium; Cell Hypoxia; Cell Survival; Cells, Cultured; Cerebral Cortex; Cyclopentanes; Deoxyglucose; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fetus; Glucose; Glutamates; Haloperidol; Neurons; Phenazocine; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sodium Azide

2002
Dopamine agonist 3-PPP fails to protect against MPTP-induced toxicity.
    Neurochemical research, 2004, Volume: 29, Issue:2

    Topics: Animals; Behavior, Animal; Cell Division; Cell Line, Tumor; Corpus Striatum; Dopamine; Dopamine Agonists; Humans; Mice; Mice, Inbred C57BL; Monoamine Oxidase; MPTP Poisoning; Neuroprotective Agents; Piperidines; Treatment Failure

2004
Phenytoin differentially modulates the affinity of agonist and antagonist ligands for sigma 1 receptors of guinea pig brain.
    Synapse (New York, N.Y.), 2005, Mar-01, Volume: 55, Issue:3

    Topics: Allosteric Regulation; Animals; Anisoles; Anticonvulsants; Binding, Competitive; Brain; Dextromethorphan; Drug Interactions; Ethylenediamines; Guinea Pigs; Haloperidol; Ligands; Male; Morpholines; Neurons; Phenazocine; Phenytoin; Piperazines; Piperidines; Progesterone; Propylamines; Receptors, sigma; Synaptic Transmission

2005
Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.
    European journal of pharmacology, 2005, May-16, Volume: 515, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Humans; Lisuride; Piperazines; Piperidines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Risperidone; Transfection; Tritium

2005
Radiosynthesis, ex vivo and in vivo evaluation of [11C]preclamol as a partial dopamine D2 agonist radioligand for positron emission tomography.
    Synapse (New York, N.Y.), 2006, Sep-15, Volume: 60, Issue:4

    Topics: Animals; Blood-Brain Barrier; Brain; Brain Chemistry; Chemical Phenomena; Chemistry, Physical; Dopamine Agonists; Indicators and Reagents; Injections, Intravenous; Isotope Labeling; Male; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2

2006
In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling.
    Journal of psychopharmacology (Oxford, England), 2007, Volume: 21, Issue:6

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Calcium Signaling; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Immunoblotting; Lisuride; MAP Kinase Signaling System; Microscopy, Confocal; Mitogen-Activated Protein Kinase 1; Phosphorylation; Piperazines; Piperidines; Quinolones; Raclopride; Receptors, Dopamine D2; Schizophrenia; Time Factors; Transfection

2007
Partial agonist actions of aripiprazole and the candidate antipsychotics S33592, bifeprunox, N-desmethylclozapine and preclamol at dopamine D(2L) receptors are modified by co-transfection of D(3) receptors: potential role of heterodimer formation.
    Journal of neurochemistry, 2007, Volume: 102, Issue:4

    Topics: Adenylyl Cyclases; Animals; Antipsychotic Agents; Aripiprazole; Benzamides; Benzoxazoles; Carrier Proteins; Chlorocebus aethiops; Clozapine; COS Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Piperazines; Piperidines; Quinolones; Receptors, Dopamine D2; Receptors, Dopamine D3; Transfection

2007
Pharmacological blockade of dopamine D2 receptors by aripiprazole is not associated with striatal sensitization.
    Naunyn-Schmiedeberg's archives of pharmacology, 2011, Volume: 383, Issue:1

    Topics: Animals; Apomorphine; Aripiprazole; Buffers; Catalepsy; Cell Membrane; Cerebral Cortex; Corpus Striatum; Domperidone; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Antagonism; Drug Partial Agonism; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Hippocampus; Male; Piperazines; Piperidines; Pyridines; Quinolones; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Stereotyped Behavior; Up-Regulation

2011
Effects of the dopamine stabilizers (S)-(-)-OSU6162 and ACR16 on prolactin secretion in drug-naive and monoamine-depleted rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2011, Volume: 384, Issue:1

    Topics: Animals; Aripiprazole; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Hyperprolactinemia; Lactotrophs; Male; Methyltyrosines; Piperazines; Piperidines; Prolactin; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reserpine

2011
Ligand-promoted C3-selective arylation of pyridines with Pd catalysts: gram-scale synthesis of (±)-preclamol.
    Journal of the American Chemical Society, 2011, Nov-30, Volume: 133, Issue:47

    Topics: Ligands; Molecular Structure; Organometallic Compounds; Palladium; Piperidines; Pyridines; Stereoisomerism

2011
A comparison of the effects of the dopamine partial agonists aripiprazole and (-)-3-PPP with quinpirole on stimulated dopamine release in the rat striatum: Studies using fast cyclic voltammetry in vitro.
    European journal of pharmacology, 2012, Jul-05, Volume: 686, Issue:1-3

    Topics: Animals; Aripiprazole; Corpus Striatum; Dopamine; Dopamine Agonists; Drug Partial Agonism; In Vitro Techniques; Male; Piperazines; Piperidines; Quinolones; Quinpirole; Rats; Rats, Wistar

2012
Regional brain imaging of vesicular acetylcholine transporter using o-[125 I]iodo-trans-decalinvesamicol as a new potential imaging probe.
    Synapse (New York, N.Y.), 2014, Volume: 68, Issue:3

    Topics: Animals; Autoradiography; Blood-Brain Barrier; Brain; Iodine Radioisotopes; Ligands; Male; Narcotic Antagonists; Pentazocine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sigma-1 Receptor; Tomography, Emission-Computed, Single-Photon; Vesicular Acetylcholine Transport Proteins

2014
The potential of o-bromo-trans-decalinvesamicol as a new PET ligand for vesicular acetylcholine transporter imaging.
    Synapse (New York, N.Y.), 2014, Volume: 68, Issue:10

    Topics: Animals; Autoradiography; Brain; Bromine Radioisotopes; Central Nervous System Agents; Male; Pentazocine; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Rats, Sprague-Dawley; Receptors, sigma; Vesicular Acetylcholine Transport Proteins

2014
Agonist and antagonist effects of aripiprazole on D₂-like receptors controlling rat brain dopamine synthesis depend on the dopaminergic tone.
    The international journal of neuropsychopharmacology, 2014, Oct-31, Volume: 18, Issue:4

    Topics: Animals; Aripiprazole; Autoreceptors; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Piperidines; Potassium; Presynaptic Terminals; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2

2014
A Cu/Pd Cooperative Catalysis for Enantioselective Allylboration of Alkenes.
    Journal of the American Chemical Society, 2015, Nov-04, Volume: 137, Issue:43

    Topics: Alkenes; Allyl Compounds; Boranes; Catalysis; Copper; Molecular Structure; Organometallic Compounds; Palladium; Piperidines; Stereoisomerism

2015
The role of kinetic context in apparent biased agonism at GPCRs.
    Nature communications, 2016, Feb-24, Volume: 7

    Topics: Animals; Aripiprazole; CHO Cells; Cricetulus; Dopamine; Dopamine Agonists; Indoles; Kinetics; Ligands; Piperazines; Piperidines; Principal Component Analysis; Protein Stability; Receptors, Dopamine D2

2016
The sigma-1 receptor mediates the beneficial effects of pridopidine in a mouse model of Huntington disease.
    Neurobiology of disease, 2017, Volume: 97, Issue:Pt A

    Topics: Aging; Animals; Calbindins; Calcium; Cations, Divalent; Coculture Techniques; Corpus Striatum; Dendritic Spines; Disease Models, Animal; Endoplasmic Reticulum; Humans; Huntington Disease; Mice; Mice, Transgenic; Neuroprotective Agents; Piperidines; Rats, Inbred SHR; Receptors, sigma; Sigma-1 Receptor; Synapses

2017
Neuroprotective Effect of σ1-Receptors on the Cell Model of Huntington's Disease.
    Bulletin of experimental biology and medicine, 2017, Volume: 164, Issue:2

    Topics: Animals; Anisoles; Calcium; Cerebral Cortex; Corpus Striatum; Dendritic Spines; Gene Expression; Homeostasis; Huntington Disease; Male; Mice; Models, Biological; Morpholines; Neurons; Piperidines; Primary Cell Culture; Propylamines; Receptors, sigma; RNA, Small Interfering; Sigma-1 Receptor; Synapses; Synaptic Transmission; Transduction, Genetic

2017