Page last updated: 2024-09-03

pre 084 and preclamol

pre 084 has been researched along with preclamol in 4 studies

Compound Research Comparison

Studies
(pre 084)
Trials
(pre 084)
Recent Studies (post-2010)
(pre 084)
Studies
(preclamol)
Trials
(preclamol)
Recent Studies (post-2010) (preclamol)
1160731200
1160732408
116073363520

Protein Interaction Comparison

ProteinTaxonomypre 084 (IC50)preclamol (IC50)
D(2) dopamine receptorRattus norvegicus (Norway rat)2.0703
DRattus norvegicus (Norway rat)0.93
D(3) dopamine receptorRattus norvegicus (Norway rat)0.93
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.93
D(4) dopamine receptorRattus norvegicus (Norway rat)0.93
Sigma non-opioid intracellular receptor 1Rattus norvegicus (Norway rat)0.1599

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowen, WD; Cao, J; George, C; Husbands, SM; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH; Williams, W1
Enache, LA; Gilardi, R; Mattson, MV; Moriarty, RM; Prakash, O; Zhao, L1
Baeyens, JM; Cobos, EJ; Del Pozo, E1
Bezprozvanny, IB; Bol'shakova, AV; Gainullina, AN; Kraskovskaya, NA; Kukanova, EO; Vlasova, OL1

Other Studies

4 other study(ies) available for pre 084 and preclamol

ArticleYear
Dual probes for the dopamine transporter and sigma1 receptors: novel piperazinyl alkyl-bis(4'-fluorophenyl)amine analogues as potential cocaine-abuse therapeutic agents.
    Journal of medicinal chemistry, 2003, Jun-19, Volume: 46, Issue:13

    Topics: Animals; Binding, Competitive; Brain; Cocaine-Related Disorders; Crystallography, X-Ray; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Structure-Activity Relationship

2003
Rigid phencyclidine analogues. Binding to the phencyclidine and sigma 1 receptors.
    Journal of medicinal chemistry, 1998, Feb-12, Volume: 41, Issue:4

    Topics: Animals; Brain; Crystallography, X-Ray; Indicators and Reagents; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Phencyclidine; Radioligand Assay; Rats; Receptors, Phencyclidine; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship

1998
Phenytoin differentially modulates the affinity of agonist and antagonist ligands for sigma 1 receptors of guinea pig brain.
    Synapse (New York, N.Y.), 2005, Mar-01, Volume: 55, Issue:3

    Topics: Allosteric Regulation; Animals; Anisoles; Anticonvulsants; Binding, Competitive; Brain; Dextromethorphan; Drug Interactions; Ethylenediamines; Guinea Pigs; Haloperidol; Ligands; Male; Morpholines; Neurons; Phenazocine; Phenytoin; Piperazines; Piperidines; Progesterone; Propylamines; Receptors, sigma; Synaptic Transmission

2005
Neuroprotective Effect of σ1-Receptors on the Cell Model of Huntington's Disease.
    Bulletin of experimental biology and medicine, 2017, Volume: 164, Issue:2

    Topics: Animals; Anisoles; Calcium; Cerebral Cortex; Corpus Striatum; Dendritic Spines; Gene Expression; Homeostasis; Huntington Disease; Male; Mice; Models, Biological; Morpholines; Neurons; Piperidines; Primary Cell Culture; Propylamines; Receptors, sigma; RNA, Small Interfering; Sigma-1 Receptor; Synapses; Synaptic Transmission; Transduction, Genetic

2017