Page last updated: 2024-09-04

pk 9084 and cl 218872

pk 9084 has been researched along with cl 218872 in 4 studies

Compound Research Comparison

Studies
(pk 9084)
Trials
(pk 9084)
Recent Studies (post-2010)
(pk 9084)
Studies
(cl 218872)
Trials
(cl 218872)
Recent Studies (post-2010) (cl 218872)
170015803

Protein Interaction Comparison

ProteinTaxonomypk 9084 (IC50)cl 218872 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.116
GABA theta subunitRattus norvegicus (Norway rat)0.116
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.116

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19903 (75.00)18.7374
1990's1 (25.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Borsini, F; Gragnani, L; Lecci, A; Meli, A; Volterra, G1
File, SE; Wilks, L1
Ator, NA; Griffiths, RR1
Gee, KW; Yamamura, HI1

Other Studies

4 other study(ies) available for pk 9084 and cl 218872

ArticleYear
Effect of psychotomimetics and some putative anxiolytics on stress-induced hyperthermia.
    Journal of neural transmission. General section, 1991, Volume: 83, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Body Temperature; Dextroamphetamine; Dizocilpine Maleate; Fever; Flumazenil; Male; Mice; Phencyclidine; Pyrazoles; Pyridazines; Quinolines; Receptors, GABA-A; Receptors, Serotonin; Single-Blind Method; Stress, Physiological

1991
Effects of acute and chronic treatment on the pro- and anti-convulsant actions of CL 218, 872, PK 8165 and PK 9084, putative ligands for the benzodiazepine receptor.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Male; Mice; Pentylenetetrazole; Picrotoxin; Pyridazines; Quinolines; Receptors, GABA-A; Time Factors

1985
Discriminative stimulus effects of atypical anxiolytics in baboons and rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepinones; Buspirone; Discrimination Learning; Flumazenil; Isoxazoles; Lorazepam; Male; Papio; Piperazines; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes?
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Cerebral Cortex; Drug Interactions; Flunitrazepam; Male; Postural Balance; Pyrazoles; Pyridazines; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Temperature

1983