Page last updated: 2024-09-03

pre 084 and dizocilpine maleate

pre 084 has been researched along with dizocilpine maleate in 10 studies

Compound Research Comparison

Studies
(pre 084)
Trials
(pre 084)
Recent Studies (post-2010)
(pre 084)
Studies
(dizocilpine maleate)
Trials
(dizocilpine maleate)
Recent Studies (post-2010) (dizocilpine maleate)
1160737,74191,449

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (20.00)18.2507
2000's6 (60.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Maurice, T; Nabeshima, T; Parish, DW; Privat, A; Su, TP1
Maurice, T; Phan, VL; Privat, A; Su, TP1
Hayashi, T; Maurice, T; Su, TP1
Maurice, T; Phan, VL; Privat, A1
Guillemain, I; Maurice, T; Phan, VL; Urani, A1
Partridge, LD; Schiess, AR1
Cortés-Montero, E; Garzón, J; Rodríguez-Muñoz, M; Sánchez-Blázquez, P1

Other Studies

10 other study(ies) available for pre 084 and dizocilpine maleate

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
PRE-084, a sigma selective PCP derivative, attenuates MK-801-induced impairment of learning in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:4

    Topics: Amnesia; Animals; Anti-Anxiety Agents; Avoidance Learning; Cholinergic Agents; Dizocilpine Maleate; Dose-Response Relationship, Drug; Haloperidol; Learning; Male; Maze Learning; Memory; Memory, Short-Term; Mice; Morpholines; Phencyclidine; Pyrimidines; Rats; Rats, Wistar; Receptors, sigma

1994
Modulation of steroidal levels by adrenalectomy/castration and inhibition of neurosteroid synthesis enzymes affect sigma1 receptor-mediated behaviour in mice.
    The European journal of neuroscience, 1999, Volume: 11, Issue:7

    Topics: Adrenalectomy; Animals; Behavior, Animal; Brain; Cerebral Cortex; Dizocilpine Maleate; Enzyme Inhibitors; Finasteride; Hippocampus; Male; Mice; Morpholines; Orchiectomy; Phenazocine; Receptors, sigma; Spatial Behavior; Steroids

1999
Ca(2+) signaling via sigma(1)-receptors: novel regulatory mechanism affecting intracellular Ca(2+) concentration.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: Animals; Bradykinin; Calcium; Calcium Signaling; Dizocilpine Maleate; Morpholines; Nifedipine; Oligonucleotides, Antisense; Pentazocine; Potassium Chloride; Pregnenolone; Rabbits; Receptors, sigma; Tumor Cells, Cultured

2000
The anti-amnesic effects of sigma1 (sigma1) receptor agonists confirmed by in vivo antisense strategy in the mouse.
    Brain research, 2001, Apr-13, Volume: 898, Issue:1

    Topics: Amnesia; Animals; Brain; Dizocilpine Maleate; Excitatory Amino Acid Agonists; In Vitro Techniques; Learning Disabilities; Male; Maze Learning; Mice; Morpholines; Nootropic Agents; Oligonucleotides, Antisense; Phenazocine; Piperazines; Receptors, sigma

2001
Differential involvement of the sigma(1) (sigma(1)) receptor in the anti-amnesic effect of neuroactive steroids, as demonstrated using an in vivo antisense strategy in the mouse.
    British journal of pharmacology, 2001, Volume: 134, Issue:8

    Topics: Amnesia; Animals; Avoidance Learning; Behavior, Animal; Binding Sites; Blotting, Western; Brain; Cerebral Cortex; Dehydroepiandrosterone; Dizocilpine Maleate; Dose-Response Relationship, Drug; Hippocampus; In Vitro Techniques; Learning Disabilities; Male; Maze Learning; Memory; Mice; Morpholines; Oligonucleotides, Antisense; Phenazocine; Pregnenolone; Receptors, sigma; Sigma-1 Receptor

2001
Pregnenolone sulfate acts through a G-protein-coupled sigma1-like receptor to enhance short term facilitation in adult hippocampal neurons.
    European journal of pharmacology, 2005, Jul-25, Volume: 518, Issue:1

    Topics: Animals; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GTP-Binding Protein alpha Subunits, Gi-Go; Hippocampus; In Vitro Techniques; Male; Morpholines; Neurons; Patch-Clamp Techniques; Pertussis Toxin; Piperazines; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sigma-1 Receptor; Synapses; Synaptic Transmission; Time Factors

2005
Sigma 1 Receptor Antagonists Inhibit Manic-Like Behaviors in Two Congenital Strains of Mice.
    The international journal of neuropsychopharmacology, 2018, 10-01, Volume: 21, Issue:10

    Topics: Animals; Animals, Outbred Strains; Antimanic Agents; Cyclopropanes; Dizocilpine Maleate; Drug Interactions; Glycogen Synthase Kinase 3 beta; Mice; Mice, Knockout; Morpholines; Motor Activity; Nerve Tissue Proteins; Piperidines; Protein Kinase Inhibitors; Receptors, sigma

2018