Page last updated: 2024-09-04

pitrazepin and flunitrazepam

pitrazepin has been researched along with flunitrazepam in 2 studies

Compound Research Comparison

Studies
(pitrazepin)
Trials
(pitrazepin)
Recent Studies (post-2010)
(pitrazepin)
Studies
(flunitrazepam)
Trials
(flunitrazepam)
Recent Studies (post-2010) (flunitrazepam)
10002,697298130

Protein Interaction Comparison

ProteinTaxonomypitrazepin (IC50)flunitrazepam (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0016
GABA theta subunitRattus norvegicus (Norway rat)0.0016
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0016

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
David, JA; Pinnock, RD; Sattelle, DB; Wafford, KA1
Gähwiler, BH; Maurer, R; Wüthrich, HJ1

Other Studies

2 other study(ies) available for pitrazepin and flunitrazepam

ArticleYear
GABA receptors on the cell-body membrane of an identified insect motor neuron.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1988, Jan-22, Volume: 232, Issue:1269

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Chlorides; Cockroaches; Dibenzazepines; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Membrane Potentials; Microelectrodes; Motor Neurons; Nipecotic Acids; Periplaneta; Picrotoxin; Receptors, GABA-A

1988
Pitrazepin, a novel GABAA antagonist.
    Neuroscience letters, 1984, Apr-06, Volume: 45, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Binding, Competitive; Culture Techniques; Dibenzazepines; Flunitrazepam; GABA Antagonists; Hippocampus; Hypothalamus; Membrane Potentials; Muscimol; Neurons; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Muscarinic

1984