Page last updated: 2024-09-04

pk 9084 and chlordiazepoxide

pk 9084 has been researched along with chlordiazepoxide in 4 studies

Compound Research Comparison

Studies
(pk 9084)
Trials
(pk 9084)
Recent Studies (post-2010)
(pk 9084)
Studies
(chlordiazepoxide)
Trials
(chlordiazepoxide)
Recent Studies (post-2010) (chlordiazepoxide)
17003,962385104

Protein Interaction Comparison

ProteinTaxonomypk 9084 (IC50)chlordiazepoxide (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.216
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)1.1
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.9967
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.216
Histamine H1 receptorHomo sapiens (human)1.795
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.216
GABA theta subunitRattus norvegicus (Norway rat)0.216
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.216

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19904 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Le Fur, G1
File, SE; Lister, RG1
Burgevin, MC; Ferris, O; Gauthier, A; Guérémy, C; Heaulme, M; Le Fur, G; Mizoule, J; Uzan, A1
File, SE1

Other Studies

4 other study(ies) available for pk 9084 and chlordiazepoxide

ArticleYear
[Anxiety receptors: new pharmacological approach (author's transl)].
    L'Encephale, 1982, Volume: 8, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Binding, Competitive; Brain; Chlordiazepoxide; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Quinolines; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Seizures

1982
Quinolines and anxiety: anxiogenic effects of CGS 8216 and partial anxiolytic profile of PK 9084.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Humans; Male; Motor Activity; Pyrazoles; Quinolines; Rats; Social Behavior

1983
Multiple benzodiazepine receptors: evidence of dissociation between anticonflict and anticonvulsant properties by PK 8165 and PK 9084 (two quinoline derivatives).
    Life sciences, 1981, Mar-30, Volume: 28, Issue:13

    Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Cerebellar Cortex; Chlordiazepoxide; Conflict, Psychological; Cyclic AMP; Cyclic GMP; Diazepam; Hypnotics and Sedatives; Kinetics; Male; Motor Activity; Piperazines; Quinolines; Rats; Receptors, Drug; Receptors, GABA-A

1981
Sedative effects of PK 9084 and PK 8165, alone and in combination with chlordiazepoxide.
    British journal of pharmacology, 1983, Volume: 79, Issue:1

    Topics: Animals; Behavior, Animal; Body Temperature; Chlordiazepoxide; Drug Interactions; Exploratory Behavior; Hypnotics and Sedatives; Male; Motor Activity; Quinolines; Rats

1983