Page last updated: 2024-09-03

pre 084 and dizocilpine

pre 084 has been researched along with dizocilpine in 2 studies

Compound Research Comparison

Studies
(pre 084)
Trials
(pre 084)
Recent Studies (post-2010)
(pre 084)
Studies
(dizocilpine)
Trials
(dizocilpine)
Recent Studies (post-2010) (dizocilpine)
11607377030

Protein Interaction Comparison

ProteinTaxonomypre 084 (IC50)dizocilpine (IC50)
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.002
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.0149
Lysosomal Pro-X carboxypeptidaseHomo sapiens (human)0.0053
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.0149
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.0149
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.0149
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.009
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.029
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.009
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.0149
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.0149
Sigma non-opioid intracellular receptor 1Rattus norvegicus (Norway rat)1.7
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.0149

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Enache, LA; Gilardi, R; Mattson, MV; Moriarty, RM; Prakash, O; Zhao, L1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1

Other Studies

2 other study(ies) available for pre 084 and dizocilpine

ArticleYear
Rigid phencyclidine analogues. Binding to the phencyclidine and sigma 1 receptors.
    Journal of medicinal chemistry, 1998, Feb-12, Volume: 41, Issue:4

    Topics: Animals; Brain; Crystallography, X-Ray; Indicators and Reagents; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Phencyclidine; Radioligand Assay; Rats; Receptors, Phencyclidine; Receptors, sigma; Sigma-1 Receptor; Structure-Activity Relationship

1998
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009