Page last updated: 2024-09-04

pk 9084 and flunitrazepam

pk 9084 has been researched along with flunitrazepam in 3 studies

Compound Research Comparison

Studies
(pk 9084)
Trials
(pk 9084)
Recent Studies (post-2010)
(pk 9084)
Studies
(flunitrazepam)
Trials
(flunitrazepam)
Recent Studies (post-2010) (flunitrazepam)
17002,697298130

Protein Interaction Comparison

ProteinTaxonomypk 9084 (IC50)flunitrazepam (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0016
GABA theta subunitRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0016

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19903 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gee, KW; Yamamura, HI1
Keane, PE; Morre, M; Simiand, J1
Brinton, RE; Gee, KW; Yamamura, HI1

Other Studies

3 other study(ies) available for pk 9084 and flunitrazepam

ArticleYear
Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes?
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Cerebral Cortex; Drug Interactions; Flunitrazepam; Male; Postural Balance; Pyrazoles; Pyridazines; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Temperature

1983
The quinolines PK 8165 and PK 9084 possess benzodiazepine-like activity in vitro but not in vivo.
    Neuroscience letters, 1984, Mar-09, Volume: 45, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Mice; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A

1984
PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam.
    Brain research, 1983, Mar-28, Volume: 264, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Diazepam; Drug Antagonism; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Quinolines; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983