Page last updated: 2024-08-17

piperoxan and yohimbine

piperoxan has been researched along with yohimbine in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-199033 (84.62)18.7374
1990's5 (12.82)18.2507
2000's1 (2.56)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andrews, PR; Craik, DJ; Martin, JL1
Caroon, JM; Clark, RD; Kluge, AF; Michel, AD; Olah, R; Repke, DB; Unger, SH; Whiting, RL1
Butler, RC; Chapleo, CB; Doxey, JC; Myers, PL; Roach, AG; Smith, CF1
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Timmermans, PB; van Zwieten, PA1
Philippu, A; Schartner, P1
Borowski, E; Ehrl, H; Endo, T; Starke, K1
Kapur, H; Mottram, DR1
Baraban, JM; Davis, M; Redmond, DE1
Dausse, J; Meyer, P; Miach, PJ1
Donabedian, RK; Gold, MS; Redmond, DE1
Antonaccio, MJ; Taylor, DG1
Bousquet, P; Feldman, J; Gonon, F; Mermet, C; Monassier, L; Tibiriça, E1
Fukuda, H; Mishima, A; Ono, H; Ono, S; Vasko, MR1
Berendsen, HH; Broekkamp, CL1
Errchidi, S; Hilaire, G; Monteau, R1
Hadjiconstantinou, M; Krajnc, D; Neff, NH; Rossetti, Z1
De Sarro, A; De Sarro, GB1
Paul, SM; Wolkowitz, OM1
Colpaert, FC; Janssen, PA2
Kassarich, J; Lien, EL; Morrison, A; Sullivan, D1
Haigler, HJ; O'Neill, TP1
Starke, K; Tanaka, T1
Anlezark, G; Horton, R; Meldrum, B1
Melchiorre, C1
Browne, RG1
Burnham, WM; King, GA1
Barsuhn, C; Humphrey, SJ; Lahti, RA; McCall, RB; Schuette, MR1
Iuvone, PM; Rauch, AL1
Gaillard, JM1
Harron, DW; Kobinger, W1
Nomura, Y; Oki, K; Segawa, T1
Sybertz, EJ; Zimmerman, BG1
Dedek, J; Scatton, B; Zivkovic, B1
Blakeley, AG; Cunnane, TC; Maskell, T; Mathie, A; Petersen, SA1
Dunn, RW; La Marca, S1
Audinot, V; Boutin, JA; Cogé, F; Cussac, D; Dekeyne, A; Galizzi, JP; Gobert, A; Lejeune, F; Millan, MJ; Newman-Tancredi, A; Nicolas, JP; Rivet, JM1

Reviews

3 review(s) available for piperoxan and yohimbine

ArticleYear
alpha 2 adrenoceptors: classification, localization, mechanisms, and targets for drugs.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:12

    Topics: Adipose Tissue; Animals; Blood Platelets; Central Nervous System; Humans; Islets of Langerhans; Melanocytes; Muscle, Smooth, Vascular; Nerve Endings; Norepinephrine; Parasympathetic Nervous System; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Serotonin; Synapses

1982
Neural and molecular mechanisms in anxiety.
    The Psychiatric clinics of North America, 1985, Volume: 8, Issue:1

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Binding, Competitive; Carbolines; Clonidine; Disease Models, Animal; Forecasting; Haplorhini; Humans; Locus Coeruleus; Piperoxan; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Purinergic; Research Design; Yohimbine

1985
Selectivity of alpha 1 and alpha 2 adrenergic agonists and antagonists.
    Il Farmaco; edizione scientifica, 1980, Volume: 35, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Disulfides; Humans; Imidazoles; Organ Specificity; Phenoxybenzamine; Piperoxan; Polyamines; Receptors, Adrenergic, alpha; Yohimbine

1980

Other Studies

36 other study(ies) available for piperoxan and yohimbine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Structure-activity relationships for 2-substituted imidazoles as alpha 2-adrenoceptor antagonists.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Chemical Phenomena; Chemistry; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rats; Structure-Activity Relationship; Vas Deferens

1982
alpha-adrenoreceptor reagents. 1. Synthesis of some 1,4-benzodioxans as selective presynaptic alpha 2-adrenoreceptor antagonists and potential antidepressants.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Dioxins; Dose-Response Relationship, Drug; Idazoxan; Male; Mice; Phenylephrine; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Synapses; Vas Deferens

1983
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Inhibition by locally applied alpha-adrenoreceptor blocking drugs of the depressor response to stimulation of the anterior hypothalamus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 295, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Electric Stimulation; Female; Hypothalamus; Hypothalamus, Anterior; Male; Phentolamine; Phenylephrine; Piperoxan; Tolazoline; Yohimbine

1976
A comparison of pre- and postsynaptic effects of alpha-adrenolytic drugs in the pulmonary artery of the rabbit.
    Neuroscience, 1977, Volume: 2, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Ergotamine; Norepinephrine; Phentolamine; Piperoxan; Pulmonary Artery; Rabbits; Yohimbine

1977
A comparative study on the pre- and post-synaptic alpha blocking activity of a series of benzodioxanes.
    Biochemical pharmacology, 1978, Volume: 27, Issue:14

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Muscle Contraction; Phentolamine; Piperidines; Piperoxan; Rats; Synapses; Yohimbine

1978
Noradrenergic agonists and antagonists: effects on conditioned fear as measured by the potentiated startle paradigm.
    Psychopharmacology, 1979, Volume: 65, Issue:2

    Topics: Animals; Clonidine; Conditioning, Operant; Fear; Male; Norepinephrine; Piperoxan; Propranolol; Rats; Reflex, Startle; Yohimbine

1979
Direct biochemical demonstration of two types of alpha-adrenoreceptor in rat brain.
    Nature, 1978, Aug-03, Volume: 274, Issue:5670

    Topics: Animals; Binding, Competitive; Brain; Clonidine; Dihydroergotoxine; Dopamine; Male; Phenoxybenzamine; Phentolamine; Piperoxan; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synaptic Membranes; Yohimbine

1978
Further evidence for alpha-2 adrenergic receptor mediated inhibition of prolactin secretion: the effect of yohimbine.
    Psychoneuroendocrinology, 1978, Volume: 3, Issue:3-4

    Topics: Animals; Haplorhini; Infusions, Parenteral; Macaca; Neural Inhibition; Piperoxan; Prolactin; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Yohimbine

1978
Effects of R-28935 on sympathetic nervous activity in anesthetized cat.
    Clinical and experimental hypertension, 1978, Volume: 1, Issue:1

    Topics: Animals; Antihypertensive Agents; Benzimidazoles; Cats; Heart; Hemodynamics; Phentolamine; Piperoxan; Pressoreceptors; Sympathetic Nervous System; Yohimbine

1978
Selectivity of rilmenidine for the nucleus reticularis lateralis, a ventrolateral medullary structure containing imidazoline-preferring receptors.
    European journal of pharmacology, 1991, Dec-17, Volume: 209, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Catecholamines; Clonidine; Dioxanes; Electrochemistry; Hemodynamics; Idazoxan; Imidazoline Receptors; Male; Medulla Oblongata; Neurons; Oxazoles; Piperoxan; Rats; Rats, Inbred WKY; Receptors, Drug; Reticular Formation; Rilmenidine; Stereotaxic Techniques; Yohimbine

1991
Inhibitory effects of clonidine and tizanidine on release of substance P from slices of rat spinal cord and antagonism by alpha-adrenergic receptor antagonists.
    Neuropharmacology, 1991, Volume: 30, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Parasympatholytics; Piperoxan; Prazosin; Radioimmunoassay; Rats; Rats, Inbred Strains; Spinal Cord; Substance P; Veratridine; Yohimbine

1991
A peripheral 5-HT1D-like receptor involved in serotonergic induced hindlimb scratching in rats.
    European journal of pharmacology, 1991, Mar-05, Volume: 194, Issue:2-3

    Topics: 5-Methoxytryptamine; Animals; Behavior, Animal; Drug Synergism; Hindlimb; Male; Piperoxan; Pruritus; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Yohimbine

1991
Permanent release of noradrenaline modulates respiratory frequency in the newborn rat: an in vitro study.
    The Journal of physiology, 1990, Volume: 429

    Topics: Animals; Animals, Newborn; Brain Stem; Desipramine; In Vitro Techniques; Methyltyrosines; Norepinephrine; Pargyline; Piperoxan; Pons; Rats; Respiration; Spinal Cord; Time Factors; Yohimbine

1990
Modulation of retinal aromatic L-amino acid decarboxylase via alpha 2 adrenoceptors.
    Journal of neurochemistry, 1989, Volume: 52, Issue:2

    Topics: Animals; Aromatic-L-Amino-Acid Decarboxylases; Clonidine; Cycloheximide; Darkness; Dihydroxyphenylalanine; Kinetics; Light; Male; Oxymetazoline; Phentolamine; Piperoxan; Pyridoxal Phosphate; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Retina; Yohimbine

1989
Antagonists of adenosine and alpha-2-adrenoceptors reverse the anticonvulsant effects of tizanidine in DBA/2 mice.
    Neuropharmacology, 1989, Volume: 28, Issue:3

    Topics: Adenosine; Adrenergic alpha-Antagonists; Aminophylline; Animals; Anticonvulsants; Clonidine; Habituation, Psychophysiologic; Methysergide; Mice; Mice, Inbred DBA; Piperoxan; Yohimbine

1989
Discriminative stimulus properties of xylazine in rat: discriminability and effects of putative alpha-2 adrenoceptor agonists and antagonists.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Discrimination Learning; Idazoxan; Lisuride; Lysergic Acid Diethylamide; Male; Piperoxan; Rats; Rats, Inbred Strains; Thiazines; Xylazine; Yohimbine

1985
Alpha-2-adrenergic control of prolactin release.
    Neuroendocrinology, 1986, Volume: 44, Issue:2

    Topics: Animals; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Female; Male; Piperoxan; Pregnancy; Prolactin; Quinolizines; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1986
Effects of clonidine on neuronal firing evoked by a noxious stimulus.
    Brain research, 1985, Feb-18, Volume: 327, Issue:1-2

    Topics: Animals; Clonidine; Electrophysiology; Isoquinolines; Male; Neurons; Norepinephrine; Pain; Physical Stimulation; Piperazines; Piperoxan; Rats; Rats, Inbred Strains; Stimulation, Chemical; Yohimbine

1985
A possible alpha 2-adrenergic component in the in vivo activity of pirenperone.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Dioxanes; Female; Idazoxan; Piperidines; Piperoxan; Postural Balance; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Reflex; Serotonin Antagonists; Tranquilizing Agents; Xylazine; Yohimbine

1984
Antagonist/agonist-preferring alpha-adrenoceptors or alpha 1/alpha 2-adrenoceptors?
    European journal of pharmacology, 1980, May-02, Volume: 63, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Clonidine; In Vitro Techniques; Male; Piperoxan; Pulmonary Artery; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Yohimbine

1980
Noradrenergic influences on sound-induced seizures.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 214, Issue:2

    Topics: Acoustic Stimulation; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Drug Interactions; Mice; Mice, Inbred DBA; Norepinephrine; Phentolamine; Piperoxan; Seizures; Yohimbine

1980
Anxiolytics antagonize yohimbine's discriminative stimulus properties.
    Psychopharmacology, 1981, Volume: 74, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Cues; Discrimination Learning; Generalization, Stimulus; Male; Piperoxan; Rats; Yohimbine

1981
alpha 2-adrenergic antagonists suppress epileptiform EEG activity in a petit mal seizure model.
    Life sciences, 1982, Jan-18, Volume: 30, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Electroencephalography; Epilepsy, Absence; Male; Mianserin; Piperoxan; Rats; Synaptic Transmission; Yohimbine

1982
Evidence for a central sympathoexcitatory action of alpha-2 adrenergic antagonists.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Brain; Cats; Denervation; Heart Rate; In Vitro Techniques; Piperoxan; Pressoreceptors; Receptors, Adrenergic, alpha; Sympathomimetics; Yohimbine

1983
Alpha 2-adrenergic receptors influence tyrosine hydroxylase activity in retinal dopamine neurons.
    Life sciences, 1983, Dec-12, Volume: 33, Issue:24

    Topics: Adaptation, Physiological; Animals; Cerebellum; Clonidine; Darkness; Dopamine; Male; Neurons; Photic Stimulation; Piperoxan; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Retina; Tyrosine 3-Monooxygenase; Yohimbine

1983
Biochemical pharmacology of paradoxical sleep.
    British journal of clinical pharmacology, 1983, Volume: 16 Suppl 2

    Topics: alpha-Methyltyrosine; Animals; Chlorpromazine; Clonidine; Humans; Hydroxydopamines; Locus Coeruleus; Membrane Fluidity; Membrane Lipids; Membrane Proteins; Methyltyrosines; Norepinephrine; Oxidopamine; Piperoxan; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Neurotransmitter; Serotonin; Sleep, REM; Synaptic Transmission; Tyrosine 3-Monooxygenase; Yohimbine

1983
Facilitation of the Bezold-Jarisch reflex by central stimulation of alpha 2 adrenoceptors in dogs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 325, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Capsaicin; Dogs; Female; Heart Rate; Male; Piperoxan; Pressoreceptors; Receptors, Adrenergic, alpha; Reflex; Respiration, Artificial; Vagus Nerve; Yohimbine

1984
Pharmacological characterization of central alpha-adrenoceptors which mediate clonidine-induced locomotor hypoactivity in the developing rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1980, Volume: 311, Issue:1

    Topics: Aging; Animals; Central Nervous System; Clonidine; Female; Male; Motor Activity; Phentolamine; Piperoxan; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Time Factors; Yohimbine

1980
The role of alpha receptors in the facilitation of the chemoreflex and inhibition of the carotid occlusion reflex by clonidine.
    Clinical and experimental hypertension, 1980, Volume: 2, Issue:6

    Topics: Animals; Blood Pressure; Carotid Arteries; Carotid Body; Clonidine; Dogs; Female; Male; Phentolamine; Piperoxan; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1980
Lack of involvement of alpha 2-adrenoceptors in the regulation of striatal dopaminergic transmission.
    European journal of pharmacology, 1983, Jan-21, Volume: 86, Issue:3-4

    Topics: Acetylcholine; Animals; Clonidine; Corpus Striatum; Dioxins; Dopamine; Idazoxan; Male; Piperoxan; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Dopamine; Yohimbine

1983
Alpha-adrenoceptors and facilitation at a sympathetic neuroeffector junction.
    Journal of autonomic pharmacology, 1984, Volume: 4, Issue:1

    Topics: Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Muscle, Smooth; Neural Conduction; Neuroeffector Junction; Piperoxan; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Yohimbine

1984
The alpha-2 antagonists idazoxan and rauwolscine but not yohimbine or piperoxan are anxiolytic in the Vogel lick-shock conflict paradigm following intravenous administration.
    Life sciences, 1994, Volume: 54, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Clonidine; Conflict, Psychological; Dioxanes; Drinking Behavior; GABA Antagonists; Idazoxan; Infusions, Intravenous; Male; Piperoxan; Rats; Rats, Sprague-Dawley; Yohimbine

1994
Agonist and antagonist actions of yohimbine as compared to fluparoxan at alpha(2)-adrenergic receptors (AR)s, serotonin (5-HT)(1A), 5-HT(1B), 5-HT(1D) and dopamine D(2) and D(3) receptors. Significance for the modulation of frontocortical monoaminergic tr
    Synapse (New York, N.Y.), 2000, Volume: 35, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Body Temperature; Frontal Lobe; Guinea Pigs; Hippocampus; Humans; Mice; Neurons; Piperoxan; Pyrroles; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Swine; Synaptic Transmission; Yohimbine

2000