Page last updated: 2024-09-03

pn 202-791 and isradipine

pn 202-791 has been researched along with isradipine in 4 studies

Compound Research Comparison

Studies
(pn 202-791)
Trials
(pn 202-791)
Recent Studies (post-2010)
(pn 202-791)
Studies
(isradipine)
Trials
(isradipine)
Recent Studies (post-2010) (isradipine)
44011,40334686

Protein Interaction Comparison

ProteinTaxonomypn 202-791 (IC50)isradipine (IC50)
Voltage-dependent L-type calcium channel subunit alpha-1COryctolagus cuniculus (rabbit)0.107
Voltage-dependent L-type calcium channel subunit alpha-1DRattus norvegicus (Norway rat)0.221
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.0022

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19902 (50.00)18.7374
1990's2 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brown, AM; Brush, K; Hamilton, SL; Schwartz, A; Yatani, A1
Kokubun, S; Porzig, H; Prod'hom, B; Reuter, H1
Fitzpatrick, LA; Maercklein, PB; Ritchie, CK1
Brauns, T; Glossmann, H; Haugland, RP; Kimball, SD; Prinz, H; Striessnig, J1

Reviews

1 review(s) available for pn 202-791 and isradipine

ArticleYear
Calcium channels in the heart. Properties and modulation by dihydropyridine enantiomers.
    Annals of the New York Academy of Sciences, 1988, Volume: 522

    Topics: Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Heart; Humans; Ion Channels; Isradipine; Nicotinic Acids; Oxadiazoles; Stereoisomerism

1988

Other Studies

3 other study(ies) available for pn 202-791 and isradipine

ArticleYear
A comparison between the binding and electrophysiological effects of dihydropyridines on cardiac membranes.
    Molecular pharmacology, 1987, Volume: 31, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Heart; Ion Channels; Isradipine; Kinetics; Membrane Potentials; Membranes; Myocardium; Nicotinic Acids; Nimodipine; Nitrendipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship

1987
Direct effect of calcium channel antagonists on osteoclast function: alterations in bone resorption and intracellular calcium concentrations.
    Endocrinology, 1994, Volume: 135, Issue:3

    Topics: Animals; Bone Resorption; Calcium; Calcium Channel Blockers; Cells, Cultured; Intracellular Membranes; Isomerism; Isradipine; Nicotinic Acids; Nifedipine; Osmolar Concentration; Osteoclasts; Oxadiazoles; Rats; Whales

1994
L-type calcium channels: binding domains for dihydropyridines and benzothiazepines are located in close proximity to each other.
    Biochemistry, 1997, Mar-25, Volume: 36, Issue:12

    Topics: Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Diltiazem; Fluorescent Dyes; Isomerism; Isradipine; Kinetics; Nicotinic Acids; Nifedipine; Nitrendipine; Oxadiazoles; Rabbits

1997