preclamol has been researched along with apomorphine in 81 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 57 (70.37) | 18.7374 |
1990's | 20 (24.69) | 18.2507 |
2000's | 2 (2.47) | 29.6817 |
2010's | 2 (2.47) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Caprathe, BW; Heffner, TG; Jaen, JC; Meltzer, LT; Parvez, M; Pugsley, TA; Wise, LD | 1 |
Bergmeier, S; Caprathe, BW; Heffner, TG; Humblet, CC; Jaen, JC; Meltzer, LT; Pugsley, TA; Tecle, H; Wise, LD | 1 |
Arnt, J; Bøgesø, KP; Lundmark, M; Sundell, S | 1 |
Arvidsson, LE; Carlsson, A; Hacksell, U; Hjorth, S; Johansson, A; Lindberg, P; Nilsson, JL; Sanchez, D; Wikström, H | 1 |
Chidester, CG; Haadsma-Svensson, SR; Lahti, RA; Lin, CH; McCall, RB; Piercey, MF; Schreur, PJ; Smith, MW; Von Voigtlander, PF | 1 |
Chidester, CG; Haadsma-Svensson, SR; Lahti, RA; Lin, CH; McCall, RB; Phillips, G; Piercey, MF; Schreur, PJ; Smith, MW; Von Voigtlander, PF | 1 |
Liljefors, T; Wikström, H | 1 |
Arvidsson, LE; Hacksell, U; Hjorth, S; Johansson, AM; Lindberg, P; Nilsson, JL; Sanchez, D; Svensson, K; Thorberg, SO; Wikström, H | 1 |
Carlsson, A; Hansson, L; Lin, CH; Smith, MW; Sonesson, C; Svensson, K; Waters, N; Wikström, H | 1 |
Pettersson, F; Pontén, H; Sonesson, C; Waters, N; Waters, S | 1 |
Hudzik, TJ | 1 |
Bohmaker, K; Bordi, F; Meller, E | 1 |
Ekman, A; Eriksson, E | 1 |
Fukamauchi, F; Shibuya, H; Yoshikawa, T | 1 |
Kruk, ZL; Millar, J; Stamford, JA | 1 |
Carlsson, A; Kujacic, M; Löfberg, L; Svensson, K | 1 |
Engberg, G; Wikström, H | 1 |
Code, RA; Tang, AH | 1 |
Svensson, L | 1 |
Bowen, WD; de Costa, BR; Hellewell, SB; Jacobson, AE; Rice, KC; Thurkauf, A; Walker, JM | 1 |
Fico, TA; Spoerlein, MT; Vanderwende, C; Wilmot, CA | 1 |
Bagetta, G; de Sarro, GB; Marra, R; Nisticò, G; Priolo, E | 1 |
Claustre, Y; Fage, D; Scatton, B; Zivkovic, B | 1 |
Sethy, VH; Wenger, D | 1 |
Carlsson, A; Clark, D; Hjorth, S | 2 |
Andersson, M; Fowler, CJ; Magnusson, O; Thorell, G | 1 |
Carnoy, P; Puech, AJ; Simon, P; Soubrie, P | 1 |
Goiny, M; Uvnäs-Moberg, K | 1 |
Nichols, NF; Schreur, PJ | 1 |
Jenner, P; Kelly, E; Marsden, CD | 2 |
Bohmaker, K; Friedhoff, AJ; Goldstein, M; Meller, E; Namba, Y | 1 |
Aihara, H; Hashimoto, S; Okuyama, S | 1 |
Bagetta, G; Nistico, G; Priolo, E | 1 |
Bagetta, G; De Sarro, G; Nisticò, G; Priolo, E | 1 |
Hiyama, T; Kikuchi, T; Suzuki, S; Tsutsui, M; Yamada, K; Yasuda, Y | 1 |
Altar, CA; Gerber, R; Hall, NR; Liebman, JM | 1 |
Christoffersen, CL; Meltzer, LT | 1 |
Di Chiara, G; Frau, R; Imperato, A; Tanda, G | 1 |
Argiolas, A; Gessa, GL; Melis, MR | 1 |
Ahlenius, S; Criborn, CO; Henriksson, C; Hillegaart, V | 1 |
Bergstrom, DA; Bromley, SD; Carlson, JH; Jackson, DM; Walters, JR | 1 |
Baldessarini, RJ; Froimowitz, M; Neumeyer, JL | 1 |
Andersson, B; Eriksson, E; Hjorth, S | 1 |
Cook, L; Steinfels, GF; Tam, SW | 1 |
Broekkamp, CL; Gower, AJ | 1 |
Carlsson, A; Clark, D; Hjorth, S; Sanchez, D; Svensson, K | 1 |
Bendesky, RJ; Jones, JH; Martin, GE | 1 |
Bacopoulos, NG; Koch, SW; Koe, BK | 1 |
Boissard, CG; Delini-Stula, A; Mogilnicka, E | 1 |
Palacios, JM; Wiederhold, KH | 1 |
Billingsley, ML; Roth, RH | 1 |
Carlsson, A; Hjorth, S; Jackson, D; Lindberg, P | 1 |
Arvidsson, LE; Carlsson, A; Clark, D; Hacksell, U; Hjorth, S; Johansson, A; Lindberg, P; Sanchez, D; Svensson, K; Wikström, H | 1 |
Carlsson, A | 1 |
Arnt, J; Hyttel, J | 1 |
Fenton, HM; Gerhardt, S; Leszczak, E; Liebman, JM | 1 |
Berendsen, HG; Broekkamp, CL; Gower, AJ; Princen, MM | 1 |
Ahlenius, S; Larsson, K | 1 |
Arvidsson, LE; Carlsson, A; Clark, D; Hacksell, U; Hjorth, S; Johansson, A; Lindberg, P; Nilsson, JL; Sanchez, D; Svensson, K; Wikström, H | 1 |
Adelung, C; Lang, JD; Späth, L; Starke, K | 1 |
Geyer, MA; Lee, EH | 1 |
Gudelsky, GA; Meltzer, HY; Mikuni, M; Simonovic, M | 1 |
Fratta, W; Gessa, GL; Napoli-Farris, L | 1 |
Ståhle, L; Ungerstedt, U | 1 |
Haubrich, DR; Martin, GE; Williams, M | 2 |
Waldmeier, PC | 1 |
Totaro, JA; Williams, M | 1 |
Meltzer, HY; Simonovic, M | 1 |
Bergstrom, DA; Gonzalez, AM; Huang, KX; Kreiss, DS; Sibley, DR; Walters, JR | 1 |
Lin, MY; Walters, DE | 1 |
Carlsson, A; Huff, RM; Kling-Petersen, T; Svensson, K; Waters, N | 1 |
Eguíbar, JR; Holmgren, B; Santos, A; Urbá-Holmgren, R | 1 |
Carlsson, A; Merello, M; Pirtosek, Z; Stern, G | 1 |
Curzon, P; Decker, MW | 1 |
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J | 1 |
Tamminga, CA | 1 |
Calas, AG; Goursaud, S; Hermans, E; Jeanjean, AP; Koener, B; Maloteaux, JM; Van De Stadt, M | 1 |
Heffner, TG; Jaen, JC; Meltzer, LT; Pugsley, TA; Wise, LD | 1 |
2 review(s) available for preclamol and apomorphine
Article | Year |
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Dopamine receptor agonists: mechanisms underlying autoreceptor selectivity. II. Theoretical considerations.
Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Corpus Striatum; Cyclic AMP; Dextroamphetamine; Dopamine; Humans; Isomerism; Lisuride; Models, Neurological; Molecular Conformation; Motor Activity; Nucleus Accumbens; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Receptors, Dopamine; Substantia Nigra; Synaptosomes | 1985 |
Partial dopamine agonists in the treatment of psychosis.
Topics: Animals; Apomorphine; Autoreceptors; Brain; Dopamine Agonists; Humans; Piperidines; Psychotic Disorders; Receptors, Dopamine | 2002 |
1 trial(s) available for preclamol and apomorphine
Article | Year |
---|---|
Preclamol and parkinsonian fluctuations.
Topics: Antiparkinson Agents; Apomorphine; Blood Pressure; Dopamine Agonists; Female; Humans; Injections, Subcutaneous; Male; Middle Aged; Movement; Parkinson Disease; Piperidines; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1993 |
78 other study(ies) available for preclamol and apomorphine
Article | Year |
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Dopamine autoreceptor agonists as potential antipsychotics. 3.6-Propyl-4,5,5a,6,7,8-hexahydrothiazolo[4,5-f]quinolin-2-amine.
Topics: Animals; Antipsychotic Agents; Dopamine Agents; Male; Molecular Structure; Rats; Stereoisomerism | 1991 |
4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties.
Topics: Animals; Apomorphine; Chemical Phenomena; Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Haloperidol; Male; Molecular Conformation; Molecular Structure; Motor Activity; Neurons; Pyridines; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Structure-Activity Relationship; Substantia Nigra; Thermodynamics; Thiazoles | 1990 |
Indolizidine and quinolizidine derivatives of the dopamine autoreceptor agonist 3-(3-hydroxyphenyl)-N-n-propylpiperidine (3-PPP).
Topics: alpha-Methyltyrosine; Animals; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Methyltyrosines; Molecular Conformation; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Structure-Activity Relationship | 1987 |
Monophenolic octahydrobenzo[f]quinolines: central dopamine- and serotonin-receptor stimulating activity.
Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Chemical Phenomena; Chemistry; Dihydroxyphenylalanine; In Vitro Techniques; Motor Activity; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin | 1982 |
Centrally acting serotonergic and dopaminergic agents. 1. Synthesis and structure-activity relationships of 2,3,3a,4,5,9b-hexahydro-1H-benz[e]indole derivatives.
Topics: Animals; Brain; Cats; Cattle; Dopamine Agents; Indoles; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Stereoisomerism; Structure-Activity Relationship | 1993 |
Centrally acting serotonergic and dopaminergic agents. 2. Synthesis and structure-activity relationships of 2,3,3a,4,9,9a-hexahydro-1H-benz[f]indole derivatives.
Topics: Animals; Binding Sites; Brain; Cats; Cattle; Dopamine Agents; Indoles; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes | 1993 |
A molecular mechanics approach to the understanding of presynaptic selectivity for centrally acting dopamine receptor agonists of the phenylpiperidine series.
Topics: Brain; Models, Molecular; Molecular Conformation; Piperidines; Receptors, Dopamine; Structure-Activity Relationship | 1986 |
Resolved 3-(3-hydroxyphenyl)-N-n-propylpiperidine and its analogues: central dopamine receptor activity.
Topics: Animals; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Male; Motor Activity; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Dopamine; Reserpine; Serotonin; X-Ray Diffraction | 1984 |
Substituted (S)-phenylpiperidines and rigid congeners as preferential dopamine autoreceptor antagonists: synthesis and structure-activity relationships.
Topics: Animals; Benzazepines; Brain; CHO Cells; Cricetinae; Dihydroxyphenylalanine; Dopamine D2 Receptor Antagonists; Habituation, Psychophysiologic; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Motor Activity; Optical Rotation; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Serotonin; Reserpine; Serotonin Antagonists; Spiperone; Structure-Activity Relationship; Transfection | 1994 |
Synthesis and evaluation of a set of 4-phenylpiperidines and 4-phenylpiperazines as D2 receptor ligands and the discovery of the dopaminergic stabilizer 4-[3-(methylsulfonyl)phenyl]-1-propylpiperidine (huntexil, pridopidine, ACR16).
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Binding, Competitive; Cell Line; Corpus Striatum; Dopamine; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Discovery; Drug Evaluation, Preclinical; Humans; Ligands; Male; Models, Chemical; Molecular Structure; Motor Activity; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2 | 2010 |
Sigma ligand-induced emesis in the pigeon.
Topics: Animals; Apomorphine; Columbidae; Dextromethorphan; Dizocilpine Maleate; Dopamine Agents; Guanidines; Haloperidol; Male; Pentobarbital; Phenazocine; Piperidines; Propranolol; Psychotropic Drugs; Pyrimidines; Receptors, Opioid; Receptors, sigma; Vomiting | 1992 |
The effects of pertussis toxin on dopamine D2 and serotonin 5-HT1A autoreceptor-mediated inhibition of neurotransmitter synthesis: relationship to receptor reserve.
Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Brain; Dopamine Agents; GTP-Binding Proteins; Levodopa; Male; Neurotransmitter Agents; Pertussis Toxin; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Ribose; Virulence Factors, Bordetella | 1992 |
Effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline on the prolactin suppression induced by a series of full and partial dopamine D2 receptor agonists in male rats.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Dopamine Agents; Ergolines; Levodopa; Male; Piperidines; Prolactin; Quinolines; Rats; Rats, Sprague-Dawley | 1992 |
Pre-synaptic dopaminergic control mechanisms for CCK-8 like immunoreactivity in the rat medial frontal cortex.
Topics: Animals; Apomorphine; Behavior, Animal; Cholecystokinin; Dopamine; Dopamine Agents; In Vitro Techniques; Male; Microinjections; N-Methylaspartate; Nerve Degeneration; Neurons; Piperidines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Dopamine | 1992 |
Differential effects of dopamine agonists upon stimulated limbic and striatal dopamine release: in vivo voltammetric data.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Bromocriptine; Corpus Striatum; Dopamine; Dopamine Agents; Electrochemistry; Electrophysiology; Ergolines; In Vitro Techniques; Limbic System; Male; Microelectrodes; Nucleus Accumbens; Pergolide; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Stereotaxic Techniques | 1991 |
Dopamine receptors, controlling dopamine levels in rat adrenal glands-comparison with central dopaminergic autoreceptors.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adrenal Medulla; Animals; Apomorphine; Azepines; Diencephalon; Domperidone; Dopamine; Dopamine Agents; Epinephrine; Ergolines; Lisuride; Male; Norepinephrine; Phenanthrenes; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Telencephalon | 1991 |
Sigma-receptors: implication for the control of neuronal activity of nigral dopamine-containing neurons.
Topics: Animals; Apomorphine; Binding, Competitive; Dizocilpine Maleate; Dopamine; Dopamine Agents; Male; Neurons; Piperidines; Quinolines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Stereotaxic Techniques; Substantia Nigra | 1991 |
Yawning produced by dopamine agonists in rhesus monkeys.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Apomorphine; Benzazepines; Dopamine; Dopamine Agents; Dopamine Antagonists; Ergolines; Macaca mulatta; Male; Physostigmine; Piperidines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Yawning | 1991 |
The role of the dopaminergic system in the modulation of the acoustic startle response in the rat.
Topics: Animals; Apomorphine; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Reflex, Startle; Stereoisomerism | 1990 |
Synthesis and evaluation of optically pure [3H]-(+)-pentazocine, a highly potent and selective radioligand for sigma receptors.
Topics: Animals; Apomorphine; Binding, Competitive; Brain; Cell Membrane; Chemical Phenomena; Chemistry; Dopamine Agents; Guanidines; Guinea Pigs; Hydroxides; Molecular Structure; Pentazocine; Phencyclidine; Piperidines; Potassium; Potassium Compounds; Receptors, Dopamine; Receptors, Opioid; Receptors, sigma; Tritium | 1989 |
Dopamine autoreceptor agonists attenuate spontaneous motor activity but not spontaneous fighting in individually-housed mice.
Topics: Aggression; Agonistic Behavior; Animals; Apomorphine; Catalepsy; Dopamine Agents; Dose-Response Relationship, Drug; Housing, Animal; Male; Mice; Motor Activity; Piperidines; Social Isolation; Stereoisomerism | 1989 |
Inhibition by pertussis toxin of the soporific effects induced by stimulation of dopamine D2 autoreceptors in the ventral tegmental area in rats.
Topics: Adenylate Cyclase Toxin; Animals; Apomorphine; Electrocardiography; Male; Pertussis Toxin; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tegmentum Mesencephali; Time Factors; Virulence Factors, Bordetella | 1989 |
Relative selectivity of 6,7-dihydroxy-2-dimethylaminotetralin, N-n-propyl-3-(3-hydroxyphenyl)piperidine, N-n-propylnorapomorphine and pergolide as agonists at striatal dopamine autoreceptors and postsynaptic dopamine receptors.
Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Ergolines; Haloperidol; Homovanillic Acid; Male; Naphthalenes; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Sodium Oxybate; Tetrahydronaphthalenes; Tyrosine 3-Monooxygenase | 1985 |
Effect of dopaminergic drugs on striatal acetylcholine concentration.
Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1985 |
Is inhibition of striatal synaptosomal tyrosine hydroxylation by dopamine agonists a measure of dopamine autoreceptor function?
Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Azepines; Corpus Striatum; Depression, Chemical; Dopamine; Ergolines; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Pergolide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter; Synaptosomes; Tyrosine 3-Monooxygenase | 1985 |
Performance deficit induced by low doses of dopamine agonists in rats. Toward a model for approaching the neurobiology of negative schizophrenic symptomatology?
Topics: Amisulpride; Animals; Antipsychotic Agents; Apomorphine; Disease Models, Animal; Male; Phenothiazines; Pimozide; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reinforcement Schedule; Reinforcement, Psychology; Schizophrenia; Schizophrenic Psychology; Sulpiride | 1986 |
Effects of dopaminomimetics on the secretion of VIP-like immunoreactivity in conscious dogs.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Apomorphine; Benzazepines; Dogs; Ergolines; Nitroglycerin; Pergolide; Piperidines; Prazosin; Receptors, Dopamine; Somatostatin; Vasoactive Intestinal Peptide | 1986 |
Two automated locomotor activity tests for dopamine autoreceptor agonists.
Topics: Amphetamine; Animals; Antipsychotic Agents; Apomorphine; Drug Evaluation, Preclinical; Exploratory Behavior; Indoles; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1986 |
Comparison of changes in locomotor activity with striatal homovanillic acid and 3,4-dihydroxyphenylacetic acid concentrations following the bilateral intranigral injection of dopamine agonist drugs in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Female; Homovanillic Acid; Motor Activity; Phenylacetates; Piperidines; Rats; Rats, Inbred Strains; Substantia Nigra; Sucrose | 1987 |
Relationship between receptor occupancy and response at striatal dopamine autoreceptors.
Topics: 4-Butyrolactone; Adrenergic alpha-Antagonists; Animals; Apomorphine; Corpus Striatum; Dihydroxyphenylalanine; Homeostasis; Hydrazines; Levodopa; Male; Piperidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1987 |
Effects of apomorphine and (+/-)-3-(3-hydroxyphenyl)-N-n-propylpiperidine, injected into the striatum, on the caudate spindle in the rat.
Topics: Animals; Antipsychotic Agents; Apomorphine; Corpus Striatum; Dopamine; Electric Stimulation; Electrophysiology; Injections; Male; Piperidines; Rats; Rats, Inbred Strains | 1987 |
Dopamine D-2 receptors in the ventral tegmental area mediate behavioural and electrocortical sleep of dopaminergic drugs in rats.
Topics: Animals; Apomorphine; Behavior, Animal; Cerebral Cortex; Dopamine Agents; Electric Stimulation; Electroencephalography; Piperidines; Rats; Receptors, Dopamine; Sleep; Tegmentum Mesencephali | 1988 |
Ventral tegmental area: site through which dopamine D2-receptor agonists evoke behavioural and electrocortical sleep in rats.
Topics: Animals; Apomorphine; Cerebral Cortex; Electroencephalography; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Sleep; Sulpiride; Tegmentum Mesencephali | 1988 |
7-[3-(4-[2,3-Dimethylphenyl]piperazinyl)propoxy]-2(1H)-quinolinone (OPC-4392), a presynaptic dopamine autoreceptor agonist and postsynaptic D2 receptor antagonist.
Topics: Animals; Apomorphine; Brain; Corpus Striatum; Diencephalon; Dihydroxyphenylalanine; Frontal Lobe; Hydroxydopamines; Kainic Acid; Kinetics; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxidopamine; Piperazines; Piperidines; Quinolines; Quinolones; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Telencephalon | 1988 |
Heterogeneous rotational responsiveness in 6-hydroxydopamine-denervated rats: pharmacological and neurochemical characterization.
Topics: Animals; Apomorphine; Benzopyrans; Brain Chemistry; Corpus Striatum; Dopamine; Ergolines; Hydroxydopamines; Male; Oxidopamine; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Rotation; Stereotyped Behavior; Sympathectomy, Chemical | 1988 |
Effects of intraperitoneal administration of apomorphine and the isomers of 3-(1-propyl-3-piperidinyl)phenol on the firing activity of substantia nigra dopamine neurons: comparison of agonist efficacies and development of acute tolerance.
Topics: Action Potentials; Animals; Apomorphine; Drug Tolerance; Injections, Intraperitoneal; Injections, Intravenous; Male; Neurons; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Substantia Nigra | 1988 |
Pharmacological profile of dopamine receptor agonists as studied by brain dialysis in behaving rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Azepines; Behavior, Animal; Benzazepines; Brain; Dialysis; Dopamine; Ergolines; Homovanillic Acid; Isomerism; Male; Motor Activity; Neurons; Pergolide; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Time Factors | 1988 |
Apomorphine-induced penile erection and yawning: site of action in brain.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Brain; Dopamine; Dopamine Antagonists; Ergolines; Male; Microinjections; Paraventricular Hypothalamic Nucleus; Penile Erection; Piperidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Yawning | 1987 |
Partial protection against hyperbaric oxygen induced convulsions by dopaminergic agents in mice: possible involvement of autoreceptors?
Topics: Animals; Antiparkinson Agents; Apomorphine; Body Temperature; Dose-Response Relationship, Drug; Haloperidol; Hyperbaric Oxygenation; Levodopa; Male; Mice; Mice, Inbred CBA; Piperidines; Reaction Time; Receptors, Dopamine; Respiration; Seizures | 1987 |
Differential electrophysiological effects of 3-PPP and its enantiomers on dopamine autoreceptors and postsynaptic receptors.
Topics: Action Potentials; Animals; Apomorphine; Electrodes, Implanted; Globus Pallidus; Male; Neurons; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Substantia Nigra; Synapses | 1986 |
A stereochemical explanation of the dopamine agonist and antagonist activity of stereoisomeric pairs.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Apomorphine; Chemical Phenomena; Chemistry; Dopamine; Dopamine Antagonists; Molecular Conformation; Naphthalenes; Piperidines; Receptors, Dopamine; Stereoisomerism; Structure-Activity Relationship; Tetrahydronaphthalenes; Thermodynamics | 1986 |
Stereoselective inhibition of prolactin secretion by (-)-HW-165, a novel 3-PPP congener; further support for similarities between central DA autoreceptors and pituitary lactotroph DA receptors.
Topics: 4-Butyrolactone; Animals; Apomorphine; Depression, Chemical; Male; Phenanthrenes; Piperidines; Pituitary Gland; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism | 1986 |
(+)-3-(3-hydroxyphenyl)-N-(1-propyl)piperidine [(+)-3-PPP] but not (-)-3-PPP produces (+)-N-allylnormetazocine-like (SKF 10,047) discriminative stimuli.
Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Isomerism; Male; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Inbred F344 | 1986 |
Dopaminergic agents including 3-PPP and its enantiomers on medial septal self-stimulation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Appetite Depressants; Benzazepines; Dextroamphetamine; Drug Interactions; Haloperidol; Male; Nomifensine; Piperidines; Rats; Receptors, Dopamine; Self Stimulation; Stereoisomerism; Sulpiride; Tetrahydronaphthalenes | 1985 |
Dopamine receptor-mediated hypothermia induced in rats by (+)-, but not by (-)-3-PPP.
Topics: Animals; Apomorphine; Biogenic Amines; Body Temperature; Brain Chemistry; Dose-Response Relationship, Drug; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism | 1985 |
Lack of effect of intranigral administration of a dopamine analogue, (+/-)-3-(3-hydroxyphenyl)-N,n-propylpiperidine [(+/-)-3-PPP], on nigrostriatal dopamine neurones.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Female; Homovanillic Acid; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra | 1985 |
(+)- and (-)-3-PPP exhibit different intrinsic activity at striatal dopamine autoreceptors controlling dopamine synthesis.
Topics: 4-Butyrolactone; Animals; Apomorphine; Corpus Striatum; Dopamine; Isomerism; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Neurotransmitter | 1984 |
Different actions of TL-99 and 3-PPP in producing contraversive turning in the 6-OHDA-lesioned rat.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apomorphine; Female; Hydroxydopamines; Motor Activity; Naphthalenes; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Substantia Nigra; Tetrahydronaphthalenes; Yohimbine | 1983 |
Differential effects of the enantiomers of 3-(3-hydroxyphenyl)-N-n-propylpiperidine (3-PPP) at dopamine receptor sites.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Corpus Striatum; Dopamine; Homovanillic Acid; Male; Mice; Molecular Conformation; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Synaptosomes; Tyrosine 3-Monooxygenase | 1983 |
Effects of apomorphine, TL-99 and 3-PPP on yawning in rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apomorphine; Behavior, Animal; Haloperidol; Male; Naphthalenes; Piperidines; Rats; Tetrahydronaphthalenes | 1984 |
Presynaptic dopaminergic agonists modify brain glucose metabolism in a way similar to the neuroleptics.
Topics: Animals; Antipsychotic Agents; Apomorphine; Brain; Catecholamines; Ergolines; Glucose; Naphthalenes; Piperidines; Rats; Reserpine; Tetrahydronaphthalenes | 1984 |
Dopamine agonists stimulate protein carboxylmethylation in striatal synaptosomes.
Topics: Animals; Apomorphine; Butaclamol; Corpus Striatum; Dopamine; Hydroxydopamines; In Vitro Techniques; Male; Nerve Tissue Proteins; Piperidines; Potassium; Protein Methyltransferases; Protein O-Methyltransferase; Rats; Rats, Inbred Strains; S-Adenosylhomocysteine; S-Adenosylmethionine; Synaptosomes | 1982 |
A behavioural study of the changes in the central nervous system of mice after subchronic treatment with the selective dopamine autoreceptor agonist 3-PPP (dl-3-[3-hydroxyphenyl]-N-n-propylpiperidine).
Topics: Animals; Apomorphine; Behavior, Animal; Dextroamphetamine; Dose-Response Relationship, Drug; Male; Motor Activity; Muridae; Piperidines; Receptors, Dopamine; Synaptic Transmission | 1982 |
Central dopamine receptor agonist and antagonist actions of the enantiomers of 3-PPP.
Topics: Animals; Apomorphine; Behavior, Animal; Biogenic Amines; Brain Chemistry; Dextroamphetamine; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism | 1983 |
Dopamine receptor agonists: intrinsic activity vs. state of receptor.
Topics: Animals; Apomorphine; Brain; Denervation; Exploratory Behavior; Hydroxydopamines; Oxidopamine; Piperidines; Prolactin; Rats; Receptors, Dopamine; Stereoisomerism; Sympathectomy, Chemical | 1983 |
Postsynaptic dopamine agonistic effects of 3-PPP enantiomers revealed by bilateral 6-hydroxy-dopamine lesions and by chronic reserpine treatment in rats.
Topics: Animals; Antiparkinson Agents; Apomorphine; Behavior, Animal; Drug Interactions; Hydroxydopamines; Male; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Reserpine; Stereoisomerism; Stimulation, Chemical | 1984 |
Evidence for heterogeneous rotational responsiveness to apomorphine, 3-PPP and SKF 38393 in 6-hydroxydopamine-denervated rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Clozapine; Ergolines; Humans; Hydroxydopamines; Male; Oxidopamine; Pergolide; Piperidines; Postural Balance; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Sympathectomy, Chemical | 1984 |
The yawning-penile erection syndrome as a model for putative dopamine autoreceptor activity.
Topics: Animals; Apomorphine; Drug Interactions; Haloperidol; Inhalation; Isomerism; Male; Models, Psychological; Penis; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Respiration; Sexual Behavior, Animal; Syndrome | 1984 |
Apomorphine and haloperidol-induced effects on male rat sexual behavior: no evidence for actions due to stimulation of central dopamine autoreceptors.
Topics: Animals; Apomorphine; Brain; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal | 1984 |
The search for selective dopaminergic autoreceptor agonists.
Topics: Animals; Apomorphine; Dextroamphetamine; Dose-Response Relationship, Drug; Motor Activity; Optical Rotation; Piperidines; Rats; Receptors, Dopamine; Reserpine | 1983 |
Further functional in vitro comparison of pre- and postsynaptic dopamine receptors in the rabbit caudate nucleus.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Apomorphine; Benzazepines; Caudate Nucleus; Choline; Clonidine; Female; Male; Piperidines; Rabbits; Receptors, Dopamine | 1983 |
Similarities of the effects of apomorphine and 3-PPP on serotonin neurons.
Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Corpus Striatum; Haloperidol; Hippocampus; Male; Neurons; Piperidines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Spectrometry, Fluorescence | 1983 |
Interaction of (+)- and (-)-3-PPP with the dopamine receptor in the anterior pituitary gland.
Topics: Animals; Apomorphine; Binding Sites; Cell Membrane; Depression, Chemical; In Vitro Techniques; Male; Methyltyrosines; Piperidines; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereoisomerism | 1984 |
Stimulation of dopamine autoreceptors elicits "premature ejaculation" in rats.
Topics: Animals; Apomorphine; Copulation; Domperidone; Dopamine Antagonists; Ejaculation; Female; Haloperidol; Lisuride; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sexual Behavior, Animal | 1984 |
Assessment of dopamine autoreceptor agonist properties of apomorphine, (+)-3-PPP and (-)-3-PPP by recording of yawning behaviour in rats.
Topics: Animals; Apomorphine; Behavior, Animal; Domperidone; Male; Motor Activity; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sulpiride | 1984 |
A pharmacological comparison of 6,7-dihydroxy-2-dimethylaminotetralin (TL-99) and N-n-propyl-3-(3-hydroxyphenyl)piperidine with (3-PPP) selected dopamine agonists.
Topics: 4-Butyrolactone; Animals; Apomorphine; Cell Membrane; Corpus Striatum; Female; Humans; Hydroxydopamines; Naphthalenes; Oxidopamine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Stereotyped Behavior; Tetrahydronaphthalenes | 1982 |
Biphasic effects of some dopamine agonists on striatal acetylcholine concentrations.
Topics: Acetylcholine; Animals; Apomorphine; Corpus Striatum; Dopamine; Male; Piperidines; Piribedil; Rats; Tetrahydronaphthalenes; Time Factors | 1983 |
Interaction of the putative dopamine autoreceptor agonists 3-PPP and TL-99 with [3H]apomorphine binding sites in rat striatal membranes.
Topics: Animals; Apomorphine; Binding Sites; Binding, Competitive; Corpus Striatum; In Vitro Techniques; Kinetics; Membranes; Naphthalenes; Piperidines; Rats; Receptors, Dopamine; Spiperone; Tetrahydronaphthalenes | 1982 |
Effect of 3-PPP, a putative dopamine autoreceptor agonist, on rat serum prolactin levels.
Topics: Animals; Apomorphine; Binding, Competitive; Humans; Male; Piperidines; Prolactin; Rats; Receptors, Dopamine; Reserpine; Spiperone; Stereotyped Behavior | 1981 |
Pharmacological profiles of the putative dopamine autoreceptor agonists 3-PPP and TL-99.
Topics: 4-Butyrolactone; Animals; Apomorphine; Brain; Dogs; Dopamine; Female; Male; Mice; Motor Activity; Naphthalenes; Piperidines; Rats; Receptors, Dopamine; Tetrahydronaphthalenes | 1981 |
Dopamine receptor agonist potencies for inhibition of cell firing correlate with dopamine D3 receptor binding affinities.
Topics: Aminoquinolines; Animals; Apomorphine; Azepines; Benzothiazoles; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Male; Neurons; Phenethylamines; Piperidines; Pramipexole; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Substantia Nigra; Tetrahydronaphthalenes; Thiazoles; Thiophenes; Transfection | 1995 |
Dopamine D2 autoreceptors in rats are behaviorally functional at 21 but not 10 days of age.
Topics: Aging; Aminoquinolines; Animals; Apomorphine; Azepines; Behavior, Animal; Benzothiazoles; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Motor Activity; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Thiazoles | 1994 |
Behavioral and neurochemical data suggest functional differences between dopamine D2 and D3 receptors.
Topics: Analysis of Variance; Animals; Apomorphine; Benzothiazoles; CHO Cells; Cricetinae; Cricetulus; Dihydroxyphenylalanine; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Male; Microdialysis; Mitogens; Motor Activity; Piperidines; Pramipexole; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Thiazoles; Transfection | 1994 |
Two inbred rat sublines that differ in spontaneous yawning behavior also differ in their responses to cholinergic and dopaminergic drugs.
Topics: Animals; Apomorphine; Dopamine Agents; Dose-Response Relationship, Drug; Male; Parasympathomimetics; Physostigmine; Pilocarpine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Receptors, Dopamine; Species Specificity; Yawning | 1993 |
Effects of phencyclidine (PCP) and (+)MK-801 on sensorimotor gating in CD-1 mice.
Topics: Acoustic Stimulation; Animals; Apomorphine; Clozapine; Dextroamphetamine; Dizocilpine Maleate; Dopamine Agonists; Dose-Response Relationship, Drug; Haloperidol; Male; Mice; Mice, Inbred Strains; Phencyclidine; Piperidines; Rats; Receptors, sigma; Reflex, Startle; Species Specificity | 1998 |
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine | 2001 |
Pharmacological blockade of dopamine D2 receptors by aripiprazole is not associated with striatal sensitization.
Topics: Animals; Apomorphine; Aripiprazole; Buffers; Catalepsy; Cell Membrane; Cerebral Cortex; Corpus Striatum; Domperidone; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Antagonism; Drug Partial Agonism; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Hippocampus; Male; Piperazines; Piperidines; Pyridines; Quinolones; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Stereotyped Behavior; Up-Regulation | 2011 |
Dopamine autoreceptor agonists as potential antipsychotics. 1. (Aminoalkoxy)anilines.
Topics: Aniline Compounds; Animals; Antipsychotic Agents; Behavior, Animal; Brain; Chemical Phenomena; Chemistry; In Vitro Techniques; Rats; Receptors, Dopamine; Saimiri; Structure-Activity Relationship | 1988 |