Page last updated: 2024-08-17

piperoxan and prazosin

piperoxan has been researched along with prazosin in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199012 (70.59)18.7374
1990's5 (29.41)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Andrews, PR; Craik, DJ; Martin, JL1
Butler, RC; Chapleo, CB; Doxey, JC; Myers, PL; Roach, AG; Smith, CF1
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Timmermans, PB; van Zwieten, PA1
Dausse, J; Meyer, P; Miach, PJ1
Cagampang, FR; Coen, CW; Maeda, K; Ohkura, S; Ota, K; Tsukamura, H1
Fukuda, H; Mishima, A; Ono, H; Ono, S; Vasko, MR1
Fukuda, H; Ono, H; Tanabe, M1
Gupta, PP; Srivastava, AK; Srivastava, YP1
Laubie, M; Schmitt, H1
Humphrey, SJ; McCall, RB1
Batink, HD; Timmermans, PB; van Kemenade, JE; van Zwieten, PA1
Grant, SJ; Jablons, D; Maas, JW; Swann, AC1
Bentley, GA; McLennan, PL1
Abrahams, TP; Liu, W; Varner, KJ1
Bricola, A; Jurkiewicz, A; Jurkiewicz, NH1

Reviews

1 review(s) available for piperoxan and prazosin

ArticleYear
alpha 2 adrenoceptors: classification, localization, mechanisms, and targets for drugs.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:12

    Topics: Adipose Tissue; Animals; Blood Platelets; Central Nervous System; Humans; Islets of Langerhans; Melanocytes; Muscle, Smooth, Vascular; Nerve Endings; Norepinephrine; Parasympathetic Nervous System; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Serotonin; Synapses

1982

Other Studies

16 other study(ies) available for piperoxan and prazosin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
alpha-adrenoreceptor reagents. 1. Synthesis of some 1,4-benzodioxans as selective presynaptic alpha 2-adrenoreceptor antagonists and potential antidepressants.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Dioxins; Dose-Response Relationship, Drug; Idazoxan; Male; Mice; Phenylephrine; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Synapses; Vas Deferens

1983
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Direct biochemical demonstration of two types of alpha-adrenoreceptor in rat brain.
    Nature, 1978, Aug-03, Volume: 274, Issue:5670

    Topics: Animals; Binding, Competitive; Brain; Clonidine; Dihydroergotoxine; Dopamine; Male; Phenoxybenzamine; Phentolamine; Piperoxan; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synaptic Membranes; Yohimbine

1978
Alpha 2-adrenergic receptors are involved in the suppression of luteinizing hormone release during acute fasting in the ovariectomized estradiol-primed rats.
    Neuroendocrinology, 1992, Volume: 56, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Dioxanes; Estradiol; Fasting; Female; Idazoxan; Luteinizing Hormone; Ovariectomy; Piperoxan; Prazosin; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha

1992
Inhibitory effects of clonidine and tizanidine on release of substance P from slices of rat spinal cord and antagonism by alpha-adrenergic receptor antagonists.
    Neuropharmacology, 1991, Volume: 30, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Parasympatholytics; Piperoxan; Prazosin; Radioimmunoassay; Rats; Rats, Inbred Strains; Spinal Cord; Substance P; Veratridine; Yohimbine

1991
Spinal alpha 1- and alpha 2-adrenoceptors mediate facilitation and inhibition of spinal motor transmission, respectively.
    Japanese journal of pharmacology, 1990, Volume: 54, Issue:1

    Topics: Animals; Clonidine; Clorgyline; Levodopa; Male; Motor Neurons; Piperoxan; Prazosin; Premedication; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Reflex, Monosynaptic; Spinal Cord; Synaptic Transmission

1990
Characterization of alpha-adrenoceptors involved in central thermoregulation in rabbits.
    Indian journal of experimental biology, 1989, Volume: 27, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Body Temperature; Body Temperature Regulation; Female; Male; Methyldopa; Piperoxan; Prazosin; Rabbits; Receptors, Adrenergic, alpha

1989
Prazosin produces a sustained and reflex-mediated increase in renal sympathetic nerve activity in anesthetized dogs.
    European journal of pharmacology, 1988, Jun-22, Volume: 151, Issue:1

    Topics: Anesthesia; Animals; Blood Pressure; Clonidine; Denervation; Dogs; Female; Heart Rate; Infusions, Intra-Arterial; Kidney; Male; Neurons; Piperoxan; Prazosin; Pressoreceptors; Reflex; Sympathetic Nervous System; Vertebral Artery

1988
Evidence for a central depressor action of postsynaptic alpha 1-adrenergic receptor antagonists.
    Journal of the autonomic nervous system, 1981, Volume: 3, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Cats; Clonidine; Depression, Chemical; Dioxanes; Hemodynamics; Phentolamine; Piperoxan; Prazosin; Pressoreceptors; Receptors, Adrenergic; Sympathetic Nervous System

1981
Selectivity of benzodioxane alpha-adrenoceptor antagonists for alpha 1- and alpha 2-adrenoceptors determined by binding affinity.
    Pharmacology, 1983, Volume: 26, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Clonidine; In Vitro Techniques; Male; Membranes; Piperidines; Piperoxan; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha

1983
Increased ouabain binding after repeated noradrenergic stimulation.
    Brain research, 1981, Jun-01, Volume: 213, Issue:2

    Topics: 4-Nitrophenylphosphatase; Animals; Cell Membrane; Cerebral Cortex; Male; Ouabain; Phosphoric Monoester Hydrolases; Piperidines; Piperoxan; Prazosin; Protein Binding; Quinazolines; Rats

1981
Effects of prazosin and piperoxan on central cardiovascular actions of St 91 in cats.
    European journal of pharmacology, 1982, Dec-17, Volume: 86, Issue:1

    Topics: Animals; Atropine; Blood Pressure; Brain; Cats; Clonidine; Female; Heart Rate; Hemodynamics; Injections, Intra-Arterial; Injections, Intravenous; Male; Piperidines; Piperoxan; Prazosin; Quinazolines; Vertebral Artery

1982
Blockade of alpha-2 adrenergic receptors in the rostral ventrolateral medulla attenuates the sympathoinhibitory response to cocaine.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Blood Pressure; Cocaine; Idazoxan; Male; Medulla Oblongata; Microinjections; Piperoxan; Prazosin; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Sympatholytics

1996
Functional study of the excitatory alpha-adrenoceptor in guinea pig ileum, in relation to the hypothesis of an atypical receptor.
    Annals of the New York Academy of Sciences, 1997, May-30, Volume: 812

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Epinephrine; Guinea Pigs; Ileum; Indoramin; Models, Biological; Muscle Contraction; Norepinephrine; Phenylephrine; Piperoxan; Prazosin; Receptors, Adrenergic, alpha

1997