pn 202-791 has been researched along with nitrendipine in 7 studies
Studies (pn 202-791) | Trials (pn 202-791) | Recent Studies (post-2010) (pn 202-791) | Studies (nitrendipine) | Trials (nitrendipine) | Recent Studies (post-2010) (nitrendipine) |
---|---|---|---|---|---|
44 | 0 | 1 | 2,170 | 378 | 83 |
Protein | Taxonomy | pn 202-791 (IC50) | nitrendipine (IC50) |
---|---|---|---|
G-protein coupled receptor 55 | Homo sapiens (human) | 1.4652 | |
Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens (human) | 0.0152 | |
Cytochrome P450 2C9 | Homo sapiens (human) | 0.3 | |
Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus (Norway rat) | 0.0013 | |
Voltage-dependent L-type calcium channel subunit alpha-1D | Rattus norvegicus (Norway rat) | 0.0013 | |
Cytochrome P450 2C19 | Homo sapiens (human) | 3 | |
Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens (human) | 0.0152 | |
Voltage-dependent L-type calcium channel subunit alpha-1S | Rattus norvegicus (Norway rat) | 0.0013 | |
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 10 | |
Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens (human) | 0.0152 | |
Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens (human) | 0.0152 | |
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C | Homo sapiens (human) | 1.85 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (57.14) | 18.7374 |
1990's | 3 (42.86) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Luchowski, EM; Rutledge, A; Su, CM; Triggle, DJ; Wei, XY | 1 |
Brown, AM; Brush, K; Hamilton, SL; Schwartz, A; Yatani, A | 1 |
Boarder, MR; Owen, PJ; Plevin, R | 1 |
Panzer-Knodle, S; Papaioannou, S; Yang, PC | 1 |
Bolger, GT; O'Neill, SK; Triggle, CR | 1 |
Christensen, JD; Fjalland, B; Jørgensen, A; Treiman, M | 1 |
Brauns, T; Glossmann, H; Haugland, RP; Kimball, SD; Prinz, H; Striessnig, J | 1 |
7 other study(ies) available for pn 202-791 and nitrendipine
Article | Year |
---|---|
Pharmacologic and radioligand binding analysis of the actions of 1,4-dihydropyridine activator-antagonist pairs in smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Calcium; Drug Synergism; Guinea Pigs; Ion Channels; Muscle Contraction; Muscle, Smooth, Vascular; Nicotinic Acids; Nitrendipine; Oxadiazoles; Potassium Chloride; Rats; Stereoisomerism | 1986 |
A comparison between the binding and electrophysiological effects of dihydropyridines on cardiac membranes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Heart; Ion Channels; Isradipine; Kinetics; Membrane Potentials; Membranes; Myocardium; Nicotinic Acids; Nimodipine; Nitrendipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship | 1987 |
Characterization of bradykinin-stimulated release of noradrenaline from cultured bovine adrenal chromaffin cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bradykinin; Calcium; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol Phosphates; Nicotinic Acids; Nitrendipine; Norepinephrine; Oxadiazoles; Potassium | 1989 |
Calcium channel blockers: correlation among receptor binding, calcium uptake and contractility in vitro.
Topics: Animals; Calcium; Calcium Channel Blockers; Muscle Contraction; Nicotinic Acids; Nitrendipine; Oxadiazoles; Potassium; Rabbits; Temperature | 1987 |
Competitive binding experiments reveal differential interactions for dihydropyridine calcium channel activators and antagonists at dihydropyridine receptors on mouse brain membranes.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Brain; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; In Vitro Techniques; Male; Membranes; Mice; Muscle Proteins; Nicotinic Acids; Nitrendipine; Oxadiazoles; Stereoisomerism; Thermodynamics | 1994 |
Dihydropyridine ligands influence the evoked release of oxytocin and vasopressin dependent on stimulation conditions.
Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Dihydropyridines; Electric Stimulation; Electrophysiology; Female; Ligands; Nicotinic Acids; Nitrendipine; Oxadiazoles; Oxytocin; Pituitary Gland, Posterior; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Stereoisomerism; Structure-Activity Relationship; Vasopressins | 1994 |
L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other.
Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Fluorescent Dyes; Isomerism; Isradipine; Kinetics; Nicotinic Acids; Nifedipine; Nitrendipine; Oxadiazoles; Rabbits | 1997 |