Page last updated: 2024-09-04

pitrazepin and baclofen

pitrazepin has been researched along with baclofen in 2 studies

Compound Research Comparison

Studies
(pitrazepin)
Trials
(pitrazepin)
Recent Studies (post-2010)
(pitrazepin)
Studies
(baclofen)
Trials
(baclofen)
Recent Studies (post-2010) (baclofen)
10006,0173721,535

Protein Interaction Comparison

ProteinTaxonomypitrazepin (IC50)baclofen (IC50)
Gamma-aminobutyric acid type B receptor subunit 2Homo sapiens (human)0.05
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.2762
Gamma-aminobutyric acid type B receptor subunit 1Homo sapiens (human)0.05
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.2762

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19901 (50.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kim, KH; Takeuchi, H1
Gähwiler, BH; Maurer, R; Wüthrich, HJ1

Other Studies

2 other study(ies) available for pitrazepin and baclofen

ArticleYear
Pharmacological characteristics of two different types of inhibitory GABA receptors on Achatina fulica neurones.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Crotonates; Diazepam; Dibenzazepines; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Muscimol; Neurons; Pentobarbital; Picrotoxin; Receptors, GABA-A; Snails

1990
Pitrazepin, a novel GABAA antagonist.
    Neuroscience letters, 1984, Apr-06, Volume: 45, Issue:3

    Topics: Animals; Baclofen; Bicuculline; Binding, Competitive; Culture Techniques; Dibenzazepines; Flunitrazepam; GABA Antagonists; Hippocampus; Hypothalamus; Membrane Potentials; Muscimol; Neurons; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Muscarinic

1984