Page last updated: 2024-09-03

pre 084 and cocaine

pre 084 has been researched along with cocaine in 10 studies

Compound Research Comparison

Studies
(pre 084)
Trials
(pre 084)
Recent Studies (post-2010)
(pre 084)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
11607332,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomypre 084 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (40.00)29.6817
2010's6 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowen, WD; Cao, J; George, C; Husbands, SM; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH; Williams, W1
Maurice, T; Phan, VL; Romieu, P; Urani, A1
Atianzar, K; Dubinett, SM; Escuadro, B; Gardner, B; Sharma, S; Tashkin, DP; Zhu, LX1
Dubinett, SM; Gardner, B; Roth, MD; Sharma, S; Tashkin, DP; Zhu, LX1
Hiranita, T; Katz, JL; Soto, PL; Tanda, G2
Garcés-Ramírez, L; Green, JL; Hiranita, T; Katz, JL; Kopajtic, TA; McCurdy, CR; Mereu, M; Mesangeau, C; Narayanan, S; Tanda, G; Thomas, AM1
Abdelazeem, AH; Hiranita, T; Katz, JL; Kopajtic, TA; McCurdy, CR; Mesangeau, C; Narayanan, S; Rice, KC1
Amara, SG; Chin, FT; Hiranita, T; Hong, WC; Katz, JL; McCurdy, CR; Su, TP; Yano, H1
Álvarez, M; Andino Norat, MC; Gorantla, S; López, OV; Meléndez, LM; Segarra, AC; Skolasky, RL1

Other Studies

10 other study(ies) available for pre 084 and cocaine

ArticleYear
Dual probes for the dopamine transporter and sigma1 receptors: novel piperazinyl alkyl-bis(4'-fluorophenyl)amine analogues as potential cocaine-abuse therapeutic agents.
    Journal of medicinal chemistry, 2003, Jun-19, Volume: 46, Issue:13

    Topics: Animals; Binding, Competitive; Brain; Cocaine-Related Disorders; Crystallography, X-Ray; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Structure-Activity Relationship

2003
Strain differences in sigma(1) receptor-mediated behaviours are related to neurosteroid levels.
    The European journal of neuroscience, 2002, Volume: 15, Issue:9

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Behavior, Animal; Binding Sites; Brain; Brain Chemistry; Cinnamates; Cocaine; Conditioning, Psychological; Cyclopropanes; Immunohistochemistry; Male; Mice; Mice, Inbred C57BL; Morpholines; Neurons; Nootropic Agents; Phenazocine; Radioligand Assay; Receptors, sigma; Sigma-1 Receptor; Steroids

2002
IL-10 mediates sigma 1 receptor-dependent suppression of antitumor immunity.
    Journal of immunology (Baltimore, Md. : 1950), 2003, Apr-01, Volume: 170, Issue:7

    Topics: Adenocarcinoma, Bronchiolo-Alveolar; Adjuvants, Immunologic; Adoptive Transfer; Animals; Antibodies, Monoclonal; Cell Division; Cocaine; Cytokines; Down-Regulation; Growth Inhibitors; Immunocompetence; Injections, Intraperitoneal; Injections, Subcutaneous; Interferon-gamma; Interleukin-10; Lung Neoplasms; Male; Mice; Mice, Inbred BALB C; Morpholines; Neoplasm Transplantation; Receptors, sigma; Sigma-1 Receptor; Spleen; Tumor Cells, Cultured; Up-Regulation

2003
Cocaine modulates cytokine and enhances tumor growth through sigma receptors.
    Journal of neuroimmunology, 2004, Volume: 147, Issue:1-2

    Topics: Adenocarcinoma, Bronchiolo-Alveolar; Anesthetics, Local; Animals; Antibodies; Cell Line, Tumor; Cell Size; Cocaine; Cytokines; Drug Interactions; Ethylenediamines; Interferon-gamma; Interleukin-10; Mice; Mice, Inbred BALB C; Morpholines; Neoplasms; Receptors, sigma; Th2 Cells; Transplants

2004
Reinforcing effects of sigma-receptor agonists in rats trained to self-administer cocaine.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:2

    Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Guanidines; Male; Morpholines; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule; Reward; Self Administration

2010
Sigma receptor agonists: receptor binding and effects on mesolimbic dopamine neurotransmission assessed by microdialysis.
    Biological psychiatry, 2011, Feb-01, Volume: 69, Issue:3

    Topics: Animals; Benzoxazoles; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Ethylenediamines; Guanidines; Male; Microdialysis; Morpholines; Nucleus Accumbens; Piperazines; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptic Transmission

2011
Lack of cocaine-like discriminative-stimulus effects of σ-receptor agonists in rats.
    Behavioural pharmacology, 2011, Volume: 22, Issue:5-6

    Topics: Animals; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Guanidines; Male; Morpholines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule; Self Administration; Time Factors

2011
Blockade of Cocaine or σ Receptor Agonist Self Administration by Subtype-Selective σ Receptor Antagonists.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 358, Issue:1

    Topics: Animals; Behavior, Animal; Brain; Cocaine; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; In Vitro Techniques; Ligands; Male; Morpholines; Pentazocine; Protein Binding; Radioligand Assay; Rats, Sprague-Dawley; Receptors, sigma; Self Administration

2016
The sigma-1 receptor modulates dopamine transporter conformation and cocaine binding and may thereby potentiate cocaine self-administration in rats.
    The Journal of biological chemistry, 2017, 07-07, Volume: 292, Issue:27

    Topics: Animals; Behavior, Animal; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Guanidines; Male; Morpholines; Protein Conformation; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptosomes

2017
Sigma-1 Receptor Antagonist (BD1047) Decreases Cathepsin B Secretion in HIV-Infected Macrophages Exposed to Cocaine.
    Journal of neuroimmune pharmacology : the official journal of the Society on NeuroImmune Pharmacology, 2019, Volume: 14, Issue:2

    Topics: Animals; Apoptosis; Brain; Caspase 3; Cathepsin B; Cell Line; Cocaine; Ethylenediamines; Female; HIV Core Protein p24; HIV Infections; Humans; Immunohistochemistry; Macrophages; Mice; Mice, Inbred ICR; Morpholines; Receptors, sigma; Sigma-1 Receptor; Young Adult

2019