Page last updated: 2024-09-03

pk 14105 and kainic acid

pk 14105 has been researched along with kainic acid in 3 studies

Compound Research Comparison

Studies
(pk 14105)
Trials
(pk 14105)
Recent Studies (post-2010)
(pk 14105)
Studies
(kainic acid)
Trials
(kainic acid)
Recent Studies (post-2010) (kainic acid)
28009,54031,775

Protein Interaction Comparison

ProteinTaxonomypk 14105 (IC50)kainic acid (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 2Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 3Rattus norvegicus (Norway rat)4.2857
Glutamate receptor 4Rattus norvegicus (Norway rat)4.2857
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 1Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.0126
Glutamate receptor ionotropic, kainate 2Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 3Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 4Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 5Homo sapiens (human)0.077
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.0126

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benavides, J; Bourdiol, F; Dubois, A; Scatton, B1
Ahier, RG; Cremer, JE; Hume, SP; Luthra, SK; Manjil, L; Myers, R; Pascali, C; Pike, VW; Price, GW1
Benavides, J; Capdeville, C; Dauphin, F; Dubois, A; Duverger, D; Fage, D; Gotti, B; MacKenzie, ET; Scatton, B1

Other Studies

3 other study(ies) available for pk 14105 and kainic acid

ArticleYear
Regional pattern of increased omega 3 (peripheral type benzodiazepine) binding site densities in the rat brain induced by systemic injection of kainic acid.
    Neuroscience letters, 1991, Apr-29, Volume: 125, Issue:2

    Topics: Affinity Labels; Animals; Autoradiography; Brain; Isoquinolines; Kainic Acid; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tritium

1991
The radiosynthesis of [18F]PK 14105 as an alternative radioligand for peripheral type benzodiazepine binding sites.
    International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes, 1990, Volume: 41, Issue:5

    Topics: Animals; Binding Sites; Corpus Striatum; Fluorine Radioisotopes; Isoquinolines; Isotope Labeling; Kainic Acid; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
The quantification of brain lesions with an omega 3 site ligand: a critical analysis of animal models of cerebral ischaemia and neurodegeneration.
    Brain research, 1990, Jul-09, Volume: 522, Issue:2

    Topics: Affinity Labels; Aging; Animals; Autoradiography; Brain; Brain Ischemia; Disease Models, Animal; Isoquinolines; Kainic Acid; Male; Mice; Nerve Degeneration; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990