pre 084 has been researched along with 1,3-ditolylguanidine in 7 studies
Studies (pre 084) | Trials (pre 084) | Recent Studies (post-2010) (pre 084) | Studies (1,3-ditolylguanidine) | Trials (1,3-ditolylguanidine) | Recent Studies (post-2010) (1,3-ditolylguanidine) |
---|---|---|---|---|---|
116 | 0 | 73 | 357 | 0 | 71 |
Protein | Taxonomy | pre 084 (IC50) | 1,3-ditolylguanidine (IC50) |
---|---|---|---|
polyadenylate-binding protein 1 | Homo sapiens (human) | 19.8 | |
Rev | Human immunodeficiency virus 1 | 8.312 | |
Female germline-specific tumor suppressor gld-1 | Caenorhabditis elegans | 5.205 | |
Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | 0.036 | |
Sigma non-opioid intracellular receptor 1 | Rattus norvegicus (Norway rat) | 0.1816 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (14.29) | 18.2507 |
2000's | 1 (14.29) | 29.6817 |
2010's | 5 (71.43) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Calderon, SN; Gutkind, JS; Heller, B; Izenwasser, S; Mattson, MV; Newman, AH; Su, TP | 1 |
Cuevas, J; Guerrero, WR; Herrera, Y; Katnik, C; Pennypacker, KR | 1 |
Hiranita, T; Katz, JL; Soto, PL; Tanda, G | 2 |
Garcés-Ramírez, L; Green, JL; Hiranita, T; Katz, JL; Kopajtic, TA; McCurdy, CR; Mereu, M; Mesangeau, C; Narayanan, S; Tanda, G; Thomas, AM | 1 |
Abdelazeem, AH; Hiranita, T; Katz, JL; Kopajtic, TA; McCurdy, CR; Mesangeau, C; Narayanan, S; Rice, KC | 1 |
Amara, SG; Chin, FT; Hiranita, T; Hong, WC; Katz, JL; McCurdy, CR; Su, TP; Yano, H | 1 |
7 other study(ies) available for pre 084 and 1,3-ditolylguanidine
Article | Year |
---|---|
Novel 1-phenylcycloalkanecarboxylic acid derivatives are potent and selective sigma 1 ligands.
Topics: Animals; Anticonvulsants; Antitussive Agents; Binding Sites; Cyclopentanes; In Vitro Techniques; Male; Myocardial Ischemia; Rats; Rats, Sprague-Dawley; Receptors, sigma; Structure-Activity Relationship | 1994 |
Sigma-1 receptor activation prevents intracellular calcium dysregulation in cortical neurons during in vitro ischemia.
Topics: Analgesics, Opioid; Animals; Brain Ischemia; Calcium; Calcium Signaling; Cerebral Cortex; Cyclopentanes; Cytophotometry; Enzyme Inhibitors; Ethylenediamines; Female; Guanidines; Morpholines; Neurons; Pentazocine; Phencyclidine; Pregnancy; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, sigma; Sigma-1 Receptor; Sodium Azide; Sodium Channel Agonists; Tetrodotoxin | 2006 |
Reinforcing effects of sigma-receptor agonists in rats trained to self-administer cocaine.
Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Guanidines; Male; Morpholines; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule; Reward; Self Administration | 2010 |
Sigma receptor agonists: receptor binding and effects on mesolimbic dopamine neurotransmission assessed by microdialysis.
Topics: Animals; Benzoxazoles; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Ethylenediamines; Guanidines; Male; Microdialysis; Morpholines; Nucleus Accumbens; Piperazines; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptic Transmission | 2011 |
Lack of cocaine-like discriminative-stimulus effects of σ-receptor agonists in rats.
Topics: Animals; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Guanidines; Male; Morpholines; Rats; Rats, Sprague-Dawley; Receptors, sigma; Reinforcement Schedule; Self Administration; Time Factors | 2011 |
Blockade of Cocaine or σ Receptor Agonist Self Administration by Subtype-Selective σ Receptor Antagonists.
Topics: Animals; Behavior, Animal; Brain; Cocaine; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; In Vitro Techniques; Ligands; Male; Morpholines; Pentazocine; Protein Binding; Radioligand Assay; Rats, Sprague-Dawley; Receptors, sigma; Self Administration | 2016 |
The sigma-1 receptor modulates dopamine transporter conformation and cocaine binding and may thereby potentiate cocaine self-administration in rats.
Topics: Animals; Behavior, Animal; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Guanidines; Male; Morpholines; Protein Conformation; Rats; Rats, Sprague-Dawley; Receptors, sigma; Synaptosomes | 2017 |