pleconaril has been researched along with pirodavir in 12 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 4 (33.33) | 29.6817 |
2010's | 8 (66.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Batugo, MR; Brown, EL; Chen, L; Dragovich, PS; Ferre, RA; Fuhrman, SA; Gleeson, JP; Guzman, MC; Hendrickson, TF; Kosa, MB; Lee, CA; Liu, B; Maldonado, FC; Matthews, DA; Meador, JW; Patick, AK; Prins, TJ; Sakata, SK; Tuntland, T; Worland, ST; Zalman, LS; Zhou, R | 1 |
Barnard, DL; Brown, RN; Cameron, R; Chalmers, DK; Hamilton, S; Jin, B; Krippner, GY; Luttick, A; McConnell, DB; Reece, PA; Ryan, J; Sidwell, RW; Stanislawski, PC; Tucker, SP; Watson, KG; Wu, WY | 1 |
Batugo, MR; Borer, BC; Brown, EL; Chen, L; Dovalsantos, EZ; Dragovich, PS; Ferre, RA; Fuhrman, SA; Gleeson, JP; Guo, M; Guzman, MC; Hua, Y; Johnson, TO; Kosa, MB; Lee, CA; Lee, S; Liese, A; Liu, B; Liu, J; Luu, HT; Maldonado, FC; Matthews, DA; McGee, K; Meador, JW; Mohajeri, M; Moran, T; Nayyar, NK; Patick, AK; Prins, TJ; Rejto, PA; Rose, PW; Sakata, SK; Tao, J; Tuntland, T; Wu, EY; Wu, ZP; Zalman, LS; Zhou, R | 1 |
Brown, RN; Cameron, R; Chalmers, DK; Hamilton, S; Krippner, GY; Luttick, A; McConnell, DB; Nearn, R; Stanislawski, PC; Tucker, SP; Watson, KG | 1 |
Gao, D; Gong, Z; Li, S; Sun, T; Wang, H; Xiao, J; Yan, H; Zhang, X | 1 |
Cook, A; Jenkinson, L; King, S; MacDonald, C; McCrae, C; Morley, A; Phillips, T; Tomkinson, N; Unitt, J; Weaver, R | 1 |
Feil, SC; Hamilton, S; Krippner, GY; Lin, B; Luttick, A; McConnell, DB; Morton, CJ; Nearn, R; Parker, MW; Ryan, J; Stanislawski, PC; Tucker, SP; Watson, KG | 1 |
Bianco, G; Caboni, P; Cottiglia, F; Distinto, S; Floris, C; Fois, B; Maccioni, E; Marras, L; Meleddu, R; Melis, C; Pompei, R; Sonar, VP | 1 |
Aguayo, E; Birkus, G; Cihlar, T; Jordan, R; Lee, G; Mello, C; Rodriguez, M | 1 |
Bernard, A; Cabiddu, MG; Lacroix, C; Leyssen, P; Neyts, J; Pompei, R | 1 |
Angius, F; Coluccia, A; Laconi, S; Lacroix, C; Leyssen, P; Neyts, J; Pompei, R; Silvestri, R | 1 |
Day, CW; Evans, WJ; Nicolaou, KC; Smee, DF; Tarbet, EB | 1 |
12 other study(ies) available for pleconaril and pirodavir
Article | Year |
---|---|
Structure-based design, synthesis, and biological evaluation of irreversible human rhinovirus 3C protease inhibitors. 6. Structure-activity studies of orally bioavailable, 2-pyridone-containing peptidomimetics.
Topics: 3C Viral Proteases; Administration, Oral; Animals; Antiviral Agents; Biological Availability; Crystallography, X-Ray; Cysteine Endopeptidases; Dogs; Drug Stability; Humans; In Vitro Techniques; Ligands; Microsomes, Liver; Models, Molecular; Molecular Mimicry; Peptides; Protease Inhibitors; Protein Binding; Pyridones; Rhinovirus; Structure-Activity Relationship; Viral Proteins | 2002 |
An orally bioavailable oxime ether capsid binder with potent activity against human rhinovirus.
Topics: Administration, Oral; Animals; Antiviral Agents; Biological Availability; Capsid; Cell Line; Ethers; Female; Humans; Male; Mice; Oximes; Piperidines; Protein Binding; Pyridazines; Rats; Rhinovirus; Structure-Activity Relationship | 2003 |
Structure-based design, synthesis, and biological evaluation of irreversible human rhinovirus 3C protease inhibitors. 8. Pharmacological optimization of orally bioavailable 2-pyridone-containing peptidomimetics.
Topics: 3C Viral Proteases; Animals; Antiviral Agents; Biological Availability; Blood Proteins; Caco-2 Cells; Cysteine Endopeptidases; Dogs; Drug Design; Half-Life; Hepatocytes; Humans; In Vitro Techniques; Indicators and Reagents; Macaca fascicularis; Magnetic Resonance Spectroscopy; Male; Microsomes, Liver; Protease Inhibitors; Protein Binding; Pyridones; Rhinovirus; Solubility; Structure-Activity Relationship; Viral Proteins | 2003 |
2-Ethoxybenzoxazole as a bioisosteric replacement of an ethyl benzoate group in a human rhinovirus (HRV) capsid binder.
Topics: Benzoates; Benzoxazoles; Capsid Proteins; Humans; Protein Binding; Rhinovirus; Stereoisomerism | 2005 |
Pharmacophore-based design, synthesis, and biological evaluation of novel chloro-pyridazine piperazines as human rhinovirus (HRV-3) inhibitors.
Topics: Antiviral Agents; Binding Sites; Computer Simulation; Drug Design; Humans; Models, Chemical; Models, Molecular; Piperazines; Pyridazines; Rhinovirus; Viral Proteins | 2011 |
Effect of lipophilicity modulation on inhibition of human rhinovirus capsid binders.
Topics: Animals; Antiviral Agents; Capsid; Capsid Proteins; Humans; Microsomes; Picornaviridae Infections; Protein Binding; Pyridazines; Rats; Rats, Sprague-Dawley; Rhinovirus; Structure-Activity Relationship | 2011 |
An Orally Available 3-Ethoxybenzisoxazole Capsid Binder with Clinical Activity against Human Rhinovirus.
Topics: | 2012 |
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders.
Topics: Antiviral Agents; Bupleurum; Capsid; Enterovirus; HeLa Cells; Humans; Models, Molecular; Molecular Structure; Monoterpenes; Phenylpropionates; Plant Leaves; Rhinovirus; Structure-Activity Relationship; Virus Replication | 2017 |
Multiple classes of antiviral agents exhibit in vitro activity against human rhinovirus type C.
Topics: Antiviral Agents; Common Cold; Dose-Response Relationship, Drug; HeLa Cells; Humans; In Vitro Techniques; Isoxazoles; Oxadiazoles; Oxazoles; Phenylalanine; Piperidines; Pyridazines; Pyrrolidinones; Replicon; Rhinovirus; RNA, Viral; Tubercidin; Valine; Virus Replication | 2014 |
Exploration of the anti-enterovirus activity of a series of pleconaril/pirodavir-like compounds.
Topics: Antiviral Agents; Dose-Response Relationship, Drug; Enterovirus; Microbial Sensitivity Tests; Oxadiazoles; Oxazoles; Piperidines; Pyridazines; Structure-Activity Relationship | 2015 |
In vitro characterisation of a pleconaril/pirodavir-like compound with potent activity against rhinoviruses.
Topics: Antiviral Agents; Capsid Proteins; Humans; Microbial Sensitivity Tests; Oxadiazoles; Oxazoles; Piperidines; Protein Binding; Pyridazines; Rhinovirus | 2015 |
Susceptibilities of enterovirus D68, enterovirus 71, and rhinovirus 87 strains to various antiviral compounds.
Topics: A549 Cells; Antimetabolites; Antiviral Agents; Benzimidazoles; Enterovirus A, Human; Enterovirus D, Human; Guanine; HeLa Cells; Humans; Oxadiazoles; Oxazoles; Oximes; Picornaviridae; Piperazines; Piperidines; Pyridazines; Rhabdomyosarcoma; Rhinovirus; Ribavirin; Sulfonamides | 2016 |