pre 084 has been researched along with dizocilpine maleate in 10 studies
Studies (pre 084) | Trials (pre 084) | Recent Studies (post-2010) (pre 084) | Studies (dizocilpine maleate) | Trials (dizocilpine maleate) | Recent Studies (post-2010) (dizocilpine maleate) |
---|---|---|---|---|---|
116 | 0 | 73 | 7,741 | 9 | 1,449 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (20.00) | 18.2507 |
2000's | 6 (60.00) | 29.6817 |
2010's | 2 (20.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L | 1 |
Maurice, T; Nabeshima, T; Parish, DW; Privat, A; Su, TP | 1 |
Maurice, T; Phan, VL; Privat, A; Su, TP | 1 |
Hayashi, T; Maurice, T; Su, TP | 1 |
Maurice, T; Phan, VL; Privat, A | 1 |
Guillemain, I; Maurice, T; Phan, VL; Urani, A | 1 |
Partridge, LD; Schiess, AR | 1 |
Cortés-Montero, E; Garzón, J; Rodríguez-Muñoz, M; Sánchez-Blázquez, P | 1 |
10 other study(ies) available for pre 084 and dizocilpine maleate
Article | Year |
---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship | 2013 |
PRE-084, a sigma selective PCP derivative, attenuates MK-801-induced impairment of learning in mice.
Topics: Amnesia; Animals; Anti-Anxiety Agents; Avoidance Learning; Cholinergic Agents; Dizocilpine Maleate; Dose-Response Relationship, Drug; Haloperidol; Learning; Male; Maze Learning; Memory; Memory, Short-Term; Mice; Morpholines; Phencyclidine; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma | 1994 |
Modulation of steroidal levels by adrenalectomy/castration and inhibition of neurosteroid synthesis enzymes affect sigma1 receptor-mediated behaviour in mice.
Topics: Adrenalectomy; Animals; Behavior, Animal; Brain; Cerebral Cortex; Dizocilpine Maleate; Enzyme Inhibitors; Finasteride; Hippocampus; Male; Mice; Morpholines; Orchiectomy; Phenazocine; Receptors, sigma; Spatial Behavior; Steroids | 1999 |
Ca(2+) signaling via sigma(1)-receptors: novel regulatory mechanism affecting intracellular Ca(2+) concentration.
Topics: Animals; Bradykinin; Calcium; Calcium Signaling; Dizocilpine Maleate; Morpholines; Nifedipine; Oligonucleotides, Antisense; Pentazocine; Potassium Chloride; Pregnenolone; Rabbits; Receptors, sigma; Tumor Cells, Cultured | 2000 |
The anti-amnesic effects of sigma1 (sigma1) receptor agonists confirmed by in vivo antisense strategy in the mouse.
Topics: Amnesia; Animals; Brain; Dizocilpine Maleate; Excitatory Amino Acid Agonists; In Vitro Techniques; Learning Disabilities; Male; Maze Learning; Mice; Morpholines; Nootropic Agents; Oligonucleotides, Antisense; Phenazocine; Piperazines; Receptors, sigma | 2001 |
Differential involvement of the sigma(1) (sigma(1)) receptor in the anti-amnesic effect of neuroactive steroids, as demonstrated using an in vivo antisense strategy in the mouse.
Topics: Amnesia; Animals; Avoidance Learning; Behavior, Animal; Binding Sites; Blotting, Western; Brain; Cerebral Cortex; Dehydroepiandrosterone; Dizocilpine Maleate; Dose-Response Relationship, Drug; Hippocampus; In Vitro Techniques; Learning Disabilities; Male; Maze Learning; Memory; Mice; Morpholines; Oligonucleotides, Antisense; Phenazocine; Pregnenolone; Receptors, sigma; Sigma-1 Receptor | 2001 |
Pregnenolone sulfate acts through a G-protein-coupled sigma1-like receptor to enhance short term facilitation in adult hippocampal neurons.
Topics: Animals; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GTP-Binding Protein alpha Subunits, Gi-Go; Hippocampus; In Vitro Techniques; Male; Morpholines; Neurons; Patch-Clamp Techniques; Pertussis Toxin; Piperazines; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sigma-1 Receptor; Synapses; Synaptic Transmission; Time Factors | 2005 |
Sigma 1 Receptor Antagonists Inhibit Manic-Like Behaviors in Two Congenital Strains of Mice.
Topics: Animals; Animals, Outbred Strains; Antimanic Agents; Cyclopropanes; Dizocilpine Maleate; Drug Interactions; Glycogen Synthase Kinase 3 beta; Mice; Mice, Knockout; Morpholines; Motor Activity; Nerve Tissue Proteins; Piperidines; Protein Kinase Inhibitors; Receptors, sigma | 2018 |