Page last updated: 2024-09-03

pramipexole and dan 2163

pramipexole has been researched along with dan 2163 in 7 studies

Compound Research Comparison

Studies
(pramipexole)
Trials
(pramipexole)
Recent Studies (post-2010)
(pramipexole)
Studies
(dan 2163)
Trials
(dan 2163)
Recent Studies (post-2010) (dan 2163)
1,103219517841189342

Protein Interaction Comparison

ProteinTaxonomypramipexole (IC50)dan 2163 (IC50)
D(2) dopamine receptorHomo sapiens (human)0.003

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (14.29)29.6817
2010's6 (85.71)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bradshaw, CM; Hou, RH; Langley, RW; Samuels, ER; Szabadi, E1
Marti, M; Morari, M; Viaro, R1
Abbott, S; Barnes, A; Bullmore, ET; Craig, KJ; Ersche, KD; Merlo-Pich, EV; Müller, U; Ooi, C; Robbins, TW; Sahakian, BJ; Shabbir, SS; Suckling, J1
Abbott, S; Bullmore, ET; Clark, L; Craig, KJ; Ersche, KD; Fineberg, NA; Merlo-Pich, EV; Müller, U; Ooi, C; Robbins, TW; Roiser, JP; Sahakian, BJ; Shabbir, SS; Suckling, J1
Ananthan, S; Głowacka, U; Kosmowska, B; Ossowska, K; Wardas, J1

Trials

2 trial(s) available for pramipexole and dan 2163

ArticleYear
Comparison of pramipexole and amisulpride on alertness, autonomic and endocrine functions in healthy volunteers.
    Psychopharmacology, 2006, Volume: 187, Issue:4

    Topics: Adult; Amisulpride; Antiparkinson Agents; Arousal; Autonomic Nervous System; Benzothiazoles; Blood Pressure; Body Temperature; Cross-Over Studies; Dopamine Agonists; Dopamine Antagonists; Double-Blind Method; Endocrine System; Heart Rate; Human Growth Hormone; Humans; Male; Pramipexole; Prolactin; Psychiatric Status Rating Scales; Pupil; Reference Values; Reflex, Pupillary; Salivation; Sulpiride; Thyrotropin

2006
Response perseveration in stimulant dependence is associated with striatal dysfunction and can be ameliorated by a D(2/3) receptor agonist.
    Biological psychiatry, 2011, Oct-15, Volume: 70, Issue:8

    Topics: Adult; Amisulpride; Amphetamine-Related Disorders; Benzothiazoles; Brain Mapping; Cocaine-Related Disorders; Compulsive Behavior; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Female; Humans; Magnetic Resonance Imaging; Male; Obsessive-Compulsive Disorder; Pramipexole; Reversal Learning; Sulpiride

2011

Other Studies

5 other study(ies) available for pramipexole and dan 2163

ArticleYear
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Dual motor response to l-dopa and nociceptin/orphanin FQ receptor antagonists in 1-methyl-4-phenyl-1,2,5,6-tetrahydropyridine (MPTP) treated mice: Paradoxical inhibition is relieved by D(2)/D(3) receptor blockade.
    Experimental neurology, 2010, Volume: 223, Issue:2

    Topics: Amisulpride; Animals; Antiparkinson Agents; Benzimidazoles; Benzothiazoles; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Drug Synergism; Levodopa; Male; Mice; Mice, Inbred C57BL; Motor Activity; Neural Inhibition; Nociceptin; Opioid Peptides; Parkinsonian Disorders; Piperidines; Pramipexole; Pyridines; Reaction Time; Receptors, Dopamine D3; Sulpiride

2010
Influence of compulsivity of drug abuse on dopaminergic modulation of attentional bias in stimulant dependence.
    Archives of general psychiatry, 2010, Volume: 67, Issue:6

    Topics: Adult; Amisulpride; Amphetamine-Related Disorders; Attention; Benzothiazoles; Bias; Cerebellar Cortex; Cocaine-Related Disorders; Compulsive Behavior; Dopamine; Dopamine Agonists; Dopamine Antagonists; England; Female; Functional Laterality; Humans; Individuality; Magnetic Resonance Imaging; Male; Pramipexole; Prefrontal Cortex; Receptors, Dopamine; Stroop Test; Substance-Related Disorders; Sulpiride; Surveys and Questionnaires

2010
Pramipexole at a Low Dose Induces Beneficial Effect in the Harmaline-induced Model of Essential Tremor in Rats.
    CNS neuroscience & therapeutics, 2016, Volume: 22, Issue:1

    Topics: Amisulpride; Animals; Anti-Dyskinesia Agents; Benzothiazoles; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Essential Tremor; Haloperidol; Harmaline; Imidazoles; Male; Movement; Nitriles; Pramipexole; Pyridines; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulpiride; Tetrahydroisoquinolines; Tetrahydronaphthalenes; Treatment Outcome

2016