Page last updated: 2024-09-03

pramipexole and physostigmine

pramipexole has been researched along with physostigmine in 3 studies

Compound Research Comparison

Studies
(pramipexole)
Trials
(pramipexole)
Recent Studies (post-2010)
(pramipexole)
Studies
(physostigmine)
Trials
(physostigmine)
Recent Studies (post-2010) (physostigmine)
1,1032195176,230252331

Protein Interaction Comparison

ProteinTaxonomypramipexole (IC50)physostigmine (IC50)
AcetylcholinesteraseElectrophorus electricus (electric eel)0.1666
AcetylcholinesteraseTetronarce californica (Pacific electric ray)0.3023
CholinesteraseHomo sapiens (human)0.3055
Cytochrome P450 2D6Homo sapiens (human)0.2
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.857
AcetylcholinesteraseMus musculus (house mouse)0.0269
AcetylcholinesteraseHomo sapiens (human)0.0853
Acetylcholinesterase Bos taurus (cattle)0.7197
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.857
Delta-type opioid receptorMus musculus (house mouse)1.1821
AcetylcholinesteraseGallus gallus (chicken)0.02
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0416
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.857
CholinesteraseEquus caballus (horse)0.4081
CholinesteraseMus musculus (house mouse)0.28
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.0189
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)0.018
Carboxylic ester hydrolase Equus caballus (horse)1.263

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andricopulo, AD; Moda, TL; Montanari, CA1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Calinski, DM; Collins, GT; Grundt, P; Newman, AH; Woods, JH1

Reviews

1 review(s) available for pramipexole and physostigmine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

2 other study(ies) available for pramipexole and physostigmine

ArticleYear
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Food restriction alters N'-propyl-4,5,6,7-tetrahydrobenzothiazole-2,6-diamine dihydrochloride (pramipexole)-induced yawning, hypothermia, and locomotor activity in rats: evidence for sensitization of dopamine D2 receptor-mediated effects.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 325, Issue:2

    Topics: Animals; Benzamides; Benzothiazoles; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Food; Hypothermia; Indoles; Male; Motor Activity; Penile Erection; Physostigmine; Piperazines; Piperidines; Pramipexole; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Yawning

2008