Page last updated: 2024-08-16

pirenzepine and darifenacin

pirenzepine has been researched along with darifenacin in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's3 (42.86)29.6817
2010's3 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bonhaus, D; Briaud, S; Choppin, A; Eglen, RM; Hegde, SS; Loeb, M; Loury, D; Moy, TM1
Challiss, RA; Nahorski, SR; Nelson, CP1
Ouyang, A; Tandon, T; Wrzos, HF1
Chapple, CR; Chess-Williams, R; Stevens, LA1
Fujino, T; Kageyama, A; Nozawa, Y; Yamada, S; Yoshida, A1
Chess-Williams, R; Moro, C; Uchiyama, J1
Arrighi, N; Bodei, S; Cosciani Cunico, S; Michel, MC; Sigala, S; Simeone, C; Spano, P; Zani, D1

Other Studies

7 other study(ies) available for pirenzepine and darifenacin

ArticleYear
Functional role of M2 and M3 muscarinic receptors in the urinary bladder of rats in vitro and in vivo.
    British journal of pharmacology, 1997, Volume: 120, Issue:8

    Topics: Adenylyl Cyclases; Animals; CHO Cells; Cricetinae; Dioxolanes; Enzyme Activation; Female; Humans; Muscarinic Antagonists; Muscle Contraction; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Urinary Bladder

1997
Constitutive activity and inverse agonism at the M2 muscarinic acetylcholine receptor.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 316, Issue:1

    Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Immunoblotting; Inositol Phosphates; Ligands; Muscarinic Agonists; Mutagenesis, Site-Directed; Radioligand Assay; Receptor, Muscarinic M2; Transfection

2006
Mechanisms mediating cholinergic antral circular smooth muscle contraction in rats.
    World journal of gastroenterology, 2004, Nov-15, Volume: 10, Issue:22

    Topics: Anesthetics, Local; Animals; Benzofurans; Bethanechol; Calcium; Calcium Channel Blockers; Cholinergic Agonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nifedipine; Pertussis Toxin; Pirenzepine; Pyloric Antrum; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Signal Transduction; Tetrodotoxin

2004
Human idiopathic and neurogenic overactive bladders and the role of M2 muscarinic receptors in contraction.
    European urology, 2007, Volume: 52, Issue:2

    Topics: Adult; Aged; Benzofurans; Carbachol; Diamines; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Piperidines; Pirenzepine; Pyrrolidines; Receptors, Muscarinic; Urinary Bladder; Urinary Bladder, Neurogenic; Urinary Bladder, Overactive

2007
Loss of muscarinic and purinergic receptors in urinary bladder of rats with hydrochloric acid-induced cystitis.
    Urology, 2010, Volume: 76, Issue:4

    Topics: Adenosine Triphosphate; Animals; Benzhydryl Compounds; Benzofurans; Cresols; Cystitis; Disease Models, Animal; Down-Regulation; Female; Hydrochloric Acid; Mandelic Acids; N-Methylscopolamine; Organophosphonates; Phenols; Phenylpropanolamine; Pirenzepine; Polycyclic Compounds; Pyridoxal Phosphate; Pyrrolidines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Purinergic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urination; Urodynamics

2010
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
    Urology, 2011, Volume: 78, Issue:6

    Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium

2011
Different muscarinic receptor subtypes modulate proliferation of primary human detrusor smooth muscle cells via Akt/PI3K and map kinases.
    Pharmacological research, 2013, Volume: 74

    Topics: Aged; Atropine; Benzofurans; Carbachol; Cell Proliferation; Cells, Cultured; Cholinergic Agonists; Gene Expression; Humans; Male; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Myocytes, Smooth Muscle; Phosphatidylinositol 3-Kinases; Piperidines; Pirenzepine; Proto-Oncogene Proteins c-akt; Pyrrolidines; Receptors, Muscarinic; RNA, Messenger; Urinary Bladder

2013